N-Acyl arylsulfonamides as novel, reversible inhibitors of human steroid sulfatase

Bioorganic and Medicinal Chemistry Letters

Volumn 15, Issue 4, 2005, Pages 1235-1238

  Lehr, Philipp ^a   Billich, Andreas ^a   Wolff, Barbara ^a   Nussbaumer, Peter ^a  

^a Novartis Inst for Biomed Research   (Austria)

Author keywords

[No Author keywords available]

Indexed keywords

ENZYME INHIBITOR; PHENYLACETYLENE; STERYL SULFATASE; SULFONAMIDE; TROPINE;

ANIMAL CELL; ARTICLE; CONTROLLED STUDY; DRUG IDENTIFICATION; DRUG POTENCY; DRUG SYNTHESIS; DRUG TARGETING; ENZYME ACTIVITY; ENZYME PURIFICATION; IC 50; NONHUMAN; STRUCTURE ACTIVITY RELATION;

EID: 16244408316     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmcl.2004.11.069     Document Type: Article

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