Oestrone 3-O-(N-acetyl)sulphamate, a potential molecular probe of the active site of oestrone sulphatase

Bioorganic and Medicinal Chemistry Letters

Volumn 7, Issue 24, 1997, Pages 3075-3080

  Woo, L W Lawrence ^a   Purohit, Atul ^b   Reed, Michael J ^b   Potter, Barry V L ^a  

^a University of Bath   (United Kingdom)

^b IMPERIAL COLLEGE SCHOOL OF MEDICINE   (United Kingdom)

Author keywords

[No Author keywords available]

Indexed keywords

ENZYME INHIBITOR; ESTROGEN; ESTRONE 3 O (N ACETYL)SULFAMATE; ESTRONE 3 SULFAMATE; STERYL SULFATASE; UNCLASSIFIED DRUG;

ARTICLE; CONTROLLED STUDY; DOSE RESPONSE; DOSE TIME EFFECT RELATION; DRUG SYNTHESIS; ENZYME INACTIVATION; FEMALE; HUMAN; HUMAN TISSUE; IN VITRO STUDY; ISOTOPE LABELING; MICROSOME; PLACENTA; REACTION ANALYSIS; STRUCTURE ACTIVITY RELATION;

EID: 0031458762     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0960-894X(97)10167-6     Document Type: Article

References (15)

1. Beatson, G. T. Lancet 1896, ii, 104-107.
2. Santner, S. J.; Feil, P. D.; Santen, R. J. J. Clin. Endocrinol. Metab. 1984, 59, 29-33.
3. Yamamoto, T.; Kitawaki, J.; Urabe, M.; Honjo, H.; Tamura, T.; Noguchi, T.; Okada, H.; Sasaki, H.; Tada, A.; Terashima, Y.; Nakamura, J.; Yoshihama, M. J. Steroid Biochem. Mol. Biol. 1993, 44, 463-468.
4. Jonat, W.; Howell, A.; Blomqvist, C.; Eiermann, W.; Winblad, G.; Tyrrell, C.; Mauriac, L.; Lundgren, S.; Hellmund, R.; Azab, M. Eur. J. Cancer, 1996, 32A, 404-412.
5. Castiglione-Gertsch, M. Eur. J. Cancer, 1996, 32A, 393-395.
6. Svenstrup, B.; Herrstedt, J.; Brünner, N.; Bennett, P.; Wachman, H.; Dombernowsky, P. Eur. J. Cancer, 1994, 30A, 1254-1258.
7. Dowsett, M.; Smithers, D.; Moore, J.; Trunet, P. F.; Coombes, R. C.; Powles, T. J.; Rubens, R.; Smith, I. E. Eur. J. Cancer, 1994, 30A, 1453-1458.
8. Johnson, S. R. D.; Smith, I. E.; Doody, D.; Jacobs, S.; Robertshaw, H.; Dowsett, M. Cancer Res. 1994, 54, 5875-5881.
9. Howarth, N. M.; Purohit, A; Reed, M. J.; Potter, B. V. L. J. Med. Chem. 1994, 37, 219-221.
10. Purohit, A.; Williams, G. J.; Howarth, N. M.; Potter, B. V. L.; Reed, M. J. Biochemistry 1995, 34, 11508-11514.
11. Purohit, A.; Dauvois, S.; Parker, M. G.; Potter, B. V. L.; Williams, G. J.; Reed, M. J. J. Steroid Biochem. Mol. Biol. 1994, 50, 101-104.
12. Dauvois, S.; Labrie, F. Breast Cancer Res. Treat. 1989, 13, 61-69.
13. Purohit, A.; Williams, G. J.; Roberts, C. J.; Potter, B. V. L.; Reed, M. J. Int. J. Cancer 1995, 63, 106-111.
14. Duncan, L.; Purohit, A.; Howarth, N. M.; Potter, B. V. L.; Reed, M. J. Cancer Res. 1993, 53, 298-303.
15. Woo, L. W. L.; Lightowler, M.; Purohit, A; Reed, M. J.; Potter, B. V. L. J. Steroid Biochem. Mol. Biol. 1996, 57, 79-88.