[3H]RS79948-197 binding to human, rat, guinea pig and pig α(2A)-, α(2B)- and α(2C)-adrenoceptors. Comparison with MK912, RX821002, rauwolscine and yohimbine

European Journal of Pharmacology

Volumn 343, Issue 1, 1998, Pages 93-101

  Uhlén, Staffan ^a   Dambrova, Maija ^a   Näsman, Johnny ^b   Schiöth, Helgi B ^a   Gu, Yuchen ^a   Wikberg Matsson, Anna ^a   Wikberg, Jarl E S ^a  

^a UPPSALA UNIVERSITY   (Sweden)

^b UPPSALA UNIVERSITY   (Sweden)

Author keywords

3H RS79948 197; Adrenoceptor, subtype; MK912

Indexed keywords

1,3,4,5',6,6',7,12B OCTAHYDRO 1',3' DIMETHYL 2H SPIRO[BENZO[B]FURO[2,3 A]QUINOLIZINE 2,4' PYRIMIDINE] 2' ONE; 12 ETHYLSULFONYL 5,8,8A,9,10,11,12,12A,13,13A DECAHYDRO 3 METHOXY 6H ISOQUINO[2,1 G][1,6]NAPHTHYRIDINE; 2 (1 METHYL 2 ISOINDOLINYLMETHYL) 2 IMIDAZOLINE; 2 (2 METHOXY 1,4 BENZODIOXAN 2 YL) 2 IMIDAZOLINE; ALPHA 2 ADRENERGIC RECEPTOR BLOCKING AGENT; ALPHA 2A ADRENERGIC RECEPTOR; ALPHA 2B ADRENERGIC RECEPTOR; ALPHA 2C ADRENERGIC RECEPTOR; RADIOLIGAND; RAUWOLSCINE; UNCLASSIFIED DRUG; YOHIMBINE; 2-METHOXYIDAZOXAN; ADRENERGIC RECEPTOR ALPHA 2B; ADRENERGIC RECEPTOR ALPHA(2C); ADRENERGIC RECEPTOR ALPHA-2B; ADRENERGIC RECEPTOR STIMULATING AGENT; ALPHA 2 ADRENERGIC RECEPTOR; DRUG DERIVATIVE; IDAZOXAN; ISOQUINOLINE DERIVATIVE; NAPHTHYRIDINE DERIVATIVE; QUINOLIZINE DERIVATIVE; RECEPTOR, ADRENERGIC, ALPHA 2A; RECEPTOR, ADRENERGIC, ALPHA-2A;

ANIMAL CELL; ANIMAL TISSUE; ARTICLE; CONTROLLED STUDY; CORPUS STRIATUM; DRUG RECEPTOR BINDING; DRUG SELECTIVITY; GUINEA PIG; HUMAN; INSECT; KIDNEY; LIGAND BINDING; NONHUMAN; PRIORITY JOURNAL; RAT; SPLEEN; ANIMAL; COMPARATIVE STUDY; METABOLISM; SWINE;

ADRENERGIC AGENTS; ANIMALS; GUINEA PIGS; HUMANS; IDAZOXAN; ISOQUINOLINES; NAPHTHYRIDINES; QUINOLIZINES; RATS; RECEPTORS, ADRENERGIC, ALPHA-2; SWINE; YOHIMBINE;

EID: 0032484715     PISSN: 00142999     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0014-2999(97)01521-5     Document Type: Article

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