Synthesis of new molecular probes for investigation of steroid biosynthesis induced by selective interaction with peripheral type benzodiazepine receptors (PBR)

Journal of Medicinal Chemistry

Volumn 45, Issue 19, 2002, Pages 4276-4281

  Campiani, Giuseppe ^a   Ramunno, Anna ^a   Fiorini, Isabella ^a   Nacci, Vito ^a   Morelli, Elena ^b   Novellino, Ettore ^b   Goegan, Mara ^c   Mennini, Tiziana ^c   Sullivan, Stephen ^d   Zisterer, Daniela M ^d   Williams, Clive D ^d  

^a UNIVERSITY OF SIENA   (Italy)

^b UNIVERSITY OF NAPLES FEDERICO II   (Italy)

^c MARIO NEGRI INSTITUTE FOR PHARMACOLOGICAL RESEARCH   (Italy)

^d TRINITY COLLEGE DUBLIN   (Ireland)

Author keywords

[No Author keywords available]

Indexed keywords

4 AMINOBUTYRIC ACID RECEPTOR; 4' CHLORODIAZEPAM; BENZODIAZEPINE RECEPTOR; BENZOTHIAZEPINE DERIVATIVE; BENZOXAZEPINE DERIVATIVE; CLONAZEPAM; FGIN 1 27; N SEC BUTYL 1 (2 CHLOROPHENYL) N METHYL 3 ISOQUINOLINECARBOXAMIDE; OXAZEPINE DERIVATIVE; STEROID; UNCLASSIFIED DRUG;

ANIMAL CELL; ANIMAL EXPERIMENT; ARTICLE; BINDING AFFINITY; BRAIN; CONTROLLED STUDY; DRUG BINDING SITE; DRUG RECEPTOR BINDING; DRUG STRUCTURE; LEYDIG CELL; MALE; MITOCHONDRION; MOLECULAR PROBE; NONHUMAN; RAT; REACTION ANALYSIS; STEROIDOGENESIS; STRUCTURE ACTIVITY RELATION;

ANIMALS; AZEPINES; BINDING SITES; BINDING, COMPETITIVE; CELL LINE; CEREBRAL CORTEX; HYDROGEN BONDING; LIGANDS; MALE; MITOCHONDRIA; MOLECULAR PROBES; OXAZEPINES; PROGESTERONE; RATS; RECEPTORS, GABA-A; STEROIDS; STRUCTURE-ACTIVITY RELATIONSHIP; TESTIS;

EID: 0037068436     PISSN: 00222623     EISSN: None     Source Type: Journal    
DOI: 10.1021/jm020849l     Document Type: Article

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