-
1
-
-
0029057703
-
Human carbonic anhydrases and carbonic anhydrase deficiencies
-
Sly W.S., Hu P.Y. Human carbonic anhydrases and carbonic anhydrase deficiencies. Annu. Rev. Biochem. 64:1995;375-401.
-
(1995)
Annu. Rev. Biochem.
, vol.64
, pp. 375-401
-
-
Sly, W.S.1
Hu, P.Y.2
-
2
-
-
0030984803
-
Expression of tumor-associated gene MN: A potential biomarker of human renal cell carcinoma
-
McKierman J.M., Buttyan R., Stifelman M.D.et al. Expression of tumor-associated gene MN: a potential biomarker of human renal cell carcinoma. Cancer Res. 57:1997;2362-2365.
-
(1997)
Cancer Res.
, vol.57
, pp. 2362-2365
-
-
McKierman, J.M.1
Buttyan, R.2
Stifelman, M.D.3
-
3
-
-
0041062296
-
Human carbonic anhydrase XII: CDNA cloning, expression and chromosomal localization of a carbonic anhydrase gene that is over expressed in some renal cancers
-
Tureci O., Sahin U., Vollmar E.et al. Human carbonic anhydrase XII: cDNA cloning, expression and chromosomal localization of a carbonic anhydrase gene that is over expressed in some renal cancers. Proc. Natl. Acad. Sci. USA. 95:1998;7608-7613.
-
(1998)
Proc. Natl. Acad. Sci. USA
, vol.95
, pp. 7608-7613
-
-
Tureci, O.1
Sahin, U.2
Vollmar, E.3
-
4
-
-
0029037972
-
Sulphonamide inhibitors of carbonic anhydrase inhibit the growth of human lymphoma cells in culture
-
Chegwidden W.R., Spencer I.M. Sulphonamide inhibitors of carbonic anhydrase inhibit the growth of human lymphoma cells in culture. Inflammopharmacology. 3:1995;231-239.
-
(1995)
Inflammopharmacology
, vol.3
, pp. 231-239
-
-
Chegwidden, W.R.1
Spencer, I.M.2
-
5
-
-
0032514685
-
Down-regulation of transmembrane carbonic anhydrases in renal cell carcinoma cell lines by wild-type von Hippel-Lindau transgenes
-
Ivanov S.V., Kuzmin I., Wei M.-H.et al. Down-regulation of transmembrane carbonic anhydrases in renal cell carcinoma cell lines by wild-type von Hippel-Lindau transgenes. Proc. Natl. Acad. Sci. USA. 95:1998;12596-12601.
-
(1998)
Proc. Natl. Acad. Sci. USA
, vol.95
, pp. 12596-12601
-
-
Ivanov, S.V.1
Kuzmin, I.2
Wei, M.-H.3
-
6
-
-
0034671307
-
Hypoxia-inducible expression of tumor-associated carbonic anhydrases
-
Wykoff C.C., Beasley N.J.P., Watson P.H.et al. Hypoxia-inducible expression of tumor-associated carbonic anhydrases. Cancer Res. 60:2000;7075-7083.
-
(2000)
Cancer Res.
, vol.60
, pp. 7075-7083
-
-
Wykoff, C.C.1
Beasley, N.J.P.2
Watson, P.H.3
-
7
-
-
0035418586
-
Carbonic anhydrase IX expression, a potential new intrinsic marker of hypoxia: Correlations with tumor oxygen measurements and prognosis in locally advanced carcinoma of the cervix
-
Loncaster J.A., Harris A.L., Davison S.E.et al. Carbonic anhydrase IX expression, a potential new intrinsic marker of hypoxia: correlations with tumor oxygen measurements and prognosis in locally advanced carcinoma of the cervix. Cancer Res. 61:2001;6394-6399.
-
(2001)
Cancer Res.
, vol.61
, pp. 6394-6399
-
-
Loncaster, J.A.1
Harris, A.L.2
Davison, S.E.3
-
8
-
-
0034842201
-
Hypoxia and oxidative stress in breast cancer
-
Knowles H.J., Harris A.L. Hypoxia and oxidative stress in breast cancer. Breast Cancer Res. 3:2001;318-322.
-
(2001)
Breast Cancer Res.
, vol.3
, pp. 318-322
-
-
Knowles, H.J.1
Harris, A.L.2
-
9
-
-
0036359548
-
Hypoxia - A key regulatory factor in tumour growth
-
Harris A.L. Hypoxia - a key regulatory factor in tumour growth. Nat. Cancer Rev. 2:2001;38-47.
-
(2001)
Nat. Cancer Rev.
, vol.2
, pp. 38-47
-
-
Harris, A.L.1
-
10
-
-
0034009497
-
Carbonic anhydrase inhibitor suppresses invasion of renal cancer cells in vitro
-
Parkkila S., Rajaniemi H., Parkkila A.-K.et al. Carbonic anhydrase inhibitor suppresses invasion of renal cancer cells in vitro. Proc. Natl. Acad. Sci. USA. 97:2000;2220-2224.
-
(2000)
Proc. Natl. Acad. Sci. USA
, vol.97
, pp. 2220-2224
-
-
Parkkila, S.1
Rajaniemi, H.2
Parkkila, A.-K.3
-
11
-
-
0027367258
-
A carbonic anhydrase inhibitor as a potential modulator of cancer therapies
-
Teicher B.A., Liu S.-D., Liu J.-T.et al. A carbonic anhydrase inhibitor as a potential modulator of cancer therapies. AntiCancer Res. 13:1993;1549-1556.
-
(1993)
AntiCancer Res.
, vol.13
, pp. 1549-1556
-
-
Teicher, B.A.1
Liu, S.-D.2
Liu, J.-T.3
-
12
-
-
0034018870
-
Carbonic anhydrase inhibitors and their therapeutic potential
-
Supuran C.T., Scozzafava A. Carbonic anhydrase inhibitors and their therapeutic potential. Exp. Opin. Ther. Patents. 10:2000;575-600.
-
(2000)
Exp. Opin. Ther. Patents
, vol.10
, pp. 575-600
-
-
Supuran, C.T.1
Scozzafava, A.2
-
13
-
-
0035106202
-
Carbonic anhydrase inhibitors: Sulfonamides as antitumor agents?
-
Supuran C.T., Briganit F., Tilli S.et al. Carbonic anhydrase inhibitors: sulfonamides as antitumor agents? Bioorg. Med. Chem. 9:2001;703-714.
-
(2001)
Bioorg. Med. Chem.
, vol.9
, pp. 703-714
-
-
Supuran, C.T.1
Briganit, F.2
Tilli, S.3
-
15
-
-
0037430638
-
Docking studies of sulphamate inhibitors of estrone sulphatase in human carbonic anhydrase II
-
Vicker N., Ho Y.T., Robinson J.et al. Docking studies of sulphamate inhibitors of estrone sulphatase in human carbonic anhydrase II. Bioorg. Med. Chem. Lett. 13:2003;863-865.
-
(2003)
Bioorg. Med. Chem. Lett.
, vol.13
, pp. 863-865
-
-
Vicker, N.1
Ho, Y.T.2
Robinson, J.3
-
16
-
-
0029620774
-
Sulfamates of various estrogens are prodrugs with increased systemic and reduced hepatic estrogenicity at oral application
-
Elger W., Schwarz S., Hedden A.et al. Sulfamates of various estrogens are prodrugs with increased systemic and reduced hepatic estrogenicity at oral application. J. Steroid Biochem. Mol. Biol. 55:1995;395-403.
-
(1995)
J. Steroid Biochem. Mol. Biol.
, vol.55
, pp. 395-403
-
-
Elger, W.1
Schwarz, S.2
Hedden, A.3
-
17
-
-
85001837381
-
Novel oestrogen sulphamates: A new approach to oral hormone therapy
-
Elger W., Palme H.-J., Schwarz S. Novel oestrogen sulphamates: a new approach to oral hormone therapy. Exp. Opin. Invest. Drugs. 7:1998;575-589.
-
(1998)
Exp. Opin. Invest. Drugs
, vol.7
, pp. 575-589
-
-
Elger, W.1
Palme, H.-J.2
Schwarz, S.3
-
18
-
-
0028879855
-
In vivo inhibition of oestrone sulphatase and dehydroepiandrosterone sulphatase by oestrone-3-O-sulphamate
-
Purohit A., Williams G.J., Howarth N.M.et al. In vivo inhibition of oestrone sulphatase and dehydroepiandrosterone sulphatase by oestrone-3-O-sulphamate. Int. J. Cancer. 62:1995;106-111.
-
(1995)
Int. J. Cancer
, vol.62
, pp. 106-111
-
-
Purohit, A.1
Williams, G.J.2
Howarth, N.M.3
-
19
-
-
0028111173
-
Cloning and characterisation of MN, a human tumor-associated protein with a domain homologous to carbonic anhydrase as a putative helix-loop-helix DNA binding segment
-
Pastorek J., Pastorekova S., Callebaut I.et al. Cloning and characterisation of MN, a human tumor-associated protein with a domain homologous to carbonic anhydrase as a putative helix-loop-helix DNA binding segment. Oncogene. 9:1994;2877-2888.
-
(1994)
Oncogene
, vol.9
, pp. 2877-2888
-
-
Pastorek, J.1
Pastorekova, S.2
Callebaut, I.3
-
20
-
-
0031040821
-
Carbonic anhydrase IX, MN/CA IX: Analysis of stomach complementary DNA sequence and expression in human and rat alimentary tracts
-
Pastorekova S., Parkkila S., Parkkila A.K.et al. Carbonic anhydrase IX, MN/CA IX: analysis of stomach complementary DNA sequence and expression in human and rat alimentary tracts. Gastroenterology. 112:1997;398-408.
-
(1997)
Gastroenterology
, vol.112
, pp. 398-408
-
-
Pastorekova, S.1
Parkkila, S.2
Parkkila, A.K.3
-
21
-
-
85031167907
-
-
Gene sequence and probe for a markar of non-small cell lung carcinoma, US Patent 5,589,579, 1996
-
R.M. Torczynski, A.P. Bollin, Gene sequence and probe for a markar of non-small cell lung carcinoma, US Patent 5,589,579, 1996.
-
-
-
Torczynski, R.M.1
Bollin, A.P.2
-
22
-
-
0027153461
-
Expression of MaTu-MN protein in human tumor cultures and in clinical specimens
-
Zavada J., Zavadova Z., Pastorekova S.et al. Expression of MaTu-MN protein in human tumor cultures and in clinical specimens. Int. J. Cancer. 54:1993;268-274.
-
(1993)
Int. J. Cancer
, vol.54
, pp. 268-274
-
-
Zavada, J.1
Zavadova, Z.2
Pastorekova, S.3
-
23
-
-
0014011587
-
Purification and properties of human erthyrocyte carbonic anhydrases
-
Armstrong J.M., Myers D.V., Verpoorte I.A.et al. Purification and properties of human erthyrocyte carbonic anhydrases. J. Biol. Chem. 241:1966;5137-5149.
-
(1966)
J. Biol. Chem.
, vol.241
, pp. 5137-5149
-
-
Armstrong, J.M.1
Myers, D.V.2
Verpoorte, I.A.3
-
25
-
-
0026463503
-
Structure of native and apo carbonic anhydrase II and some of its anion-ligand complexes
-
Hakansson K., Carlsson M., Svensson L.A.et al. Structure of native and apo carbonic anhydrase II and some of its anion-ligand complexes. J. Mol. Biol. 227:1992;1192-1204.
-
(1992)
J. Mol. Biol.
, vol.227
, pp. 1192-1204
-
-
Hakansson, K.1
Carlsson, M.2
Svensson, L.A.3
-
26
-
-
0035859892
-
Crystal structure of the dimeric extracellular domain of human carbonic anhydrase XII, a bitopic membrane protein over expressed in certain cancer tumor cells
-
Whittington D.A., Waheed A., Ulmasou B.et al. Crystal structure of the dimeric extracellular domain of human carbonic anhydrase XII, a bitopic membrane protein over expressed in certain cancer tumor cells. Proc. Soc. Natl. Acad. Sci. USA. 98:2001;9545-9550.
-
(2001)
Proc. Soc. Natl. Acad. Sci. USA
, vol.98
, pp. 9545-9550
-
-
Whittington, D.A.1
Waheed, A.2
Ulmasou, B.3
-
27
-
-
85031165102
-
-
Sybyl 6.8 Tripos, Inc., St. Louis, 170, 2000
-
Sybyl 6.8 Tripos, Inc., St. Louis, 170, 2000.
-
-
-
-
28
-
-
0037571112
-
Merck molecular force field I. Basis, form, scope, parameterization, and performance with MMFF94
-
Halgren T.A. Merck molecular force field I. Basis, form, scope, parameterization, and performance with MMFF94. J. Comput. Chem. 17:1996;490-519.
-
(1996)
J. Comput. Chem.
, vol.17
, pp. 490-519
-
-
Halgren, T.A.1
-
29
-
-
0030599010
-
A fast flexible docking method using an incremental construction algorithm
-
Rarey M., Kramer B., Laugenauer T.et al. A fast flexible docking method using an incremental construction algorithm. J. Mol. Biol. 261:1996;470-489.
-
(1996)
J. Mol. Biol.
, vol.261
, pp. 470-489
-
-
Rarey, M.1
Kramer, B.2
Laugenauer, T.3
-
30
-
-
85031167300
-
-
MOE - Molecular Operating Environment, Chemical Computing Group Inc., Quebec, Canada
-
MOE - Molecular Operating Environment, Chemical Computing Group Inc., Quebec, Canada.
-
-
-
-
31
-
-
0028854034
-
Molecular recognition of a receptor sites using a genetic algorithm with a description of desolvation
-
Jones G., Willet P., Glen R.C. Molecular recognition of a receptor sites using a genetic algorithm with a description of desolvation. J. Mol. Biol. 245:1995;43-53.
-
(1995)
J. Mol. Biol.
, vol.245
, pp. 43-53
-
-
Jones, G.1
Willet, P.2
Glen, R.C.3
-
32
-
-
0031552362
-
Development and validation of a genetic algorithm for flexible docking
-
Jones G., Willet P., Glen R.C.et al. Development and validation of a genetic algorithm for flexible docking. J. Mol. Biol. 267:1997;727-748.
-
(1997)
J. Mol. Biol.
, vol.267
, pp. 727-748
-
-
Jones, G.1
Willet, P.2
Glen, R.C.3
-
33
-
-
0033780686
-
Potent active site-directed inhibition of steroid sulphatase by tricyclic coumarin-based sulphamates
-
Woo L.W.L., Purohit A., Malini B.et al. Potent active site-directed inhibition of steroid sulphatase by tricyclic coumarin-based sulphamates. Chem. Biol. 7:2000;773-791.
-
(2000)
Chem. Biol.
, vol.7
, pp. 773-791
-
-
Woo, L.W.L.1
Purohit, A.2
Malini, B.3
-
34
-
-
0038303879
-
Milanese, Development and pharmacological characterization of a modified procedure for the measurement of carbonic anhydrase activity
-
Landolfi C., Marchetti M., Ciocci G.et al. Milanese, Development and pharmacological characterization of a modified procedure for the measurement of carbonic anhydrase activity. Anal. Biochem. 185:1990;254-264.
-
(1990)
Anal. Biochem.
, vol.185
, pp. 254-264
-
-
Landolfi, C.1
Marchetti, M.2
Ciocci, G.3
-
36
-
-
0027399723
-
Synthesis and biochemical studies of estrone sulphatase inhibitors
-
Li P.-K., Pillai R., Young B.L.et al. Synthesis and biochemical studies of estrone sulphatase inhibitors. Steroids. 58:1993;106-111.
-
(1993)
Steroids
, vol.58
, pp. 106-111
-
-
Li, P.-K.1
Pillai, R.2
Young, B.L.3
-
38
-
-
0033598320
-
Discovery of novel antitumor sulfonamides targeting G1 phase of the cell cycle
-
Owa T., Yoshino H., Okauchi T.et al. Discovery of novel antitumor sulfonamides targeting G1 phase of the cell cycle. J. Med. Chem. 42:1999;3789-3799.
-
(1999)
J. Med. Chem.
, vol.42
, pp. 3789-3799
-
-
Owa, T.1
Yoshino, H.2
Okauchi, T.3
-
39
-
-
0037315480
-
Indisulam - An anticancer sulfonamide in clinical development
-
Supuran C.T. Indisulam - an anticancer sulfonamide in clinical development. Exp. Opin. Invest. Drugs. 12:2003;283-287.
-
(2003)
Exp. Opin. Invest. Drugs
, vol.12
, pp. 283-287
-
-
Supuran, C.T.1
-
40
-
-
0027397024
-
Inhibition of estrone sulfatase activity by estrone-3-methylethiophosphonate: A potential therapeutic agent in breast cancer
-
Duncan L.J., Purohit A., Howarth N.M.et al. Inhibition of estrone sulfatase activity by estrone-3-methylethiophosphonate: a potential therapeutic agent in breast cancer. Cancer Res. 53:1993;298-303.
-
(1993)
Cancer Res.
, vol.53
, pp. 298-303
-
-
Duncan, L.J.1
Purohit, A.2
Howarth, N.M.3
-
41
-
-
0344193512
-
Carbonic anhydrase inhibitors: SAR and X-ray crystallographic study for the interaction of sugar sulfamates/sulphamides with isoenzymes I, II and IV
-
Casini A., Antel J., Abbate F.et al. Carbonic anhydrase inhibitors: SAR and X-ray crystallographic study for the interaction of sugar sulfamates/sulphamides with isoenzymes I, II and IV. Bioorg. Med. Lett. 13:2003;841-845.
-
(2003)
Bioorg. Med. Lett.
, vol.13
, pp. 841-845
-
-
Casini, A.1
Antel, J.2
Abbate, F.3
-
43
-
-
0034719437
-
Carbonic anhydrase inhibitors: Synthesis of membrane-impermeant low molecular weight sulfonamides possessing in vivo selectivity for the membrane-bound versus cytosolic isozymes
-
Scozzafava A., Briganti F., Ilies M.A.et al. Carbonic anhydrase inhibitors: synthesis of membrane-impermeant low molecular weight sulfonamides possessing in vivo selectivity for the membrane-bound versus cytosolic isozymes. J. Med. Chem. 43:2000;292-300.
-
(2000)
J. Med. Chem.
, vol.43
, pp. 292-300
-
-
Scozzafava, A.1
Briganti, F.2
Ilies, M.A.3
-
45
-
-
0037434582
-
Surflex: Fully automated flexible molecular docking using a molecular similarity-based search engine
-
Jain A.N. Surflex: Fully automated flexible molecular docking using a molecular similarity-based search engine. J. Med. Chem. 46:2003;499-511.
-
(2003)
J. Med. Chem.
, vol.46
, pp. 499-511
-
-
Jain, A.N.1
|