-
1
-
-
0023554261
-
The peripheral-type benzodiazepine receptor: a protein of mitochondrial outer membranes utilizing porphyrins as endogenous ligands
-
Oct
-
S.H.Snyder, A.Verma, R.R.Trifiletti The peripheral-type benzodiazepine receptor:a protein of mitochondrial outer membranes utilizing porphyrins as endogenous ligands. Faseb J. 1987 Oct;1(4):282–288.
-
(1987)
Faseb J
, vol.1
, Issue.4
, pp. 282-288
-
-
Snyder, S.H.1
Verma, A.2
Trifiletti, R.R.3
-
2
-
-
33746035655
-
Translocator protein (18kDa): new nomenclature for the peripheral-type benzodiazepine receptor based on its structure and molecular function
-
Aug
-
V.Papadopoulos, M.Baraldi, T.R.Guilarte, et al. Translocator protein (18kDa):new nomenclature for the peripheral-type benzodiazepine receptor based on its structure and molecular function. Trends Pharmacol Sci. 2006 Aug;27(8):402–409.
-
(2006)
Trends Pharmacol Sci
, vol.27
, Issue.8
, pp. 402-409
-
-
Papadopoulos, V.1
Baraldi, M.2
Guilarte, T.R.3
-
3
-
-
0017730392
-
High-densities of benzodiazepine receptors in human cortical areas
-
C.Braestrup, R.Albrechtsen, R.F.Squires. High-densities of benzodiazepine receptors in human cortical areas. Nature. 1977;269(5630):702–704.
-
(1977)
Nature
, vol.269
, Issue.5630
, pp. 702-704
-
-
Braestrup, C.1
Albrechtsen, R.2
Squires, R.F.3
-
4
-
-
0000114680
-
Specific benzodiazepine receptors in rat brain characterized by high-affinity (3H)diazepam binding
-
C.Braestrup, R.F.Squires. Specific benzodiazepine receptors in rat brain characterized by high-affinity (3H)diazepam binding. Proc Natl Acad Sci U S A. 1977;74(9):3805–3809.
-
(1977)
Proc Natl Acad Sci U S A
, vol.74
, Issue.9
, pp. 3805-3809
-
-
Braestrup, C.1
Squires, R.F.2
-
5
-
-
20844451376
-
Peripheral-type benzodiazepine receptor-mediated action of steroidogenic acute regulatory protein on cholesterol entry into Leydig cell mitochondria
-
Feb
-
T.Hauet, Z.-X.Yao, H.S.Bose, et al. Peripheral-type benzodiazepine receptor-mediated action of steroidogenic acute regulatory protein on cholesterol entry into Leydig cell mitochondria. Mol Endocrinol. 2005 Feb;19(2):540–554.
-
(2005)
Mol Endocrinol
, vol.19
, Issue.2
, pp. 540-554
-
-
Hauet, T.1
Yao, Z.-X.2
Bose, H.S.3
-
6
-
-
84860279460
-
The role of 18 kDa mitochondrial translocator protein (TSPO) in programmed cell death, and effects of steroids on TSPO expression
-
May
-
L.Veenman, M.Gavish. The role of 18 kDa mitochondrial translocator protein (TSPO) in programmed cell death, and effects of steroids on TSPO expression. Curr Mol Med. 2012 May;12(4):398–412.
-
(2012)
Curr Mol Med
, vol.12
, Issue.4
, pp. 398-412
-
-
Veenman, L.1
Gavish, M.2
-
7
-
-
0032707529
-
Enigma of the peripheral benzodiazepine receptor
-
Dec
-
M.Gavish, I.Bachman, R.Shoukrun, et al. Enigma of the peripheral benzodiazepine receptor. Pharmacol Rev. 1999 Dec;51(4):629–650.
-
(1999)
Pharmacol Rev
, vol.51
, Issue.4
, pp. 629-650
-
-
Gavish, M.1
Bachman, I.2
Shoukrun, R.3
-
8
-
-
0024590270
-
Effects of peripheral benzodiazepines upon the O2 consumption of neuro-blastoma cells
-
Feb
-
J.C.Larcher, J.L.Vayssiere, F.J.Lemarquer, et al. Effects of peripheral benzodiazepines upon the O2 consumption of neuro-blastoma cells. Eur J Pharmacol. 1989 Feb 28;161(2–3):197–202.
-
(1989)
Eur J Pharmacol
, vol.161
, Issue.2-3
, pp. 197-202
-
-
Larcher, J.C.1
Vayssiere, J.L.2
Lemarquer, F.J.3
-
9
-
-
67649613018
-
Effect of peripheral benzodiazepine receptor (PBR/TSPO) ligands on opening of Ca2+-induced pore and phosphorylation of 3.5-kDa polypeptide in rat brain mitochondria
-
Apr
-
O.V.Krestinina, D.E.Grachev, I.V.Odinokova, et al. Effect of peripheral benzodiazepine receptor (PBR/TSPO) ligands on opening of Ca2+-induced pore and phosphorylation of 3.5-kDa polypeptide in rat brain mitochondria. Biochemistry-Moscow+. 2009 Apr;74(4):421–429.
-
(2009)
Biochemistry-Moscow+
, vol.74
, Issue.4
, pp. 421-429
-
-
Krestinina, O.V.1
Grachev, D.E.2
Odinokova, I.V.3
-
10
-
-
84923241444
-
Positron emission tomography and functional characterization of a complete PBR/TSPO knockout
-
R.B.Banati, R.J.Middleton, R.Chan, et al. Positron emission tomography and functional characterization of a complete PBR/TSPO knockout. Nat Commun. 2014;5:5452.
-
(2014)
Nat Commun
, vol.5
, pp. 5452
-
-
Banati, R.B.1
Middleton, R.J.2
Chan, R.3
-
11
-
-
84892892196
-
The role of allopregnanolone in depression and anxiety
-
Feb
-
C.Schüle, C.Nothdurfter, R.Rupprecht. The role of allopregnanolone in depression and anxiety. Prog Neurobiol. 2014 Feb;113:79–87.
-
(2014)
Prog Neurobiol
, vol.113
, pp. 79-87
-
-
Schüle, C.1
Nothdurfter, C.2
Rupprecht, R.3
-
12
-
-
84924173806
-
Enhancing neurosteroid synthesis–relationship to the pharmacology of translocator protein (18 kDa) (TSPO) ligands and benzodiazepines
-
Mar
-
L.Wolf, A.Bauer, D.Melchner, et al. Enhancing neurosteroid synthesis–relationship to the pharmacology of translocator protein (18 kDa) (TSPO) ligands and benzodiazepines. Pharmacopsychiatry. 2015 Mar;48(2):72–77.
-
(2015)
Pharmacopsychiatry
, vol.48
, Issue.2
, pp. 72-77
-
-
Wolf, L.1
Bauer, A.2
Melchner, D.3
-
13
-
-
84907293074
-
Peripheral benzodiazepine receptor/translocator protein global knock-out mice are viable with no effects on steroid hormone biosynthesis
-
Oct
-
L.N.Tu, K.Morohaku, P.R.Manna, et al. Peripheral benzodiazepine receptor/translocator protein global knock-out mice are viable with no effects on steroid hormone biosynthesis. J Biol Chem. 2014 Oct 3;289(40):27444–27454.
-
(2014)
J Biol Chem
, vol.289
, Issue.40
, pp. 27444-27454
-
-
Tu, L.N.1
Morohaku, K.2
Manna, P.R.3
-
14
-
-
84931274608
-
Conditional steroidogenic cell-targeted deletion of TSPO unveils a crucial role in viability and hormone-dependent steroid formation
-
Jun
-
J.Fan, E.Campioli, A.Midzak, et al. Conditional steroidogenic cell-targeted deletion of TSPO unveils a crucial role in viability and hormone-dependent steroid formation. Proc Natl Acad Sci U S A. 2015 Jun 9;112(23):7261–7266.
-
(2015)
Proc Natl Acad Sci U S A
, vol.112
, Issue.23
, pp. 7261-7266
-
-
Fan, J.1
Campioli, E.2
Midzak, A.3
-
15
-
-
0026538576
-
The mitochondrial benzodiazepine receptor: evidence for association with the voltage-dependent anion channel (VDAC)
-
Feb
-
M.W.McEnery. The mitochondrial benzodiazepine receptor:evidence for association with the voltage-dependent anion channel (VDAC). J Bioenerg Biomembr. 1992 Feb;24(1):63–69.
-
(1992)
J Bioenerg Biomembr
, vol.24
, Issue.1
, pp. 63-69
-
-
McEnery, M.W.1
-
16
-
-
84934907493
-
Parkin-mediated responses against infection and wound involve TSPO-VDAC complex in Drosophila
-
Jul
-
J.H.Cho, J.H.Park, C.G.Chung, et al. Parkin-mediated responses against infection and wound involve TSPO-VDAC complex in Drosophila. Biochem Biophys Res Commun. 2015 Jul 17–24;463(1–2):1–6.
-
(2015)
Biochem Biophys Res Commun
, vol.463
, Issue.1-2
, pp. 1-6
-
-
Cho, J.H.1
Park, J.H.2
Chung, C.G.3
-
17
-
-
84865682758
-
The mitochondrial permeability transition pore (PTP) - an example of multiple molecular exaptation?
-
Nov
-
A.Vianello, V.Casolo, E.Petrussa, et al. The mitochondrial permeability transition pore (PTP) - an example of multiple molecular exaptation? Biochim Biophys Acta. 2012 Nov;1817(11):2072–2086.
-
(2012)
Biochim Biophys Acta
, vol.1817
, Issue.11
, pp. 2072-2086
-
-
Vianello, A.1
Casolo, V.2
Petrussa, E.3
-
18
-
-
67349117275
-
What is the mitochondrial permeability transition pore?
-
Jun
-
A.P.Halestrap. What is the mitochondrial permeability transition pore? J Mol Cell Cardiol. 2009 Jun;46(6):821–831.
-
(2009)
J Mol Cell Cardiol
, vol.46
, Issue.6
, pp. 821-831
-
-
Halestrap, A.P.1
-
19
-
-
84901008605
-
Regulation of the mitochondrial permeability transition pore by the outer membrane does not involve the peripheral benzodiazepine receptor (translocator protein of 18 kDa (TSPO))
-
May
-
J.Šileikytė, E.Blachly-Dyson, R.Sewell, et al. Regulation of the mitochondrial permeability transition pore by the outer membrane does not involve the peripheral benzodiazepine receptor (translocator protein of 18 kDa (TSPO)). J Biol Chem. 2014 May 16;289(20):13769–13781.
-
(2014)
J Biol Chem
, vol.289
, Issue.20
, pp. 13769-13781
-
-
Šileikytė, J.1
Blachly-Dyson, E.2
Sewell, R.3
-
20
-
-
77955415606
-
Regulation of translocator protein 18 kDa (TSPO) expression in health and disease states
-
Oct
-
A.Batarseh, V.Papadopoulos. Regulation of translocator protein 18 kDa (TSPO) expression in health and disease states. Mol Cell Endocrinol. 2010 Oct 7;327(1–2):1–12.
-
(2010)
Mol Cell Endocrinol
, vol.327
, Issue.1-2
, pp. 1-12
-
-
Batarseh, A.1
Papadopoulos, V.2
-
21
-
-
34548238745
-
Channel-like functions of the 18-kDa translocator protein (TSPO): regulation of apoptosis and steroidogenesis as part of the host-defense response
-
L.Veenman, V.Papadopoulos, M.Gavish. Channel-like functions of the 18-kDa translocator protein (TSPO):regulation of apoptosis and steroidogenesis as part of the host-defense response. Curr Pharm Des. 2007;13(23):2385–2405.
-
(2007)
Curr Pharm Des
, vol.13
, Issue.23
, pp. 2385-2405
-
-
Veenman, L.1
Papadopoulos, V.2
Gavish, M.3
-
22
-
-
52449115923
-
VDAC activation by the 18 kDa translocator protein (TSPO), implications for apoptosis
-
Jun
-
L.Veenman, Y.Shandalov, M.Gavish. VDAC activation by the 18 kDa translocator protein (TSPO), implications for apoptosis. J Bioenerg Biomembr. 2008 Jun;40(3):199–205.
-
(2008)
J Bioenerg Biomembr
, vol.40
, Issue.3
, pp. 199-205
-
-
Veenman, L.1
Shandalov, Y.2
Gavish, M.3
-
23
-
-
84892174249
-
Translocator protein (18 kDa) (TSPO) is expressed in reactive retinal microglia and modulates microglial inflammation and phagocytosis
-
M.Karlstetter, C.Nothdurfter, A.Aslanidis, et al. Translocator protein (18 kDa) (TSPO) is expressed in reactive retinal microglia and modulates microglial inflammation and phagocytosis. J Neuroinflammation. 2014;11:3.
-
(2014)
J Neuroinflammation
, vol.11
, pp. 3
-
-
Karlstetter, M.1
Nothdurfter, C.2
Aslanidis, A.3
-
24
-
-
84896333770
-
The translocator protein as a drug target in Alzheimer’s disease
-
Apr
-
S.W.Chua, M.Kassiou, L.M.Ittner. The translocator protein as a drug target in Alzheimer’s disease. Expert Rev Neurother. 2014 Apr;14(4):439–448.• This article highlighted TSPO as a promising drug target for AD.
-
(2014)
Expert Rev Neurother
, vol.14
, Issue.4
, pp. 439-448
-
-
Chua, S.W.1
Kassiou, M.2
Ittner, L.M.3
-
25
-
-
84971650049
-
TSPO as a target for treatments of diseases, including neuropathological disorders
-
L.Veenman, A.Vainshtein, M.Gavish. TSPO as a target for treatments of diseases, including neuropathological disorders. Cell Death Dis. 2015;6:e1911.
-
(2015)
Cell Death Dis
, vol.6
, pp. e1911
-
-
Veenman, L.1
Vainshtein, A.2
Gavish, M.3
-
26
-
-
28944443373
-
Extragonadal synthesis of estradiol is protective against kainic acid excitotoxic damage to the hippocampus
-
Sep
-
S.Veiga, I.Azcoitia, L.M.Garcia-Segura. Extragonadal synthesis of estradiol is protective against kainic acid excitotoxic damage to the hippocampus. Neuroreport. 2005 Sep 28;16(14):1599–1603.
-
(2005)
Neuroreport
, vol.16
, Issue.14
, pp. 1599-1603
-
-
Veiga, S.1
Azcoitia, I.2
Garcia-Segura, L.M.3
-
27
-
-
78649687576
-
Translocator protein (18 kDa) (TSPO) as a therapeutic target for neurological and psychiatric disorders
-
Dec
-
R.Rupprecht, V.Papadopoulos, G.Rammes, et al. Translocator protein (18 kDa) (TSPO) as a therapeutic target for neurological and psychiatric disorders. Nat Rev Drug Discov. 2010 Dec;9(12):971–988.•• This review provides a summary of TSPO function.
-
(2010)
Nat Rev Drug Discov
, vol.9
, Issue.12
, pp. 971-988
-
-
Rupprecht, R.1
Papadopoulos, V.2
Rammes, G.3
-
28
-
-
84896998596
-
Structure of the mitochondrial translocator protein in complex with a diagnostic ligand
-
Mar
-
L.Jaremko, M.Jaremko, K.Giller, et al. Structure of the mitochondrial translocator protein in complex with a diagnostic ligand. Science. 2014 Mar 21;343(6177):1363–1366.
-
(2014)
Science
, vol.343
, Issue.6177
, pp. 1363-1366
-
-
Jaremko, L.1
Jaremko, M.2
Giller, K.3
-
29
-
-
84946027944
-
Conformational flexibility in the transmembrane protein TSPO
-
Nov
-
Ł.Jaremko, M.Jaremko, K.Giller, et al. Conformational flexibility in the transmembrane protein TSPO. Chemistry. 2015 Nov 9;21(46):16555–16563.
-
(2015)
Chemistry
, vol.21
, Issue.46
, pp. 16555-16563
-
-
Jaremko, Ł.1
Jaremko, M.2
Giller, K.3
-
30
-
-
84921829870
-
Crystal structures of translocator protein (TSPO) and mutant mimic of a human polymorphism
-
Jan
-
F.Li, J.Liu, Y.Zheng, et al. Crystal structures of translocator protein (TSPO) and mutant mimic of a human polymorphism. Science. 2015 Jan 30;347(6221):555–558.
-
(2015)
Science
, vol.347
, Issue.6221
, pp. 555-558
-
-
Li, F.1
Liu, J.2
Zheng, Y.3
-
31
-
-
77953560009
-
Three-dimensional structure of TspO by electron cryomicroscopy of helical crystals
-
Jun
-
V.M.Korkhov, C.Sachse, J.M.Short, et al. Three-dimensional structure of TspO by electron cryomicroscopy of helical crystals. Structure. 2010 Jun 9;18(6):677–687.
-
(2010)
Structure
, vol.18
, Issue.6
, pp. 677-687
-
-
Korkhov, V.M.1
Sachse, C.2
Short, J.M.3
-
32
-
-
84921931701
-
Protein structure. Structure and activity of tryptophan-rich TSPO proteins
-
Jan
-
Y.Z.Guo, R.C.Kalathur, Q.Liu, et al. Protein structure. Structure and activity of tryptophan-rich TSPO proteins. Science. 2015 Jan 30;347(6221):551–555.
-
(2015)
Science
, vol.347
, Issue.6221
, pp. 551-555
-
-
Guo, Y.Z.1
Kalathur, R.C.2
Liu, Q.3
-
33
-
-
0031755752
-
Peripheral-type benzodiazepine receptor function in cholesterol transport. Identification of a putative cholesterol recognition/interaction amino acid sequence and consensus pattern
-
Dec
-
H.Li, V.Papadopoulos. Peripheral-type benzodiazepine receptor function in cholesterol transport. Identification of a putative cholesterol recognition/interaction amino acid sequence and consensus pattern. Endocrinology. 1998 Dec;139(12):4991–4997.
-
(1998)
Endocrinology
, vol.139
, Issue.12
, pp. 4991-4997
-
-
Li, H.1
Papadopoulos, V.2
-
34
-
-
59649098348
-
PET imaging of the peripheral benzodiazepine receptor: monitoring disease progression and therapy response in neurodegenerative disorders
-
J.Doorduin, E.F.J.de Vries, R.A.Dierckx, et al. PET imaging of the peripheral benzodiazepine receptor:monitoring disease progression and therapy response in neurodegenerative disorders. Curr Pharm Des. 2008;14(31):3297–3315.
-
(2008)
Curr Pharm Des
, vol.14
, Issue.31
, pp. 3297-3315
-
-
Doorduin, J.1
de Vries, E.F.J.2
Dierckx, R.A.3
-
35
-
-
0027238911
-
Radioligands for PET studies of central benzodiazepine receptors and PK (peripheral benzodiazepine) binding sites–current status
-
May
-
V.W.Pike, C.Halldin, C.Crouzel, et al. Radioligands for PET studies of central benzodiazepine receptors and PK (peripheral benzodiazepine) binding sites–current status. Nucl Med Biol. 1993 May;20(4):503–525.
-
(1993)
Nucl Med Biol
, vol.20
, Issue.4
, pp. 503-525
-
-
Pike, V.W.1
Halldin, C.2
Crouzel, C.3
-
36
-
-
0036355229
-
The concept of in vivo imaging of neuroinflammation with [11C](R)-PK11195 PET
-
A.Cagnin, A.Gerhard, R.B.Banati. The concept of in vivo imaging of neuroinflammation with [11C](R)-PK11195 PET. Ernst Schering Res Found Workshop. 2002;39:179–191.
-
(2002)
Ernst Schering Res Found Workshop
, Issue.39
, pp. 179-191
-
-
Cagnin, A.1
Gerhard, A.2
Banati, R.B.3
-
37
-
-
36249003354
-
Neuroinflammation in the pathophysiology of Parkinson’s disease: evidence from animal models to human in vivo studies with [11C]-PK11195 PET
-
Oct
-
A.L.Bartels, K.L.Leenders. Neuroinflammation in the pathophysiology of Parkinson’s disease:evidence from animal models to human in vivo studies with [11C]-PK11195 PET. Mov Disord. 2007 Oct 15;22(13):1852–1856.
-
(2007)
Mov Disord
, vol.22
, Issue.13
, pp. 1852-1856
-
-
Bartels, A.L.1
Leenders, K.L.2
-
38
-
-
10744230035
-
Evaluation of three quinoline-carboxamide derivatives as potential radioligands for the in vivo pet imaging of neurodegeneration
-
May
-
S.Belloli, R.M.Moresco, M.Matarrese, et al. Evaluation of three quinoline-carboxamide derivatives as potential radioligands for the in vivo pet imaging of neurodegeneration. Neurochem Int. 2004 May;44(6):433–440.
-
(2004)
Neurochem Int
, vol.44
, Issue.6
, pp. 433-440
-
-
Belloli, S.1
Moresco, R.M.2
Matarrese, M.3
-
39
-
-
25144465870
-
Ro5-4864, a synthetic ligand of peripheral benzodiazepine receptor, reduces aging-associated myelin degeneration in the sciatic nerve of male rats
-
Nov
-
E.Leonelli, J.G.Yague, M.Ballabio, et al. Ro5-4864, a synthetic ligand of peripheral benzodiazepine receptor, reduces aging-associated myelin degeneration in the sciatic nerve of male rats. Mech Ageing Dev. 2005 Nov;126(11):1159–1163.
-
(2005)
Mech Ageing Dev
, vol.126
, Issue.11
, pp. 1159-1163
-
-
Leonelli, E.1
Yague, J.G.2
Ballabio, M.3
-
40
-
-
84877753769
-
Ligand for translocator protein reverses pathology in a mouse model of Alzheimer’s disease
-
May
-
A.M.Barron, L.M.Garcia-Segura, D.Caruso, et al. Ligand for translocator protein reverses pathology in a mouse model of Alzheimer’s disease. J Neurosci. 2013 May 15;33(20):8891–8897.
-
(2013)
J Neurosci
, vol.33
, Issue.20
, pp. 8891-8897
-
-
Barron, A.M.1
Garcia-Segura, L.M.2
Caruso, D.3
-
41
-
-
4143123246
-
Antianxiety and antidepressant-like effects of AC-5216, a novel mitochondrial benzodiazepine receptor ligand
-
Aug
-
A.Kita, H.Kohayakawa, T.Kinoshita, et al. Antianxiety and antidepressant-like effects of AC-5216, a novel mitochondrial benzodiazepine receptor ligand. Br J Pharmacol. 2004 Aug;142(7):1059–1072.
-
(2004)
Br J Pharmacol
, vol.142
, Issue.7
, pp. 1059-1072
-
-
Kita, A.1
Kohayakawa, H.2
Kinoshita, T.3
-
42
-
-
52449100136
-
Anxiolytic-like effects of N,N-dialkyl-2-phenylindol-3-ylglyoxylamides by modulation of translocator protein promoting neurosteroid biosynthesis
-
Sep
-
F.Da Settimo, F.Simorini, S.Taliani, et al. Anxiolytic-like effects of N,N-dialkyl-2-phenylindol-3-ylglyoxylamides by modulation of translocator protein promoting neurosteroid biosynthesis. J Med Chem. 2008 Sep 25;51(18):5798–5806.
-
(2008)
J Med Chem
, vol.51
, Issue.18
, pp. 5798-5806
-
-
Da Settimo, F.1
Simorini, F.2
Taliani, S.3
-
43
-
-
67651117272
-
Translocator protein (18 kD) as target for anxiolytics without benzodiazepine-like side effects
-
Jul
-
R.Rupprecht, G.Rammes, D.Eser, et al. Translocator protein (18 kD) as target for anxiolytics without benzodiazepine-like side effects. Science. 2009 Jul 24;325(5939):490–493.
-
(2009)
Science
, vol.325
, Issue.5939
, pp. 490-493
-
-
Rupprecht, R.1
Rammes, G.2
Eser, D.3
-
44
-
-
67650075027
-
Quantitative analysis of peripheral benzodiazepine receptor in the human brain using PET with (11)C-AC-5216
-
Jul
-
M.Miyoshi, H.Ito, R.Arakawa, et al. Quantitative analysis of peripheral benzodiazepine receptor in the human brain using PET with (11)C-AC-5216. J Nucl Med. 2009 Jul;50(7):1095–1101.
-
(2009)
J Nucl Med
, vol.50
, Issue.7
, pp. 1095-1101
-
-
Miyoshi, M.1
Ito, H.2
Arakawa, R.3
-
45
-
-
0025121160
-
Pharmacological and behavioral profile of alpidem as an anxiolytic
-
May
-
B.Zivkovic, E.Morel, D.Joly, et al. Pharmacological and behavioral profile of alpidem as an anxiolytic. Pharmacopsychiatry. 1990 May;23:108–113.
-
(1990)
Pharmacopsychiatry
, vol.23
, pp. 108-113
-
-
Zivkovic, B.1
Morel, E.2
Joly, D.3
-
46
-
-
0028319015
-
Comparison of the efficacy, safety and withdrawal of alpidem and alprazolam in anxious patients
-
Jul
-
L.Frattola, M.Garreau, R.Piolti, et al. Comparison of the efficacy, safety and withdrawal of alpidem and alprazolam in anxious patients. Brit J Psychiat. 1994 Jul;165:94–100.
-
(1994)
Brit J Psychiat
, vol.165
, pp. 94-100
-
-
Frattola, L.1
Garreau, M.2
Piolti, R.3
-
47
-
-
0034768233
-
Toxicity of alpidem, a peripheral benzodiazepine receptor ligand, but not zolpidem, in rat hepatocytes: role of mitochondrial permeability transition and metabolic activation
-
Nov
-
A.Berson, V.Descatoire, A.Sutton, et al. Toxicity of alpidem, a peripheral benzodiazepine receptor ligand, but not zolpidem, in rat hepatocytes:role of mitochondrial permeability transition and metabolic activation. J Pharmacol Exp Ther. 2001 Nov;299(2):793–800.
-
(2001)
J Pharmacol Exp Ther
, vol.299
, Issue.2
, pp. 793-800
-
-
Berson, A.1
Descatoire, V.2
Sutton, A.3
-
48
-
-
0026806389
-
2-Aryl-3-indoleacetamides (Fgin-1) - a new class of potent and specific ligands for the mitochondrial Dbi receptor (Mdr)
-
Sep
-
E.Romeo, J.Auta, A.P.Kozikowski, et al. 2-Aryl-3-indoleacetamides (Fgin-1) - a new class of potent and specific ligands for the mitochondrial Dbi receptor (Mdr). J Pharmacol Exp Ther. 1992 Sep;262(3):971–978.
-
(1992)
J Pharmacol Exp Ther
, vol.262
, Issue.3
, pp. 971-978
-
-
Romeo, E.1
Auta, J.2
Kozikowski, A.P.3
-
49
-
-
0027443448
-
Stimulation of brain steroidogenesis by 2-aryl-indole-3-acetamide derivatives acting at the mitochondrial diazepam-binding inhibitor receptor complex
-
Oct
-
E.Romeo, S.Cavallaro, A.Korneyev, et al. Stimulation of brain steroidogenesis by 2-aryl-indole-3-acetamide derivatives acting at the mitochondrial diazepam-binding inhibitor receptor complex. J Pharmacol Exp Ther. 1993 Oct;267(1):462–471.
-
(1993)
J Pharmacol Exp Ther
, vol.267
, Issue.1
, pp. 462-471
-
-
Romeo, E.1
Cavallaro, S.2
Korneyev, A.3
-
50
-
-
0036264571
-
SSR180575 (7-chloro-N,N,5-trimethyl-4-oxo-3-phenyl-3,5-dihydro-4H-pyridazino[4,5-b]indole-1 -acetamide), a peripheral benzodiazepine receptor ligand, promotes neuronal survival and repair
-
Jun
-
B.Ferzaz, E.Brault, G.Bourliaud, et al. SSR180575 (7-chloro-N,N,5-trimethyl-4-oxo-3-phenyl-3,5-dihydro-4H-pyridazino[4,5-b]indole-1 -acetamide), a peripheral benzodiazepine receptor ligand, promotes neuronal survival and repair. J Pharmacol Exp Ther. 2002 Jun;301(3):1067–1078.
-
(2002)
J Pharmacol Exp Ther
, vol.301
, Issue.3
, pp. 1067-1078
-
-
Ferzaz, B.1
Brault, E.2
Bourliaud, G.3
-
51
-
-
79953737531
-
In vivo imaging of neuroinflammation in the rodent brain with [11C]SSR180575, a novel indoleacetamide radioligand of the translocator protein (18 kDa)
-
Mar
-
F.Chauveau, H.Boutin, N.Van Camp, et al. In vivo imaging of neuroinflammation in the rodent brain with [11C]SSR180575, a novel indoleacetamide radioligand of the translocator protein (18 kDa). Eur J Nucl Med Mol Imaging. 2011 Mar;38(3):509–514.
-
(2011)
Eur J Nucl Med Mol Imaging
, vol.38
, Issue.3
, pp. 509-514
-
-
Chauveau, F.1
Boutin, H.2
Van Camp, N.3
-
52
-
-
84894427619
-
[F-18]fluoromethyl-PBR28 as a potential radiotracer for TSPO: preclinical comparison with [C-11]PBR28 in a rat model of neuroinflammation
-
Feb
-
B.S.Moon, B.S.Kim, C.Park, et al. [F-18]fluoromethyl-PBR28 as a potential radiotracer for TSPO:preclinical comparison with [C-11]PBR28 in a rat model of neuroinflammation. Bioconjugate Chem. 2014 Feb;25(2):442–450.
-
(2014)
Bioconjugate Chem
, vol.25
, Issue.2
, pp. 442-450
-
-
Moon, B.S.1
Kim, B.S.2
Park, C.3
-
53
-
-
38149021285
-
The high affinity peripheral benzodiazepine receptor ligand DAA1106 binds to activated and infected brain macrophages in areas of synaptic degeneration: implications for PET imaging of neuroinflammation in lentiviral encephalitis
-
Feb
-
S.Venneti, G.Wang, C.A.Wiley. The high affinity peripheral benzodiazepine receptor ligand DAA1106 binds to activated and infected brain macrophages in areas of synaptic degeneration:implications for PET imaging of neuroinflammation in lentiviral encephalitis. Neurobiol Dis. 2008 Feb;29(2):232–241.
-
(2008)
Neurobiol Dis
, vol.29
, Issue.2
, pp. 232-241
-
-
Venneti, S.1
Wang, G.2
Wiley, C.A.3
-
54
-
-
34547123812
-
Identification and characterization of cholest-4-en-3-one, oxime (TRO19622), a novel drug candidate for amyotrophic lateral sclerosis
-
Aug
-
T.Bordet, B.Buisson, M.Michaud, et al. Identification and characterization of cholest-4-en-3-one, oxime (TRO19622), a novel drug candidate for amyotrophic lateral sclerosis. J Pharmacol Exp Ther. 2007 Aug;322(2):709–720.
-
(2007)
J Pharmacol Exp Ther
, vol.322
, Issue.2
, pp. 709-720
-
-
Bordet, T.1
Buisson, B.2
Michaud, M.3
-
55
-
-
84885920071
-
TRO19622 promotes myelin repair in a rat model of demyelination
-
Nov
-
Y.Q.Li, Y.Y.Zhang, W.W.Han, et al. TRO19622 promotes myelin repair in a rat model of demyelination. Int J Neurosci. 2013 Nov;123(11):810–822.
-
(2013)
Int J Neurosci
, vol.123
, Issue.11
, pp. 810-822
-
-
Li, Y.Q.1
Zhang, Y.Y.2
Han, W.W.3
-
56
-
-
84892373557
-
Molecular therapeutic strategies for spinal muscular atrophies: current and future clinical trials
-
Jan
-
C.Zanetta, M.Nizzardo, C.Simone, et al. Molecular therapeutic strategies for spinal muscular atrophies:current and future clinical trials. Clin Ther. 2014 Jan;36(1):128–140.
-
(2014)
Clin Ther
, vol.36
, Issue.1
, pp. 128-140
-
-
Zanetta, C.1
Nizzardo, M.2
Simone, C.3
-
57
-
-
43849100475
-
Secondary and tertiary structures of the transmembrane domains of the translocator protein TSPO determined by NMR. Stabilization of the TSPO tertiary fold upon ligand binding
-
Jun
-
S.Murail, J.C.Robert, Y.M.Coic, et al. Secondary and tertiary structures of the transmembrane domains of the translocator protein TSPO determined by NMR. Stabilization of the TSPO tertiary fold upon ligand binding. Biochim Biophys Acta. 2008 Jun;1778(6):1375–1381.
-
(2008)
Biochim Biophys Acta
, vol.1778
, Issue.6
, pp. 1375-1381
-
-
Murail, S.1
Robert, J.C.2
Coic, Y.M.3
-
58
-
-
0028585940
-
Site-directed mutagenesis of the peripheral benzodiazepine receptor: identification of amino acids implicated in the binding site of Ro5-4864
-
Dec
-
R.Farges, E.Joseph-Liauzun, D.Shire, et al. Site-directed mutagenesis of the peripheral benzodiazepine receptor:identification of amino acids implicated in the binding site of Ro5-4864. Mol Pharmacol. 1994 Dec;46(6):1160–1167.
-
(1994)
Mol Pharmacol
, vol.46
, Issue.6
, pp. 1160-1167
-
-
Farges, R.1
Joseph-Liauzun, E.2
Shire, D.3
-
59
-
-
84856429837
-
Computational studies on translocator protein (TSPO) and its ligands
-
G.Ortore, T.Tuccinardi, A.Martinelli. Computational studies on translocator protein (TSPO) and its ligands. Curr Top Med Chem. 2012;12(4):352–359.
-
(2012)
Curr Top Med Chem
, vol.12
, Issue.4
, pp. 352-359
-
-
Ortore, G.1
Tuccinardi, T.2
Martinelli, A.3
-
60
-
-
84883234112
-
Characterization and modeling of the oligomeric state and ligand binding behavior of purified translocator protein 18 kDa from Rhodobacter sphaeroides
-
Aug
-
F.Li, Y.Xia, J.Meiler, et al. Characterization and modeling of the oligomeric state and ligand binding behavior of purified translocator protein 18 kDa from Rhodobacter sphaeroides. Biochemistry-Us. 2013 Aug 27;52(34):5884–5899.
-
(2013)
Biochemistry-Us
, vol.52
, Issue.34
, pp. 5884-5899
-
-
Li, F.1
Xia, Y.2
Meiler, J.3
-
61
-
-
85029236421
-
Identification of novel ligands targeted to the cholesterol recognition/interaction amino acid consensus (CRAC) domain of the translocator protein (TSPO)
-
Jun
-
A.S.Midzak, N.Akula, L.Lecanu, et al. Identification of novel ligands targeted to the cholesterol recognition/interaction amino acid consensus (CRAC) domain of the translocator protein (TSPO). Endocr Rev. 2010 Jun;31(3):S2494–S94.
-
(2010)
Endocr Rev
, vol.31
, Issue.3
, pp. S2494
-
-
Midzak, A.S.1
Akula, N.2
Lecanu, L.3
-
62
-
-
84940724646
-
Evolving understanding of translocator protein 18 kDa (TSPO)
-
Sep
-
F.Li, J.Liu, R.M.Garavito, et al. Evolving understanding of translocator protein 18 kDa (TSPO). Pharmacol Res. 2015 Sep;99:404–409.
-
(2015)
Pharmacol Res
, vol.99
, pp. 404-409
-
-
Li, F.1
Liu, J.2
Garavito, R.M.3
-
63
-
-
84868087742
-
Identification of a dynamic mitochondrial protein complex driving cholesterol import, trafficking, and metabolism to steroid hormones
-
Nov
-
M.B.Rone, A.S.Midzak, L.Issop, et al. Identification of a dynamic mitochondrial protein complex driving cholesterol import, trafficking, and metabolism to steroid hormones. Mol Endocrinol. 2012 Nov;26(11):1868–1882.
-
(2012)
Mol Endocrinol
, vol.26
, Issue.11
, pp. 1868-1882
-
-
Rone, M.B.1
Midzak, A.S.2
Issop, L.3
-
64
-
-
79851473610
-
Mixed-affinity binding in humans with 18-kDa translocator protein ligands
-
Jan
-
D.R.J.Owen, R.N.Gunn, E.A.Rabiner, et al. Mixed-affinity binding in humans with 18-kDa translocator protein ligands. J Nucl Med. 2011 Jan;52(1):24–32.• This article contains a summary of the mixed binding affinity.
-
(2011)
J Nucl Med
, vol.52
, Issue.1
, pp. 24-32
-
-
Owen, D.R.J.1
Gunn, R.N.2
Rabiner, E.A.3
-
65
-
-
84979031920
-
Translocator protein 18 kDa (TSPO): an old protein with new functions?
-
May
-
F.Li, J.Liu, N.Liu, et al. Translocator protein 18 kDa (TSPO):an old protein with new functions? Biochemistry. 2016 May 9;55(20):2821–2831.
-
(2016)
Biochemistry
-
-
Li, F.1
Liu, J.2
Liu, N.3
-
66
-
-
84945410815
-
Comment on “Crystal structures of translocator protein (TSPO) and mutant mimic of a human polymorphism
-
Oct
-
J.Wang. Comment on “Crystal structures of translocator protein (TSPO) and mutant mimic of a human polymorphism”. Science. 2015 Oct 30;350(6260):519.
-
(2015)
Science
, vol.350
, Issue.6260
, pp. 519
-
-
Wang, J.1
-
67
-
-
84945410815
-
Response to comment on “Crystal structures of translocator protein (TSPO) and mutant mimic of a human polymorphism
-
Oct
-
F.Li, J.Liu, Y.Zheng, et al. Response to comment on “Crystal structures of translocator protein (TSPO) and mutant mimic of a human polymorphism”. Science. 2015 Oct 30;350(6260):519.
-
(2015)
Science
, vol.350
, Issue.6260
, pp. 519
-
-
Li, F.1
Liu, J.2
Zheng, Y.3
-
68
-
-
84878158934
-
[11C]PK11195 PET imaging of spinal glial activation after nerve injury in rats
-
Oct
-
N.Imamoto, S.Momosaki, M.Fujita, et al. [11C]PK11195 PET imaging of spinal glial activation after nerve injury in rats. NeuroImage. 2013 Oct 1;79:121–128.
-
(2013)
NeuroImage
, vol.79
, pp. 121-128
-
-
Imamoto, N.1
Momosaki, S.2
Fujita, M.3
-
70
-
-
77949270219
-
Human biodistribution and radiation dosimetry of 11C-(R)-PK11195, the prototypic PET ligand to image inflammation
-
Mar
-
J.Hirvonen, A.Roivainen, J.Virta, et al. Human biodistribution and radiation dosimetry of 11C-(R)-PK11195, the prototypic PET ligand to image inflammation. Eur J Nucl Med Mol Imaging. 2010 Mar;37(3):606–612.
-
(2010)
Eur J Nucl Med Mol Imaging
, vol.37
, Issue.3
, pp. 606-612
-
-
Hirvonen, J.1
Roivainen, A.2
Virta, J.3
-
71
-
-
25844495011
-
Medicinal chemical properties of successful central nervous system drugs
-
Oct
-
H.Pajouhesh, G.R.Lenz. Medicinal chemical properties of successful central nervous system drugs. NeuroRx. 2005 Oct;2(4):541–553.
-
(2005)
NeuroRx
, vol.2
, Issue.4
, pp. 541-553
-
-
Pajouhesh, H.1
Lenz, G.R.2
-
72
-
-
0035865790
-
Labeling and evaluation of N-[11C]methylated quinoline-2-carboxamides as potential radioligands for visualization of peripheral benzodiazepine receptors
-
Feb
-
M.Matarrese, R.M.Moresco, A.Cappelli, et al. Labeling and evaluation of N-[11C]methylated quinoline-2-carboxamides as potential radioligands for visualization of peripheral benzodiazepine receptors. J Med Chem. 2001 Feb 15;44(4):579–585.
-
(2001)
J Med Chem
, vol.44
, Issue.4
, pp. 579-585
-
-
Matarrese, M.1
Moresco, R.M.2
Cappelli, A.3
-
73
-
-
0042732948
-
Structure-activity relationships in carboxamide derivatives based on the targeted delivery of radionuclides and boron atoms by means of peripheral benzodiazepine receptor ligands
-
Aug
-
A.Cappelli, G.Pericot Mohr, A.Gallelli, et al. Structure-activity relationships in carboxamide derivatives based on the targeted delivery of radionuclides and boron atoms by means of peripheral benzodiazepine receptor ligands. J Med Chem. 2003 Aug 14;46(17):3568–3571.
-
(2003)
J Med Chem
, vol.46
, Issue.17
, pp. 3568-3571
-
-
Cappelli, A.1
Pericot Mohr, G.2
Gallelli, A.3
-
74
-
-
33646199161
-
Synthesis, labeling, and biological evaluation of halogenated 2-quinolinecarboxamides as potential radioligands for the visualization of peripheral benzodiazepine receptors
-
Jun
-
A.Cappelli, M.Matarrese, R.M.Moresco, et al. Synthesis, labeling, and biological evaluation of halogenated 2-quinolinecarboxamides as potential radioligands for the visualization of peripheral benzodiazepine receptors. Bioorg Med Chem. 2006 Jun 15;14(12):4055–4066.
-
(2006)
Bioorg Med Chem
, vol.14
, Issue.12
, pp. 4055-4066
-
-
Cappelli, A.1
Matarrese, M.2
Moresco, R.M.3
-
75
-
-
44449123579
-
Synthesis, fluorine-18 radiolabeling, and in vitro characterization of 1-iodophenyl-N-methyl-N-fluoroalkyl-3-isoquinoline carboxamide derivatives as potential PET radioligands for imaging peripheral benzodiazepine receptor
-
Jun
-
W.Yu, E.Wang, R.J.Voll, et al. Synthesis, fluorine-18 radiolabeling, and in vitro characterization of 1-iodophenyl-N-methyl-N-fluoroalkyl-3-isoquinoline carboxamide derivatives as potential PET radioligands for imaging peripheral benzodiazepine receptor. Bioorg Med Chem. 2008 Jun 1;16(11):6145–6155.
-
(2008)
Bioorg Med Chem
, vol.16
, Issue.11
, pp. 6145-6155
-
-
Yu, W.1
Wang, E.2
Voll, R.J.3
-
77
-
-
0242299669
-
Expression of peripheral benzodiazepine receptor (PBR) in human tumors: relationship to breast, colorectal, and prostate tumor progression
-
Z.Han, R.S.Slack, W.Li, et al. Expression of peripheral benzodiazepine receptor (PBR) in human tumors:relationship to breast, colorectal, and prostate tumor progression. J Recept Signal Transduct Res. 2003;23(2–3):225–238.
-
(2003)
J Recept Signal Transduct Res
, vol.23
, Issue.2-3
, pp. 225-238
-
-
Han, Z.1
Slack, R.S.2
Li, W.3
-
78
-
-
79951534507
-
TSPO 18 kDa (PBR) targeted photosensitizers for cancer imaging (PET) and PDT
-
Feb
-
Y.Chen, M.Sajjad, Y.Wang, et al. TSPO 18 kDa (PBR) targeted photosensitizers for cancer imaging (PET) and PDT. ACS Med Chem Lett. 2011 Feb 10;2(2):136–141.
-
(2011)
ACS Med Chem Lett
, vol.2
, Issue.2
, pp. 136-141
-
-
Chen, Y.1
Sajjad, M.2
Wang, Y.3
-
79
-
-
84897411408
-
Structure-activity relationship refinement and further assessment of 4-phenylquinazoline-2-carboxamide translocator protein ligands as antiproliferative agents in human glioblastoma tumors
-
Mar
-
S.Castellano, S.Taliani, M.Viviano, et al. Structure-activity relationship refinement and further assessment of 4-phenylquinazoline-2-carboxamide translocator protein ligands as antiproliferative agents in human glioblastoma tumors. J Med Chem. 2014 Mar 27;57(6):2413–2428.
-
(2014)
J Med Chem
, vol.57
, Issue.6
, pp. 2413-2428
-
-
Castellano, S.1
Taliani, S.2
Viviano, M.3
-
80
-
-
84861054375
-
Synthesis and biological evaluation of 4-phenylquinazoline-2-carboxamides designed as a novel class of potent ligands of the translocator protein
-
May
-
S.Castellano, S.Taliani, C.Milite, et al. Synthesis and biological evaluation of 4-phenylquinazoline-2-carboxamides designed as a novel class of potent ligands of the translocator protein. J Med Chem. 2012 May 10;55(9):4506–4510.
-
(2012)
J Med Chem
, vol.55
, Issue.9
, pp. 4506-4510
-
-
Castellano, S.1
Taliani, S.2
Milite, C.3
-
82
-
-
84937397405
-
Design, synthesis and anxiolytic-like activity of 1-arylpyrrolo[1,2-a]pyrazine-3-carboxamides
-
Jul
-
G.V.Mokrov, O.A.Deeva, T.A.Gudasheva, et al. Design, synthesis and anxiolytic-like activity of 1-arylpyrrolo[1,2-a]pyrazine-3-carboxamides. Bioorg Med Chem. 2015 Jul 1;23(13):3368–3378.
-
(2015)
Bioorg Med Chem
, vol.23
, Issue.13
, pp. 3368-3378
-
-
Mokrov, G.V.1
Deeva, O.A.2
Gudasheva, T.A.3
-
83
-
-
0022374863
-
Validation of open: closedarm entries in an elevated plus-maze as a measure of anxiety in the rat
-
Aug
-
S.Pellow, P.Chopin, S.E.File, et al. Validation of open:closedarm entries in an elevated plus-maze as a measure of anxiety in the rat. J Neurosci Methods. 1985 Aug;14(3):149–167.
-
(1985)
J Neurosci Methods
, vol.14
, Issue.3
, pp. 149-167
-
-
Pellow, S.1
Chopin, P.2
File, S.E.3
-
86
-
-
0033548505
-
Neuropharmacological profile of peripheral benzodiazepine receptor agonists, DAA1097 and DAA1106
-
S.Okuyama, S.Chaki, R.Yoshikawa, et al. Neuropharmacological profile of peripheral benzodiazepine receptor agonists, DAA1097 and DAA1106. Life Sci. 1999;64(16):1455–1464.
-
(1999)
Life Sci
, vol.64
, Issue.16
, pp. 1455-1464
-
-
Okuyama, S.1
Chaki, S.2
Yoshikawa, R.3
-
88
-
-
0346690184
-
Design, synthesis and structure-affinity relationships of aryloxyanilide derivatives as novel peripheral benzodiazepine receptor ligands
-
Jan
-
T.Okubo, R.Yoshikawa, S.Chaki, et al. Design, synthesis and structure-affinity relationships of aryloxyanilide derivatives as novel peripheral benzodiazepine receptor ligands. Bioorg Med Chem. 2004 Jan 15;12(2):423–438.
-
(2004)
Bioorg Med Chem
, vol.12
, Issue.2
, pp. 423-438
-
-
Okubo, T.1
Yoshikawa, R.2
Chaki, S.3
-
90
-
-
79953660905
-
Structural requirements to obtain highly potent and selective 18 kDa translocator protein (TSPO) ligands
-
S.Taliani, I.Pugliesi, F.Da Settimo. Structural requirements to obtain highly potent and selective 18 kDa translocator protein (TSPO) ligands. Curr Top Med Chem. 2011;11(7):860–886.
-
(2011)
Curr Top Med Chem
, vol.11
, Issue.7
, pp. 860-886
-
-
Taliani, S.1
Pugliesi, I.2
Da Settimo, F.3
-
91
-
-
37849053628
-
Synthesis and evaluation in monkey of two sensitive 11C-labeled aryloxyanilide ligands for imaging brain peripheral benzodiazepine receptors in vivo
-
Jan
-
E.Briard, S.S.Zoghbi, M.Imaizumi, et al. Synthesis and evaluation in monkey of two sensitive 11C-labeled aryloxyanilide ligands for imaging brain peripheral benzodiazepine receptors in vivo. J Med Chem. 2008 Jan 10;51(1):17–30.
-
(2008)
J Med Chem
, vol.51
, Issue.1
, pp. 17-30
-
-
Briard, E.1
Zoghbi, S.S.2
Imaizumi, M.3
-
92
-
-
79851499878
-
Quantitative, preclinical PET of translocator protein expression in glioma using F-18-N-fluoroacetyl-N-(2,5-dimethoxybenzyl)-2-phenoxyaniline
-
Jan
-
J.R.Buck, E.T.McKinley, M.R.Hight, et al. Quantitative, preclinical PET of translocator protein expression in glioma using F-18-N-fluoroacetyl-N-(2,5-dimethoxybenzyl)-2-phenoxyaniline. J Nucl Med. 2011 Jan 1;52(1):107–114.
-
(2011)
J Nucl Med
, vol.52
, Issue.1
, pp. 107-114
-
-
Buck, J.R.1
McKinley, E.T.2
Hight, M.R.3
-
93
-
-
80052707691
-
Synthesis of [C-11]PBR06 and [F-18]PBR06 as agents for positron emission tomographic (PET) imaging of the translocator protein (TSPO)
-
Nov
-
M.Wang, M.Z.Gao, K.D.Miller, et al. Synthesis of [C-11]PBR06 and [F-18]PBR06 as agents for positron emission tomographic (PET) imaging of the translocator protein (TSPO). Steroids. 2011 Nov;76(12):1331–1340.
-
(2011)
Steroids
, vol.76
, Issue.12
, pp. 1331-1340
-
-
Wang, M.1
Gao, M.Z.2
Miller, K.D.3
-
94
-
-
0037212103
-
[18F]FMDAA1106 and [18F]FEDAA1106: two positron-emitter labeled ligands for peripheral benzodiazepine receptor (PBR)
-
Jan
-
M.R.Zhang, J.Maeda, K.Furutsuka, et al. [18F]FMDAA1106 and [18F]FEDAA1106:two positron-emitter labeled ligands for peripheral benzodiazepine receptor (PBR). Bioorg Med Chem Lett. 2003 Jan 20;13(2):201–204.
-
(2003)
Bioorg Med Chem Lett
, vol.13
, Issue.2
, pp. 201-204
-
-
Zhang, M.R.1
Maeda, J.2
Furutsuka, K.3
-
95
-
-
84878784892
-
In vivo TSPO imaging in patients with multiple sclerosis: a brain PET study with [18F]FEDAA1106
-
A.Takano, F.Piehl, J.Hillert, et al. In vivo TSPO imaging in patients with multiple sclerosis:a brain PET study with [18F]FEDAA1106. EJNMMI Res. 2013;3(1):30.
-
(2013)
EJNMMI Res
, vol.3
, Issue.1
, pp. 30
-
-
Takano, A.1
Piehl, F.2
Hillert, J.3
-
96
-
-
84891702940
-
In vivo imaging of the 18-kDa translocator protein (TSPO) with [18F]FEDAA1106 and PET does not show increased binding in Alzheimer’s disease patients
-
Jun
-
A.Varrone, P.Mattsson, A.Forsberg, et al. In vivo imaging of the 18-kDa translocator protein (TSPO) with [18F]FEDAA1106 and PET does not show increased binding in Alzheimer’s disease patients. Eur J Nucl Med Mol Imaging. 2013 Jun;40(6):921–931.
-
(2013)
Eur J Nucl Med Mol Imaging
, vol.40
, Issue.6
, pp. 921-931
-
-
Varrone, A.1
Mattsson, P.2
Forsberg, A.3
-
97
-
-
84937763794
-
(11)C-PBR28 imaging in multiple sclerosis patients and healthy controls: test-retest reproducibility and focal visualization of active white matter areas
-
Jun
-
E.Park, J.-D.Gallezot, A.Delgadillo, et al. (11)C-PBR28 imaging in multiple sclerosis patients and healthy controls:test-retest reproducibility and focal visualization of active white matter areas. Eur J Nucl Med Mol Imaging. 2015 Jun;42(7):1081–1092.
-
(2015)
Eur J Nucl Med Mol Imaging
, vol.42
, Issue.7
, pp. 1081-1092
-
-
Park, E.1
Gallezot, J.-D.2
Delgadillo, A.3
-
100
-
-
40749142849
-
Radiosynthesis and initial evaluation of [18F]-FEPPA for PET imaging of peripheral benzodiazepine receptors
-
Apr
-
A.A.Wilson, A.Garcia, J.Parkes, et al. Radiosynthesis and initial evaluation of [18F]-FEPPA for PET imaging of peripheral benzodiazepine receptors. Nucl Med Biol. 2008 Apr;35(3):305–314.
-
(2008)
Nucl Med Biol
, vol.35
, Issue.3
, pp. 305-314
-
-
Wilson, A.A.1
Garcia, A.2
Parkes, J.3
-
101
-
-
84885710671
-
Neuroinflammation in healthy aging: a PET study using a novel translocator protein 18kDa (TSPO) radioligand, [(18)F]-FEPPA
-
Jan
-
I.Suridjan, P.M.Rusjan, A.N.Voineskos, et al. Neuroinflammation in healthy aging:a PET study using a novel translocator protein 18kDa (TSPO) radioligand, [(18)F]-FEPPA. NeuroImage. 2014 Jan 1;84:868–875.
-
(2014)
NeuroImage
, vol.84
, pp. 868-875
-
-
Suridjan, I.1
Rusjan, P.M.2
Voineskos, A.N.3
-
102
-
-
84908510509
-
Quantitative imaging of neuroinflammation in human white matter: a positron emission tomography study with translocator protein 18 kDa radioligand, [18F]-FEPPA
-
Nov
-
I.Suridjan, P.M.Rusjan, M.Kenk, et al. Quantitative imaging of neuroinflammation in human white matter:a positron emission tomography study with translocator protein 18 kDa radioligand, [18F]-FEPPA. Synapse. 2014 Nov;68(11):536–547.
-
(2014)
Synapse
, vol.68
, Issue.11
, pp. 536-547
-
-
Suridjan, I.1
Rusjan, P.M.2
Kenk, M.3
-
103
-
-
84947615776
-
In-vivo imaging of grey and white matter neuroinflammation in Alzheimer’s disease: a positron emission tomography study with a novel radioligand, [18F]-FEPPA
-
Feb
-
I.Suridjan, B.G.Pollock, N.P.Verhoeff, et al. In-vivo imaging of grey and white matter neuroinflammation in Alzheimer’s disease:a positron emission tomography study with a novel radioligand, [18F]-FEPPA. Mol Psychiatry. 2015 Feb 24;20(12):1579–1587.
-
(2015)
Mol Psychiatry
-
-
Suridjan, I.1
Pollock, B.G.2
Verhoeff, N.P.3
-
104
-
-
84920171026
-
Image derived input function for [18F]-FEPPA: application to quantify translocator protein (18 kDa) in the human brain
-
R.Mabrouk, P.M.Rusjan, R.Mizrahi, et al. Image derived input function for [18F]-FEPPA:application to quantify translocator protein (18 kDa) in the human brain. PLoS One. 2014;9(12):e115768.
-
(2014)
PLoS One
, vol.9
, Issue.12
, pp. e115768
-
-
Mabrouk, R.1
Rusjan, P.M.2
Mizrahi, R.3
-
105
-
-
84928798486
-
Imaging neuroinflammation in gray and white matter in schizophrenia: an in-vivo PET study with [18F]-FEPPA
-
Jan
-
M.Kenk, T.Selvanathan, N.Rao, et al. Imaging neuroinflammation in gray and white matter in schizophrenia:an in-vivo PET study with [18F]-FEPPA. Schizophr Bull. 2015 Jan;41(1):85–93.
-
(2015)
Schizophr Bull
, vol.41
, Issue.1
, pp. 85-93
-
-
Kenk, M.1
Selvanathan, T.2
Rao, N.3
-
108
-
-
17744386969
-
Ro5-4864, a peripheral benzodiazepine receptor ligand, reduces reactive gliosis and protects hippocampal hilar neurons from kainic acid excitotoxicity
-
Apr
-
S.Veiga, I.Azcoitia, L.M.Garcia-Segura. Ro5-4864, a peripheral benzodiazepine receptor ligand, reduces reactive gliosis and protects hippocampal hilar neurons from kainic acid excitotoxicity. J Neurosci Res. 2005 Apr 1;80(1):129–137.
-
(2005)
J Neurosci Res
, vol.80
, Issue.1
, pp. 129-137
-
-
Veiga, S.1
Azcoitia, I.2
Garcia-Segura, L.M.3
-
109
-
-
56749175080
-
Neuroprotective effect of Ro5-4864 following brain injury
-
Dec
-
J.F.Soustiel, M.Zaaroor, E.Vlodavsky, et al. Neuroprotective effect of Ro5-4864 following brain injury. Exp Neurol. 2008 Dec;214(2):201–208.
-
(2008)
Exp Neurol
, vol.214
, Issue.2
, pp. 201-208
-
-
Soustiel, J.F.1
Zaaroor, M.2
Vlodavsky, E.3
-
111
-
-
9544219672
-
Synthesis, biological activity, and SARs of pyrrolobenzoxazepine derivatives, a new class of specific “peripheral-type” benzodiazepine receptor ligands
-
Aug
-
G.Campiani, V.Nacci, I.Fiorini, et al. Synthesis, biological activity, and SARs of pyrrolobenzoxazepine derivatives, a new class of specific “peripheral-type” benzodiazepine receptor ligands. J Med Chem. 1996 Aug 30;39(18):3435–3450.
-
(1996)
J Med Chem
, vol.39
, Issue.18
, pp. 3435-3450
-
-
Campiani, G.1
Nacci, V.2
Fiorini, I.3
-
112
-
-
0037068436
-
Synthesis of new molecular probes for investigation of steroid biosynthesis induced by selective interaction with peripheral type benzodiazepine receptors (PBR)
-
Sep
-
G.Campiani, A.Ramunno, I.Fiorini, et al. Synthesis of new molecular probes for investigation of steroid biosynthesis induced by selective interaction with peripheral type benzodiazepine receptors (PBR). J Med Chem. 2002 Sep 12;45(19):4276–4281.
-
(2002)
J Med Chem
, vol.45
, Issue.19
, pp. 4276-4281
-
-
Campiani, G.1
Ramunno, A.2
Fiorini, I.3
-
115
-
-
33745596837
-
5-aryl-imidazo[2,1-c][1,4]benzodiazepine derivatives as tricyclic constrained analogues of diazepam and Ro5-4864. Synthesis and binding properties at peripheral and central benzodiazepine receptors
-
Jun
-
E.Rizzetto, S.Castellano, C.Florio, et al. 5-aryl-imidazo[2,1-c][1,4]benzodiazepine derivatives as tricyclic constrained analogues of diazepam and Ro5-4864. Synthesis and binding properties at peripheral and central benzodiazepine receptors. Die Pharmazie. 2006 Jun;61(6):505–510.
-
(2006)
Die Pharmazie
, vol.61
, Issue.6
, pp. 505-510
-
-
Rizzetto, E.1
Castellano, S.2
Florio, C.3
-
116
-
-
0029793981
-
Molecular basis of peripheral vs central benzodiazepine receptor selectivity in a new class of peripheral benzodiazepine receptor ligands related to alpidem
-
Oct
-
M.Anzini, A.Cappelli, S.Vomero, et al. Molecular basis of peripheral vs central benzodiazepine receptor selectivity in a new class of peripheral benzodiazepine receptor ligands related to alpidem. J Med Chem. 1996 Oct 11;39(21):4275–4284.
-
(1996)
J Med Chem
, vol.39
, Issue.21
, pp. 4275-4284
-
-
Anzini, M.1
Cappelli, A.2
Vomero, S.3
-
117
-
-
84930209686
-
2-Phenylimidazo[1,2-a]pyridine-containing ligands of the 18-kDa translocator protein (TSPO) behave as agonists and antagonists of steroidogenesis in a mouse leydig tumor cell line
-
Aug
-
A.Midzak, N.Denora, V.Laquintana, et al. 2-Phenylimidazo[1,2-a]pyridine-containing ligands of the 18-kDa translocator protein (TSPO) behave as agonists and antagonists of steroidogenesis in a mouse leydig tumor cell line. Eur J Pharm Sci. 2015 Aug 30;76:231–237.
-
(2015)
Eur J Pharm Sci
, vol.76
, pp. 231-237
-
-
Midzak, A.1
Denora, N.2
Laquintana, V.3
-
118
-
-
56249143493
-
2-Phenyl-imidazo[1,2-a]pyridine compounds containing hydrophilic groups as potent and selective ligands for peripheral benzodiazepine receptors: synthesis, binding affinity and electrophysiological studies
-
Nov
-
N.Denora, V.Laquintana, M.G.Pisu, et al. 2-Phenyl-imidazo[1,2-a]pyridine compounds containing hydrophilic groups as potent and selective ligands for peripheral benzodiazepine receptors:synthesis, binding affinity and electrophysiological studies. J Med Chem. 2008 Nov 13;51(21):6876–6888.
-
(2008)
J Med Chem
, vol.51
, Issue.21
, pp. 6876-6888
-
-
Denora, N.1
Laquintana, V.2
Pisu, M.G.3
-
119
-
-
84866743619
-
Novel codrugs with GABAergic activity for dopamine delivery in the brain
-
Nov
-
N.Denora, T.Cassano, V.Laquintana, et al. Novel codrugs with GABAergic activity for dopamine delivery in the brain. Int J Pharm. 2012 Nov 1;437(1–2):221–231.
-
(2012)
Int J Pharm
, vol.437
, Issue.1-2
, pp. 221-231
-
-
Denora, N.1
Cassano, T.2
Laquintana, V.3
-
120
-
-
84957818686
-
A novel PET imaging probe for the detection and monitoring of translocator protein 18 kDa expression in pathological disorders
-
M.Perrone, B.S.Moon, H.S.Park, et al. A novel PET imaging probe for the detection and monitoring of translocator protein 18 kDa expression in pathological disorders. Sci Rep. 2016;6:20422.
-
(2016)
Sci Rep
, vol.6
, pp. 20422
-
-
Perrone, M.1
Moon, B.S.2
Park, H.S.3
-
121
-
-
40949117086
-
Synthesis and structure-activity relationship studies in peripheral benzodiazepine receptor ligands related to alpidem
-
Mar
-
A.Cappelli, G.Giuliani, S.Valenti, et al. Synthesis and structure-activity relationship studies in peripheral benzodiazepine receptor ligands related to alpidem. Bioorg Med Chem. 2008 Mar 15;16(6):3428–3437.
-
(2008)
Bioorg Med Chem
, vol.16
, Issue.6
, pp. 3428-3437
-
-
Cappelli, A.1
Giuliani, G.2
Valenti, S.3
-
122
-
-
80054954224
-
Synthesis and structure-activity relationship studies in translocator protein ligands based on a pyrazolo[3,4-b]quinoline scaffold
-
Oct
-
A.Cappelli, G.Bini, S.Valenti, et al. Synthesis and structure-activity relationship studies in translocator protein ligands based on a pyrazolo[3,4-b]quinoline scaffold. J Med Chem. 2011 Oct 27;54(20):7165–7175.
-
(2011)
J Med Chem
, vol.54
, Issue.20
, pp. 7165-7175
-
-
Cappelli, A.1
Bini, G.2
Valenti, S.3
-
124
-
-
84992022223
-
-
R.Yang, Y.Li, Y.Li, et al. 2-Aryl imidazo[1,2-a]pyridine-3-acetamide derivatives, preparation methods and uses thereof.US20130203754 A1. 2013.
-
(2013)
2-Aryl imidazo[1,2-a]pyridine-3-acetamide derivatives, preparation methods and uses thereof
-
-
Yang, R.1
Li, Y.2
Li, Y.3
-
125
-
-
0034846643
-
2-Arylpyrazolo[1,5-a]pyrimidin-3-yl acetamides. New potent and selective peripheral benzodiazepine receptor ligands
-
Oct
-
S.Selleri, F.Bruni, C.Costagli, et al. 2-Arylpyrazolo[1,5-a]pyrimidin-3-yl acetamides. New potent and selective peripheral benzodiazepine receptor ligands. Bioorg Med Chem. 2001 Oct;9(10):2661–2671.
-
(2001)
Bioorg Med Chem
, vol.9
, Issue.10
, pp. 2661-2671
-
-
Selleri, S.1
Bruni, F.2
Costagli, C.3
-
126
-
-
44149118198
-
DPA-714, a new translocator protein-specific ligand: synthesis, radiofluorination, and pharmacologic characterization
-
May
-
M.L.James, R.R.Fulton, J.Vercoullie, et al. DPA-714, a new translocator protein-specific ligand:synthesis, radiofluorination, and pharmacologic characterization. J Nucl Med. 2008 May;49(5):814–822.
-
(2008)
J Nucl Med
, vol.49
, Issue.5
, pp. 814-822
-
-
James, M.L.1
Fulton, R.R.2
Vercoullie, J.3
-
128
-
-
84922883622
-
In vivo imaging and characterization of [(18)F]DPA-714, a potential new TSPO ligand, in mouse brain and peripheral tissues using small-animal PET
-
Mar
-
C.Vicidomini, M.Panico, A.Greco, et al. In vivo imaging and characterization of [(18)F]DPA-714, a potential new TSPO ligand, in mouse brain and peripheral tissues using small-animal PET. Nucl Med Biol. 2015 Mar;42(3):309–316.
-
(2015)
Nucl Med Biol
, vol.42
, Issue.3
, pp. 309-316
-
-
Vicidomini, C.1
Panico, M.2
Greco, A.3
-
129
-
-
84895829890
-
Preparation and evaluation of novel pyrazolo[1,5-a]pyrimidine acetamides, closely related to DPA-714, as potent ligands for imaging the TSPO 18kDa with PET
-
Mar
-
V.Médran-Navarrete, A.Damont, M.-A.Peyronneau, et al. Preparation and evaluation of novel pyrazolo[1,5-a]pyrimidine acetamides, closely related to DPA-714, as potent ligands for imaging the TSPO 18kDa with PET. Bioorg Med Chem Lett. 2014 Mar 15;24(6):1550–1556.
-
(2014)
Bioorg Med Chem Lett
, vol.24
, Issue.6
, pp. 1550-1556
-
-
Médran-Navarrete, V.1
Damont, A.2
Peyronneau, M.-A.3
-
130
-
-
84925490787
-
[18F]DPA-714 PET imaging of translocator protein TSPO (18 kDa) in the normal and excitotoxically-lesioned nonhuman primate brain
-
Mar
-
S.Lavisse, K.Inoue, C.Jan, et al. [18F]DPA-714 PET imaging of translocator protein TSPO (18 kDa) in the normal and excitotoxically-lesioned nonhuman primate brain. Eur J Nucl Med Mol Imaging. 2015 Mar;42(3):478–494.
-
(2015)
Eur J Nucl Med Mol Imaging
, vol.42
, Issue.3
, pp. 478-494
-
-
Lavisse, S.1
Inoue, K.2
Jan, C.3
-
131
-
-
84876883279
-
Synthesis and structure-activity relationships of 5,6,7-substituted pyrazolopyrimidines: discovery of a novel TSPO PET ligand for cancer imaging
-
Apr
-
D.Tang, E.T.McKinley, M.R.Hight, et al. Synthesis and structure-activity relationships of 5,6,7-substituted pyrazolopyrimidines:discovery of a novel TSPO PET ligand for cancer imaging. J Med Chem. 2013 Apr 25;56(8):3429–3433.
-
(2013)
J Med Chem
, vol.56
, Issue.8
, pp. 3429-3433
-
-
Tang, D.1
McKinley, E.T.2
Hight, M.R.3
-
132
-
-
84923556920
-
Ether analogues of DPA-714 with subnanomolar affinity for the translocator protein (TSPO)
-
Mar
-
S.D.Banister, C.Beinat, S.M.Wilkinson, et al. Ether analogues of DPA-714 with subnanomolar affinity for the translocator protein (TSPO). Eur J Med Chem. 2015 Mar 26;93:392–400.
-
(2015)
Eur J Med Chem
, vol.93
, pp. 392-400
-
-
Banister, S.D.1
Beinat, C.2
Wilkinson, S.M.3
-
133
-
-
84942284228
-
Novel pyrazolo[1,5-a]pyrimidines as translocator protein 18 kDa (TSPO) ligands: synthesis, in vitro biological evaluation, [(18)F]-labeling, and in vivo neuroinflammation PET images
-
Sep
-
A.Damont, V.Médran-Navarrete, F.Cacheux, et al. Novel pyrazolo[1,5-a]pyrimidines as translocator protein 18 kDa (TSPO) ligands:synthesis, in vitro biological evaluation, [(18)F]-labeling, and in vivo neuroinflammation PET images. J Med Chem. 2015 Sep 24;58(18):7449–7464.
-
(2015)
J Med Chem
, vol.58
, Issue.18
, pp. 7449-7464
-
-
Damont, A.1
Médran-Navarrete, V.2
Cacheux, F.3
-
135
-
-
0036184049
-
Tay-Sachs and Sandhoff diseases: enzymatic diagnosis in dried blood spots on filter paper: retrospective diagnoses in newborn-screening cards
-
Apr
-
N.A.Chamoles, M.Blanco, D.Gaggioli, et al. Tay-Sachs and Sandhoff diseases:enzymatic diagnosis in dried blood spots on filter paper:retrospective diagnoses in newborn-screening cards. Clin Chim Acta. 2002 Apr;318(1–2):133–137.
-
(2002)
Clin Chim Acta
, vol.318
, Issue.1-2
, pp. 133-137
-
-
Chamoles, N.A.1
Blanco, M.2
Gaggioli, D.3
-
138
-
-
84992141718
-
-
T.Murata, K.Masumoto, K.Kondo, et al. 2-aryl-8-oxodihydropurine derivative, process for the producing the same, medicinal compositions containing the same, and intermediates thereof.US6372740 B1. 2002.
-
(2002)
2-aryl-8-oxodihydropurine derivative, process for the producing the same, medicinal compositions containing the same, and intermediates thereof
-
-
Murata, T.1
Masumoto, K.2
Kondo, K.3
-
139
-
-
84926671031
-
Anxiolytic-like effects of translocator protein (TSPO) ligand ZBD-2 in an animal model of chronic pain
-
D.-S.Wang, Z.Tian, -Y.-Y.Guo, et al. Anxiolytic-like effects of translocator protein (TSPO) ligand ZBD-2 in an animal model of chronic pain. Mol Pain. 2015;11:16.
-
(2015)
Mol Pain
, vol.11
, pp. 16
-
-
Wang, D.-S.1
Tian, Z.2
Guo, -Y.-Y.3
-
141
-
-
84866240889
-
Design, synthesis and structure-activity relationships of novel benzoxazolone derivatives as 18 kDa translocator protein (TSPO) ligands
-
Sep
-
T.Fukaya, T.Kodo, T.Ishiyama, et al. Design, synthesis and structure-activity relationships of novel benzoxazolone derivatives as 18 kDa translocator protein (TSPO) ligands. Bioorg Med Chem. 2012 Sep 15;20(18):5568–5582.
-
(2012)
Bioorg Med Chem
, vol.20
, Issue.18
, pp. 5568-5582
-
-
Fukaya, T.1
Kodo, T.2
Ishiyama, T.3
-
142
-
-
84886552984
-
Identification of a novel benzoxazolone derivative as a selective, orally active 18 kDa translocator protein (TSPO) ligand
-
Oct
-
T.Fukaya, T.Ishiyama, S.Baba, et al. Identification of a novel benzoxazolone derivative as a selective, orally active 18 kDa translocator protein (TSPO) ligand. J Med Chem. 2013 Oct 24;56(20):8191–8195.
-
(2013)
J Med Chem
, vol.56
, Issue.20
, pp. 8191-8195
-
-
Fukaya, T.1
Ishiyama, T.2
Baba, S.3
-
143
-
-
84873721829
-
Design, synthesis and structure-activity relationship of novel tricyclic benzimidazolone derivatives as potent 18 kDa translocator protein (TSPO) ligands
-
Mar
-
T.Fukaya, T.Kodo, T.Ishiyama, et al. Design, synthesis and structure-activity relationship of novel tricyclic benzimidazolone derivatives as potent 18 kDa translocator protein (TSPO) ligands. Bioorg Med Chem. 2013 Mar 1;21(5):1257–1267.
-
(2013)
Bioorg Med Chem
, vol.21
, Issue.5
, pp. 1257-1267
-
-
Fukaya, T.1
Kodo, T.2
Ishiyama, T.3
-
144
-
-
84899486540
-
Characterization of a novel acetamidobenzoxazolone-based PET ligand for translocator protein (18 kDa) imaging of neuroinflammation in the brain
-
May
-
A.K.Tiwari, J.Yui, M.Fujinaga, et al. Characterization of a novel acetamidobenzoxazolone-based PET ligand for translocator protein (18 kDa) imaging of neuroinflammation in the brain. J Neurochem. 2014 May;129(4):712–720.
-
(2014)
J Neurochem
, vol.129
, Issue.4
, pp. 712-720
-
-
Tiwari, A.K.1
Yui, J.2
Fujinaga, M.3
-
145
-
-
84910020373
-
Synthesis and evaluation of new (18)F-labelled acetamidobenzoxazolone-based radioligands for imaging of the translocator protein (18 kDa, TSPO) in the brain
-
Dec
-
A.K.Tiwari, M.Fujinaga, J.Yui, et al. Synthesis and evaluation of new (18)F-labelled acetamidobenzoxazolone-based radioligands for imaging of the translocator protein (18 kDa, TSPO) in the brain. Org Biomol Chem. 2014 Dec 21;12(47):9621–9630.
-
(2014)
Org Biomol Chem
, vol.12
, Issue.47
, pp. 9621-9630
-
-
Tiwari, A.K.1
Fujinaga, M.2
Yui, J.3
-
146
-
-
84945936058
-
[18F]FEBMP: positron emission tomography imaging of TSPO in a model of neuroinflammation in rats, and in vitro autoradiograms of the human brain
-
A.K.Tiwari, B.Ji, J.Yui, et al. [18F]FEBMP:positron emission tomography imaging of TSPO in a model of neuroinflammation in rats, and in vitro autoradiograms of the human brain. Theranostics. 2015;5(9):961–969.
-
(2015)
Theranostics
, vol.5
, Issue.9
, pp. 961-969
-
-
Tiwari, A.K.1
Ji, B.2
Yui, J.3
-
148
-
-
84971602793
-
Tetrapyrroles as endogenous TSPO ligands in eukaryotes and prokaryotes: comparisons with synthetic ligands
-
L.Veenman, A.Vainshtein, N.Yasin, et al. Tetrapyrroles as endogenous TSPO ligands in eukaryotes and prokaryotes:comparisons with synthetic ligands. Int J Mol Sci. 2016;17(6):880.
-
(2016)
Int J Mol Sci
, vol.17
, Issue.6
-
-
Veenman, L.1
Vainshtein, A.2
Yasin, N.3
-
149
-
-
84860303350
-
PK11195 inhibits mitophagy targeting the F1Fo-ATPsynthase in Bcl-2 knock-down cells
-
May
-
M.S.Seneviratne, D.Faccenda, V.De Biase, et al. PK11195 inhibits mitophagy targeting the F1Fo-ATPsynthase in Bcl-2 knock-down cells. Curr Mol Med. 2012 May;12(4):476–482.
-
(2012)
Curr Mol Med
, vol.12
, Issue.4
, pp. 476-482
-
-
Seneviratne, M.S.1
Faccenda, D.2
De Biase, V.3
-
150
-
-
84939161869
-
Protein-ligand and membrane-ligand interactions in pharmacology: the case of the translocator protein (TSPO)
-
Oct
-
C.R.Hatty, R.B.Banati. Protein-ligand and membrane-ligand interactions in pharmacology:the case of the translocator protein (TSPO). Pharmacol Res. 2015 Oct;100:58–63.
-
(2015)
Pharmacol Res
, vol.100
, pp. 58-63
-
-
Hatty, C.R.1
Banati, R.B.2
|