Multisteric TRPV1 nocisensor: A target for analgesics

Trends in Pharmacological Sciences

Volumn 33, Issue 12, 2012, Pages 646-655

  Szolcsányi, János ^a   Sándor, Zoltán ^b  

^a UNIVERSITY OF PÉCS   (Hungary)

^b UNIVERSITY OF PÉCS   (Hungary)

Author keywords

[No Author keywords available]

Indexed keywords

(5 TERT BUTYL 2,3 DIHYDRO 1H INDEN 1 YL) 3 (1H INDAZOL 4 YL)UREA; 1 (2 BROMOPHENYL) 3 [1 (5 TRIFLUOROMETHYL 2 PYRIDINYL) 3 PYRROLIDINYL]UREA; ALGR 4975; ANALGESIC AGENT; AS 1928370; AZD 1386; BRADYKININ; CALCITONIN GENE RELATED PEPTIDE; CALCIUM ION; CAPSAICIN; CAPSAICIN ADLEA; CIS CAPSAICIN; ENDOCANNABINOID; ION CHANNEL; JNJ 39729209; LIGAND; LYSOPHOSPHATIDIC ACID; MK 2295; MRS 1477; NERVE GROWTH FACTOR; PF 4065463; PROSTAGLANDIN E2; PROTEIN TYROSINE KINASE A; PROTON; RESINIFERATOXIN; SOMATOSTATIN; TACHYKININ; TRANSIENT RECEPTOR POTENTIAL CHANNEL A1; UNCLASSIFIED DRUG; UNINDEXED DRUG; VANILLOID RECEPTOR 1; VANILLOID RECEPTOR 1 ANTAGONIST;

AMINO TERMINAL SEQUENCE; ANALGESIA; BURN; CARBOXY TERMINAL SEQUENCE; CHANNEL GATING; CHEMORECEPTOR; CHRONIC DRUG ADMINISTRATION; CLUSTER HEADACHE; DRUG MECHANISM; DRUG STRUCTURE; HEAT SENSITIVITY; HUMAN; HYPERTHERMIA; LIGAND BINDING; MOLECULAR BIOLOGY; MOLECULAR CLONING; MUTAGENESIS; NERVOUS SYSTEM ELECTROPHYSIOLOGY; NEUROMODULATION; NEUROPATHIC PAIN; NONHUMAN; OSTEOARTHRITIS; PAIN; PAIN RECEPTOR; PRIORITY JOURNAL; PROTEIN EXPRESSION; PROTEIN FUNCTION; PROTEIN PHOSPHORYLATION; PROTEIN STRUCTURE; REVIEW; SENSORY NERVE CELL; SENSORY STIMULATION;

ANALGESICS; ANIMALS; HUMANS; NOCICEPTORS; TRPV CATION CHANNELS;

EID: 84869219281     PISSN: 01656147     EISSN: 18733735     Source Type: Journal    
DOI: 10.1016/j.tips.2012.09.002     Document Type: Review

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