Nortropinyl-arylsulfonylureas as novel, reversible inhibitors of human steroid sulfatase

Bioorganic and Medicinal Chemistry Letters

Volumn 13, Issue 21, 2003, Pages 3673-3677

  Nussbaumer, Peter ^a   Geyl, Dieter ^b   Horvath, Amarylla ^a   Lehr, Philipp ^a   Wolff, Barbara ^a   Billich, Andreas ^a  

^a Research Institute of the Vienna   (Austria)

^b NOVARTIS PHARMA AG   (Switzerland)

Author keywords

[No Author keywords available]

Indexed keywords

ANDROGEN; BROMINE DERIVATIVE; ENZYME INHIBITOR; FLUORENE DERIVATIVE; METHYL GROUP; NORTROPINYL ARYLSULFONYLUREA; STERYL SULFATASE; UNCLASSIFIED DRUG; UREA DERIVATIVE;

ARTICLE; CHO CELL; DRUG IDENTIFICATION; DRUG SCREENING; DRUG SYNTHESIS; ENDOCRINE DISEASE; ENZYME INHIBITION; ESTROGEN DEFICIENCY; HUMAN; HUMAN CELL; STRUCTURE ACTIVITY RELATION;

EID: 0141545127     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmcl.2003.08.019     Document Type: Article

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