Pharmacological profile of histaprodifens at four recombinant histamine H1 receptor species isoforms

Journal of Pharmacology and Experimental Therapeutics

Volumn 324, Issue 1, 2008, Pages 60-71

  Straßer, Andrea ^a   Striegl, Birgit ^a   Wittmann, Hans Joachim ^a   Seifert, Roland ^a  

^a UNIVERSITY OF REGENSBURG   (Germany)

Author keywords

[No Author keywords available]

Indexed keywords

ASPARTIC ACID; COMPLEMENTARY DNA; GLUTAMIC ACID; GUANOSINE TRIPHOSPHATASE; HISTAMINE H1 RECEPTOR; HISTAPRODIFEN DERIVATIVE; ISOPROTEIN; LYSINE; MEPYRAMINE; PHENYL GROUP; PHENYLHISTAMINE DERIVATIVE; RGS4 PROTEIN; SERINE; TYROSINE; UNCLASSIFIED DRUG;

ANIMAL CELL; ANIMAL EXPERIMENT; ANIMAL MODEL; ANIMAL TISSUE; ARTICLE; BINDING AFFINITY; BINDING SITE; CHIRALITY; CONTROLLED STUDY; DIMERIZATION; DRUG POTENCY; DRUG RECEPTOR BINDING; ELECTRICITY; GUINEA PIG; HISTAMINE RELEASE; HYDROGEN BOND; MOLECULAR DYNAMICS; NONHUMAN; NUCLEOTIDE SEQUENCE; PRIORITY JOURNAL; PROTEIN INTERACTION; SIMULATION; SPECIES DIFFERENCE; STRUCTURAL HOMOLOGY;

AMINO ACID SEQUENCE; ANIMALS; BINDING, COMPETITIVE; CATTLE; CLONING, MOLECULAR; GTP PHOSPHOHYDROLASES; GUINEA PIGS; HISTAMINE; HISTAMINE AGONISTS; HISTAMINE H1 ANTAGONISTS; HUMANS; MOLECULAR SEQUENCE DATA; PHYLOGENY; PYRILAMINE; RATS; RECEPTORS, HISTAMINE H1; RECOMBINANT PROTEINS; SEQUENCE ALIGNMENT;

EID: 37349122184     PISSN: 00223565     EISSN: 15210103     Source Type: Journal    
DOI: 10.1124/jpet.107.129601     Document Type: Article

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