Mutational analysis of the antagonist-binding site of the histamine H1 receptor

Journal of Biological Chemistry

Volumn 274, Issue 42, 1999, Pages 29994-30000

  Wieland, Kerstin ^a   Ter Laak, Anton M ^b   Smit, Martine J ^a   Kühne, Ronald ^b   Timmerman, Henk ^a   Leurs, Rob ^a  

^a VU UNIVERSITY AMSTERDAM   (Netherlands)

^b LEIBNIZ INSTITUT FÜR MOLEKULARE PHARMAKOLOGIE   (Germany)

Author keywords

[No Author keywords available]

Indexed keywords

ACRIVASTINE; AMINO ACID; CARBOXYLIC ACID DERIVATIVE; CETIRIZINE; HISTAMINE H1 RECEPTOR; HISTAMINE H1 RECEPTOR ANTAGONIST; MECLOZINE; TRIPROLIDINE;

ANIMAL CELL; ARTICLE; BINDING AFFINITY; BINDING SITE; CERCOPITHECIDAE; HUMAN; HUMAN CELL; MUTATION; NONHUMAN; PHARMACOPHORE; PRIORITY JOURNAL; RECEPTOR BINDING; SITE DIRECTED MUTAGENESIS;

ANIMALS; CELL LINE; CELL MEMBRANE; CETIRIZINE; GUINEA PIGS; HISTAMINE; HISTAMINE H1 ANTAGONISTS; HUMANS; INOSITOL PHOSPHATES; LIGANDS; LYSINE; MODELS, MOLECULAR; MUTAGENESIS, SITE-DIRECTED; RECEPTORS, HISTAMINE H1; TRIPROLIDINE;

ANIMALIA; CERCOPITHECIDAE;

EID: 0033569709     PISSN: 00219258     EISSN: None     Source Type: Journal    
DOI: 10.1074/jbc.274.42.29994     Document Type: Article

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