-
1
-
-
67650230587
-
Irreversible inhibition of serine proteasesdesign and in vivo activity of diaryl α-aminophosphonate derivatives
-
Sieαczyk, M.; Oleksyszyn, J. Irreversible inhibition of serine proteasesdesign and in vivo activity of diaryl α-aminophosphonate derivatives. Curr. Med. Chem. 2009, 16, 1673-1687.
-
(2009)
Curr. Med. Chem.
, vol.16
, pp. 1673-1687
-
-
Sieαczyk, M.1
Oleksyszyn, J.2
-
2
-
-
0003563365
-
-
Aminophosphonic and Aminophosphinic Acids., Kukhar, VP.; Hudson, H, R., Eds.; John Wiley & Sons: Chichester, UK
-
Aminophosphonic and Aminophosphinic Acids. Chemistry and Biological Activity; Kukhar, V. P.; Hudson, H. R., Eds.; John Wiley & Sons: Chichester, UK, 2000.
-
(2000)
Chemistry and Biological Activity
-
-
-
3
-
-
84913150907
-
Biological activity of aminophosphonic acids. βPhosphorus, Sulfur Silicon Relat
-
Kafarski, P.; Lejczak, B. Biological activity of aminophosphonic acids. βPhosphorus, Sulfur Silicon Relat. Elem. 1991, 63, 193-215.
-
(1991)
Elem.
, vol.63
, pp. 193-215
-
-
Kafarski, P.1
Lejczak, B.2
-
4
-
-
0000899405
-
Optically active 1-aminoalkylphosphonic acids
-
Dhawan, B.; Redmore, D. Optically active 1-aminoalkylphosphonic acids. Phosphorus Sulfur 1987, 32, 119-144.
-
(1987)
Phosphorus Sulfur
, vol.32
, pp. 119-144
-
-
Dhawan, B.1
Redmore, D.2
-
5
-
-
0347625851
-
Contribution of molecular modeling and site-directed mutagenesis to the identification of a new residue, glutamate 215, involve in the exopeptidase specificity of aminopeptidase A
-
Rozenfeld, R.; Iturrioz, X.; Okada, M.; Maigret, B.; Llorents-Cortes, C. Contribution of molecular modeling and site-directed mutagenesis to the identification of a new residue, glutamate 215, involve in the exopeptidase specificity of aminopeptidase A. Biochemistry 2003, 42, 14785-14793.
-
(2003)
Biochemistry
, vol.42
, pp. 14785-14793
-
-
Rozenfeld, R.1
Iturrioz, X.2
Okada, M.3
Maigret, B.4
Llorents-Cortes, C.5
-
6
-
-
0030818538
-
Phosphonate diester and phosphonamide synthesis Reaction coordinate analysis by 31P NMR spectroscopy: Identification of pyrophosphonate anhydrides and highly reactive phosphonylammonium salts
-
Hirschmann, R.; Yager, K. M.; Taylor, C. M.; Witherington, J.; Sprengler, P. A.; Phillips, B. W.; Moore, W.; Smith, III, A. B. Phosphonate diester and phosphonamide synthesis. Reaction coordinate analysis by 31P NMR spectroscopy: identification of pyrophosphonate anhydrides and highly reactive phosphonylammonium salts. J. Am. Chem. Soc. 1997, 119, 8177-8190.
-
(1997)
J. Am. Chem. Soc.
, vol.119
, pp. 8177-8190
-
-
Hirschmann, R.1
Yager, K.M.2
Taylor, C.M.3
Witherington, J.4
Sprengler, P.A.5
Phillips, B.W.6
Moore, W.7
Smith III, A.B.8
-
7
-
-
0028131354
-
Peptide synthesis catalyzed by an antibody containing a binding site for variable amino acids
-
Hirschmann, R.; Smith, III, A. B.; Taylor, C. M.; Benkovic, P. A.; Taylor, S. D.; Yager, K. M.; Sprengler, P. A.; Benkovic, S. J. Peptide synthesis catalyzed by an antibody containing a binding site for variable amino acids. Science 1994, 265, 234-237.
-
(1994)
Science
, vol.265
, pp. 234-237
-
-
Hirschmann, R.1
Smith III, A.B.2
Taylor, C.M.3
Benkovic, P.A.4
Taylor, S.D.5
Yager, K.M.6
Sprengler, P.A.7
Benkovic, S.J.8
-
8
-
-
0025979246
-
Irreversible inhibition of serine proteases by peptide derivatives of (α-aminoalkyl)phosphonate diphenyl esters
-
Oleksyszyn, J.; Powers, J. C. Irreversible inhibition of serine proteases by peptide derivatives of (α-aminoalkyl)phosphonate diphenyl esters. Biochemistry 1991, 30, 485-493.
-
(1991)
Biochemistry
, vol.30
, pp. 485-493
-
-
Oleksyszyn, J.1
Powers, J.C.2
-
9
-
-
0024409372
-
Renin inhibitors Synthesis of transition-state analog inhibitors containing phosphorus acid derivatives at the scissile bond
-
Allen, M. C.; Fuhrer, W.; Tuck, B.; Wade, R.; Wood, J. M. Renin inhibitors. Synthesis of transition-state analog inhibitors containing phosphorus acid derivatives at the scissile bond. J. Med. Chem. 1989, 32, 1652-1661.
-
(1989)
J. Med. Chem.
, vol.32
, pp. 1652-1661
-
-
Allen, M.C.1
Fuhrer, W.2
Tuck, B.3
Wade, R.4
Wood, J.M.5
-
10
-
-
0023277991
-
Phosphorus amino acid analogues as inhibitors of leucine aminopeptidase
-
Giannousis, P. P.; Bartlett, P. A. Phosphorus amino acid analogues as inhibitors of leucine aminopeptidase. J. Med. Chem. 1987, 30, 1603-1609.
-
(1987)
J. Med. Chem.
, vol.30
, pp. 1603-1609
-
-
Giannousis, P.P.1
Bartlett, P.A.2
-
11
-
-
0141786949
-
Rapid parallel synthesis of dipeptide diphenyl phosphonate esters as inhibitors of dipeptidyl peptidases
-
For some examples on the synthesis of phosphono-peptides see
-
For some examples on the synthesis of phosphono-peptides see Senten, K.; Daniëls, L.; Van der Veken, P.; De Meester, I.; Lambeir, A.-M.; Scharpé, S.; Haemers, A.; Augustyns, K. Rapid parallel synthesis of dipeptide diphenyl phosphonate esters as inhibitors of dipeptidyl peptidases. J. Comb. Chem. 2003, 5, 336-344.
-
(2003)
J. Comb. Chem.
, vol.5
, pp. 336-344
-
-
Senten, K.1
Daniëls, L.2
van der Veken, P.3
de Meester, I.4
Lambeir, A.-M.5
Scharpé, S.6
Haemers, A.7
Augustyns, K.8
-
12
-
-
0035945011
-
Polymer-assisted solution-phase parallel synthesis of dipeptide p-nitroanilides and dipeptide diphenyl phosphonates
-
Senten, K.; Van der Veken, P.; Bal. G.; Hae mers, A.; Augustyns, K. Polymer-assisted solution-phase parallel synthesis of dipeptide p-nitroanilides and dipeptide diphenyl phosphonates. Tetrahedron Lett. 2001, 42, 9135-9138.
-
(2001)
Tetrahedron Lett.
, vol.42
, pp. 9135-9138
-
-
Senten, K.1
van der Veken, P.2
Bal, G.3
Hae mers, A.4
Augustyns, K.5
-
13
-
-
0035906032
-
OEthyl 1-azidoalkylphosphonic acids-versatile reagents for the synthesis of protected phosphonamidate peptides
-
Sikora, D.; Nonas, T.; Gajda, T. OEthyl 1-azidoalkylphosphonic acids-versatile reagents for the synthesis of protected phosphonamidate peptides. Tetrahedron 2001, 57, 1619-1625.
-
(2001)
Tetrahedron
, vol.57
, pp. 1619-1625
-
-
Sikora, D.1
Nonas, T.2
Gajda, T.3
-
14
-
-
0028134093
-
Solid-phase synthesis of peptidylphosphonates
-
Cambell, D. A.; Bermak, J. C. Solid-phase synthesis of peptidylphosphonates. J. Am. Chem. Soc. 1994, 116, 6039-6040.
-
(1994)
J. Am. Chem. Soc.
, vol.116
, pp. 6039-6040
-
-
Cambell, D.A.1
Bermak, J.C.2
-
15
-
-
33845278913
-
Synthesis of phosphonic acid derivatives by oxidative activation of phosphinate esters
-
Sampson, N. S.; Batlett, P. A. Synthesis of phosphonic acid derivatives by oxidative activation of phosphinate esters. J. Org. Chem. 1988, 53, 4500-4503.
-
(1988)
J. Org. Chem.
, vol.53
, pp. 4500-4503
-
-
Sampson, N.S.1
Batlett, P.A.2
-
16
-
-
0020616474
-
Phosphonopeptides as substrates for peptide transport systems and peptidases of Escherichia coli
-
Atherton, F. R.; Hall, M. J.; Hassall, C. H.; Lambert, R. W.; Lloyd, W. J.; Lord, A. V.; Ringrose, P. S.; Westmacott, D. Phosphonopeptides as substrates for peptide transport systems and peptidases of Escherichia coli. Antimicrob. Agents Chemother. 1983, 24, 522-528.
-
(1983)
Antimicrob. Agents Chemother.
, vol.24
, pp. 522-528
-
-
Atherton, F.R.1
Hall, M.J.2
Hassall, C.H.3
Lambert, R.W.4
Lloyd, W.J.5
Lord, A.V.6
Ringrose, P.S.7
Westmacott, D.8
-
17
-
-
0020400143
-
Antibacterial activity and mechanism of action of phosphonopeptides based on aminomethylphosphonic acid
-
Atherton, F. R.; Hall, M. J.; Hassall, C. H.; Lambert, R. W.; Lloyd, W. J.; Ringrose, P. S.; Westmacott, D. Antibacterial activity and mechanism of action of phosphonopeptides based on aminomethylphosphonic acid. Antimicrob. Agents Chemother. 1982, 22, 571-578.
-
(1982)
Antimicrob. Agents Chemother.
, vol.22
, pp. 571-578
-
-
Atherton, F.R.1
Hall, M.J.2
Hassall, C.H.3
Lambert, R.W.4
Lloyd, W.J.5
Ringrose, P.S.6
Westmacott, D.7
-
18
-
-
0001700634
-
Studies on the synthesis of chemotherapeutics. Part XI Synthesis and antibacterial activities of phosphono-peptides
-
Kametani, T.; Kigasawa, K.; Hiiragi, M.; Wakisaka, K.; Haga, S.; Sugi, H.; Tanigawa, K.; Suzuki, Y.; Fukawa, K.; Irino, O.; Saita, O.; Yamabe, S. Studies on the synthesis of chemotherapeutics. Part XI. Synthesis and antibacterial activities of phosphono-peptides. Heterocycles 1981, 16, 1205-1241.
-
(1981)
Heterocycles
, vol.16
, pp. 1205-1241
-
-
Kametani, T.1
Kigasawa, K.2
Hiiragi, M.3
Wakisaka, K.4
Haga, S.5
Sugi, H.6
Tanigawa, K.7
Suzuki, Y.8
Fukawa, K.9
Irino, O.10
Saita, O.11
Yamabe, S.12
-
19
-
-
0034083373
-
Synthesis of N-alkyl-(α-aminoalkyl)phosphine oxides and phosphonic esters as potential HIVprotease inhibitors, starting from α-aminoacids
-
Alonso, E.; Solis, A.; del Pozo, C. Synthesis of N-alkyl-(α-aminoalkyl)phosphine oxides and phosphonic esters as potential HIVprotease inhibitors, starting from α-aminoacids. Synlett 2000, 698-700.
-
(2000)
Synlett
, pp. 698-700
-
-
Alonso, E.1
Solis, A.2
del Pozo, C.3
-
21
-
-
0026438772
-
Synthesis of stereochemically defined phosphonamidate-containing peptides: Inhibitors for the HIV-1 proteinase
-
Camp, N. P.; Hawkins, P. C. D.; Hitchcock, P. B.; Gani, D. Synthesis of stereochemically defined phosphonamidate-containing peptides: inhibitors for the HIV-1 proteinase. Bioorg. Med. Chem. Lett. 1992, 2, 1047-1052.
-
(1992)
Bioorg. Med. Chem. Lett.
, vol.2
, pp. 1047-1052
-
-
Camp, N.P.1
Hawkins, P.C.D.2
Hitchcock, P.B.3
Gani, D.4
-
22
-
-
0017853042
-
Phosphonopeptides, a new class of synthetic antibacterial agents
-
Allen, J. G.; Atherton, F. R.; Hall, M. J.; Hassall, C. H.; Holmes, S. W.; Lambert, R. W.; Nisbet, L. J.; Ringrose, P. S. Phosphonopeptides, a new class of synthetic antibacterial agents. Nature 1978, 272, 56-58.
-
(1978)
Nature
, vol.272
, pp. 56-58
-
-
Allen, J.G.1
Atherton, F.R.2
Hall, M.J.3
Hassall, C.H.4
Holmes, S.W.5
Lambert, R.W.6
Nisbet, L.J.7
Ringrose, P.S.8
-
23
-
-
0022577081
-
Synthesis and structure-activity relationships of antibacterial phosphonopeptides incorporating (1-aminoethyl)phosphonic acid and (aminomethyl)phosphonic acid
-
Atherton, F. R.; Hassall, C. H.; Lambert, R. W. Synthesis and structure-activity relationships of antibacterial phosphonopeptides incorporating (1-aminoethyl)phosphonic acid and (aminomethyl)phosphonic acid. J. Med. Chem. 1986, 29, 29-40.
-
(1986)
J. Med. Chem.
, vol.29
, pp. 29-40
-
-
Atherton, F.R.1
Hassall, C.H.2
Lambert, R.W.3
-
24
-
-
0023034922
-
Antibacterial activity of phosphonodipeptides related to alafosfalin
-
Lejczak, B.; Kafarski, P.; Sztajer, H.; Mastalerz, P. Antibacterial activity of phosphonodipeptides related to alafosfalin. J. Med. Chem. 1986, 29, 2212-2217.
-
(1986)
J. Med. Chem.
, vol.29
, pp. 2212-2217
-
-
Lejczak, B.1
Kafarski, P.2
Sztajer, H.3
Mastalerz, P.4
-
25
-
-
31544482713
-
Prodrug forms of N-[(4-deoxy-4-amino-10-methyl)pteroyl]glutamate-γ-[ωP(O)(OH)]-glutarate, a potent inhibitor of folypoly-γ-glutamate synthetase: Synthesis and hydrolytic stability
-
Feng, Y.; Coward, J. K. Prodrug forms of N-[(4-deoxy-4-amino-10-methyl)pteroyl]glutamate-γ-[ωP(O)(OH)]-glutarate, a potent inhibitor of folypoly-γ-glutamate synthetase: synthesis and hydrolytic stability. J. Med. Chem. 2006, 49, 770-788.
-
(2006)
J. Med. Chem.
, vol.49
, pp. 770-788
-
-
Feng, Y.1
Coward, J.K.2
-
26
-
-
0001624368
-
Aminophosphonic acids of potential medical importance
-
Kafarski, P.; Lejczak, B. Aminophosphonic acids of potential medical importance. Curr. Med. Chem. 2001, 1, 301-312.
-
(2001)
Curr. Med. Chem.
, vol.1
, pp. 301-312
-
-
Kafarski, P.1
Lejczak, B.2
-
27
-
-
0025879040
-
New α-aminophosphonic acid derivatives of vinblastine: Chemistry and antitumor activity
-
Lavielle, G.; Hautefaye, P.; Schaeffer, C.; Boutin, J. A.; Cudennec, C. A.; Pierré, A. New α-aminophosphonic acid derivatives of vinblastine: chemistry and antitumor activity. J. Med. Chem. 1991, 34, 1998-2003.
-
(1991)
J. Med. Chem.
, vol.34
, pp. 1998-2003
-
-
Lavielle, G.1
Hautefaye, P.2
Schaeffer, C.3
Boutin, J.A.4
Cudennec, C.A.5
Pierré, A.6
-
28
-
-
0034499290
-
An overview of recent advances on the synthesis and biological activity of α-aminophosphonic acid derivatives
-
Huang, J.; Chen, R. An overview of recent advances on the synthesis and biological activity of α-aminophosphonic acid derivatives. Heteroatom. Chem. 2000, 11, 480-492.
-
(2000)
Heteroatom. Chem.
, vol.11
, pp. 480-492
-
-
Huang, J.1
Chen, R.2
-
29
-
-
82855179830
-
Organic phosphorus compounds: Preparation, physical and biological properties of aminoarylmethylphosphonic and phosphonous acids
-
Maier, L.; Diel, P. J. Organic phosphorus compounds: preparation, physical and biological properties of aminoarylmethylphosphonic and phosphonous acids. Phosphorus, Sulfur Silicon Relat. Elem. 1991, 57, 57-64.
-
(1991)
Phosphorus, Sulfur Silicon Relat. Elem.
, vol.57
, pp. 57-64
-
-
Maier, L.1
Diel, P.J.2
-
30
-
-
0001570391
-
Binding ability of pesticides X-ray, spectroscopic, and polarographic studies of the copper (II) interaction with acifluorfen
-
Kozlowski, H.; Pusino, A.; Swiatek, J.; Spychala, J.; Glowiak, T.; Micera, G.; Gessa, C. Binding ability of pesticides. X-ray, spectroscopic, and polarographic studies of the copper (II) interaction with acifluorfen. J. Agric. Food Chem. 1990, 38, 1989-1992.
-
(1990)
J. Agric. Food Chem.
, vol.38
, pp. 1989-1992
-
-
Kozlowski, H.1
Pusino, A.2
Swiatek, J.3
Spychala, J.4
Glowiak, T.5
Micera, G.6
Gessa, C.7
-
31
-
-
0036420749
-
Antioxidative activity of some phenoxy and organophosphorous compounds
-
Nska, H.; Bonarska, D.; Bielecki, K.; Sarapuk, J. Antioxidative activity of some phenoxy and organophosphorous compounds. Cell. Mol. Biol. Lett. 2002, 7, 929-935.
-
(2002)
Cell. Mol. Biol. Lett.
, vol.7
, pp. 929-935
-
-
Nska, H.1
Bonarska, D.2
Bielecki, K.3
Sarapuk, J.4
-
32
-
-
0040931016
-
Synthesis and properties of a novel aminophosphonic acid as an extracting agent for metals
-
Jagodic, V.; Herak, M. J. Synthesis and properties of a novel aminophosphonic acid as an extracting agent for metals. J. Inorg. Nucl. Chem. 1970, 32, 1323-1332.
-
(1970)
J. Inorg. Nucl. Chem.
, vol.32
, pp. 1323-1332
-
-
Jagodic, V.1
Herak, M.J.2
-
33
-
-
0141506639
-
Transition metal complexes of dialkyl α-hydroxyiminophosphonates, a novel class of metal complexes
-
and references cited therein
-
Bligh, S. W. A.; Choi, N.; Green, D. St. C.; Hudson, H. R.; McGrath, C. M.; McPartlin, M.; Pianka, M. Transition metal complexes of dialkyl α-hydroxyiminophosphonates, a novel class of metal complexes. Polyhedron 1993, 12, 2887-2890 and references cited therein.
-
(1993)
Polyhedron
, vol.12
, pp. 2887-2890
-
-
Bligh, S.W.A.1
Choi, N.2
StGreen, D.C.3
Hudson, H.R.4
McGrath, C.M.5
McPartlin, M.6
Pianka, M.7
-
34
-
-
0001576843
-
-
In, Priest, N. O.; Van de Vyver, F. L. Eds., CRC Press: Boca Raton, FL
-
Bulman, R. A. In Trace Metals and Fluoride in Bones and Teeth, Priest, N. O.; Van de Vyver, F. L. Eds., CRC Press: Boca Raton, FL, 1990; p. 271.
-
(1990)
Trace Metals and Fluoride in Bones and Teeth
, pp. 271
-
-
Bulman, R.A.1
-
35
-
-
1542690351
-
Phosphonates as analogues of natural phosphates
-
Engel, R. Phosphonates as analogues of natural phosphates. Chem. Rev. 1977, 77, 349-367.
-
(1977)
Chem. Rev.
, vol.77
, pp. 349-367
-
-
Engel, R.1
-
36
-
-
56949101063
-
An overview of stereoselective synthesis of α-aminophosphonic acids and derivatives
-
Ordóñez, M.; Rojas-Cabrera, H.; Cativiela, C. An overview of stereoselective synthesis of α-aminophosphonic acids and derivatives. Tetrahedron 2009, 65, 17-49.
-
(2009)
Tetrahedron
, vol.65
, pp. 17-49
-
-
Ordóñez, M.1
Rojas-Cabrera, H.2
Cativiela, C.3
-
37
-
-
47749154512
-
Some potential chiral catalysts for preparation of asymmetric α-aminophosphonates
-
Bhadury, P. S.; Song, B.-A.; Yang, S.; Zhang, Y.; Zhang, S. Some potential chiral catalysts for preparation of asymmetric α-aminophosphonates. Curr. Org. Synth. 2008, 5, 134-150.
-
(2008)
Curr. Org. Synth.
, vol.5
, pp. 134-150
-
-
Bhadury, P.S.1
Song, B.-A.2
Yang, S.3
Zhang, Y.4
Zhang, S.5
-
38
-
-
49249117085
-
Catalytic enantioselective hydrophosphonylation of aldehydes and imines
-
Merino, P.; Marqués-López, E.; Herrera, R. P. Catalytic enantioselective hydrophosphonylation of aldehydes and imines. Adv. Synth. Catal. 2008, 350, 1195-1208.
-
(2008)
Adv. Synth. Catal.
, vol.350
, pp. 1195-1208
-
-
Merino, P.1
Marqués-López, E.2
Herrera, R.P.3
-
39
-
-
33745390196
-
Catalytic asymmetric synthesis of α-and α-aminoalkanephosphonic acid derivatives
-
Ma, J.-A. Catalytic asymmetric synthesis of α-and α-aminoalkanephosphonic acid derivatives. Chem. Soc. Rev. 2006, 35, 630-636.
-
(2006)
Chem. Soc. Rev.
, vol.35
, pp. 630-636
-
-
Ma, J.-A.1
-
40
-
-
0008307835
-
Synthesis of racemic and optically active α-aminophosphonic acids
-
Uziel, J.; Genêt, J. P. Synthesis of racemic and optically active α-aminophosphonic acids. Russ. J. Org. Chem. 1997, 33, 1521-1542.
-
(1997)
Russ. J. Org. Chem.
, vol.33
, pp. 1521-1542
-
-
Uziel, J.1
Genêt, J.P.2
-
41
-
-
84953500772
-
Asymmetric synthesis of phosphorus analogs of amino acids
-
Kukhar, V. P.; Soloshonok, V. A.; Solodenko, V. A. Asymmetric synthesis of phosphorus analogs of amino acids. Phosphorus, Sulfur Silicon Relat. Elem. 1994, 92, 239-264.
-
(1994)
Phosphorus, Sulfur Silicon Relat. Elem.
, vol.92
, pp. 239-264
-
-
Kukhar, V.P.1
Soloshonok, V.A.2
Solodenko, V.A.3
-
42
-
-
0042665702
-
Stereoselective synthesis of 1-aminoalkanephosphonic acids with two chiral centers and their activity towards leucine aminopeptidase
-
Drag, M.; Pawelczak, M.; Kafarski, P. Stereoselective synthesis of 1-aminoalkanephosphonic acids with two chiral centers and their activity towards leucine aminopeptidase. Chirality 2003, 15, S104-S107.
-
(2003)
Chirality
, vol.15
-
-
Drag, M.1
Pawelczak, M.2
Kafarski, P.3
-
43
-
-
0013610276
-
1-Aminoalkylphosphonous acids. Part 1. Isosteres of the protein amino acids
-
Baylis, E. K.; Campbell, C. D.; Dingwall, J. G. 1-Aminoalkylphosphonous acids. Part 1. Isosteres of the protein amino acids. J. Chem. Soc., Perkin Trans 1 1984, 2845-2853.
-
(1984)
J. Chem. Soc., Perkin Trans 1
, pp. 2845-2853
-
-
Baylis, E.K.1
Campbell, C.D.2
Dingwall, J.G.3
-
44
-
-
0018774396
-
Phosphonopeptides as antibacterial agents: Mechanism of action of alaphosphin
-
Atherton, F. R.; Hall, M. J.; Hassall, C. H.; Lambert, R. W.; Lloyd, W. J.; Ringrose, P. S. Phosphonopeptides as antibacterial agents: mechanism of action of alaphosphin. Antimicrob. Agents Chemother. 1979, 15, 696-705.
-
(1979)
Antimicrob. Agents Chemother.
, vol.15
, pp. 696-705
-
-
Atherton, F.R.1
Hall, M.J.2
Hassall, C.H.3
Lambert, R.W.4
Lloyd, W.J.5
Ringrose, P.S.6
-
45
-
-
84861165589
-
Glyphosate, weed control methods Handbook
-
Tu, M.; Hurd, C.; Robinson, R.; Randall, J. M. Glyphosate, weed control methods. Handbook. Nat. Conservancy 2001, 11, 123-144.
-
(2001)
Nat. Conservancy
, vol.11
, pp. 123-144
-
-
Tu, M.1
Hurd, C.2
Robinson, R.3
Randall, J.M.4
-
46
-
-
0034792021
-
The membrane-disrupting activity of α-aminoalkanephosphonic acids and their derivatives
-
and references cited therein
-
Deron, A.; Dziamska, A.; Pawlaczyk, I.; Bielecki, K.; Kleszczyska, H.; Gancarz, R.; Sarapuk, J. The membrane-disrupting activity of α-aminoalkanephosphonic acids and their derivatives. Cell. Mol. Biol. Lett. 2001, 6, 291-297 and references cited therein.
-
(2001)
Cell. Mol. Biol. Lett.
, vol.6
, pp. 291-297
-
-
Deron, A.1
Dziamska, A.2
Pawlaczyk, I.3
Bielecki, K.4
Kleszczyska, H.5
Gancarz, R.6
Sarapuk, J.7
-
47
-
-
41849092226
-
Aminomethylphosphonic acid accumulation in plant species trated with glyphosate
-
Reddy, K. N.; Rimando, A. M.; Duke, S. O.; Nandula, V. K. Aminomethylphosphonic acid accumulation in plant species trated with glyphosate. J. Agric. Food Chem. 2008, 56, 2125-2130.
-
(2008)
J. Agric. Food Chem.
, vol.56
, pp. 2125-2130
-
-
Reddy, K.N.1
Rimando, A.M.2
Duke, S.O.3
Nandula, V.K.4
-
48
-
-
0037226084
-
Isoflavone, glyphosate, and aminomethyl-phosphonic acid levels in seeds of glyphosate-treated, glyphosateresistant soybean
-
Duke, S. O.; Rimando, A. M.; Pace, P. F.; Reddy, K. N.; Smeda, R. J. Isoflavone, glyphosate, and aminomethyl-phosphonic acid levels in seeds of glyphosate-treated, glyphosateresistant soybean. J. Agric. Food Chem. 2003, 51, 340-344.
-
(2003)
J. Agric. Food Chem.
, vol.51
, pp. 340-344
-
-
Duke, S.O.1
Rimando, A.M.2
Pace, P.F.3
Reddy, K.N.4
Smeda, R.J.5
-
49
-
-
0037716457
-
Simultaneous analysis of biologically active aminoalkanephosphonic acids
-
and references cited therein
-
Kudzin, Z. H.; Gralak, D. K.; Adrijewski, G.; Drabowicz, J.; Uczak, J. Simultaneous analysis of biologically active aminoalkanephosphonic acids. J. Chromatogr. A 2003, 998, 183-199 and references cited therein.
-
(2003)
J. Chromatogr. A
, vol.998
, pp. 183-199
-
-
Kudzin, Z.H.1
Gralak, D.K.2
Adrijewski, G.3
Drabowicz, J.4
Uczak, J.5
-
50
-
-
0034628537
-
Potent and selective nonpeptidic inhibitors of endothelin-converting enzyme-1 with sustained duration of action
-
De Lombaert, S.; Blanchard, L.; Stamford, L. B.; Tan, J.; Wallace, E. M.; Satoh, Y.; Fitt, J.; Hoyer, D.; Simonsbergen, D.; Moliterni, J.; Marcopoulos, N.; Savage, P.; Chou, M.; Trapani, A. J.; Jeng, A. Y. Potent and selective nonpeptidic inhibitors of endothelin-converting enzyme-1 with sustained duration of action. J. Med. Chem. 2000, 43, 488-504.
-
(2000)
J. Med. Chem.
, vol.43
, pp. 488-504
-
-
de Lombaert, S.1
Blanchard, L.2
Stamford, L.B.3
Tan, J.4
Wallace, E.M.5
Satoh, Y.6
Fitt, J.7
Hoyer, D.8
Simonsbergen, D.9
Moliterni, J.10
Marcopoulos, N.11
Savage, P.12
Chou, M.13
Trapani, A.J.14
Jeng, A.Y.15
-
51
-
-
0030818538
-
Phosphonate diester and phosphonamide synthesis Reaction coordinate analysis by 31P NMR spectroscopy: Identification of pyrophosphonate anhydrides and highly reactive phosphonylammonium salts
-
Hirschmann, R.; Yager, K. M.; Taylor, C. M.; Witherington, J.; Sprengler, P. A.; Phillips, B. W.; Moore, W.; Smith, III, A. B. Phosphonate diester and phosphonamide synthesis. Reaction coordinate analysis by 31P NMR spectroscopy: identification of pyrophosphonate anhydrides and highly reactive phosphonylammonium salts. J. Am. Chem. Soc. 1997, 119, 8177-8190.
-
(1997)
J. Am. Chem. Soc.
, vol.119
, pp. 8177-8190
-
-
Hirschmann, R.1
Yager, K.M.2
Taylor, C.M.3
Witherington, J.4
Sprengler, P.A.5
Phillips, B.W.6
Moore, W.7
Smith III, A.B.8
-
52
-
-
0001718823
-
Peptides containing aminophosphonic acids 3. Synthesis of tripeptide containing aminomethylphosphonic acid
-
Yamauchi, K.; Mitsuda, Y.; Kinoshita, M. Peptides containing aminophosphonic acids 3. Synthesis of tripeptide containing aminomethylphosphonic acid. Bull. Chem. Soc. Jpn. 1975, 48, 3285-3286.
-
(1975)
Bull. Chem. Soc. Jpn.
, vol.48
, pp. 3285-3286
-
-
Yamauchi, K.1
Mitsuda, Y.2
Kinoshita, M.3
-
53
-
-
0000185336
-
Peptides containing aminophosphonic acids II The synthesis of tripeptide analogs
-
Yamauchi, K.; Kinoshita, M.; Imoto, M. Peptides containing aminophosphonic acids II. The synthesis of tripeptide analogs. Bull. Chem. Soc. Jpn. 1972, 45, 2531-2534.
-
(1972)
Bull. Chem. Soc. Jpn.
, vol.45
, pp. 2531-2534
-
-
Yamauchi, K.1
Kinoshita, M.2
Imoto, M.3
-
54
-
-
0027976825
-
Characterization of covalently bound enzyme inhibitors as transition-state analogs by protein stability measurements: Phosphonate monoester inhibitors of β-lactamase
-
Rahil, J.; Pratt, F. R. Characterization of covalently bound enzyme inhibitors as transition-state analogs by protein stability measurements: phosphonate monoester inhibitors of β-lactamase. Biochemistry 1994, 33, 116-125.
-
(1994)
Biochemistry
, vol.33
, pp. 116-125
-
-
Rahil, J.1
Pratt, F.R.2
-
55
-
-
0027495528
-
Structure-activity relationships in the inhibition of serine β-lactamases by phosphonic acid derivatives
-
Rahil, J.; Pratt R. F. Structure-activity relationships in the inhibition of serine β-lactamases by phosphonic acid derivatives. Biochem. J. 1993, 296, 389-393.
-
(1993)
Biochem. J.
, vol.296
, pp. 389-393
-
-
Rahil, J.1
Pratt, R.F.2
-
56
-
-
0024370749
-
Inhibition of a class C β-lactamase by a specific phosphonate monoester
-
Pratt, R. F. Inhibition of a class C β-lactamase by a specific phosphonate monoester. Science 1989, 246, 917-919.
-
(1989)
Science
, vol.246
, pp. 917-919
-
-
Pratt, R.F.1
-
57
-
-
0023667707
-
Possible role for water dissociation in the slow binding of phosphorus-containing transition-state-analog inhibitors of thermolysin
-
Bartlett, P. A.; Marlowe, C. K. Possible role for water dissociation in the slow binding of phosphorus-containing transition-state-analog inhibitors of thermolysin. Biochemistry 1987, 26, 8553-8561.
-
(1987)
Biochemistry
, vol.26
, pp. 8553-8561
-
-
Bartlett, P.A.1
Marlowe, C.K.2
-
58
-
-
0029865582
-
Phosphonamidate analogues of dipeptides with carboxypeptidase A and β-lactamase-inhibitory activity: Elucidation of the mechanism of β-lactamase inhibition by electrospray mass spectrometry
-
Payne, D. J.; Bateson, J. H.; Tolson, D. A.; Gasson, B. C.; Khushi, T.; Ledent, P.; Fere, J. M. Phosphonamidate analogues of dipeptides with carboxypeptidase A and β-lactamase-inhibitory activity: elucidation of the mechanism of β-lactamase inhibition by electrospray mass spectrometry. Biochem. J. 1996, 314, 457-461.
-
(1996)
Biochem. J.
, vol.314
, pp. 457-461
-
-
Payne, D.J.1
Bateson, J.H.2
Tolson, D.A.3
Gasson, B.C.4
Khushi, T.5
Ledent, P.6
Fere, J.M.7
-
59
-
-
0027932588
-
The synthesis and serine β-lactamase inhibitory activity of some phosphonamidate analogues of dipeptides
-
Bateson, J. H.; Gasson, B. C.; Khushi, T.; Neale, J. E.; Payne D. J.; Tolson, D. A.; Walker, G. The synthesis and serine β-lactamase inhibitory activity of some phosphonamidate analogues of dipeptides. Bioorg. Med. Chem. Lett. 1994, 4, 1667-1672.
-
(1994)
Bioorg. Med. Chem. Lett.
, vol.4
, pp. 1667-1672
-
-
Bateson, J.H.1
Gasson, B.C.2
Khushi, T.3
Neale, J.E.4
Payne, D.J.5
Tolson, D.A.6
Walker, G.7
-
60
-
-
0030847769
-
Structure-activity studies of the inhibition of serine β-lactamases by phosphonate monoesters
-
Li, N.; Rahil, J.; Wright, M. E.; Pratt, R. F. Structure-activity studies of the inhibition of serine β-lactamases by phosphonate monoesters. Bioorg. Med. Chem. 1997, 5, 1783-1788.
-
(1997)
Bioorg. Med. Chem.
, vol.5
, pp. 1783-1788
-
-
Li, N.1
Rahil, J.2
Wright, M.E.3
Pratt, R.F.4
-
63
-
-
0000176550
-
Comments on the synthesis of aminomethylphosphonic acid
-
Soroka, M. Comments on the synthesis of aminomethylphosphonic acid. Synthesis 1989, 547-548.
-
(1989)
Synthesis
, pp. 547-548
-
-
Soroka, M.1
-
64
-
-
84953999914
-
A convenient synthesis of aminomethylphosphonic acid
-
Pulwer, M. J.; Balthazor, T. M. A convenient synthesis of aminomethylphosphonic acid. Synth. Commun. 1986, 16, 733-739.
-
(1986)
Synth. Commun.
, vol.16
, pp. 733-739
-
-
Pulwer, M.J.1
Balthazor, T.M.2
-
65
-
-
84986418178
-
Aminomethanephosphonic acid and its diphenyl ester
-
Oleksyszyn, J.; Subotkowska, L. Aminomethanephosphonic acid and its diphenyl ester. Synthesis 1980, 906-906.
-
(1980)
Synthesis
, pp. 906
-
-
Oleksyszyn, J.1
Subotkowska, L.2
-
66
-
-
0015750978
-
Total synthesis of β-lactam antibiotics I α-thioformamido-diethylphosphonoacetates
-
Ratcliffe, R. W.; Christensen, B. G. Total synthesis of β-lactam antibiotics I. α-thioformamido-diethylphosphonoacetates. Tetrahedron Lett. 1973, 14, 4645-4648.
-
(1973)
Tetrahedron Lett.
, vol.14
, pp. 4645-4648
-
-
Ratcliffe, R.W.1
Christensen, B.G.2
-
67
-
-
0012835444
-
Stabilization demands of diethyl phosphonate substituted carbocations as revealed by substituent effects
-
For the synthesis of diethyl phosphonomethyl-triflate, see
-
For the synthesis of diethyl phosphonomethyl-triflate, see: Creary, X.; Underiner, T. L. Stabilization demands of diethyl phosphonate substituted carbocations as revealed by substituent effects. J. Org. Chem. 1985, 50, 2165-2170.
-
(1985)
J. Org. Chem.
, vol.50
, pp. 2165-2170
-
-
Creary, X.1
Underiner, T.L.2
-
68
-
-
0000444481
-
Synthesis and reactivity of diethyl phosphonomethyltriflate
-
Phillion, D. P.; Andrew, S. S. Synthesis and reactivity of diethyl phosphonomethyltriflate. Tetrahedron Lett. 1986, 27, 1477-1480.
-
(1986)
Tetrahedron Lett.
, vol.27
, pp. 1477-1480
-
-
Phillion, D.P.1
Andrew, S.S.2
-
69
-
-
84986674101
-
Synthesis of 1-aminoalkylphosphonic acids via amidoalkylation of phosphorous acid by N, N'-alkylidenebisamides
-
Soroka, M.; Jaworska, D.; Szczsny, Z. Synthesis of 1-aminoalkylphosphonic acids via amidoalkylation of phosphorous acid by N, N'-alkylidenebisamides. Liebigs Ann. Chem. 1990, 1153-1155.
-
(1990)
Liebigs Ann. Chem.
, pp. 1153-1155
-
-
Soroka, M.1
Jaworska, D.2
Szczsny, Z.3
-
70
-
-
84986706380
-
The synthesis of 1-aminoalkylphosphonic acids. A revised mechanism of the reaction of phosphorus trichloride, amides and aldehydes or ketones in acetic acid (Oleksyszyn reaction)
-
Soroka, M. The synthesis of 1-aminoalkylphosphonic acids. A revised mechanism of the reaction of phosphorus trichloride, amides and aldehydes or ketones in acetic acid (Oleksyszyn reaction). Liebigs Ann. Chem. 1990, 331-334.
-
(1990)
Liebigs Ann. Chem.
, pp. 331-334
-
-
Soroka, M.1
-
71
-
-
2442688922
-
Transport of the phosphonodipeptide alafosfalin by the H+/peptide cotransporters PEPT1 and PEPT2 in intestinal and renal epithelial cells
-
For the biological activity of (S, R)-alafosfalin, see
-
For the biological activity of (S, R)-alafosfalin, see: Neumann, J.; Bruch, M.; Gebauer, S.; Brandsch, M. Transport of the phosphonodipeptide alafosfalin by the H+/peptide cotransporters PEPT1 and PEPT2 in intestinal and renal epithelial cells. Eur. J. Biochem. 2004, 271, 2012-2017.
-
(2004)
Eur. J. Biochem.
, vol.271
, pp. 2012-2017
-
-
Neumann, J.1
Bruch, M.2
Gebauer, S.3
Brandsch, M.4
-
72
-
-
0036840003
-
Alafosfalin as a selective agent for isolation of salmonella from clinical samples
-
Perry, J. D.; Riley, G.; Gould, F. K.; Perez, J. M.; Boissier, E.; Ouedraogo, R. T.; Freydière, A. M. Alafosfalin as a selective agent for isolation of salmonella from clinical samples. J. Clin. Microbiol. 2002, 40, 3913-3916.
-
(2002)
J. Clin. Microbiol.
, vol.40
, pp. 3913-3916
-
-
Perry, J.D.1
Riley, G.2
Gould, F.K.3
Perez, J.M.4
Boissier, E.5
Ouedraogo, R.T.6
Freydière, A.M.7
-
73
-
-
0019128997
-
Phosphonopeptide antibacterial agents related to alafosfalin: Design, synthesis, and structure-activity relationships
-
Atherton, F. R.; Hall, M. J.; Hassall, C. H.; Lambert, R. W.; Lloyd, W. J.; Ringrose, P. S. Phosphonopeptide antibacterial agents related to alafosfalin: design, synthesis, and structure-activity relationships. Antimicrob. Agents Chemother. 1980, 18, 897-905.
-
(1980)
Antimicrob. Agents Chemother.
, vol.18
, pp. 897-905
-
-
Atherton, F.R.1
Hall, M.J.2
Hassall, C.H.3
Lambert, R.W.4
Lloyd, W.J.5
Ringrose, P.S.6
-
74
-
-
53749093104
-
Preparation and transmetallation of enantioenriched α-aminoorganostannanes derived from N-Boc phenylglycinol: Application to the synthesis of alafosfalin
-
Coeffard, V.; Beaudet, I.; Evain, M.; Grognec, E. L.; Quintard, J.-P. Preparation and transmetallation of enantioenriched α-aminoorganostannanes derived from N-Boc phenylglycinol: application to the synthesis of alafosfalin. Eur. J. Org. Chem. 2008, 3344-3351.
-
(2008)
Eur. J. Org. Chem.
, pp. 3344-3351
-
-
Coeffard, V.1
Beaudet, I.2
Evain, M.3
Grognec, E.L.4
Quintard, J.-P.5
-
75
-
-
56249120996
-
Synthesis of alafosfalin and its phosphinic analogue and their fungicidal activity
-
Khomutov, R. M.; Osipova, T. I.; Khurs, E. N.; Dzhavakhiya, V. G. Synthesis of alafosfalin and its phosphinic analogue and their fungicidal activity. Mendeleev Commun. 2008, 18, 295-296.
-
(2008)
Mendeleev Commun.
, vol.18
, pp. 295-296
-
-
Khomutov, R.M.1
Osipova, T.I.2
Khurs, E.N.3
Dzhavakhiya, V.G.4
-
76
-
-
0025895388
-
Preparation of N-acylated phosphonopeptides with free phosphonic group
-
Solodenko, V.; Kasheva, T.; Kukhar, V. P. Preparation of N-acylated phosphonopeptides with free phosphonic group. Synth. Commun. 1991, 21, 1631-1641.
-
(1991)
Synth. Commun.
, vol.21
, pp. 1631-1641
-
-
Solodenko, V.1
Kasheva, T.2
Kukhar, V.P.3
-
77
-
-
0024843404
-
Stereoselective papain-catalyzed synthesis of alafosfalin
-
Solodenko, V. A.; Kukhar, V. P. Stereoselective papain-catalyzed synthesis of alafosfalin. Tetrahedron Lett. 1989, 30, 6917-6918.
-
(1989)
Tetrahedron Lett.
, vol.30
, pp. 6917-6918
-
-
Solodenko, V.A.1
Kukhar, V.P.2
-
78
-
-
0010622452
-
Phosphonodipeptides: Synthesis and separation of diastereoisomers
-
Kafarski, P.; Lejzak, B.; Mastalerz, P.; Szewczyk, J.; Wasielewski, C. Phosphonodipeptides: synthesis and separation of diastereoisomers. Can. J. Chem. 1982, 60, 3081-3084.
-
(1982)
Can. J. Chem.
, vol.60
, pp. 3081-3084
-
-
Kafarski, P.1
Lejzak, B.2
Mastalerz, P.3
Szewczyk, J.4
Wasielewski, C.5
-
79
-
-
0016422783
-
Synthesis and antimicrobial evaluation of N-D-alanyl-1-aminoethylphosphonic acid
-
Huber, III, J. W.; Gilmore, W. F. Synthesis and antimicrobial evaluation of N-D-alanyl-1-aminoethylphosphonic acid. J. Med. Chem. 1975, 18, 106-108.
-
(1975)
J. Med. Chem.
, vol.18
, pp. 106-108
-
-
Huber III, J.W.1
Gilmore, W.F.2
-
80
-
-
0023764098
-
Inhibition of alanine racemase by alanine phosphonate: Detection of an imine linkage to pyridoxal 5'-phosphate in the enzyme-inhibitor complex by solid-state nitrogen-15 nuclear magnetic resonance
-
Copie, V.; Faraci, W. S.; Walsh, C. T.; Griffin, R. G. Inhibition of alanine racemase by alanine phosphonate: detection of an imine linkage to pyridoxal 5'-phosphate in the enzyme-inhibitor complex by solid-state nitrogen-15 nuclear magnetic resonance. Biochemistry 1988, 27, 4966-4970.
-
(1988)
Biochemistry
, vol.27
, pp. 4966-4970
-
-
Copie, V.1
Faraci, W.S.2
Walsh, C.T.3
Griffin, R.G.4
-
81
-
-
0017853042
-
Phosphonopeptides, a new class of synthetic antibacterial agents
-
Allen, J. G.; Atherton, F. R.; Hall, M. J.; Hassall, C. H.; Holmes, S. W.; Lambert, R. W.; Nisbet, L. J.; Ringrose, P. S. Phosphonopeptides, a new class of synthetic antibacterial agents. Nature 1978, 272, 56-58.
-
(1978)
Nature
, vol.272
, pp. 56-58
-
-
Allen, J.G.1
Atherton, F.R.2
Hall, M.J.3
Hassall, C.H.4
Holmes, S.W.5
Lambert, R.W.6
Nisbet, L.J.7
Ringrose, P.S.8
-
82
-
-
0022577081
-
Synthesis and structureactivity relationships of antibacterial phosphonopeptides incorporating (1-aminoethyl)phosphonic acid and (aminomethyl)phosphonic acid
-
Atherton, F. R.; Hassall, C. H.; Lambert, R. W. Synthesis and structureactivity relationships of antibacterial phosphonopeptides incorporating (1-aminoethyl)phosphonic acid and (aminomethyl)phosphonic acid. J. Med. Chem. 1986, 29, 29-40.
-
(1986)
J. Med. Chem.
, vol.29
, pp. 29-40
-
-
Atherton, F.R.1
Hassall, C.H.2
Lambert, R.W.3
-
83
-
-
0018774396
-
Phosphonopeptides as antibacterial agents: Mechanism of action of alaphosphin
-
Atherton, F. R.; Hall, M. J.; Hassall, C. H.; Lambert, R. W.; Lloyd, W. J.; Ringrose, P. S. Phosphonopeptides as antibacterial agents: mechanism of action of alaphosphin. Antimicrob. Agents Chemother. 1979, 15, 696-705.
-
(1979)
Antimicrob. Agents Chemother.
, vol.15
, pp. 696-705
-
-
Atherton, F.R.1
Hall, M.J.2
Hassall, C.H.3
Lambert, R.W.4
Lloyd, W.J.5
Ringrose, P.S.6
-
84
-
-
0018419355
-
Phosphonopeptides as antibacterial agents: Alaphosphin and related phosphonopeptides
-
Allen, J. G.; Atherton, F. R.; Hall, M. J.; Hassall, C. H.; Holmes, S. W.; Lambert, R. W.; Nisbet, L. J.; Ringrose, P. S. Phosphonopeptides as antibacterial agents: alaphosphin and related phosphonopeptides. Antimicrob. Agents Chemother. 1979, 15, 684-695.
-
(1979)
Antimicrob. Agents Chemother.
, vol.15
, pp. 684-695
-
-
Allen, J.G.1
Atherton, F.R.2
Hall, M.J.3
Hassall, C.H.4
Holmes, S.W.5
Lambert, R.W.6
Nisbet, L.J.7
Ringrose, P.S.8
-
85
-
-
0037343936
-
Synthesis and biological evaluation of fotemustine analogues on human melanoma cell lines
-
Winum, J.-Y.; Bouissière, J.-L.; Passagne, I.; Evrard, A.; Montero, V.; Cuq, P.; Montero, J.-L. Synthesis and biological evaluation of fotemustine analogues on human melanoma cell lines. Eur. J. Med. Chem. 2003, 38, 319-324.
-
(2003)
Eur. J. Med. Chem.
, vol.38
, pp. 319-324
-
-
Winum, J.-Y.1
Bouissière, J.-L.2
Passagne, I.3
Evrard, A.4
Montero, V.5
Cuq, P.6
Montero, J.-L.7
-
86
-
-
0028113292
-
Phase II trial of fotemustine in patients with metastatic malignant melanoma
-
Falkson, C. I.; Falkson, G.; Falkson, H. C. Phase II trial of fotemustine in patients with metastatic malignant melanoma. Invest. News Drugs 1994, 12, 251-254.
-
(1994)
Invest. News Drugs
, vol.12
, pp. 251-254
-
-
Falkson, C.I.1
Falkson, G.2
Falkson, H.C.3
-
87
-
-
0029877012
-
Molecular mechanisms of toxic effects of fotemustine in rat hepatocytes and subcellular rat liver fractions
-
Brakenhoff, J. P. G.; Commandeur, J. N. M.; Wormhoudt, L. W.; Groot, E. J.; Vermeulen, N. P. E. Molecular mechanisms of toxic effects of fotemustine in rat hepatocytes and subcellular rat liver fractions. Carcinogenesis 1996, 17, 715-724.
-
(1996)
Carcinogenesis
, vol.17
, pp. 715-724
-
-
Brakenhoff, J.P.G.1
Commandeur, J.N.M.2
Wormhoudt, L.W.3
Groot, E.J.4
Vermeulen, N.P.E.5
-
88
-
-
0029994657
-
Pharmacokinetics and pharmacodynamics of nitrosourea fotemustine: A French cancer centre multicentric study
-
Iliadis, A.; Launay-Iliadis, M.-C.; Lucas, C.; Fety, R.; Lokiec, F.; Tranchand, B.; Milano, G. Pharmacokinetics and pharmacodynamics of nitrosourea fotemustine: a French cancer centre multicentric study. Eur. J. Cancer 1996, 32A, 455-460.
-
(1996)
Eur. J. Cancer
, vol.32 A
, pp. 455-460
-
-
Iliadis, A.1
Launay-Iliadis, M.-C.2
Lucas, C.3
Fety, R.4
Lokiec, F.5
Tranchand, B.6
Milano, G.7
-
89
-
-
0037108173
-
Aminophosphonate inhibitors of dialkylglycine decarboxylase: Structural basis for slow binding inhibition
-
Liu, W.; Rogers, C. J.; Fisher, A. J.; Toney, M. D. Aminophosphonate inhibitors of dialkylglycine decarboxylase: structural basis for slow binding inhibition. Biochemistry 2002, 41, 12320-12328.
-
(2002)
Biochemistry
, vol.41
, pp. 12320-12328
-
-
Liu, W.1
Rogers, C.J.2
Fisher, A.J.3
Toney, M.D.4
-
90
-
-
0021928231
-
Purification of an alanine racemase from Streptococcus faecalis and analysis of its inactivation by (1-aminoethyl)phosphonic acid enantiomers
-
Badet, B.; Walsh, C. Purification of an alanine racemase from Streptococcus faecalis and analysis of its inactivation by (1-aminoethyl)phosphonic acid enantiomers. Biochemistry 1985, 24, 1333-1341.
-
(1985)
Biochemistry
, vol.24
, pp. 1333-1341
-
-
Badet, B.1
Walsh, C.2
-
91
-
-
0037041183
-
5-Phosphonomethylquinoxalinediones as competitive NMDA receptor antagonists with a preference for the human 1A/2A, rather than 1A/2B receptor composition
-
Auberson, Y. P.; Allgeier, H.; Bischoff, S.; Lingenhoehl, K.; Moretti, R.; Schmutz, M. 5-Phosphonomethylquinoxalinediones as competitive NMDA receptor antagonists with a preference for the human 1A/2A, rather than 1A/2B receptor composition. Bioorg. Med. Chem. Lett. 2002, 12, 1099-1102.
-
(2002)
Bioorg. Med. Chem. Lett.
, vol.12
, pp. 1099-1102
-
-
Auberson, Y.P.1
Allgeier, H.2
Bischoff, S.3
Lingenhoehl, K.4
Moretti, R.5
Schmutz, M.6
-
92
-
-
0033579923
-
N-phosphonoalkyl-5-aminomethylquinoxaline-2,3-diones: In vivo active AMPA and NMDA (glycine) antagonists
-
Auberson, Y. P.; Acklin, P.; Bischoff, S.; Moretti, R.; Ofner, S.; Schmutz, M.; Veenstra, S. J. N-phosphonoalkyl-5-aminomethylquinoxaline-2,3-diones: In vivo active AMPA and NMDA (glycine) antagonists. Bioorg. Med. Chem. 1999, 9, 249-254.
-
(1999)
Bioorg. Med. Chem.
, vol.9
, pp. 249-254
-
-
Auberson, Y.P.1
Acklin, P.2
Bischoff, S.3
Moretti, R.4
Ofner, S.5
Schmutz, M.6
Veenstra, S.J.7
-
93
-
-
0032793783
-
Differential in vitro association of vinca alkaloid-induced tubulin spiral filaments into aggregated spirals
-
Verdier-Pinard, P.; Garès, M.; Wright, M. Differential in vitro association of vinca alkaloid-induced tubulin spiral filaments into aggregated spirals. Biochem. Pharmacol. 1999, 58, 959-971.
-
(1999)
Biochem. Pharmacol.
, vol.58
, pp. 959-971
-
-
Verdier-Pinard, P.1
Garès, M.2
Wright, M.3
-
94
-
-
84987480058
-
Nucleophilic additions to N-glycosylnitrones: Asymmetric synthesis of α-aminophosphonic acids
-
Huber, R.; Knierzinger, A.; Obrecht, J.-P.; Vasella, A. Nucleophilic additions to N-glycosylnitrones: asymmetric synthesis of α-aminophosphonic acids. Helv. Chim. Acta 1985, 68, 1730-1747.
-
(1985)
Helv. Chim. Acta
, vol.68
, pp. 1730-1747
-
-
Huber, R.1
Knierzinger, A.2
Obrecht, J.-P.3
Vasella, A.4
-
95
-
-
0024835884
-
Preparation of optically active 1-aminoalkylphosphonic acids from chiral carbamates and chiral ureas
-
Oshikawa, T.; Yamashita, M. Preparation of optically active 1-aminoalkylphosphonic acids from chiral carbamates and chiral ureas. Bull. Chem. Soc. Jpn. 1989, 62, 3177-3181.
-
(1989)
Bull. Chem. Soc. Jpn.
, vol.62
, pp. 3177-3181
-
-
Oshikawa, T.1
Yamashita, M.2
-
96
-
-
0001195570
-
Asymmetric synthesis of α-aminophosphonic acids by diastereoselective addition of trimethyl phosphite onto chiral oxazolidines
-
Maury, C.; Gharbaoui, T.; Royer, J.; Husson, H.-P. Asymmetric synthesis of α-aminophosphonic acids by diastereoselective addition of trimethyl phosphite onto chiral oxazolidines. J. Org. Chem. 1996, 61, 3687-3693.
-
(1996)
J. Org. Chem.
, vol.61
, pp. 3687-3693
-
-
Maury, C.1
Gharbaoui, T.2
Royer, J.3
Husson, H.-P.4
-
97
-
-
84985225807
-
Asymmetrische synthese von (S)-(1-aminoalkyl)phosphonsäure-diethylestern unter verwendung von (+)-campher als chiralem hilfsreagens
-
Schöllkopf, U.; Schütze, R. Asymmetrische synthese von (S)-(1-aminoalkyl)phosphonsäure-diethylestern unter verwendung von (+)-campher als chiralem hilfsreagens. Liebigs Ann. Chem. 1987, 45-49.
-
(1987)
Liebigs Ann. Chem.
, pp. 45-49
-
-
Schöllkopf, U.1
Schütze, R.2
-
98
-
-
0026663281
-
A simple and general method for the asymmetric synthesis of α-aminophosphonic acids
-
Maury, C.; Royer, J.; Husson, H.-P. A simple and general method for the asymmetric synthesis of α-aminophosphonic acids. Tetrahedron Lett. 1992, 33, 6127-6130.
-
(1992)
Tetrahedron Lett.
, vol.33
, pp. 6127-6130
-
-
Maury, C.1
Royer, J.2
Husson, H.-P.3
-
99
-
-
0025187520
-
A versatile asymmetric synthesis of α-amino α-alkylphosphonic acids of high enantiomeric purity
-
Hanessian, S.; Bennani, Y. L. A versatile asymmetric synthesis of α-amino α-alkylphosphonic acids of high enantiomeric purity. Tetrahedron Lett. 1990, 31, 6465-6468.
-
(1990)
Tetrahedron Lett.
, vol.31
, pp. 6465-6468
-
-
Hanessian, S.1
Bennani, Y.L.2
-
100
-
-
30744461593
-
Facile and efficient asymmetric synthesis of α-aminoalkylphosphonic acids
-
Yuan, C.-Y.; Chen, Q.-Y. Facile and efficient asymmetric synthesis of α-aminoalkylphosphonic acids. Chin. J. Chem. 2005, 23, 1671-1676.
-
(2005)
Chin. J. Chem.
, vol.23
, pp. 1671-1676
-
-
Yuan, C.-Y.1
Chen, Q.-Y.2
-
101
-
-
0036020828
-
Asymmetric synthesis of aminophosphonic acids and trifluoromethylated derivatives thereof
-
Yuan, C.-Y.; Li, J. X.; Cui, S.; Wang, G. Asymmetric synthesis of aminophosphonic acids and trifluoromethylated derivatives thereof. Phosphorus Sulfur 2002, 177, 1731-1734.
-
(2002)
Phosphorus Sulfur
, vol.177
, pp. 1731-1734
-
-
Yuan, C.-Y.1
Li, J.X.2
Cui, S.3
Wang, G.4
-
102
-
-
0026516860
-
Recent advances in the Staudinger reaction
-
Gololobov, Y. G.; Kasukhin, L. F. Recent advances in the Staudinger reaction. Tetrahedron 1992, 48, 1353-1406.
-
(1992)
Tetrahedron
, vol.48
, pp. 1353-1406
-
-
Gololobov, Y.G.1
Kasukhin, L.F.2
-
103
-
-
3042698861
-
Mechanisms of Staudinger reactions within density functional theory
-
and references cited therein
-
Tian, W. Q.; Wang, Y. A. Mechanisms of Staudinger reactions within density functional theory. J. Org. Chem. 2004, 69, 4299-4308 and references cited therein.
-
(2004)
J. Org. Chem.
, vol.69
, pp. 4299-4308
-
-
Tian, W.Q.1
Wang, Y.A.2
-
104
-
-
0034499739
-
A new and efficient asymmetric synthesis of 1-amino-1-alkylphosphonic acids
-
Yuan, C.; Li, S.; Wang, G. A new and efficient asymmetric synthesis of 1-amino-1-alkylphosphonic acids. Heteroatom. Chem. 2000, 11, 528-535.
-
(2000)
Heteroatom. Chem.
, vol.11
, pp. 528-535
-
-
Yuan, C.1
Li, S.2
Wang, G.3
-
105
-
-
84986691327
-
Phosphoranalogue von aminosäuren III. Synthese optisch aktiver 1-aminoalkylphosphonsäuren der (S)-und (R)-reihe mit hilfe von (-)-ephedrin als auxiliar
-
Sting, M.; Steglich, W. Phosphoranalogue von aminosäuren III. Synthese optisch aktiver 1-aminoalkylphosphonsäuren der (S)-und (R)-reihe mit hilfe von (-)-ephedrin als auxiliar. Synthesis 1990, 132-134.
-
(1990)
Synthesis
, pp. 132-134
-
-
Sting, M.1
Steglich, W.2
-
106
-
-
0028618170
-
Electrophilic amination and azidation of chiral α-alkyl phosphonamides: Asymmetric syntheses of α-amino α-alkyl phosphonic acids
-
Hanessian, S.; Bennani, Y. F. Electrophilic amination and azidation of chiral α-alkyl phosphonamides: asymmetric syntheses of α-amino α-alkyl phosphonic acids. Synthesis 1994, 1272-1274.
-
(1994)
Synthesis
, pp. 1272-1274
-
-
Hanessian, S.1
Bennani, Y.F.2
-
107
-
-
0001551678
-
Synthesis of α-amino phosphonic acids by asymmetric hydrogenation
-
Kitamura, M.; Yoshimura, M.; Tsukamoto, M.; Noyori, R. Synthesis of α-amino phosphonic acids by asymmetric hydrogenation. Enantiomer 1996, 1, 281-303.
-
(1996)
Enantiomer
, vol.1
, pp. 281-303
-
-
Kitamura, M.1
Yoshimura, M.2
Tsukamoto, M.3
Noyori, R.4
-
108
-
-
84985186249
-
Enantioselective synthesis of L-(1-aminoethyl)phosphonic acid by asymmetric catalytic hydrogenation of N-[1-(dimethoxy-phosphoryl)ethenyl]formamide
-
Schöllkopf, U.; Hoppe, I.; Thiele, A. Enantioselective synthesis of L-(1-aminoethyl)phosphonic acid by asymmetric catalytic hydrogenation of N-[1-(dimethoxy-phosphoryl)ethenyl]formamide. Liebigs Ann. Chem. 1985, 555-559.
-
(1985)
Liebigs Ann. Chem.
, pp. 555-559
-
-
Schöllkopf, U.1
Hoppe, I.2
Thiele, A.3
-
109
-
-
0018745481
-
Phosphonopeptides as antibacterial agents: Rationale, chemistry, and structure-activity relationships
-
Atherton, F. R.; Hall, M. J.; Hassall, C. H.; Lambert, R. W.; Ringrose, P. S. Phosphonopeptides as antibacterial agents: rationale, chemistry, and structure-activity relationships. Antimicrob. Agents Chemother. 1979, 15, 677-683.
-
(1979)
Antimicrob. Agents Chemother.
, vol.15
, pp. 677-683
-
-
Atherton, F.R.1
Hall, M.J.2
Hassall, C.H.3
Lambert, R.W.4
Ringrose, P.S.5
-
110
-
-
0000726942
-
Optically active 1-aminoalkanephosphonic acids. Dibenzoyl-L-tartaric anhydride as an effective agent for the resolution of racemic diphenyl 1-aminoalkanephosphonates
-
Kafarski, P.; Lejczak, B.; Szewczyk, J. Optically active 1-aminoalkanephosphonic acids. Dibenzoyl-L-tartaric anhydride as an effective agent for the resolution of racemic diphenyl 1-aminoalkanephosphonates. Can. J. Chem. 1983, 61, 2425-2030.
-
(1983)
Can. J. Chem.
, vol.61
, pp. 2030-2425
-
-
Kafarski, P.1
Lejczak, B.2
Szewczyk, J.3
-
111
-
-
0343449134
-
Determination of absolute configuration of optically active 1-aminoalkanephosphonic acids by chemical correlations
-
Kowalik, J.; Zygmunt, J.; Mastalerz, P. Determination of absolute configuration of optically active 1-aminoalkanephosphonic acids by chemical correlations. Phosphorus Sulfur 1983, 18, 393-396.
-
(1983)
Phosphorus Sulfur
, vol.18
, pp. 393-396
-
-
Kowalik, J.1
Zygmunt, J.2
Mastalerz, P.3
-
112
-
-
13344267040
-
Chromatographic assigment of the configuration of 1-aminoalkanephosphonic acids
-
Lejczak, B.; Kafarski, P.; Mastalerz, P. Chromatographic assigment of the configuration of 1-aminoalkanephosphonic acids. J. Chromatogr. A 1985, 324, 455-461.
-
(1985)
J. Chromatogr. A
, vol.324
, pp. 455-461
-
-
Lejczak, B.1
Kafarski, P.2
Mastalerz, P.3
-
113
-
-
0025843366
-
Preparation of optically active 1-aminoalkylphosphonic acids by stereoselective anzymatic hydrolysis of racemic N-acylated 1-aminoalkylphosphonic acids
-
Solodenko, V. A.; Kasheva, T. N.; Kukhar, V. P.; Kozlova, E. V.; Mironenko, D. A.; Vedas, V. K. Preparation of optically active 1-aminoalkylphosphonic acids by stereoselective anzymatic hydrolysis of racemic N-acylated 1-aminoalkylphosphonic acids. Tetrahedron 1991, 47, 3989-3998.
-
(1991)
Tetrahedron
, vol.47
, pp. 3989-3998
-
-
Solodenko, V.A.1
Kasheva, T.N.2
Kukhar, V.P.3
Kozlova, E.V.4
Mironenko, D.A.5
Vedas, V.K.6
-
114
-
-
0029992442
-
Synthesis of phosphorus-containing amino acid analogs as inhibitors of nitric oxide synthase
-
Cowart, M.; Kowaluk, E. A.; Kohlhaas, K. L.; Alexander, K. M.; Kerwin, Jr. J. F. Synthesis of phosphorus-containing amino acid analogs as inhibitors of nitric oxide synthase. Bioorg. Med. Chem. Lett. 1996, 6, 999-1002.
-
(1996)
Bioorg. Med. Chem. Lett.
, vol.6
, pp. 999-1002
-
-
Cowart, M.1
Kowaluk, E.A.2
Kohlhaas, K.L.3
Alexander, K.M.4
Kerwin Jr., J.F.5
-
115
-
-
0026677017
-
Synthesis of phosphonopeptides as thrombin inhibitors
-
Wang, C.-L. J.; Taylor, T. L.; Mical, A. J.; Spitz, S.; Reilly, T. M. Synthesis of phosphonopeptides as thrombin inhibitors. Tetrahedron Lett. 1992, 33, 7667-7670.
-
(1992)
Tetrahedron Lett.
, vol.33
, pp. 7667-7670
-
-
Wang, C.-L.J.1
Taylor, T.L.2
Mical, A.J.3
Spitz, S.4
Reilly, T.M.5
-
116
-
-
2342618859
-
Development of irreversible diphenyl phosphonate inhibitors for urokinase plasminogen activator
-
Joossens, J.; Van der Veken, P.; Lambeir, A.-M.; Augustyns, K.; Haemers, A. Development of irreversible diphenyl phosphonate inhibitors for urokinase plasminogen activator. J. Med. Chem. 2004, 47, 2411-2413.
-
(2004)
J. Med. Chem.
, vol.47
, pp. 2411-2413
-
-
Joossens, J.1
van der Veken, P.2
Lambeir, A.-M.3
Augustyns, K.4
Haemers, A.5
-
117
-
-
0022200175
-
In the search for new anticancer drugs. 13. Phosphonic and phosphinic analogues of ornithine
-
Sosnovsky, G.; Lukszo, J.; Gravela, E.; Zuretti, M. F. In the search for new anticancer drugs. 13. Phosphonic and phosphinic analogues of ornithine. J. Med. Chem. 1985, 28, 1350-1354.
-
(1985)
J. Med. Chem.
, vol.28
, pp. 1350-1354
-
-
Sosnovsky, G.1
Lukszo, J.2
Gravela, E.3
Zuretti, M.F.4
-
118
-
-
0027230517
-
A convenient synthesis of N-protected diphenyl phosphonate ester analogues of ornithine, lysine and homolysine
-
Hamilton, R.; Walker, B. J.; Walker, B. A convenient synthesis of N-protected diphenyl phosphonate ester analogues of ornithine, lysine and homolysine. Tetrahedron Lett. 1993, 34, 2847-2850.
-
(1993)
Tetrahedron Lett.
, vol.34
, pp. 2847-2850
-
-
Hamilton, R.1
Walker, B.J.2
Walker, B.3
-
119
-
-
33749107229
-
Zinc (II) complexes of phosphonic acid analogues of aspartic acid and asparagine
-
Matczak-Jon, E.; Kurzak, B.; Sawka-Dobrowolska, W.; Lejczak, B.; Kafarski, P. Zinc (II) complexes of phosphonic acid analogues of aspartic acid and asparagine. J. Chem. Soc., Dalton Trans. 1998, 161-169.
-
(1998)
J. Chem. Soc., Dalton Trans.
, pp. 161-169
-
-
Matczak-Jon, E.1
Kurzak, B.2
Sawka-Dobrowolska, W.3
Lejczak, B.4
Kafarski, P.5
-
120
-
-
33749086361
-
Zinc (II) complexes of phosphonic acid analogues of glutamic acid
-
Matczak-Jon, E.; Kurzak, B.; Sawka-Dobrowolska, W.; Kafarski, P.; Lejczak, B. Zinc (II) complexes of phosphonic acid analogues of glutamic acid. J. Chem. Soc., Dalton Trans. 1996, 3455-3464.
-
(1996)
J. Chem. Soc., Dalton Trans.
, pp. 3455-3464
-
-
Matczak-Jon, E.1
Kurzak, B.2
Sawka-Dobrowolska, W.3
Kafarski, P.4
Lejczak, B.5
-
121
-
-
0242575091
-
Utilisation of structurally diverse organophosphonates by Streptomycetes
-
Obojska, A.; Lejczak, B. Utilisation of structurally diverse organophosphonates by Streptomycetes. Appl. Microbiol. Biotechnol. 2003, 62, 557-563.
-
(2003)
Appl. Microbiol. Biotechnol.
, vol.62
, pp. 557-563
-
-
Obojska, A.1
Lejczak, B.2
-
122
-
-
33847660883
-
Isolation and characterization of two new microbial strains capable of degradation of the naturally occurring organophosphonate-ciliatine
-
Klimeck-Ochab, M.; Obojska, A.; Lejczak, B.; Picco, A. N. Isolation and characterization of two new microbial strains capable of degradation of the naturally occurring organophosphonate-ciliatine. Biodegradation 2007, 18, 223-231.
-
(2007)
Biodegradation
, vol.18
, pp. 223-231
-
-
Klimeck-Ochab, M.1
Obojska, A.2
Lejczak, B.3
Picco, A.N.4
-
123
-
-
84985087355
-
Asymmetric synthesis of α-aminophosphonic acids by cycloaddition of N-glycosyl-C-dialkoxyphosphonoylnitrones
-
Vasella, A.; Voeffray, R. Asymmetric synthesis of α-aminophosphonic acids by cycloaddition of N-glycosyl-C-dialkoxyphosphonoylnitrones. Helv. Chim. Acta 1982, 65, 1953-1964.
-
(1982)
Helv. Chim. Acta
, vol.65
, pp. 1953-1964
-
-
Vasella, A.1
Voeffray, R.2
-
124
-
-
0019958810
-
Aminophosphonic and aminophosphinic acid analogues of aspartic acid
-
Campell, M. M.; Carruthers, N. I.; Mickel, S. J. Aminophosphonic and aminophosphinic acid analogues of aspartic acid. Tetrahedron 1982, 38, 2513-2524.
-
(1982)
Tetrahedron
, vol.38
, pp. 2513-2524
-
-
Campell, M.M.1
Carruthers, N.I.2
Mickel, S.J.3
-
125
-
-
37049104232
-
Synthesis of α-aminophosphonic and α-aminophosphinic acids and derived dipeptides from 4-acetoxyazetidin-2-ones
-
Campell, M. M.; Carruthers, N. I. Synthesis of α-aminophosphonic and α-aminophosphinic acids and derived dipeptides from 4-acetoxyazetidin-2-ones. J. Chem. Soc., Chem. Commun. 1980, 730-731.
-
(1980)
J. Chem. Soc., Chem. Commun.
, pp. 730-731
-
-
Campell, M.M.1
Carruthers, N.I.2
-
126
-
-
0032493326
-
Synthesis and proteinase inhibitory properties of diphenyl phosphonate analogues of aspartic and glutamic acids
-
Hamilton, R.; Walker, B.; Walker, B. J. Synthesis and proteinase inhibitory properties of diphenyl phosphonate analogues of aspartic and glutamic acids. Bioorg. Med. Chem. Lett. 1998, 9, 1655-1660.
-
(1998)
Bioorg. Med. Chem. Lett.
, vol.9
, pp. 1655-1660
-
-
Hamilton, R.1
Walker, B.2
Walker, B.J.3
-
127
-
-
0022408355
-
N-(Phosphonoacetyl)amino phosphonates Phosphonate analogues of N (phosphonoacetyl)-L-aspartic acid (PALA)
-
Kafarski, P.; Lejczak, B.; Mastalerz, P.; Du, D.; Radzikowski, C. N-(Phosphonoacetyl)amino phosphonates. Phosphonate analogues of N (phosphonoacetyl)-L-aspartic acid (PALA). J. Med. Chem. 1995, 28, 1555-1558.
-
(1995)
J. Med. Chem.
, vol.28
, pp. 1555-1558
-
-
Kafarski, P.1
Lejczak, B.2
Mastalerz, P.3
Du, D.4
Radzikowski, C.5
-
128
-
-
0027433691
-
Inhibition of aminopeptidases by phosphonic acid and phosphinic acid analogues of aspartic and glutamic acids
-
Lejczak, B.; Popiel de Choszczak, M.; Kafarski, P. Inhibition of aminopeptidases by phosphonic acid and phosphinic acid analogues of aspartic and glutamic acids. J. Enzyme Inhib. Med. Chem. 1993, 7, 97-103.
-
(1993)
J. Enzyme Inhib. Med. Chem.
, vol.7
, pp. 97-103
-
-
Lejczak, B.1
Popiel de Choszczak, M.2
Kafarski, P.3
-
129
-
-
84989719185
-
Herbicidal activity of phosphonic and phosphinic acid analogues of glutamic and aspartic acids
-
Miliszkiewicz, D.; Wieczorek, P.; Lejczak, B.; Kowalik, E.; Kafarski, P. Herbicidal activity of phosphonic and phosphinic acid analogues of glutamic and aspartic acids. Pestic. Sci. 1992, 34, 349-354.
-
(1992)
Pestic. Sci.
, vol.34
, pp. 349-354
-
-
Miliszkiewicz, D.1
Wieczorek, P.2
Lejczak, B.3
Kowalik, E.4
Kafarski, P.5
-
130
-
-
0009225758
-
Complexes of aminophosphonates. II Transition metal complexes of aminophosphonic acid analogues of aspartic acid and glutamic acid
-
Kiss, T.; Farkas, E. Complexes of aminophosphonates. II. Transition metal complexes of aminophosphonic acid analogues of aspartic acid and glutamic acid. Inorg. Chim. Acta 1989, 155, 281-287.
-
(1989)
Inorg. Chim. Acta
, vol.155
, pp. 281-287
-
-
Kiss, T.1
Farkas, E.2
-
131
-
-
84986374290
-
Phosphonocysteine and phosphonohomocysteine; synthesis and isolation
-
Kudzin, Z. H. Phosphonocysteine and phosphonohomocysteine; synthesis and isolation. Synthesis 1983, 812-813.
-
(1983)
Synthesis
, pp. 812-813
-
-
Kudzin, Z.H.1
-
132
-
-
0001523922
-
Aziridine-2-phosphonic acid, the valuable synthon for synthesis of 1-amino-2-functionalized ethanephosphonic acids
-
Zygmunt, J. Aziridine-2-phosphonic acid, the valuable synthon for synthesis of 1-amino-2-functionalized ethanephosphonic acids. Tetrahedron 1985, 41, 4979-4982.
-
(1985)
Tetrahedron
, vol.41
, pp. 4979-4982
-
-
Zygmunt, J.1
-
133
-
-
5144221294
-
1-Amino-2-mercaptoethanephosphonic acid, the phosphonic analog of cysteine
-
Kowalik, J.; Zygmunt, J.; Mastalerz, P. 1-Amino-2-mercaptoethanephosphonic acid, the phosphonic analog of cysteine. Pol. J. Chem. 1981, 55, 713-715.
-
(1981)
Pol. J. Chem.
, vol.55
, pp. 713-715
-
-
Kowalik, J.1
Zygmunt, J.2
Mastalerz, P.3
-
134
-
-
5144221340
-
Optically active diethyl N-(ptoluenesulfonyl)-aziridine-2-phosphonates as chiral synthons for the synthesis of γ-substituted ω-aminophosphonates
-
Dolence, E. K.; Roylance, J. B. Optically active diethyl N-(ptoluenesulfonyl)-aziridine-2-phosphonates as chiral synthons for the synthesis of γ-substituted ω-aminophosphonates. Tetrahedron: Asymmetry 2004, 15, 3307-3322.
-
(2004)
Tetrahedron: Asymmetry
, vol.15
, pp. 3307-3322
-
-
Dolence, E.K.1
Roylance, J.B.2
-
135
-
-
0019881070
-
Inhibition of rat liver glutamine synthetase by phosphonic analogues of glutamic acid
-
Lejczak, B.; Starzemska, H.; Mastalerz, P. Inhibition of rat liver glutamine synthetase by phosphonic analogues of glutamic acid. Experientia 1981, 37, 461-462.
-
(1981)
Experientia
, vol.37
, pp. 461-462
-
-
Lejczak, B.1
Starzemska, H.2
Mastalerz, P.3
-
136
-
-
0002157166
-
Organische phosphorverbindungen 79 herstellung und eigenschaften von ω-amino-carboxyalkylphosphon-und-phosphinsäuren
-
Diel, P. J.; Maier, L. Organische phosphorverbindungen 79 herstellung und eigenschaften von ω-amino-carboxyalkylphosphon-und-phosphinsäuren. Phosphorus Sulfur 1987, 29, 201-209.
-
(1987)
Phosphorus Sulfur
, vol.29
, pp. 201-209
-
-
Diel, P.J.1
Maier, L.2
-
137
-
-
0030713348
-
A tyrosine residue essential for catalytic activity in aminopeptidase A
-
Vazeux, G.; Iturrioz, X.; Corvol, P.; Llorens-Cortès, C. A tyrosine residue essential for catalytic activity in aminopeptidase A. Biochem. J. 1997, 327, 883-889.
-
(1997)
Biochem. J.
, vol.327
, pp. 883-889
-
-
Vazeux, G.1
Iturrioz, X.2
Corvol, P.3
Llorens-Cortès, C.4
-
138
-
-
0029609299
-
Enantioselective synthesis of diverse ω-aminophosphonate diesters
-
Smith, III, A. B.; Yager, K. M.; Taylor, C. M. Enantioselective synthesis of diverse ω-aminophosphonate diesters. J. Am. Chem. Soc. 1995, 117, 10879-10888.
-
(1995)
J. Am. Chem. Soc.
, vol.117
, pp. 10879-10888
-
-
Smith III, A.B.1
Yager, K.M.2
Taylor, C.M.3
-
139
-
-
28644431674
-
Catalytic enantioselective Michael addition in the synthesis of ω-aminophosphonates
-
Jászay, Z. M.; Németh, G.; Pham, T. S.; Petneházy, I.; Grün, A.; Tγke, L. Catalytic enantioselective Michael addition in the synthesis of ω-aminophosphonates. Tetrahedron: Asymmetry 2005, 16, 3837-3840.
-
(2005)
Tetrahedron: Asymmetry
, vol.16
, pp. 3837-3840
-
-
Jászay, Z.M.1
Németh, G.2
Pham, T.S.3
Petneházy, I.4
Grün, A.5
Tγke, L.6
-
140
-
-
0028898313
-
ω-Aminophosphonate derivatives as nucleophiles in diastereoselective and enantioselective palladium catalysed allylic substitution reactions
-
For the catalytic enantioselective synthesis of ω-aminophosphonates from 92, see
-
For the catalytic enantioselective synthesis of ω-aminophosphonates from 92, see: Baldwin, I. C.; Williams, J. M. J.; Beckett, R. P. ω-Aminophosphonate derivatives as nucleophiles in diastereoselective and enantioselective palladium catalysed allylic substitution reactions. Tetrahedron: Asymmetry 1995, 6, 679-682.
-
(1995)
Tetrahedron: Asymmetry
, vol.6
, pp. 679-682
-
-
Baldwin, I.C.1
Williams, J.M.J.2
Beckett, R.P.3
-
141
-
-
3543122090
-
Separation of racemic phosphonic analogues of glutamic acid
-
Antczak, K.; Szewczyk, J. Separation of racemic phosphonic analogues of glutamic acid. Phosphorus Sulfur 1985, 22, 247-251.
-
(1985)
Phosphorus Sulfur
, vol.22
, pp. 247-251
-
-
Antczak, K.1
Szewczyk, J.2
-
142
-
-
0020406531
-
New phosphonic analogs of aspartic and glutamic acid by aminoalkylation of trivalent phosphorus chlorides with ethyl acetyloacetate or ethyl levulinate and benzyl carbamate
-
For the synthesis of 100, see
-
For the synthesis of 100, see: Oleksyszyn, J.; Gruszecka, E.; Kafarski, P.; Mastalerz, P. New phosphonic analogs of aspartic and glutamic acid by aminoalkylation of trivalent phosphorus chlorides with ethyl acetyloacetate or ethyl levulinate and benzyl carbamate. Monatsh. Chem. 1982, 113, 59-71.
-
(1982)
Monatsh. Chem.
, vol.113
, pp. 59-71
-
-
Oleksyszyn, J.1
Gruszecka, E.2
Kafarski, P.3
Mastalerz, P.4
-
143
-
-
0028258788
-
1-Amino-2-imidazol-4'-ylethylphosphonic acid is a potent reversible inhibitor of Pseudomonas putida histidine ammonia-lyase
-
Hernandez, D.; Phillips, A. T.; Zon, J. 1-Amino-2-imidazol-4'-ylethylphosphonic acid is a potent reversible inhibitor of Pseudomonas putida histidine ammonia-lyase. Biochem. Mol. Biol. Int. 1994, 32, 189-194.
-
(1994)
Biochem. Mol. Biol. Int.
, vol.32
, pp. 189-194
-
-
Hernandez, D.1
Phillips, A.T.2
Zon, J.3
-
144
-
-
0042572071
-
ω-Amino-(4-imidazoil)-ethylphosphonic acid, the phosphonoisostere of histidine
-
Wu, Y. Y.-L.; Tishler, M. ω-Amino-(4-imidazoil)-ethylphosphonic acid, the phosphonoisostere of histidine. Chin. Chem. Lett. 1991, 2, 95-98.
-
(1991)
Chin. Chem. Lett.
, vol.2
, pp. 95-98
-
-
Wu, Y.Y.-L.1
Tishler, M.2
-
145
-
-
0027174063
-
Inhibitory effect of synthetic aminophosphonic acid derivatives on human carbonic anhydrase
-
Ösapay, G.; Csiba, A. Inhibitory effect of synthetic aminophosphonic acid derivatives on human carbonic anhydrase. Eur. J. Med. Chem. 1993, 28, 355-361.
-
(1993)
Eur. J. Med. Chem.
, vol.28
, pp. 355-361
-
-
Ösapay, G.1
Csiba, A.2
-
146
-
-
50949112789
-
Chemical target validation studies of aminopeptidase in malaria parasites using ω-aminoalkylphosphonate and phosphonopeptide inhibitors
-
Cunningham, E.; Drag, M.; Kafarski, P.; Bell, A. Chemical target validation studies of aminopeptidase in malaria parasites using ω-aminoalkylphosphonate and phosphonopeptide inhibitors. Antimicrob. Agents Chemother. 2008, 52, 3221-3228.
-
(2008)
Antimicrob. Agents Chemother.
, vol.52
, pp. 3221-3228
-
-
Cunningham, E.1
Drag, M.2
Kafarski, P.3
Bell, A.4
-
147
-
-
0033532313
-
Enzymes in organic chemistry Part 9: Chemo-enzymatic synthesis of phosphonic acid analogues of L-valine, Lleucine, L-isoleucine, L-methionine and L-ω-aminobutyric acid of high enantiomeric excess
-
Hammerschmidt, F.; Wuggenig, F. Enzymes in organic chemistry. Part 9: chemo-enzymatic synthesis of phosphonic acid analogues of L-valine, Lleucine, L-isoleucine, L-methionine and L-ω-aminobutyric acid of high enantiomeric excess. Tetrahedron: Asymmetry 1999, 10, 1709-1721.
-
(1999)
Tetrahedron: Asymmetry
, vol.10
, pp. 1709-1721
-
-
Hammerschmidt, F.1
Wuggenig, F.2
-
148
-
-
0028960436
-
Enzymes in organic chemistry, part 2: Lipase-catalysed hydrolysis of 1-acyloxy-2-aryethylphosphonates and synthesis of phosphonic acid analogues of L-phenylalanine and L-tyrosine
-
Drescher, M.; Li, Y.-F.; Hammerschmidt, F. Enzymes in organic chemistry, part 2: lipase-catalysed hydrolysis of 1-acyloxy-2-aryethylphosphonates and synthesis of phosphonic acid analogues of L-phenylalanine and L-tyrosine. Tetrahedron 1995, 51, 4933-4946.
-
(1995)
Tetrahedron
, vol.51
, pp. 4933-4946
-
-
Drescher, M.1
Li, Y.-F.2
Hammerschmidt, F.3
-
149
-
-
85077634689
-
The use of diethyl azodicarboxylate and triphenylphosphine in synthesis and transformation of natural products
-
Mitsunobu, O. The use of diethyl azodicarboxylate and triphenylphosphine in synthesis and transformation of natural products. Synthesis 1981, 1-28.
-
(1981)
Synthesis
, pp. 1-28
-
-
Mitsunobu, O.1
-
150
-
-
0002779608
-
Replacement of alcoholic hydroxyl groups by halogens and other nucleophiles via oxyphosphonium intermediates
-
Castro, B. R. Replacement of alcoholic hydroxyl groups by halogens and other nucleophiles via oxyphosphonium intermediates. Org. React. 1983, 29, 1-162.
-
(1983)
Org. React.
, vol.29
, pp. 1-162
-
-
Castro, B.R.1
-
151
-
-
0000414496
-
The Mitsunobu reaction
-
Hughess, D. L. The Mitsunobu reaction. Org. React. 1992, 42, 335-356.
-
(1992)
Org. React.
, vol.42
, pp. 335-356
-
-
Hughess, D.L.1
-
152
-
-
0001640928
-
Progress in the Mitsunobu reaction A review
-
Hughess, D. L. Progress in the Mitsunobu reaction. A review. Org. Prep. Proced. Int. 1996, 28, 127-164.
-
(1996)
Org. Prep. Proced. Int.
, vol.28
, pp. 127-164
-
-
Hughess, D.L.1
-
153
-
-
0001088596
-
Advances in the Mitsunobu reaction for the stereochemical inversion of hindered secondary alcohols
-
Dodge, J. A.; Jones, S. A. Advances in the Mitsunobu reaction for the stereochemical inversion of hindered secondary alcohols. Rec. Res. Dev. Org. Chem. 1997, 1, 273-283.
-
(1997)
Rec. Res. Dev. Org. Chem.
, vol.1
, pp. 273-283
-
-
Dodge, J.A.1
Jones, S.A.2
-
154
-
-
4143084064
-
Recent advances in the Mitsunobu reaction: Modified reagents and the quest for chromatography-free separation
-
Dembinski, R. Recent advances in the Mitsunobu reaction: modified reagents and the quest for chromatography-free separation. Eur. J. Org. Chem. 2004, 2763-2772.
-
(2004)
Eur. J. Org. Chem.
, pp. 2763-2772
-
-
Dembinski, R.1
-
155
-
-
0037071231
-
Fluorous Mitsunobu reagents and reactions
-
Dandapani, S.; Curran, D. P. Fluorous Mitsunobu reagents and reactions. Tetrahedron 2002, 58, 3855-3864.
-
(2002)
Tetrahedron
, vol.58
, pp. 3855-3864
-
-
Dandapani, S.1
Curran, D.P.2
-
156
-
-
33750902195
-
Simplification of the Mitsunobu reaction Di-p-chlorobenzyl azodicarboxylate: A new azodicarboxylate
-
Lipshutz, B. H.; Chung, D. W.; Rich, B.; Corral, R. Simplification of the Mitsunobu reaction. Di-p-chlorobenzyl azodicarboxylate: a new azodicarboxylate. Org. Lett. 2006, 8, 5069-5072.
-
(2006)
Org. Lett.
, vol.8
, pp. 5069-5072
-
-
Lipshutz, B.H.1
Chung, D.W.2
Rich, B.3
Corral, R.4
-
157
-
-
0037467898
-
A convenient synthesis of 1-aminophosphonates from 1-hydroxyphosphonates
-
For the synthesis of non-chiral ω-aminophosphonates from ω-hydroxyphosphonates under solvent-free conditions using microwave irradiation, see
-
For the synthesis of non-chiral ω-aminophosphonates from ω-hydroxyphosphonates under solvent-free conditions using microwave irradiation, see: Kaboudin, B. A convenient synthesis of 1-aminophosphonates from 1-hydroxyphosphonates. Tetrahedron Lett. 2003, 44, 1051-1053.
-
(2003)
Tetrahedron Lett.
, vol.44
, pp. 1051-1053
-
-
Kaboudin, B.1
-
158
-
-
23944516347
-
ω-Aminoalkylphosphonates as a tool in experimental optimisation of P1 side chain shape of potential inhibitors in S1 pocket of leucine-and neutral aminopeptidases
-
Drαg, M.; Grembecka, J.; Paweαczak, M.; Kafarski, P. ω-Aminoalkylphosphonates as a tool in experimental optimisation of P1 side chain shape of potential inhibitors in S1 pocket of leucine-and neutral aminopeptidases. Eur. J. Med. Chem. 2005, 40, 764-771.
-
(2005)
Eur. J. Med. Chem.
, vol.40
, pp. 764-771
-
-
Drαg, M.1
Grembecka, J.2
Paweαczak, M.3
Kafarski, P.4
-
159
-
-
0035912827
-
Inhibition of the aminopeptidase from Aeromonas proteolytica by L-leucinephosphonic acid Spectroscopic and crystallographic characterization of the transition state of peptide hydrolysis
-
Stamper, C.; Bennett, B.; Edwards, T.; Holz, R. C.; Ringe, D.; Petsko, G. Inhibition of the aminopeptidase from Aeromonas proteolytica by L-leucinephosphonic acid. Spectroscopic and crystallographic characterization of the transition state of peptide hydrolysis. Biochemistry 2001, 40, 7035-7046.
-
(2001)
Biochemistry
, vol.40
, pp. 7035-7046
-
-
Stamper, C.1
Bennett, B.2
Edwards, T.3
Holz, R.C.4
Ringe, D.5
Petsko, G.6
-
160
-
-
0141649386
-
A new enzyme model for enantioselective esterases based on molecularly imprinted polymers
-
Emgenbroich, M.; Wulff, G. A new enzyme model for enantioselective esterases based on molecularly imprinted polymers. Chem. Eur. J. 2003, 9, 4106-4117.
-
(2003)
Chem. Eur. J.
, vol.9
, pp. 4106-4117
-
-
Emgenbroich, M.1
Wulff, G.2
-
161
-
-
0038115341
-
The most potent organophosphorus inhibitors of leucine aminopeptidase Structure-based design, chemistry, and activity
-
Grembecka, J.; Mucha, A.; Cierpicki, T.; Kafarski, P. The most potent organophosphorus inhibitors of leucine aminopeptidase. Structure-based design, chemistry, and activity. J. Med. Chem. 2003, 46, 2641-2655.
-
(2003)
J. Med. Chem.
, vol.46
, pp. 2641-2655
-
-
Grembecka, J.1
Mucha, A.2
Cierpicki, T.3
Kafarski, P.4
-
162
-
-
0032567158
-
Inhibition of the aminopeptidase from Aeromonas proteolytica by L-leucinephosphonic acid, a transition state analogue of peptide hydrolysis
-
Bennett, B.; Holz, R. C. Inhibition of the aminopeptidase from Aeromonas proteolytica by L-leucinephosphonic acid, a transition state analogue of peptide hydrolysis. J. Am. Chem. Soc. 1998, 120, 12139-12140.
-
(1998)
J. Am. Chem. Soc.
, vol.120
, pp. 12139-12140
-
-
Bennett, B.1
Holz, R.C.2
-
163
-
-
0029025424
-
A highly convenient route to optically pure ω-aminophosphonic acids
-
Hamilton, R.; Walker, B.; Walker, B. J. A highly convenient route to optically pure ω-aminophosphonic acids. Tetrahedron Lett. 1995, 36, 4451-4454.
-
(1995)
Tetrahedron Lett.
, vol.36
, pp. 4451-4454
-
-
Hamilton, R.1
Walker, B.2
Walker, B.J.3
-
164
-
-
0036020811
-
The computer-aided design, synthesis, and activity prediction of new leucine aminopeptidase inhibitors
-
Drag, M.; Grembecka, J.; Kafarski, P. The computer-aided design, synthesis, and activity prediction of new leucine aminopeptidase inhibitors. Phosphorus, Sulfur Silicon Relat. Elem. 2002, 177, 1591-1595.
-
(2002)
Phosphorus, Sulfur Silicon Relat. Elem.
, vol.177
, pp. 1591-1595
-
-
Drag, M.1
Grembecka, J.2
Kafarski, P.3
-
165
-
-
1842555199
-
Thiourea-catalyzed enantioselective hydrophosphonylation of imines: Practical access to enantiomerically enriched ω-amino phosphonic acids
-
Joly, G. D.; Jacobsen, E. N. Thiourea-catalyzed enantioselective hydrophosphonylation of imines: practical access to enantiomerically enriched ω-amino phosphonic acids. J. Am. Chem. Soc. 2004, 126, 4102-4103.
-
(2004)
J. Am. Chem. Soc.
, vol.126
, pp. 4102-4103
-
-
Joly, G.D.1
Jacobsen, E.N.2
-
166
-
-
0026551174
-
Enantioselective synthesis of ω-aminophosphonic acids by an application of stereoselective opening of homochiral dioxane acetals with triethyl phosphite
-
Yokomatsu, T.; Shibuya, S. Enantioselective synthesis of ω-aminophosphonic acids by an application of stereoselective opening of homochiral dioxane acetals with triethyl phosphite. Tetrahedron: Asymmetry 1992, 3, 377-378.
-
(1992)
Tetrahedron: Asymmetry
, vol.3
, pp. 377-378
-
-
Yokomatsu, T.1
Shibuya, S.2
-
167
-
-
0032543521
-
Synthesis and evaluation of diphenyl phosphonate esters as inhibitors of the trypsin-like granzymes A and K and mast cell tryptase
-
Jackson, D. S.; Fraser, S. A.; Ni, L.-M.; Kam, C.-M.; Winkler, U.; Johnson, D. A.; Froelich, C. J.; Hudig, D.; Powers, J. C. Synthesis and evaluation of diphenyl phosphonate esters as inhibitors of the trypsin-like granzymes A and K and mast cell tryptase. J. Med. Chem. 1998, 41, 2289-2301.
-
(1998)
J. Med. Chem.
, vol.41
, pp. 2289-2301
-
-
Jackson, D.S.1
Fraser, S.A.2
Ni, L.-M.3
Kam, C.-M.4
Winkler, U.5
Johnson, D.A.6
Froelich, C.J.7
Hudig, D.8
Powers, J.C.9
-
168
-
-
33646059852
-
Development of activity-based probes for trypsinfamily serine proteases
-
Pan, Z.; Jeffery, D. A.; Chehade, K.; Beltman, J.; Clark, J. M.; Grothaus, P.; Bogyo, M.; Baruch, A. Development of activity-based probes for trypsinfamily serine proteases. Bioorg. Med. Chem. Lett. 2006, 16, 2882-2885.
-
(2006)
Bioorg. Med. Chem. Lett.
, vol.16
, pp. 2882-2885
-
-
Pan, Z.1
Jeffery, D.A.2
Chehade, K.3
Beltman, J.4
Clark, J.M.5
Grothaus, P.6
Bogyo, M.7
Baruch, A.8
-
169
-
-
0034512642
-
Syntheses of new racemic N-(1-iminoethyl)phosphalysine derivatives as potential inhibitors of nitric oxide synthase
-
Massa, M. A.; Pitzele, B. S.; Jerome, G. M.; Moore, W. M.; Manning, P. T.; Sikorski, J. A. Syntheses of new racemic N-(1-iminoethyl)phosphalysine derivatives as potential inhibitors of nitric oxide synthase. Heteroatom Chem. 2000, 11, 505-511.
-
(2000)
Heteroatom Chem.
, vol.11
, pp. 505-511
-
-
Massa, M.A.1
Pitzele, B.S.2
Jerome, G.M.3
Moore, W.M.4
Manning, P.T.5
Sikorski, J.A.6
-
170
-
-
0013610276
-
1-Aminoalkylphosphonous acids. Part 1. Isosteres of the protein amino acids
-
Keith, B. E.; Campbell, C. D.; Dingwall, J. G. 1-Aminoalkylphosphonous acids. Part 1. Isosteres of the protein amino acids. J. Chem. Soc., Perkin Trans. 1 1984, 2845-2853.
-
(1984)
J. Chem. Soc., Perkin Trans. 1
, pp. 2845-2853
-
-
Keith, B.E.1
Campbell, C.D.2
Dingwall, J.G.3
-
171
-
-
0024847293
-
Synthesis of new phosphonate inhibitors of serine proteases
-
Fastrez, J.; Jespers, L.; Lison, D.; Renard, M.; Sonveaux, E. Synthesis of new phosphonate inhibitors of serine proteases. Tetrahedron Lett. 1989, 30, 6861-6864.
-
(1989)
Tetrahedron Lett.
, vol.30
, pp. 6861-6864
-
-
Fastrez, J.1
Jespers, L.2
Lison, D.3
Renard, M.4
Sonveaux, E.5
-
172
-
-
33646513265
-
Synthesis of isocyanide derivatives of ω-aminoalkylphosphonate diphenyl esters
-
For the synthesis of protected LysP, see
-
For the synthesis of protected LysP, see: Sieβczyk, M.; Kliszczak, M.; Oleksyszyn, J. Synthesis of isocyanide derivatives of ω-aminoalkylphosphonate diphenyl esters. Tetrahedron Lett. 2006, 47, 4209-4211.
-
(2006)
Tetrahedron Lett.
, vol.47
, pp. 4209-4211
-
-
Sießczyk, M.1
Kliszczak, M.2
Oleksyszyn, J.3
-
173
-
-
0033539594
-
Insights into the mechanism of Escherichia coli methionine aminopeptidase from the structural analysis of reaction products and phosphorus-based transition-state analogues
-
Lowther, W. T.; Zhang, Y.; Sampson, P. B.; Honek, J. F.; Matthews, B. W. Insights into the mechanism of Escherichia coli methionine aminopeptidase from the structural analysis of reaction products and phosphorus-based transition-state analogues. Biochemistry 1999, 38, 14810-14819.
-
(1999)
Biochemistry
, vol.38
, pp. 14810-14819
-
-
Lowther, W.T.1
Zhang, Y.2
Sampson, P.B.3
Honek, J.F.4
Matthews, B.W.5
-
174
-
-
0031571612
-
Synthesis and kinetic studies of diphenyl 1-(N-peptidylamino)alkanephosphonate esters and their biotinylated derivatives as inhibitors of serine proteases and probes for lymphocyte granzymes
-
Abuelyaman, A. S.; Jackson, D. S.; Hudig, D.; Woodard, S. L.; Powers, J. C. Synthesis and kinetic studies of diphenyl 1-(N-peptidylamino)alkanephosphonate esters and their biotinylated derivatives as inhibitors of serine proteases and probes for lymphocyte granzymes. Arch. Biochem. Biophys. 1997, 344, 271-280.
-
(1997)
Arch. Biochem. Biophys.
, vol.344
, pp. 271-280
-
-
Abuelyaman, A.S.1
Jackson, D.S.2
Hudig, D.3
Woodard, S.L.4
Powers, J.C.5
-
175
-
-
0028512603
-
Fluorescent derivatives of diphenyl[1-(Npeptidylamino) alkyl]phosphonate esters: Synthesis and use in the inhibition and cellular localization of serine proteases
-
Abuelyaman, A. S.; Hudig, D.; Woodard, S. L.; Powers, J. C. Fluorescent derivatives of diphenyl[1-(Npeptidylamino) alkyl]phosphonate esters: synthesis and use in the inhibition and cellular localization of serine proteases. Bioconjugate Chem. 1994, 5, 400-405.
-
(1994)
Bioconjugate Chem.
, vol.5
, pp. 400-405
-
-
Abuelyaman, A.S.1
Hudig, D.2
Woodard, S.L.3
Powers, J.C.4
-
176
-
-
0025979246
-
Irreversible inhibition of serine proteases by peptide derivatives of (ω-aminoalkyl)phosphonate diphenyl esters
-
Oleksyszyn, J.; Powers, J. C. Irreversible inhibition of serine proteases by peptide derivatives of (ω-aminoalkyl)phosphonate diphenyl esters. Biochemistry 1991, 30, 485-493.
-
(1991)
Biochemistry
, vol.30
, pp. 485-493
-
-
Oleksyszyn, J.1
Powers, J.C.2
-
177
-
-
0037059912
-
Synthesis of an ω-aminophosphonate nucleoside as an inhibitor of S-adenosyl-L-homocysteine hydrolase
-
Steere, J. A.; Sampson, P. B.; Honek, J. F. Synthesis of an ω-aminophosphonate nucleoside as an inhibitor of S-adenosyl-L-homocysteine hydrolase. Bioorg. Med. Chem. Lett. 2002, 12, 457-460.
-
(2002)
Bioorg. Med. Chem. Lett.
, vol.12
, pp. 457-460
-
-
Steere, J.A.1
Sampson, P.B.2
Honek, J.F.3
-
178
-
-
0001357755
-
Nucleophilic additions to N-glycosylnitrones: Asymmetric synthesis of N-hydroxy-ω-aminophosphonic and ω-aminophosphonic acids
-
Huber, R.; Vasella, A. Nucleophilic additions to N-glycosylnitrones: asymmetric synthesis of N-hydroxy-ω-aminophosphonic and ω-aminophosphonic acids. Helv. Chim. Acta 1987, 70, 1461-1476.
-
(1987)
Helv. Chim. Acta
, vol.70
, pp. 1461-1476
-
-
Huber, R.1
Vasella, A.2
-
179
-
-
0019545487
-
Dual effects of phenylalanine analogs on rabbit-muscle pyruvate kinase activity
-
Izbicka-Dimitrjevic, E.; Mastalerz, P.; Kochman, M. Dual effects of phenylalanine analogs on rabbit-muscle pyruvate kinase activity. Eur. J. Biochem. 1981, 114, 565-568.
-
(1981)
Eur. J. Biochem.
, vol.114
, pp. 565-568
-
-
Izbicka-Dimitrjevic, E.1
Mastalerz, P.2
Kochman, M.3
-
180
-
-
0030272641
-
Phosphatase inhibitors-III Benzylaminophosphonic acids as potent inhibitors of human prostatic acid phosphatase
-
Beers, S. A.; Schwender, C. F.; Loughney, D. A.; Malloy, E.; Demarest, K.; Jordan, J. Phosphatase inhibitors-III. Benzylaminophosphonic acids as potent inhibitors of human prostatic acid phosphatase. Bioorg. Med. Chem. 1996, 4, 1693-1701.
-
(1996)
Bioorg. Med. Chem.
, vol.4
, pp. 1693-1701
-
-
Beers, S.A.1
Schwender, C.F.2
Loughney, D.A.3
Malloy, E.4
Demarest, K.5
Jordan, J.6
-
181
-
-
84963145245
-
Organic phosphorus compounds Synthesis and properties of 1-amino-2-arylethylphosphonic and phosphinic acids as well as phosphine oxides
-
Maier, L. Organic phosphorus compounds. Synthesis and properties of 1-amino-2-arylethylphosphonic and phosphinic acids as well as phosphine oxides. Phosphorus Sulfur 1990, 53, 43-67.
-
(1990)
Phosphorus Sulfur
, vol.53
, pp. 43-67
-
-
Maier, L.1
-
182
-
-
0029929790
-
Synthesis of five enantiomerically pure haptens designed for in vitro evolution of antibodies with peptidase activity
-
Wagner, J.; Lerner, R. A.; Barbas, III, C. F. Synthesis of five enantiomerically pure haptens designed for in vitro evolution of antibodies with peptidase activity. Bioorg. Med. Chem. 1996, 4, 901-916.
-
(1996)
Bioorg. Med. Chem.
, vol.4
, pp. 901-916
-
-
Wagner, J.1
Lerner, R.A.2
Barbas III, C.F.3
-
183
-
-
0030598676
-
Design and synthesis of phosphinic acids that triply inhibit endothelin converting enzyme, angiotensin converting enzyme and neutral endopeptidase 24.11
-
McKittrick, B. A.; Stamford, A. W.; Weng, X.; Ma, K.; Chackalamannil, S.; Czarniecki, M.; Cleven, R. M.; Fawzi, A. B. Design and synthesis of phosphinic acids that triply inhibit endothelin converting enzyme, angiotensin converting enzyme and neutral endopeptidase 24.11. Bioorg. Med. Chem. Lett. 1996, 6, 1629-1634.
-
(1996)
Bioorg. Med. Chem. Lett.
, vol.6
, pp. 1629-1634
-
-
McKittrick, B.A.1
Stamford, A.W.2
Weng, X.3
Ma, K.4
Chackalamannil, S.5
Czarniecki, M.6
Cleven, R.M.7
Fawzi, A.B.8
-
184
-
-
0026438772
-
Synthesis of stereochemically defined phosphonamidate-containing peptides: Inhibitors for the HIV-1 proteinase
-
Camp, N. P.; Hawkins, P. C. D.; Hitchcock, P. B.; Gani, D. Synthesis of stereochemically defined phosphonamidate-containing peptides: inhibitors for the HIV-1 proteinase. Bioorg. Med. Chem. Lett. 1992, 2, 1047-1050.
-
(1992)
Bioorg. Med. Chem. Lett.
, vol.2
, pp. 1047-1050
-
-
Camp, N.P.1
Hawkins, P.C.D.2
Hitchcock, P.B.3
Gani, D.4
-
185
-
-
0032236435
-
Synthesis of phosphono dipeptides, inhibitors of cathepsin C
-
Pawelczak, M.; Nowak, K.; Kafarski, P. Synthesis of phosphono dipeptides, inhibitors of cathepsin C. Phosphorus Sulfur 1998, 132, 65-71.
-
(1998)
Phosphorus Sulfur
, vol.132
, pp. 65-71
-
-
Pawelczak, M.1
Nowak, K.2
Kafarski, P.3
-
186
-
-
0037169268
-
Chymase inhibitor suppresses adhesion formation in a hamster experimental model
-
Okamoto, Y.; Takai, S.; Miyazaki, M. Chymase inhibitor suppresses adhesion formation in a hamster experimental model. Eur. J. Pharmacol. 2002, 435, 265-267.
-
(2002)
Eur. J. Pharmacol.
, vol.435
, pp. 265-267
-
-
Okamoto, Y.1
Takai, S.2
Miyazaki, M.3
-
187
-
-
0030934793
-
Potent non-peptidic dual inhibitors of endothelin-converting enzyme and neutral endopeptidase 24.11
-
De Lombaert, S.; Stamford, L. B.; Blanchard, L.; Tan, J.; Hoyer, D.; Diefenbacher, C. G.; Wei, D.; Wallace, E. M.; Moskal, M. A.; Paula Savage, P.; Jeng, A. Y. Potent non-peptidic dual inhibitors of endothelin-converting enzyme and neutral endopeptidase 24.11. Bioorg. Med. Chem. Lett. 1997, 7, 1059-1064.
-
(1997)
Bioorg. Med. Chem. Lett.
, vol.7
, pp. 1059-1064
-
-
de Lombaert, S.1
Stamford, L.B.2
Blanchard, L.3
Tan, J.4
Hoyer, D.5
Diefenbacher, C.G.6
Wei, D.7
Wallace, E.M.8
Moskal, M.A.9
Paula Savage, P.10
Jeng, A.Y.11
-
188
-
-
0034194353
-
A one-pot multistep approach to γ-azidophosphonate and phosphonothioate diesters: Key intermediates in the synthesis of haptens for the generation of antibody ligases
-
Harwig, C. W.; Hoffman, T. Z.; Wentworth, A. D.; Janda, K. D. A one-pot multistep approach to γ-azidophosphonate and phosphonothioate diesters: key intermediates in the synthesis of haptens for the generation of antibody ligases. Bioorg. Med. Chem. Lett. 2000, 10, 915-918.
-
(2000)
Bioorg. Med. Chem. Lett.
, vol.10
, pp. 915-918
-
-
Harwig, C.W.1
Hoffman, T.Z.2
Wentworth, A.D.3
Janda, K.D.4
-
189
-
-
0021749522
-
Phosphorous-containing analogues of aspartame
-
Nelson, V.; Mastalerz, P. Phosphorous-containing analogues of aspartame. J. Pharm. Sci. 1984, 73, 1844-1846.
-
(1984)
J. Pharm. Sci.
, vol.73
, pp. 1844-1846
-
-
Nelson, V.1
Mastalerz, P.2
-
190
-
-
52749098178
-
Stereoselective synthesis of enantiopure cyclic γ-aminophosphonic acids: Direct observation of inversion at phosphorus in phosphonate ester silyldealkylation by bromotrimethylsilane
-
For diastereoselectivity explication, see
-
For diastereoselectivity explication, see: Alfonsov, V. A.; McKenna, C. E.; Bayandina, E. V.; Kashemirov, B. A.; Yarmieva, L. N.; Punegova, L. N.; Kataeva, O. N. Stereoselective synthesis of enantiopure cyclic γ-aminophosphonic acids: direct observation of inversion at phosphorus in phosphonate ester silyldealkylation by bromotrimethylsilane. Heteroatom. Chem. 2008, 19, 575-582.
-
(2008)
Heteroatom. Chem.
, vol.19
, pp. 575-582
-
-
Alfonsov, V.A.1
McKenna, C.E.2
Bayandina, E.V.3
Kashemirov, B.A.4
Yarmieva, L.N.5
Punegova, L.N.6
Kataeva, O.N.7
-
191
-
-
0001750272
-
Asymmetric synthesis of 1-aminoalkylphosphonic acids
-
Jacquier, R.; Lhassani, M.; Petrus, C.; Petrus, F. Asymmetric synthesis of 1-aminoalkylphosphonic acids. Phosphorus Sulfur 1993, 81, 83-87.
-
(1993)
Phosphorus Sulfur
, vol.81
, pp. 83-87
-
-
Jacquier, R.1
Lhassani, M.2
Petrus, C.3
Petrus, F.4
-
192
-
-
0024544078
-
Asymmetric synthesis of (1-aminoalkyl)phosphonic acids via asymmetric aldol reaction of (isocyanomethyl) phosphonates catalyzed by a chiral ferrocenyl-phosphine-gold(I) complex
-
Sawamura, M.; Ito, Y.; Hayashi, T. Asymmetric synthesis of (1-aminoalkyl)phosphonic acids via asymmetric aldol reaction of (isocyanomethyl) phosphonates catalyzed by a chiral ferrocenyl-phosphine-gold(I) complex. Tetrahedron Lett. 1989, 30, 2247-2250.
-
(1989)
Tetrahedron Lett.
, vol.30
, pp. 2247-2250
-
-
Sawamura, M.1
Ito, Y.2
Hayashi, T.3
-
193
-
-
0029929790
-
Synthesis of five enantiomerically pure haptens designed for in vitro evolution of antibodies with peptidase activity
-
Wagner, J.; Lerner, R. A.; Barbas, III, C. F. Synthesis of five enantiomerically pure haptens designed for in vitro evolution of antibodies with peptidase activity. Bioorg. Med. Chem. 1996, 4, 901-916.
-
(1996)
Bioorg. Med. Chem.
, vol.4
, pp. 901-916
-
-
Wagner, J.1
Lerner, R.A.2
Barbas III, C.F.3
-
194
-
-
37049105484
-
Synthesis, molecular structure, and absolute configuration of an optically active (1-amino-2-phenylethyl)phosphonic acid monohydrate
-
Kowalik, J.; Sawka-Dobrowolska, W.; Gβowiak, T. Synthesis, molecular structure, and absolute configuration of an optically active (1-amino-2-phenylethyl)phosphonic acid monohydrate. J. Chem. Soc., Chem. Commun. 1984, 446-447.
-
(1984)
J. Chem. Soc., Chem. Commun.
, pp. 446-447
-
-
Kowalik, J.1
Sawka-Dobrowolska, W.2
Gßowiak, T.3
-
196
-
-
33744814981
-
Aminophosphonates as organocatalysts in the direct asymmetric aldol reaction: Towards syn selectivity in the presence of Lewis bases
-
Dinér, P.; Amedjkouh, M. Aminophosphonates as organocatalysts in the direct asymmetric aldol reaction: towards syn selectivity in the presence of Lewis bases. Org. Biomol. Chem. 2006, 4, 2091-2096.
-
(2006)
Org. Biomol. Chem.
, vol.4
, pp. 2091-2096
-
-
Dinér, P.1
Amedjkouh, M.2
-
197
-
-
58649104900
-
Asymmetric conjugate addition of unmodified cyclic ketones to nitroolefins using aminophosphonate as the organocatalyst
-
Chen, G.; Wang, Z.; Ding, K. Asymmetric conjugate addition of unmodified cyclic ketones to nitroolefins using aminophosphonate as the organocatalyst. Chin. J. Chem. 2009, 27, 163-168.
-
(2009)
Chin. J. Chem.
, vol.27
, pp. 163-168
-
-
Chen, G.1
Wang, Z.2
Ding, K.3
-
198
-
-
45849103527
-
γ-Aminophosphonates as novel organocatalysts for asymmetric Michael addition of carbonyl compounds to nitroolefins
-
Tao, Q.; Tang, G.; Lin, K.; Zhao, Y.-F. γ-Aminophosphonates as novel organocatalysts for asymmetric Michael addition of carbonyl compounds to nitroolefins. Chirality 2008, 20, 833-838.
-
(2008)
Chirality
, vol.20
, pp. 833-838
-
-
Tao, Q.1
Tang, G.2
Lin, K.3
Zhao, Y.-F.4
-
199
-
-
50649112343
-
Asymmetric conjugate addition of nitroalkanes to enones with a chiral γ-aminophosphonate catalyst
-
Malmgren, M.; Granander, J.; Amedjkouh, M. Asymmetric conjugate addition of nitroalkanes to enones with a chiral γ-aminophosphonate catalyst. Tetrahedron: Asymmetry 2008, 19, 1934-1940.
-
(2008)
Tetrahedron: Asymmetry
, vol.19
, pp. 1934-1940
-
-
Malmgren, M.1
Granander, J.2
Amedjkouh, M.3
-
200
-
-
25444463074
-
Copper-catalyzed arylation of amines using diphenyl pyrrolidine-2-phosphonate as the new ligand
-
Rao, H.; Fu, H.; Jiang, Y.; Zhao, Y. Copper-catalyzed arylation of amines using diphenyl pyrrolidine-2-phosphonate as the new ligand. J. Org. Chem. 2005, 70, 8107-8109.
-
(2005)
J. Org. Chem.
, vol.70
, pp. 8107-8109
-
-
Rao, H.1
Fu, H.2
Jiang, Y.3
Zhao, Y.4
-
201
-
-
33745171752
-
Dipeptide proline diphenyl phosphonates are potent, irreversible inhibitors of seprase (FAPγ)
-
Gilmore, B. F.; Lynas, J. F.; Scott, C. J.; McGooham, C.; Martin, L.; Walker, B. Dipeptide proline diphenyl phosphonates are potent, irreversible inhibitors of seprase (FAPγ). Biochem. Biophys. Res. Commun. 2006, 346, 436-446.
-
(2006)
Biochem. Biophys. Res. Commun.
, vol.346
, pp. 436-446
-
-
Gilmore, B.F.1
Lynas, J.F.2
Scott, C.J.3
McGooham, C.4
Martin, L.5
Walker, B.6
-
202
-
-
0141786949
-
Rapid parallel synthesis of dipeptide diphenyl phosphonate esters as inhibitors of dipeptidyl peptidases
-
Sesten, K.; Danils, L.; Van der Veken, P.; De Meester, I.; Lambeir, A.-M.; Sharpe, S.; Haemers, A.; Augustyns, K. Rapid parallel synthesis of dipeptide diphenyl phosphonate esters as inhibitors of dipeptidyl peptidases. J. Comb. Chem. 2003, 5, 336-344.
-
(2003)
J. Comb. Chem.
, vol.5
, pp. 336-344
-
-
Sesten, K.1
Danils, L.2
van der Veken, P.3
de Meester, I.4
Lambeir, A.-M.5
Sharpe, S.6
Haemers, A.7
Augustyns, K.8
-
203
-
-
0033602521
-
Structure-activity relationship of diaryl phosphonate esters as potent irreversible dipeptidyl peptidase IV inhibitors
-
Belyaev, A.; Zhang, X.; Augustyns, K.; Lambeir, A.-M.; De Meester, I.; Vedernikova, I.; Sharpe, S.; Haemers, A. Structure-activity relationship of diaryl phosphonate esters as potent irreversible dipeptidyl peptidase IV inhibitors. J. Med. Chem. 1999, 42, 1041-1050.
-
(1999)
J. Med. Chem.
, vol.42
, pp. 1041-1050
-
-
Belyaev, A.1
Zhang, X.2
Augustyns, K.3
Lambeir, A.-M.4
de Meester, I.5
Vedernikova, I.6
Sharpe, S.7
Haemers, A.8
-
204
-
-
0030612395
-
In vivo inhibition of dipeptidyl peptidase IV activity by pro-pro-diphenylphosphonate (prodipine)
-
De Meester, I.; Belyaev, A.; Lambeir, A.-M.; De Meyer, G. R. Y.; Van Osselaer, N.; Haemers, A.; Sharpe, S. In vivo inhibition of dipeptidyl peptidase IV activity by pro-pro-diphenylphosphonate (prodipine). Biochem. Pharm. 1997, 54, 173-179.
-
(1997)
Biochem. Pharm.
, vol.54
, pp. 173-179
-
-
de Meester, I.1
Belyaev, A.2
Lambeir, A.-M.3
de Meyer, G.R.Y.4
van Osselaer, N.5
Haemers, A.6
Sharpe, S.7
-
205
-
-
0028075874
-
Dipeptide phosphonates as inhibitors of dipeptidyl peptidase IV
-
Boduszek, B.; Oleksyszyn, J.; Kam, C.-M.; Selzler, J.; Smith, R. E.; Powers, J. C. Dipeptide phosphonates as inhibitors of dipeptidyl peptidase IV. J. Med. Chem. 1994, 37, 3969-3976.
-
(1994)
J. Med. Chem.
, vol.37
, pp. 3969-3976
-
-
Boduszek, B.1
Oleksyszyn, J.2
Kam, C.-M.3
Selzler, J.4
Smith, R.E.5
Powers, J.C.6
-
206
-
-
0001356419
-
Synthesis of 2-phosphonopyrrolidine and its substitution for proline in an inhibitor of angiotensin-converting enzyme
-
Petrillo, Jr., E. W.; Spitzmiller, E. R. Synthesis of 2-phosphonopyrrolidine and its substitution for proline in an inhibitor of angiotensin-converting enzyme. Tetrahedron Lett. 1979, 4929-4930.
-
(1979)
Tetrahedron Lett.
, pp. 4929-4930
-
-
Petrillo Jr., E.W.1
Spitzmiller, E.R.2
-
207
-
-
0021793924
-
Synthesis and biological activity of carboxylic acid replacement analogues of the potent angiotensin converting enzyme inhibitor 5(S)-benzamido-4-oxo-6-phenylhexanoyl-L-proline
-
Almquist, R. G.; Chao, W.-R.; Jennings-White, C. Synthesis and biological activity of carboxylic acid replacement analogues of the potent angiotensin converting enzyme inhibitor 5(S)-benzamido-4-oxo-6-phenylhexanoyl-L-proline. J. Med. Chem. 1985, 28, 1067-1071.
-
(1985)
J. Med. Chem.
, vol.28
, pp. 1067-1071
-
-
Almquist, R.G.1
Chao, W.-R.2
Jennings-White, C.3
-
208
-
-
37049166036
-
A synthesis of tropinone
-
Robinson, R. A synthesis of tropinone. J. Chem. Soc. 1917, 111, 762-768.
-
(1917)
J. Chem. Soc.
, vol.111
, pp. 762-768
-
-
Robinson, R.1
-
209
-
-
0001519457
-
Die synthese von naturstoffen, insbesondere von alkaloiden, unter physiolo-gischen
-
Schopf, C. Die synthese von naturstoffen, insbesondere von alkaloiden, unter physiolo-gischen. Angew. Chem. 1937, 50, 779-787.
-
(1937)
Angew. Chem.
, vol.50
, pp. 779-787
-
-
Schopf, C.1
-
210
-
-
0000566807
-
Stereochemistry of the Robinson-Schoepf reaction A stereospecific total synthesis of the ladybug defense alkaloids precoccinelline and coccinelline
-
Stevens, R. V.; Lee, A. W. M. Stereochemistry of the Robinson-Schoepf reaction. A stereospecific total synthesis of the ladybug defense alkaloids precoccinelline and coccinelline. J. Am. Chem. Soc. 1979, 101, 7032-7035.
-
(1979)
J. Am. Chem. Soc.
, vol.101
, pp. 7032-7035
-
-
Stevens, R.V.1
Lee, A.W.M.2
-
211
-
-
56949105334
-
A stable chiral 1,4-dihydropyridine equivalent for the asymmetric synthesis of substituted piperidines: 2-cyano-6-phenyl-oxazolopiperidine
-
Bonin, M.; Grierson, D. S.; Royer, J.; Husson H.-P. A stable chiral 1,4-dihydropyridine equivalent for the asymmetric synthesis of substituted piperidines: 2-cyano-6-phenyl-oxazolopiperidine. Org. Synth. Coll. 1998, 9, 176-180.
-
(1998)
Org. Synth. Coll.
, vol.9
, pp. 176-180
-
-
Bonin, M.1
Grierson, D.S.2
Royer, J.3
Husson, H.-P.4
-
212
-
-
0033583019
-
Asymmetric syntheses of 2-substituted and 2,5-disubstituted pyrrolidines from (3S,5R,7aR)-5-(benzotriazol-1-yl)-3-phenyl[2,1-b]oxazolopyrrolidine
-
Katritzky, A. R.; Cui, X.-L.; Yang, B.; Steel, P. J. Asymmetric syntheses of 2-substituted and 2,5-disubstituted pyrrolidines from (3S,5R,7aR)-5-(benzotriazol-1-yl)-3-phenyl[2,1-b]oxazolopyrrolidine. J. Org. Chem. 1999, 64, 1979-1985.
-
(1999)
J. Org. Chem.
, vol.64
, pp. 1979-1985
-
-
Katritzky, A.R.1
Cui, X.-L.2
Yang, B.3
Steel, P.J.4
-
213
-
-
0035795103
-
Synthesis of novel (R)-and (S)-piperidazine-3-phosphonic acids and transformation into (R)-and (S)-pyrrolidine-2-phosphonic acids
-
Kaname, M.; Arakawa, Y.; Yoshifuji, S. Synthesis of novel (R)-and (S)-piperidazine-3-phosphonic acids and transformation into (R)-and (S)-pyrrolidine-2-phosphonic acids. Tetrahedron Lett. 2001, 42, 2713-2716.
-
(2001)
Tetrahedron Lett.
, vol.42
, pp. 2713-2716
-
-
Kaname, M.1
Arakawa, Y.2
Yoshifuji, S.3
-
214
-
-
67650745031
-
Potential neuroprotective drugs in cerebral ischemia: New saturated and polyunsaturated lipids coupled to hydrophilic moieties: Synthesis and biological activity
-
Biraboneye, A. C.; Madonna, S.; Laras, Y.; Krantic, S.; Maher, P.; Kraus, J.-L. Potential neuroprotective drugs in cerebral ischemia: new saturated and polyunsaturated lipids coupled to hydrophilic moieties: synthesis and biological activity. J. Med. Chem. 2009, 52, 4358-4369.
-
(2009)
J. Med. Chem.
, vol.52
, pp. 4358-4369
-
-
Biraboneye, A.C.1
Madonna, S.2
Laras, Y.3
Krantic, S.4
Maher, P.5
Kraus, J.-L.6
-
215
-
-
0037008687
-
Direct calcium binding results in activation of brain serine racemase
-
Cook, S. P.; Galve-Roperh, I.; Martínez del Pozo, A.; Rodríguez-Crespos, I. Direct calcium binding results in activation of brain serine racemase. J. Biol. Chem. 2002, 277, 27782-27792.
-
(2002)
J. Biol. Chem.
, vol.277
, pp. 27782-27792
-
-
Cook, S.P.1
Galve-Roperh, I.2
Martínez del Pozo, A.3
Rodríguez-Crespos, I.4
-
216
-
-
84986704022
-
Absolute konfiguration der (2-amino-1-hydroxyethyl) phosphon-säure aus Acanthamoeba castellanii (Neff)-darstellung der phosphonsäure-analoga von (+)-und (-)-serin
-
Hammerschmidt, F.; Völlenkle, H. Absolute konfiguration der (2-amino-1-hydroxyethyl) phosphon-säure aus Acanthamoeba castellanii (Neff)-darstellung der phosphonsäure-analoga von (+)-und (-)-serin. Liebigs Ann. Chem. 1989, 577-583.
-
(1989)
Liebigs Ann. Chem.
, pp. 577-583
-
-
Hammerschmidt, F.1
Völlenkle, H.2
-
217
-
-
0034725687
-
Enzymes in organic chemistry Part 10: Chemo-enzymatic synthesis of L-phosphaserine and L-phosphaisoserine and enantioseparation of aminohydroxyethylphosphonic acids by non-aqueous capillary electrophoresis with quinine carbamate as chiral ion pair agent
-
Hammerschmidt, F.; Lindner, W.; Wuggenig, F.; Zarbl, E. Enzymes in organic chemistry. Part 10: chemo-enzymatic synthesis of L-phosphaserine and L-phosphaisoserine and enantioseparation of aminohydroxyethylphosphonic acids by non-aqueous capillary electrophoresis with quinine carbamate as chiral ion pair agent. Tetrahedron: Asymmetry 2000, 11, 2955-2964.
-
(2000)
Tetrahedron: Asymmetry
, vol.11
, pp. 2955-2964
-
-
Hammerschmidt, F.1
Lindner, W.2
Wuggenig, F.3
Zarbl, E.4
-
218
-
-
0000033249
-
γ-Alkylation of serine with self-reproduction of the center of chirality
-
Seebach, D.; Aebi, J. D. γ-Alkylation of serine with self-reproduction of the center of chirality. Tetrahedron Lett. 1984, 25, 2545-2548.
-
(1984)
Tetrahedron Lett.
, vol.25
, pp. 2545-2548
-
-
Seebach, D.1
Aebi, J.D.2
-
219
-
-
84985571847
-
Preparation of chiral building blocks from amino acids and peptides via electrolytic decarboxylation and TiCl4-induced aminoalkylation
-
Renaud, P.; Seebach, D. Preparation of chiral building blocks from amino acids and peptides via electrolytic decarboxylation and TiCl4-induced aminoalkylation. Angew. Chem. Int. Ed. Engl. 1986, 25, 843-844.
-
(1986)
Angew. Chem. Int. Ed. Engl.
, vol.25
, pp. 843-844
-
-
Renaud, P.1
Seebach, D.2
-
220
-
-
85004823274
-
Synthesis of the phosphonic acid analog of serine
-
Lejczak, B.; Kafarski, P.; Soroka, M.; Mastalerz, P. Synthesis of the phosphonic acid analog of serine. Synthesis 1984, 577-580.
-
(1984)
Synthesis
, pp. 577-580
-
-
Lejczak, B.1
Kafarski, P.2
Soroka, M.3
Mastalerz, P.4
-
221
-
-
0029903192
-
Efficient synthesis of the four diastereomers of phosphothreonine from lactaldehyde
-
Bongini, A.; Camerini, R.; Panunzio, M. Efficient synthesis of the four diastereomers of phosphothreonine from lactaldehyde. Tetrahedron: Asymmetry 1996, 7, 1467-1476.
-
(1996)
Tetrahedron: Asymmetry
, vol.7
, pp. 1467-1476
-
-
Bongini, A.1
Camerini, R.2
Panunzio, M.3
-
222
-
-
0027949155
-
Synthesis of (1S,2S)-phosphothreonine via Ntrimethylsilylimine of (S)-lactic aldehyde
-
Bongini, A.; Camerini, R.; Hofman, S.; Panunzio, M. Synthesis of (1S,2S)-phosphothreonine via Ntrimethylsilylimine of (S)-lactic aldehyde. Tetrahedron Lett. 1994, 35, 8045-8048.
-
(1994)
Tetrahedron Lett.
, vol.35
, pp. 8045-8048
-
-
Bongini, A.1
Camerini, R.2
Hofman, S.3
Panunzio, M.4
-
223
-
-
85047671655
-
Asymmetric synthesis of γ-amino α-hydroxy phosphonic acids via BINAP-ruthenium catalyzed hydrogenation
-
Kitamura, M.; Tokunaga, M.; Pham, T.; Lubell, W. D.; Noyori, R. Asymmetric synthesis of γ-amino α-hydroxy phosphonic acids via BINAP-ruthenium catalyzed hydrogenation. Tetrahedron Lett. 1995, 36, 5769-5772.
-
(1995)
Tetrahedron Lett.
, vol.36
, pp. 5769-5772
-
-
Kitamura, M.1
Tokunaga, M.2
Pham, T.3
Lubell, W.D.4
Noyori, R.5
-
224
-
-
84986409622
-
50 Elektrochemische decarboxylierung von L-threonin-und oligopeptidderivaten unter bildung von N-acyl-N, O-acetalen: Herstellung von oligopeptiden mit carboxamid-oder phosphonat-C-terminus
-
Seebach, D.; Charczuk, R.; Geber, C.; Renaud, P.; Berner, H.; Schneider, H. 50. Elektrochemische decarboxylierung von L-threonin-und oligopeptidderivaten unter bildung von N-acyl-N, O-acetalen: herstellung von oligopeptiden mit carboxamid-oder phosphonat-C-terminus. Helv. Chim. Acta 1989, 72, 401-425.
-
(1989)
Helv. Chim. Acta
, vol.72
, pp. 401-425
-
-
Seebach, D.1
Charczuk, R.2
Geber, C.3
Renaud, P.4
Berner, H.5
Schneider, H.6
-
225
-
-
13844296531
-
Synthesis and evaluation of new tripeptide phosphonate inhibitors of MMP-8 and MMP-2
-
Agamennone, M.; Campestre, C.; Preziuso, S.; Consalvi, V.; Crucianelli, M.; Mazza, F.; Politi, V.; Ragno, R.; Tortorella, P.; Gallina, C. Synthesis and evaluation of new tripeptide phosphonate inhibitors of MMP-8 and MMP-2. Eur. J. Med. Chem. 2005, 40, 271-279.
-
(2005)
Eur. J. Med. Chem.
, vol.40
, pp. 271-279
-
-
Agamennone, M.1
Campestre, C.2
Preziuso, S.3
Consalvi, V.4
Crucianelli, M.5
Mazza, F.6
Politi, V.7
Ragno, R.8
Tortorella, P.9
Gallina, C.10
-
226
-
-
0036520839
-
Computational study of the catalytic domain of human neutrophil collagenase Specific role of the S3 and S'3 subsites in the interaction with a phosphonate inhibitor
-
Aschi, M.; Roccatano, D.; Di Nola, A.; Gallina, C.; Gavuzzo, E.; Pochetti, G.; Pieper, M.; Tschesche, H.; Mazza, F. Computational study of the catalytic domain of human neutrophil collagenase. Specific role of the S3 and S'3 subsites in the interaction with a phosphonate inhibitor. J. Comput.-Aided Mol. Des. 2002, 16, 213-225.
-
(2002)
J. Comput.-Aided Mol. Des.
, vol.16
, pp. 213-225
-
-
Aschi, M.1
Roccatano, D.2
Di Nola, A.3
Gallina, C.4
Gavuzzo, E.5
Pochetti, G.6
Pieper, M.7
Tschesche, H.8
Mazza, F.9
-
227
-
-
0032980326
-
Inhibition of adamalysin II and MMPs by phosphonate analogues of snake venom peptides
-
D'Alessio, S.; Gallina, C.; Gavuzzo, E.; Giordano, C.; Gorini, B.; Mazza, F.; Paradisi, M. P.; Panini, G.; Pochetti, G.; Sella, A. Inhibition of adamalysin II and MMPs by phosphonate analogues of snake venom peptides. Bioorg. Med. Chem. Lett. 1999, 7, 389-394.
-
(1999)
Bioorg. Med. Chem. Lett.
, vol.7
, pp. 389-394
-
-
D'Alessio, S.1
Gallina, C.2
Gavuzzo, E.3
Giordano, C.4
Gorini, B.5
Mazza, F.6
Paradisi, M.P.7
Panini, G.8
Pochetti, G.9
Sella, A.10
-
228
-
-
0034618636
-
Two crystal structures of human neutrophil collagenase, one complexed with a primed-and the other with an unprimed-side inhibitor: Implications for drug design
-
Gavuzzo, E.; Pochetti, G.; Mazza, F.; Gallina, C.; Gorini, B.; D'Alessio, S.; Pieper, M.; Tschesche, H.; Tucker, P. A. Two crystal structures of human neutrophil collagenase, one complexed with a primed-and the other with an unprimed-side inhibitor: implications for drug design. J. Med. Chem. 2000, 43, 3377-3385.
-
(2000)
J. Med. Chem.
, vol.43
, pp. 3377-3385
-
-
Gavuzzo, E.1
Pochetti, G.2
Mazza, F.3
Gallina, C.4
Gorini, B.5
D'Alessio, S.6
Pieper, M.7
Tschesche, H.8
Tucker, P.A.9
-
229
-
-
85064410120
-
An improved synthesis of the phosphonic acid analog of tryptophan
-
Rogers, R. S.; Sterm, M. K. An improved synthesis of the phosphonic acid analog of tryptophan. Synlett 1992, 708-708.
-
(1992)
Synlett
, pp. 708
-
-
Rogers, R.S.1
Sterm, M.K.2
-
230
-
-
0001877222
-
The synthesis of D, L-phosphotryptophan
-
Chen, S. F.; Kumar, S. D.; Tishler, M. The synthesis of D, L-phosphotryptophan. Tetrahedron Lett. 1983, 24, 5461-5464.
-
(1983)
Tetrahedron Lett.
, vol.24
, pp. 5461-5464
-
-
Chen, S.F.1
Kumar, S.D.2
Tishler, M.3
-
231
-
-
0010038769
-
The phosphonic analog of tryptophan
-
Subotkowski, W.; Kowalik, J.; Tyka, R.; Mastalerz, P. The phosphonic analog of tryptophan. Pol. J. Chem. 1981, 55, 853-857.
-
(1981)
Pol. J. Chem.
, vol.55
, pp. 853-857
-
-
Subotkowski, W.1
Kowalik, J.2
Tyka, R.3
Mastalerz, P.4
-
232
-
-
0021224327
-
Isolation and characterization of I5B2, a new phosphorus containing inhibitor of angiotensin I converting enzyme produced by Actinomadura sp
-
Kido, Y.; Hamakado, T.; Anno, M.; Miyagawa, E.; Motoki, Y.; Wakamiya, T.; Shiba, T. Isolation and characterization of I5B2, a new phosphorus containing inhibitor of angiotensin I converting enzyme produced by Actinomadura sp. J. Antibiot. 1984, 37, 965-969.
-
(1984)
J. Antibiot.
, vol.37
, pp. 965-969
-
-
Kido, Y.1
Hamakado, T.2
Anno, M.3
Miyagawa, E.4
Motoki, Y.5
Wakamiya, T.6
Shiba, T.7
-
233
-
-
43549111368
-
Identification of ACE pharmacophore in the phosphonopeptide metabolite K-26
-
Ntai, I.; Bachmann, B. O. Identification of ACE pharmacophore in the phosphonopeptide metabolite K-26. Bioorg. Med. Chem. Lett. 2008, 18, 3068-3071.
-
(2008)
Bioorg. Med. Chem. Lett.
, vol.18
, pp. 3068-3071
-
-
Ntai, I.1
Bachmann, B.O.2
-
234
-
-
33750440778
-
Phosphonopeptide K-26 biosynthetic intermediates in Astrosporangium hypotensionis
-
Ntai, I.; Vanessa V. Phelan, V. V.; Bachmann, B. O. Phosphonopeptide K-26 biosynthetic intermediates in Astrosporangium hypotensionis. Chem. Commun. 2006, 4518-4520.
-
(2006)
Chem. Commun.
, pp. 4518-4520
-
-
Ntai, I.1
Vanessa, V.2
Phelan, V.V.3
Bachmann, B.O.4
-
235
-
-
0022631409
-
K-26, a novel inhibitor of angiotensin I converting enzyme produced by an actinomycete K-26
-
Yamato, M.; Koguchi, T.; Okachi, R.; Yamada, K.; Nakayama, K.; Kase, H.; Karasawa, A.; Shuto, K. K-26, a novel inhibitor of angiotensin I converting enzyme produced by an actinomycete K-26. J. Antibiot. 1986, 39, 44-52.
-
(1986)
J. Antibiot.
, vol.39
, pp. 44-52
-
-
Yamato, M.1
Koguchi, T.2
Okachi, R.3
Yamada, K.4
Nakayama, K.5
Kase, H.6
Karasawa, A.7
Shuto, K.8
-
236
-
-
0025890985
-
Structure and conformation of a novel inhibitor of angiotensin I converting enzyme: A tripeptide containing phosphonic acid
-
Hirayama, N.; Kasai, M.; Shirahata, K. Structure and conformation of a novel inhibitor of angiotensin I converting enzyme: a tripeptide containing phosphonic acid. Int. J. Pept. Prot. Res. 1991, 38, 20-24.
-
(1991)
Int. J. Pept. Prot. Res.
, vol.38
, pp. 20-24
-
-
Hirayama, N.1
Kasai, M.2
Shirahata, K.3
-
237
-
-
0343449134
-
Determination of absolute configuration of optically active 1-aminoalkanephosphonic acids by chemical correlations
-
Kowalik, J.; Zygmunt, J.; Mastalerz, P. Determination of absolute configuration of optically active 1-aminoalkanephosphonic acids by chemical correlations. Phosphorus Sulfur 1983, 18, 393-396.
-
(1983)
Phosphorus Sulfur
, vol.18
, pp. 393-396
-
-
Kowalik, J.1
Zygmunt, J.2
Mastalerz, P.3
-
238
-
-
0022570993
-
K-4, a novel inhibitor of angiotensin I converting enzyme produced by Actinomadura spiculosospora
-
Koguchi, T.; Yamada, K.; Yamoto, M.; Okachi, R.; Nakayama, K.; Kase, K. K-4, a novel inhibitor of angiotensin I converting enzyme produced by Actinomadura spiculosospora. J. Antibiot. 1986, 39, 364-371.
-
(1986)
J. Antibiot.
, vol.39
, pp. 364-371
-
-
Koguchi, T.1
Yamada, K.2
Yamoto, M.3
Okachi, R.4
Nakayama, K.5
Kase, K.6
-
239
-
-
0023143082
-
Phosphonic analogues of tyrosine and 3,4-dihydroxyphenylalanine (dopa) influence mushroom tyrosinase activity
-
Lejczak, B.; Kafarski, P.; Makowiecka, E. Phosphonic analogues of tyrosine and 3,4-dihydroxyphenylalanine (dopa) influence mushroom tyrosinase activity. Biochem. J. 1987, 242, 81-88.
-
(1987)
Biochem. J.
, vol.242
, pp. 81-88
-
-
Lejczak, B.1
Kafarski, P.2
Makowiecka, E.3
-
240
-
-
0014189785
-
Recherches sur les acides aminoalkylphosphoniques. I Action de la tyrosinase sur l'analogue phosphonique de la tyrosine
-
Cassaigne, A.; Lacoste, A. M.; Neuzil, E. Recherches sur les acides aminoalkylphosphoniques. I. Action de la tyrosinase sur l'analogue phosphonique de la tyrosine. Bull. Soc. Chim. Biol. 1967, 49, 1813-1825.
-
(1967)
Bull. Soc. Chim. Biol.
, vol.49
, pp. 1813-1825
-
-
Cassaigne, A.1
Lacoste, A.M.2
Neuzil, E.3
-
241
-
-
0033710749
-
Interaction of tyrosine phenol-lyase with phosphoro-organic analogues of substrate amino acids
-
Faleev, N. G.; Zhukov, Y. N.; Khurs, E. N.; Gogoleva, O. I.; Barbolina, M. V.; Bazhulina, N. P.; Belikov, V. M.; Demidkina, T. V.; Khomutov, R. D. Interaction of tyrosine phenol-lyase with phosphoro-organic analogues of substrate amino acids. Eur. J. Biochem. 2000, 267, 6897-6902.
-
(2000)
Eur. J. Biochem.
, vol.267
, pp. 6897-6902
-
-
Faleev, N.G.1
Zhukov, Y.N.2
Khurs, E.N.3
Gogoleva, O.I.4
Barbolina, M.V.5
Bazhulina, N.P.6
Belikov, V.M.7
Demidkina, T.V.8
Khomutov, R.D.9
-
242
-
-
0346539486
-
1-Amino-2-(4-hydroxyphenyl) ethyl phosphinic acid: A novel substrate of tyrosine phenol-lyase
-
Khomutov, R. M.; Faleev, N. G.; Belyankin, A. V.; Khurs, E. N.; Khomutov, A. R.; Peryshkova, O. E.; Belikov, V. M. 1-Amino-2-(4-hydroxyphenyl) ethyl phosphinic acid: a novel substrate of tyrosine phenol-lyase. Bioorg. Khim. (Russ.) 1997, 23, 919-921.
-
(1997)
Bioorg. Khim. (Russ.)
, vol.23
, pp. 919-921
-
-
Khomutov, R.M.1
Faleev, N.G.2
Belyankin, A.V.3
Khurs, E.N.4
Khomutov, A.R.5
Peryshkova, O.E.6
Belikov, V.M.7
-
243
-
-
33845283570
-
α-Biphenylsulfonylamino 2-methylpropyl phosphonates: Enantioselective synthesis and selective inhibition of MMPs
-
Biasone, A.; Tortorella, P.; Campestre, C.; Agamennone, M.; Preziuso, S.; Chiappini, M.; Nuti, E.; Carelli, P.; Rossello, A.; Mazza, F.; Gallina, C. α-Biphenylsulfonylamino 2-methylpropyl phosphonates: enantioselective synthesis and selective inhibition of MMPs. Bioorg. Med. Chem. 2007, 15, 791-799.
-
(2007)
Bioorg. Med. Chem.
, vol.15
, pp. 791-799
-
-
Biasone, A.1
Tortorella, P.2
Campestre, C.3
Agamennone, M.4
Preziuso, S.5
Chiappini, M.6
Nuti, E.7
Carelli, P.8
Rossello, A.9
Mazza, F.10
Gallina, C.11
-
244
-
-
32344433663
-
Structural insight into the stereoselective inhibition of MMP-8 by enantiomeric sulfonamide phosphonates
-
Pochetti, G.; Gavuzzo, E.; Campestre, C.; Agamennone, M.; Tortorella, P.; Consalvi, V.; Gallina, C.; Hiller, O.; Tschesche, H.; Tucker, P. A.; Mazza, F. Structural insight into the stereoselective inhibition of MMP-8 by enantiomeric sulfonamide phosphonates. J. Med. Chem. 2006, 49, 923-931.
-
(2006)
J. Med. Chem.
, vol.49
, pp. 923-931
-
-
Pochetti, G.1
Gavuzzo, E.2
Campestre, C.3
Agamennone, M.4
Tortorella, P.5
Consalvi, V.6
Gallina, C.7
Hiller, O.8
Tschesche, H.9
Tucker, P.A.10
Mazza, F.11
-
245
-
-
0007929196
-
Absolute configuration of optically active aminophosphonic acids
-
Gαowiak, T.; Sawka-Dobrowolska, W.; Kowalik, J.; Mastalerz, P.; Soroka, M.; Zoα, J. Absolute configuration of optically active aminophosphonic acids. Tetrahedron Lett. 1977, 45, 3965-3968.
-
(1977)
Tetrahedron Lett.
, vol.45
, pp. 3965-3968
-
-
Gαowiak, T.1
Sawka-Dobrowolska, W.2
Kowalik, J.3
Mastalerz, P.4
Soroka, M.5
Zoα, J.6
-
246
-
-
33751154738
-
Catalytic Asymmetric Synthesis of α-aminophosphonates using lanthanoid-potassium-BINOL complexes
-
Sasai, H.; Arai, S.; Tahara, Y.; Shibasaki, M. Catalytic Asymmetric Synthesis of α-aminophosphonates using lanthanoid-potassium-BINOL complexes. J. Org. Chem. 1995, 60, 6656-6657.
-
(1995)
J. Org. Chem.
, vol.60
, pp. 6656-6657
-
-
Sasai, H.1
Arai, S.2
Tahara, Y.3
Shibasaki, M.4
|