RX 821002 as a tool for physiological investigation of α2-adrenoceptors

CNS Drug Reviews

Volumn 8, Issue 2, 2002, Pages 177-192

  Clarke, R W ^a,b   Harris, J ^a  

^a UNIVERSITY OF NOTTINGHAM   (United Kingdom)

^b Alcocer School of Biosciences Sutton Bonington Campus   (United Kingdom)

Author keywords

5 HT1A receptor; Imidazoline receptor; Nociceptive processing; RX 821002; Spinal cord; 2 Adrenoceptors

Indexed keywords

1,3,4,5',6,6',7,12B OCTAHYDRO 1',3' DIMETHYL 2H SPIRO[BENZO[B]FURO[2,3 A]QUINOLIZINE 2,4' PYRIMIDINE] 2' ONE; 12 ETHYLSULFONYL 5,8,8A,9,10,11,12,12A,13,13A DECAHYDRO 3 METHOXY 6H ISOQUINO[2,1 G][1,6]NAPHTHYRIDINE; 2 (2 ETHOXY 1,4 BENZODIOXAN 2 YL) 2 IMIDAZOLINE; 2 (2 METHOXY 1,4 BENZODIOXAN 2 YL) 2 IMIDAZOLINE; 2 [(2 DIMETHYLAMINO 2 METHYLPROPYL)THIO] 3 PHENYLQUINOLINE; ALPHA 2 ADRENERGIC RECEPTOR; ALPHA 2 ADRENERGIC RECEPTOR BLOCKING AGENT; ALPHA 2A ADRENERGIC RECEPTOR; ATIPAMEZOLE; BRIMONIDINE; FENTANYL; IDAZOXAN; IMIDAZOLINE RECEPTOR; MU OPIATE RECEPTOR AGONIST; N [2 [4 (2 METHOXYPHENYL) 1 PIPERAZINYL]ETHYL] N (2 PYRIDYL)CYCLOHEXANECARBOXAMIDE; NORADRENALIN; PRAZOSIN; RAUWOLSCINE; RECEPTOR SUBTYPE; SEROTONIN 1A ANTAGONIST; SEROTONIN 1A RECEPTOR; SEROTONIN 2 ANTAGONIST; UNCLASSIFIED DRUG; YOHIMBINE; 2-METHOXYIDAZOXAN; ALPHA ADRENERGIC RECEPTOR BLOCKING AGENT; ALPHA ADRENERGIC RECEPTOR STIMULATING AGENT; DRUG DERIVATIVE; DRUG RECEPTOR; IMIDAZOLINE RECEPTORS; SEROTONIN 1 RECEPTOR; SEROTONIN RECEPTOR;

BRAIN; CELL CULTURE; DRINKING BEHAVIOR; DRUG ANTAGONISM; DRUG BINDING SITE; DRUG DISTRIBUTION; DRUG ELIMINATION; DRUG RECEPTOR BINDING; DRUG SELECTIVITY; FRONTAL CORTEX; HUMAN; NERVE CELL INHIBITION; NOCICEPTION; NONHUMAN; NORADRENALIN RELEASE; PREGANGLIONIC NERVE CELL; RECEPTOR AFFINITY; REVIEW; SPINAL CORD; WITHDRAWAL REFLEX; ANIMAL; ANIMAL BEHAVIOR; DRUG EFFECT; METABOLISM; PAIN ASSESSMENT; PHYSIOLOGY; RABBIT; RAT;

ADRENERGIC ALPHA-AGONISTS; ADRENERGIC ALPHA-ANTAGONISTS; ANIMALS; BEHAVIOR, ANIMAL; BRAIN; IDAZOXAN; NOREPINEPHRINE; PAIN MEASUREMENT; RABBITS; RATS; RECEPTORS, ADRENERGIC, ALPHA-2; RECEPTORS, DRUG; RECEPTORS, SEROTONIN; RECEPTORS, SEROTONIN, 5-HT1; SPINAL CORD;

EID: 0036023388     PISSN: 1080563X     EISSN: None     Source Type: Journal    
DOI: 10.1111/j.1527-3458.2002.tb00222.x     Document Type: Review

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