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Tremblay, C.1
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76
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68549102641
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PFIZER LTD (Basford PA, Stephenson PT, Taylor SCJ, Wood A): Tropane derivatives as CCR5 modulators. WO-00084954 (2003).
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PFIZER LTD (Basford PA, Stephenson PT, Taylor SCJ, Wood A): Tropane derivatives as CCR5 modulators. WO-00084954 (2003).
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77
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68549102587
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ONO PHARMACEUTICALS CO LTD (Takaoka Y, Okamoto M, Genba Y, Ohie K): Novel crystals of triazaspiro[5.5]undecane derivative. WO-2004026874 (2004).
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ONO PHARMACEUTICALS CO LTD (Takaoka Y, Okamoto M, Genba Y, Ohie K): Novel crystals of triazaspiro[5.5]undecane derivative. WO-2004026874 (2004).
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78
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68549084396
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SCHERING-PLOUGH CORP (Palani A, Miller MA, Scott JD): Piperidine derivatives useful as CCR5 antagonists. US-00010008 (2004).
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SCHERING-PLOUGH CORP (Palani A, Miller MA, Scott JD): Piperidine derivatives useful as CCR5 antagonists. US-00010008 (2004).
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79
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68549093429
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SCHERING-PLOUGH CORP (Baroudu BM, Clader JW, Josien HB, McCombie SW, McKittrick BA, Miller MW, Neustadt BR, Palani A, Smith EM, Steensma R, Tagat JR et al): Piperazine derivatives useful as CCR5 antagonists. US-00069252 (2003).
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SCHERING-PLOUGH CORP (Baroudu BM, Clader JW, Josien HB, McCombie SW, McKittrick BA, Miller MW, Neustadt BR, Palani A, Smith EM, Steensma R, Tagat JR et al): Piperazine derivatives useful as CCR5 antagonists. US-00069252 (2003).
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80
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68549138468
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SCHERING-PLOUGH (Baroudu BM, Clader JW, Josien HB, McCombie SW, McKittrick BA, Miller MW, Neustadt BR, Palani A, Smith EM, Steensma R, Tagat JR et al): Piperidine derivatives useful as CCR5 antagonists. US-00004185 (2003).
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SCHERING-PLOUGH (Baroudu BM, Clader JW, Josien HB, McCombie SW, McKittrick BA, Miller MW, Neustadt BR, Palani A, Smith EM, Steensma R, Tagat JR et al): Piperidine derivatives useful as CCR5 antagonists. US-00004185 (2003).
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81
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68549095233
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SCHERING-PLOUGH CORP (Miller MW): CCR5 antagonists useful for treating AIDS. US-00008877 (2003).
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SCHERING-PLOUGH CORP (Miller MW): CCR5 antagonists useful for treating AIDS. US-00008877 (2003).
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82
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68549100706
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SCHERING-PLOUGH CORP (Palani A, Miller MA, Scott JD): Piperidine derivatives useful as CCR5 antagonists. WO-00020716 (2003).
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SCHERING-PLOUGH CORP (Palani A, Miller MA, Scott JD): Piperidine derivatives useful as CCR5 antagonists. WO-00020716 (2003).
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83
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68549105103
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SCHERING-PLOUGH CORP (Leong W, Chen M, D'Sa B, Zhu M, Xiao T, Shi X, Tang S, Gala S, Goodman A, Nielsen CM, Lee GM et al, The synthesis of piperidine and piperazine compounds as CCR5 antagonists. WO-00084950 2003
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SCHERING-PLOUGH CORP (Leong W, Chen M, D'Sa B, Zhu M, Xiao T, Shi X, Tang S, Gala S, Goodman A, Nielsen CM, Lee GM et al): The synthesis of piperidine and piperazine compounds as CCR5 antagonists. WO-00084950 (2003).
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84
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68549141020
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SCHERING-PLOUGH CORP (Dunning L, Jaroch S, Kochanny M, Lee W, Lian X, Liang M, Lu S-F, Onuffer J, Phillips G, Wei G-P, Ye B): Substituted quinoline CCR5 receptor antagonists. WO-00002960 (2004).
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SCHERING-PLOUGH CORP (Dunning L, Jaroch S, Kochanny M, Lee W, Lian X, Liang M, Lu S-F, Onuffer J, Phillips G, Wei G-P, Ye B): Substituted quinoline CCR5 receptor antagonists. WO-00002960 (2004).
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85
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68549126125
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MERCK & CO INC (Kim R, Chang J, Chapman KT, Mills SG): Modulators of CCR5 chemokine receptor activity. WO-03030898 (2003).
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MERCK & CO INC (Kim R, Chang J, Chapman KT, Mills SG): Modulators of CCR5 chemokine receptor activity. WO-03030898 (2003).
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86
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68549105101
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MERCK & CO INC (Willoughby CA, Matawan KR, Chapman KT, Mills SG, Shen D-M, Shu M): Pyrrolidine modulators of CCR5 chemokine receptor activity. US-06531484 (2003).
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MERCK & CO INC (Willoughby CA, Matawan KR, Chapman KT, Mills SG, Shen D-M, Shu M): Pyrrolidine modulators of CCR5 chemokine receptor activity. US-06531484 (2003).
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87
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68549129711
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MERCK & CO INC (Finke RE, Loebach JL, Maccross M, Mills SG): Cyclopentyl modulators of chemokine receptor activity. US-06506777 (2003).
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MERCK & CO INC (Finke RE, Loebach JL, Maccross M, Mills SG): Cyclopentyl modulators of chemokine receptor activity. US-06506777 (2003).
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88
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68549129539
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NORVARTIS-ERFINDUNGEN VERWALTUNGSGESELLSCHAFT GMBH (Albert R, Bruns C, Nuninger F, Streiff M, Thoma G, Zerwes H-G): Piperidine derivative chemokine receptor inhibitors useful for the treatment of inflammatory, allergic and autoimmune diseases. WO-02081449 (2002).
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NORVARTIS-ERFINDUNGEN VERWALTUNGSGESELLSCHAFT GMBH (Albert R, Bruns C, Nuninger F, Streiff M, Thoma G, Zerwes H-G): Piperidine derivative chemokine receptor inhibitors useful for the treatment of inflammatory, allergic and autoimmune diseases. WO-02081449 (2002).
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89
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68549141019
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TAKEDA CHEMICAL INDUSTRIES LTD (Shiraishi M, Baba M, Aikawa K, Kanzaki N, Seto M, Iizawa Y): Bicyclic compound, production and use thereof. WO-03014105 (2003).
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TAKEDA CHEMICAL INDUSTRIES LTD (Shiraishi M, Baba M, Aikawa K, Kanzaki N, Seto M, Iizawa Y): Bicyclic compound, production and use thereof. WO-03014105 (2003).
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90
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68549117893
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TAKEDA CHEMICAL INDUSTRIES LTD (Shiraishi M, Baba M, Seto M, Kanzaki N, Nishimura O): Cyclic compounds and uses thereof. US-06627651 (2003).
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TAKEDA CHEMICAL INDUSTRIES LTD (Shiraishi M, Baba M, Seto M, Kanzaki N, Nishimura O): Cyclic compounds and uses thereof. US-06627651 (2003).
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91
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68549102640
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TAKEDA C HEMICAL INDUSTRIES LTD (Imamura S, Hashiguchi S, Hattori T, Nishimura O, Kanzaki N, Baba M, Sugihara Y): Cyclic amine compounds as CCR5 antagonists. US-20030114443 (2003).
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TAKEDA C HEMICAL INDUSTRIES LTD (Imamura S, Hashiguchi S, Hattori T, Nishimura O, Kanzaki N, Baba M, Sugihara Y): Cyclic amine compounds as CCR5 antagonists. US-20030114443 (2003).
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92
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68549139124
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TAKEDA CHEMICAL INDUSTRIES LTD (Imamura S, Hashiguchi S, Hattori T, Nishimura O, Kanzaki N, Baba M, Sugihara Y): Cyclic amine compounds as CCR5 antagonists. US-06562978 (2003).
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TAKEDA CHEMICAL INDUSTRIES LTD (Imamura S, Hashiguchi S, Hattori T, Nishimura O, Kanzaki N, Baba M, Sugihara Y): Cyclic amine compounds as CCR5 antagonists. US-06562978 (2003).
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93
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68549139074
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ANORMED INC (Bridger GJ, Skerlj RT, Kaller A, Harwig C, Bogucki D, Wilson T, Crawford J, McEachern EJ, Atsma B, Nan S, Zhou Y et al, Novel heterocyclic compounds are modulators of chemokine receptors CXCR4 or CCR-5 useful for the treatment of HIV infection. WO-00222599 2002
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ANORMED INC (Bridger GJ, Skerlj RT, Kaller A, Harwig C, Bogucki D, Wilson T, Crawford J, McEachern EJ, Atsma B, Nan S, Zhou Y et al): Novel heterocyclic compounds are modulators of chemokine receptors CXCR4 or CCR-5 useful for the treatment of HIV infection. WO-00222599 (2002).
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94
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68549086113
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ASTRAZENECA AB (Cumming J, Winter J): Novel piperidinyl derivatives as CCR5 modulators, useful for the treatment of autoimmune, proliferative or immunologically-mediated diseases including transplant rejection and AIDS. WO-2004018425 (2004).
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ASTRAZENECA AB (Cumming J, Winter J): Novel piperidinyl derivatives as CCR5 modulators, useful for the treatment of autoimmune, proliferative or immunologically-mediated diseases including transplant rejection and AIDS. WO-2004018425 (2004).
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95
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68549105104
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ASTRAZENECA AB (Cumming J, Piperidine or 8-aza-bicyclo[3.2.1]oct-3-yl derivatives useful as modulators of chemokine receptor activity (especially CCR5, WO-03080574 2003
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ASTRAZENECA AB (Cumming J): Piperidine or 8-aza-bicyclo[3.2.1]oct-3-yl derivatives useful as modulators of chemokine receptor activity (especially CCR5). WO-03080574 (2003).
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96
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68549086114
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ASTRAZENECA AB (Tucker H): Preparation of N- piperidin-4-yl amides and ureas and their use as modulators of chemokine receptor activity (especially CCR5). WO-03042205 (2003).
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ASTRAZENECA AB (Tucker H): Preparation of N- piperidin-4-yl amides and ureas and their use as modulators of chemokine receptor activity (especially CCR5). WO-03042205 (2003).
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97
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68549127749
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ASTRAZENECA AB (Cumming J): Novel piperidine derivatives as modulators of chemokine CCR5 activity. WO-00042178 (2003).
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ASTRAZENECA AB (Cumming J): Novel piperidine derivatives as modulators of chemokine CCR5 activity. WO-00042178 (2003).
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98
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68549106812
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ASTRAZENECA AB (Cumming J, Tucker H): Piperidine derivatives and their use as modulators of chemokine CCR5 activity. WO-03042177 (2003).
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ASTRAZENECA AB (Cumming J, Tucker H): Piperidine derivatives and their use as modulators of chemokine CCR5 activity. WO-03042177 (2003).
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99
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68549087958
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ASTRAZENECA AB (Burrows J, Cumming J): Novel 3-[4-(phenylacetylamino)piperidin-1-yl]propane derivatives as chemokine receptor modulators useful for treating immune and inflammatory and inflammatory disorders and HIV infection. WO-02079156 (2002).
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ASTRAZENECA AB (Burrows J, Cumming J): Novel 3-[4-(phenylacetylamino)piperidin-1-yl]propane derivatives as chemokine receptor modulators useful for treating immune and inflammatory and inflammatory disorders and HIV infection. WO-02079156 (2002).
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100
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68549084397
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ASTRAZENECA AB (Burrows J, Cumming J): Novel N-acyl-N-(2-[4-(2-phenylacetylamino)piperidin-1-yl] ethyl)aniline derivatives. WO-02076948 (2002).
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ASTRAZENECA AB (Burrows J, Cumming J): Novel N-acyl-N-(2-[4-(2-phenylacetylamino)piperidin-1-yl] ethyl)aniline derivatives. WO-02076948 (2002).
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101
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68549091649
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SMITHKLINE B EECHAM CORP (Bondinell WE, Neeb MJ): Novel substituted benzanilides useful as CCR5 modulators for treating inflammatory and autoimmune diseases. WO-2004011427 (2004).
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SMITHKLINE B EECHAM CORP (Bondinell WE, Neeb MJ): Novel substituted benzanilides useful as CCR5 modulators for treating inflammatory and autoimmune diseases. WO-2004011427 (2004).
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102
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68549137534
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SMITHKLINE BEECHAM CORP (Bondinell WE, Neeb MJ): Novel substituted benzanilide compounds as CCR5 chemokine modulators useful for the treatment of inflammatory, autoimmune and other disorders. WO-2004010943 (2004).
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SMITHKLINE BEECHAM CORP (Bondinell WE, Neeb MJ): Novel substituted benzanilide compounds as CCR5 chemokine modulators useful for the treatment of inflammatory, autoimmune and other disorders. WO-2004010943 (2004).
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