Novel designer receptors to probe GPCR signaling and physiology

Trends in Pharmacological Sciences

Volumn 34, Issue 7, 2013, Pages 385-392

  Wess, Jürgen ^a   Nakajima, Kenichiro ^a   Jain, Shalini ^a  

^a NATIONAL INSTITUTE OF DIABETES AND DIGESTIVE AND KIDNEY DISEASES   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

ACETYLCHOLINE; CLOZAPINE; CLOZAPINE N OXIDE; DESIGNER DRUG; DESIGNER RECEPTOR; DESIGNER RECEPTORS EXCLUSIVELY ACTIVATED BY DESIGNER DRUG; G PROTEIN COUPLED RECEPTOR; MUSCARINIC RECEPTOR; RETINA S ANTIGEN; TIOTROPIUM BROMIDE; UNCLASSIFIED DRUG;

BIOTECHNOLOGY; DRUG EFFICACY; DRUG HALF LIFE; DRUG METABOLISM; DRUG POTENCY; HUMAN; IN VIVO STUDY; MOLECULAR DOCKING; MOLECULAR INTERACTION; NONHUMAN; PRIORITY JOURNAL; PROTEIN EXPRESSION; PROTEIN FUNCTION; RECEPTOR BINDING; REVIEW; SIGNAL TRANSDUCTION;

ANIMALS; HUMANS; LIGANDS; MEMBRANE TRANSPORT MODULATORS; MODELS, MOLECULAR; MOLECULAR STRUCTURE; PROTEIN CONFORMATION; RECEPTORS, G-PROTEIN-COUPLED; SIGNAL TRANSDUCTION; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 84879787863     PISSN: 01656147     EISSN: 18733735     Source Type: Journal    
DOI: 10.1016/j.tips.2013.04.006     Document Type: Review

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