Interactions of recombinant human histamine H 1, H 2, H 3, and H 4 receptors with 34 antidepressants and antipsychotics

Naunyn-Schmiedeberg's Archives of Pharmacology

Volumn 385, Issue 2, 2012, Pages 145-170

  Appl, Heidrun ^a   Holzammer, Tobias ^a   Dove, Stefan ^a   Haen, Ekkehard ^a   Straer, Andrea ^a   Seifert, Roland ^b  

^a UNIVERSITY OF REGENSBURG   (Germany)

^b HANNOVER MEDICAL SCHOOL   (Germany)

Author keywords

Antidepressants; Antipsychotics; Clozapine; Histamine receptors; Therapeutic reference range; Trimipramine

Indexed keywords

AMITRIPTYLINE; ANTIDEPRESSANT AGENT; ASTEMIZOLE; CHLORPROMAZINE; CHLORPROTHIXENE; CLOMIPRAMINE; CLOZAPINE; CYPROHEPTADINE; DESIPRAMINE; DEXCHLORPHENIRAMINE; DIBENZEPIN; DIPHENHYDRAMINE; DOXEPIN; FLUPHENAZINE; HISTAMINE H1 RECEPTOR; HISTAMINE H2 RECEPTOR; HISTAMINE H3 RECEPTOR; HISTAMINE H4 RECEPTOR; IMIPRAMINE; KETOTIFEN; LEVOMEPROMAZINE; LOFEPRAMINE; LOXAPINE; MAPROTILINE; MEPYRAMINE; MIANSERIN; NEUROLEPTIC AGENT; TRIMIPRAMINE; TRIPROLIDINE; UNINDEXED DRUG;

AGRANULOCYTOSIS; ANIMAL CELL; ANIMAL TISSUE; ARTICLE; BINDING AFFINITY; BINDING COMPETITION; DISSOCIATION CONSTANT; DRUG ANTAGONISM; DRUG EFFICACY; DRUG POTENCY; DRUG RECEPTOR BINDING; ENZYME ASSAY; HUMAN; INSECT CELL; LIGAND BINDING; MOLECULAR DOCKING; NEUTROPENIA; NONHUMAN; STEADY STATE;

ANTIDEPRESSIVE AGENTS; ANTIPSYCHOTIC AGENTS; BINDING, COMPETITIVE; HISTAMINE AGONISTS; HISTAMINE ANTAGONISTS; HUMANS; MODELS, MOLECULAR; PROTEIN BINDING; RADIOLIGAND ASSAY; RECEPTORS, HISTAMINE; RECOMBINANT PROTEINS;

EID: 84857030583     PISSN: 00281298     EISSN: 14321912     Source Type: Journal    
DOI: 10.1007/s00210-011-0704-0     Document Type: Article

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