Steroid sulfatase inhibitors: Their potential in the therapy of breast cancer

Current Medicinal Chemistry - Anti-Cancer Agents

Volumn 5, Issue 5, 2005, Pages 507-528

  Nussbaumer, Peter ^a   Billich, Andreas ^a  

^a Novartis Institutes for BioMedical Research Vienna   (Austria)

Author keywords

Arylsulfatase; Breast cancer; Desulfation; Steroid sulfatase; Sulfamate

Indexed keywords

2 PHENYLINDOLE DERIVATIVE; 7 HYDROXYBENZOCOUMARIN; ACETIC ACID DERIVATIVE; ALCOHOL DERIVATIVE; ALDEHYDE DERIVATIVE; ANGIOGENESIS INHIBITOR; ANTINEOPLASTIC AGENT; AROMATASE; AROMATASE INHIBITOR; BENZOPHENONE DERIVATIVE; BIPHENYL DERIVATIVE; CARBAMIC ACID DERIVATIVE; CARBOXYLIC ACID DERIVATIVE; COUMARIN DERIVATIVE; CYANIC ACID DERIVATIVE; ENZYME PRECURSOR; ESTER DERIVATIVE; ESTRADIOL DERIVATIVE; ESTROGEN; ESTRONE 3 O SULFAMATE; ESTRONE DERIVATIVE; ESTRONE SULFATE; KETOL; PRASTERONE SULFATE; STEROID; STERYL SULFATASE; STERYL SULFATASE INHIBITOR; SULFATE; THIOCARBAMIC ACID DERIVATIVE; UNCLASSIFIED DRUG; UNINDEXED DRUG;

BIOCHEMISTRY; BREAST CANCER; BREAST TUMOR; CLINICAL CHEMISTRY; DRUG BIOAVAILABILITY; DRUG BLOOD LEVEL; DRUG EFFICACY; DRUG MECHANISM; DRUG POTENCY; DRUG SCREENING; DRUG STABILITY; ENDOMETRIUM CANCER; ENZYME INHIBITION; ENZYME STRUCTURE; ESTROGEN SYNTHESIS; HORMONE SYNTHESIS; HUMAN; IC 50; NONHUMAN; PROTEIN EXPRESSION; REVIEW; SULFATION; SURVIVAL; TUMOR GROWTH;

ANIMALS; BREAST NEOPLASMS; ENZYME INHIBITORS; FEMALE; HUMANS; MOLECULAR STRUCTURE; STEREOISOMERISM; STERYL-SULFATASE; STRUCTURE-ACTIVITY RELATIONSHIP; TIME FACTORS;

EID: 23844509596     PISSN: 15680118     EISSN: None     Source Type: Journal    
DOI: 10.2174/1568011054866955     Document Type: Review

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