Molecular pharmacology of store-operated CRAC channels

Channels

Volumn 7, Issue 5, 2013, Pages 402-414

  Jairaman, Amit ^a   Prakriya, Murali ^a  

^a NORTHWESTERN UNIVERSITY   (United States)

Author keywords

CRAC channel; Orai1; Pharmacology; SOCE; STIM1

Indexed keywords

1 (5 CHLORO 1 NAPHTHALENESULFONYL)HEXAHYDRO 1H 1,4 DIAZEPINE; 1 [2 (4 METHOXYPHENYL) 2 [3 (4 METHOXYPHENYL)PROPOXY]ETHYL] 1H IMIDAZOLE; 2 AMINOETHYLDIPHENYL BORATE; CALCIUM ION; CALCIUM RELEASE ACTIVATED CALCIUM CHANNEL; CALCIUM RELEASE ACTIVATED CALCIUM CHANNEL 1; CM 2489; CM 3457; DPB 162AE; DPB 163AE; ECONAZOLE; GSK 5503A; GSK 7975A; IMIDAZOLE DERIVATIVE; LANTHANIDE; MICONAZOLE; PYRAZOLE DERIVATIVE; RO 2959; STROMAL INTERACTION MOLECULE 1; SYNTA 66; TRANSCRIPTION FACTOR NFAT; UNCLASSIFIED DRUG;

ARTICLE; AUTOIMMUNITY; BINDING AFFINITY; BINDING SITE; CELL MEMBRANE; CHANNEL GATING; CONCENTRATION (PARAMETERS); CONFORMATIONAL TRANSITION; CRYSTAL STRUCTURE; CYTOSOL; DIMERIZATION; DRUG MECHANISM; ENDOPLASMIC RETICULUM; GENE OVEREXPRESSION; IC 50; INFLAMMATORY BOWEL DISEASE; MOLECULAR SENSOR; NONHUMAN; NOSE POLYP; OLIGOMERIZATION; PHARMACOLOGY; POINT MUTATION; PROTEIN DEPHOSPHORYLATION; PROTEIN PROTEIN INTERACTION; RNA INTERFERENCE; SEVERE COMBINED IMMUNODEFICIENCY;

CRAC CHANNEL; ORAI1; PHARMACOLOGY; SOCE; STIM1;

ANIMALS; CALCIUM CHANNEL BLOCKERS; CALCIUM CHANNELS; CALCIUM SIGNALING; ENDOPLASMIC RETICULUM; HUMANS; MEMBRANE PROTEINS; NEOPLASM PROTEINS; PROTEIN CONFORMATION;

EID: 84892148550     PISSN: 19336950     EISSN: 19336969     Source Type: Journal    
DOI: 10.4161/chan.25292     Document Type: Article

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