Inhibiting the deubiquitinating enzymes (DUBs)

Journal of Medicinal Chemistry

Volumn 58, Issue 4, 2015, Pages 1581-1595

  Ndubaku, Chudi ^a   Tsui, Vickie ^a  

^a GENENTECH INC   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

DEUBIQUITINATING ENZYME INHIBITOR; SMALL MOLECULE TRANSPORT AGENT; UNCLASSIFIED DRUG; DEUBIQUITINASE; ENZYME INHIBITOR;

DRUG IDENTIFICATION; DRUG POTENCY; DRUG SCREENING; DRUG STRUCTURE; HUMAN; NONHUMAN; REVIEW; VALIDATION STUDY; ANTAGONISTS AND INHIBITORS; CHEMICAL STRUCTURE; CHEMISTRY; DRUG DEVELOPMENT; METABOLISM; STRUCTURE ACTIVITY RELATION; X RAY CRYSTALLOGRAPHY;

CRYSTALLOGRAPHY, X-RAY; DRUG DISCOVERY; ENZYME INHIBITORS; HUMANS; MODELS, MOLECULAR; MOLECULAR STRUCTURE; STRUCTURE-ACTIVITY RELATIONSHIP; UBIQUITIN-SPECIFIC PROTEASES;

EID: 84924082223     PISSN: 00222623     EISSN: 15204804     Source Type: Journal    
DOI: 10.1021/jm501061a     Document Type: Review

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