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Volumn 4, Issue 3, 2011, Pages 214-247

Chemical and radiochemical considerations in radiolabeling with α-emitting radionuclides

Author keywords

Actinium 225; Alpha emitter; Astatine 211; Bismuth 212; Bismuth 213; Chelate; Fermium 255; Radioimmunotherapy; Radiolabeling; Radium 223; Radium 224; Targeted alpha radiotherapy; Terbium 149; Thorium 226; Thorium 227

Indexed keywords

1,4,7,10 TETRAAZACYCLODODECANE 1,4,7,10 TETRAACETIC ACID; 1,4,7,10 TETRAAZACYCLODODECANE 1,4,7,10 TETRAACETIC ACID AC 225; 1,4,7,10 TETRAAZACYCLODODECANE 1,4,7,10 TETRAKIS(METHYLENEPHOSPHONIC ACID); ACTINIUM 225; ASTATINE 211; BISMUTH 212; BISMUTH 213; BORON DERIVATIVE; CHELATING AGENT; EDETIC ACID DERIVATIVE; FERMIUM 255; FULLERENE DERIVATIVE; LANTHANIDE; LIPOSOME; MONOCLONAL ANTIBODY; NANOPARTICLE; PENTETATE INDIUM IN 111; PENTETIC ACID DERIVATIVE; POLYMER; RADIOISOTOPE; RADIOPHARMACEUTICAL AGENT; RADIUM 223; RADIUM 224; SINGLE WALLED NANOTUBE; TERBIUM 149; THORIUM 226; THORIUM 227; UNCLASSIFIED DRUG;

EID: 79959556136     PISSN: 18744710     EISSN: 18744729     Source Type: Journal    
DOI: 10.2174/1874471011104030214     Document Type: Review
Times cited : (48)

References (329)
  • 1
    • 14844359242 scopus 로고    scopus 로고
    • Radiobiologic principles in radionuclide therapy
    • Kassis, A.I.; Adelstein, S.J. Radiobiologic principles in radionuclide therapy. J. Nucl. Med., 2005, 46 Suppl. 1, 4S-12S.
    • (2005) J. Nucl. Med. , vol.46 , Issue.SUPPL. 1
    • Kassis, A.I.1    Adelstein, S.J.2
  • 2
    • 0029784810 scopus 로고    scopus 로고
    • Targeted therapy using alpha emitters
    • Vaidyanathan, G.; Zalutsky, M.R. Targeted therapy using alpha emitters. Phys. Med. Biol., 1996, 41, 1915-1931.
    • (1996) Phys. Med. Biol. , vol.41 , pp. 1915-1931
    • Vaidyanathan, G.1    Zalutsky, M.R.2
  • 4
    • 0032726066 scopus 로고    scopus 로고
    • Targeted alpha therapy: Evidence for potential efficacy of alpha-immunoconjugates in the management of micrometastatic cancer
    • Allen, B.J. Targeted alpha therapy: Evidence for potential efficacy of alpha-immunoconjugates in the management of micrometastatic cancer. Australas Radiol., 1999, 43, 480-486.
    • (1999) Australas Radiol. , vol.43 , pp. 480-486
    • Allen, B.J.1
  • 5
    • 0035451674 scopus 로고    scopus 로고
    • Advancements in cancer therapy with alpha-emitters: A review
    • Imam, S.K. Advancements in cancer therapy with alpha-emitters: A review. Int. J. Rad. Oncol. Biol. Phys., 2001, 51, 271-278.
    • (2001) Int. J. Rad. Oncol. Biol. Phys. , vol.51 , pp. 271-278
    • Imam, S.K.1
  • 7
    • 14844340282 scopus 로고    scopus 로고
    • The promise of targeted alpha-particle therapy
    • Mulford, D.A.; Scheinberg, D.A.; Jurcic, J.G. The promise of targeted alpha-particle therapy. J. Nucl. Med., 2005, 46 Suppl. 1, 199S-204S.
    • (2005) J. Nucl. Med. , vol.46 , Issue.SUPPL. 1
    • Mulford, D.A.1    Scheinberg, D.A.2    Jurcic, J.G.3
  • 9
    • 35549000927 scopus 로고    scopus 로고
    • Targeted alpha-therapy: Past, present, future?
    • Brechbiel, M.W. Targeted alpha-therapy: Past, present, future? Dalton Trans., 2007, 4918-4928.
    • (2007) Dalton Trans. , pp. 4918-4928
    • Brechbiel, M.W.1
  • 10
    • 77949897111 scopus 로고    scopus 로고
    • Cancer therapy with alpha-emitters labeled peptides
    • Dadachova, E. Cancer therapy with alpha-emitters labeled peptides. Semin. Nucl. Med., 2010, 40, 204-8.
    • (2010) Semin. Nucl. Med. , vol.40 , pp. 204-208
    • Dadachova, E.1
  • 11
    • 46949107981 scopus 로고    scopus 로고
    • Realizing the potential of the actinium-225 radionuclide generator in targeted alpha particle therapy applications
    • Miederer, M.; Scheinberg, D.A.; McDevitt, M.R. Realizing the potential of the actinium-225 radionuclide generator in targeted alpha particle therapy applications. Adv. Drug Deliv. Rev., 2008, 60, 1371-1382.
    • (2008) Adv. Drug Deliv. Rev. , vol.60 , pp. 1371-1382
    • Miederer, M.1    Scheinberg, D.A.2    McDevitt, M.R.3
  • 12
    • 0036255688 scopus 로고    scopus 로고
    • Targeted therapy of cancer with radiolabeled antibodies
    • Goldenberg, D.M. Targeted therapy of cancer with radiolabeled antibodies. J. Nucl. Med., 2002, 43, 693-713.
    • (2002) J. Nucl. Med. , vol.43 , pp. 693-713
    • Goldenberg, D.M.1
  • 13
    • 27144449009 scopus 로고    scopus 로고
    • Monoclonal antibody therapy of cancer
    • Adams, G.P.; Weiner, L.M. Monoclonal antibody therapy of cancer. Nat. Biotechnol., 2005, 23, 1147-1157.
    • (2005) Nat. Biotechnol. , vol.23 , pp. 1147-1157
    • Adams, G.P.1    Weiner, L.M.2
  • 14
    • 15244351004 scopus 로고    scopus 로고
    • Overview of monoclonal antibodies in cancer therapy: Present and promise
    • Stern, M.; Herrmann, R. Overview of monoclonal antibodies in cancer therapy: Present and promise. Crit. Rev. Oncol. Hematol., 2005, 54, 11-29.
    • (2005) Crit. Rev. Oncol. Hematol. , vol.54 , pp. 11-29
    • Stern, M.1    Herrmann, R.2
  • 15
    • 33746836894 scopus 로고    scopus 로고
    • Targeted therapy of cancer: New prospects for antibodies and immunoconjugates
    • Sharkey, R.M.; Goldenberg, D.M. Targeted therapy of cancer: New prospects for antibodies and immunoconjugates. CA Cancer J. Clin., 2006, 56, 226-243.
    • (2006) CA Cancer J. Clin. , vol.56 , pp. 226-243
    • Sharkey, R.M.1    Goldenberg, D.M.2
  • 16
    • 0022515047 scopus 로고
    • Chelating agents for the binding of metal ions to antibodies
    • Meares, C.F. Chelating agents for the binding of metal ions to antibodies. Nucl. Med. Biol., 1986, 13, 311-318.
    • (1986) Nucl. Med. Biol. , vol.13 , pp. 311-318
    • Meares, C.F.1
  • 17
    • 44949283598 scopus 로고
    • Newer approaches to the radiolabeling of monoclonal antibodies by use of metal chelates
    • Gansow, O.A. Newer approaches to the radiolabeling of monoclonal antibodies by use of metal chelates. Nucl. Med. Biol., 1991, 18, 369-381.
    • (1991) Nucl. Med. Biol. , vol.18 , pp. 369-381
    • Gansow, O.A.1
  • 18
    • 33746361782 scopus 로고    scopus 로고
    • Labelling monoclonal antibodies with macrocyclic radiometal complexes. A challenge for coordination chemists
    • Kaden, T.A. Labelling monoclonal antibodies with macrocyclic radiometal complexes. A challenge for coordination chemists. Dalton Trans., 2006, 3617-23.
    • (2006) Dalton Trans. , pp. 3617-3623
    • Kaden, T.A.1
  • 19
    • 1842579039 scopus 로고    scopus 로고
    • Radiolabeling of peptides for diagnosis and therapy of non-oncological diseases
    • Sosabowski, J.; Melendez-Alafort, L.; Mather, S. Radiolabeling of peptides for diagnosis and therapy of non-oncological diseases. Q. J. Nucl. Med., 2003, 47, 223-237.
    • (2003) Q. J. Nucl. Med. , vol.47 , pp. 223-237
    • Sosabowski, J.1    Melendez-Alafort, L.2    Mather, S.3
  • 20
    • 0037262667 scopus 로고    scopus 로고
    • Synthesis of target-specific radiolabeled peptides for diagnostic imaging
    • Fichna, J.; Janecka, A. Synthesis of target-specific radiolabeled peptides for diagnostic imaging. Bioconjugate Chem., 2003, 14, 3-17.
    • (2003) Bioconjugate Chem. , vol.14 , pp. 3-17
    • Fichna, J.1    Janecka, A.2
  • 21
    • 14844354089 scopus 로고    scopus 로고
    • Candidates for peptide receptor radiotherapy today and in the future
    • Reubi, J.C.; Macke, H.R.; Krenning, E.P. Candidates for peptide receptor radiotherapy today and in the future. J. Nucl. Med., 2005, 46 Suppl. 1, 67S-75S.
    • (2005) J. Nucl. Med. , vol.46 , Issue.SUPPL. 1
    • Reubi, J.C.1    Macke, H.R.2    Krenning, E.P.3
  • 22
    • 22244439233 scopus 로고    scopus 로고
    • Radiolabeled peptides in oncology: Role in diagnosis and treatment
    • Weiner, R.E.; Thakur, M.L. Radiolabeled peptides in oncology: Role in diagnosis and treatment. BioDrugs, 2005, 19, 145-63.
    • (2005) BioDrugs , vol.19 , pp. 145-163
    • Weiner, R.E.1    Thakur, M.L.2
  • 24
    • 38649126592 scopus 로고    scopus 로고
    • Peptide-based radiopharmaceuticals and cytotoxic conjugates: Potential tools against cancer
    • Okarvi, S.M. Peptide-based radiopharmaceuticals and cytotoxic conjugates: Potential tools against cancer. Cancer Treat. Rev., 2008, 34, 13-26.
    • (2008) Cancer Treat. Rev. , vol.34 , pp. 13-26
    • Okarvi, S.M.1
  • 28
    • 0034980926 scopus 로고    scopus 로고
    • Effects of 2,3-dimercapto-1-propanesulfonic acid (DMPS) on tissue and urine mercury levels following prolonged methylmercury exposure in rats
    • Pingree, S.D.; Simmonds, P.L.; Woods, J.S. Effects of 2,3-dimercapto-1-propanesulfonic acid (DMPS) on tissue and urine mercury levels following prolonged methylmercury exposure in rats. Toxicol. Sci., 2001, 61, 224-233.
    • (2001) Toxicol. Sci. , vol.61 , pp. 224-233
    • Pingree, S.D.1    Simmonds, P.L.2    Woods, J.S.3
  • 29
    • 78549263790 scopus 로고    scopus 로고
    • Conventional and pretargeted radioimmunotherapy using bismuth-213 to target and treat non-hodgkin lymphomas expressing CD20: A preclinical model toward optimal consolidation therapy to eradicate minimal residual disease
    • Park, S.I.; Shenoi, J.; Pagel, J.M.; Hamlin, D.K.; Wilbur, D.S.; Orgun, N.; Kenoyer, A.L.; Frayo, S.; Axtman, A.; Back, T.; Lin, Y.; Fisher, D.R.; Gopal, A.K.; Green, D.J.; Press, O.W. Conventional and pretargeted radioimmunotherapy using bismuth-213 to target and treat non-hodgkin lymphomas expressing CD20: A preclinical model toward optimal consolidation therapy to eradicate minimal residual disease. Blood, 2010, 116, 4231-4239.
    • (2010) Blood , vol.116 , pp. 4231-4239
    • Park, S.I.1    Shenoi, J.2    Pagel, J.M.3    Hamlin, D.K.4    Wilbur, D.S.5    Orgun, N.6    Kenoyer, A.L.7    Frayo, S.8    Axtman, A.9    Back, T.10    Lin, Y.11    Fisher, D.R.12    Gopal, A.K.13    Green, D.J.14    Press, O.W.15
  • 32
    • 0003466026 scopus 로고
    • General properties of astatine
    • In, 8th ed.; Kugler, H. K.; Keller, C., Eds. Springer-Verlag: Berlin
    • Vasáros, L.; Berei, K., General properties of astatine. In Gmelin handbook of inorganic chemistry. Astatine, 8th ed.; Kugler, H. K.; Keller, C., Eds. Springer-Verlag: Berlin, 1985, pp. 107-128.
    • (1985) Gmelin handbook of inorganic chemistry. Astatine , pp. 107-128
    • Vasáros, L.1    Berei, K.2
  • 33
    • 0022446458 scopus 로고
    • Disposition of metals in rats: A comparative study of fecal, urinary, and biliary excretion and tissue distribution of eighteen metals
    • Gregus, Z.; Klaassen, C.D. Disposition of metals in rats: A comparative study of fecal, urinary, and biliary excretion and tissue distribution of eighteen metals. Toxicol. Appl. Pharmacol., 1986, 85, 24-38.
    • (1986) Toxicol. Appl. Pharmacol. , vol.85 , pp. 24-38
    • Gregus, Z.1    Klaassen, C.D.2
  • 35
    • 0023261787 scopus 로고
    • Tissue and subcellular distribution of bismuth radiotracer in the rat: Considerations of cytotoxicity and microdosimetry for bismuth radiopharmaceuticals
    • Zidenberg-Cherr, S.; Parks, N.J.; Keen, C.L. Tissue and subcellular distribution of bismuth radiotracer in the rat: Considerations of cytotoxicity and microdosimetry for bismuth radiopharmaceuticals. Radiat. Res., 1987, 111, 119-129.
    • (1987) Radiat. Res. , vol.111 , pp. 119-129
    • Zidenberg-Cherr, S.1    Parks, N.J.2    Keen, C.L.3
  • 37
    • 45249131181 scopus 로고
    • Relation between the location of elements in the periodic table and various organ-uptake rates
    • Ando, A.; Ando, I.; Hiraki, T.; Hisada, K. Relation between the location of elements in the periodic table and various organ-uptake rates. Nucl. Med. Biol., 1989, 16, 57-80.
    • (1989) Nucl. Med. Biol. , vol.16 , pp. 57-80
    • Ando, A.1    Ando, I.2    Hiraki, T.3    Hisada, K.4
  • 40
    • 63749118446 scopus 로고    scopus 로고
    • 211At]astatide and development of labeling reagents to increase stability
    • 211At]astatide and development of labeling reagents to increase stability. Curr. Radiopharm., 2008, 1, 144-176.
    • (2008) Curr. Radiopharm. , vol.1 , pp. 144-176
    • Wilbur, D.S.1
  • 41
    • 0035155042 scopus 로고    scopus 로고
    • Bifunctional chelators for therapeutic lanthanide radiopharmaceuticals
    • Liu, S.; Edwards, D.S. Bifunctional chelators for therapeutic lanthanide radiopharmaceuticals. Bioconj. Chem., 2001, 12, 7-34.
    • (2001) Bioconj. Chem. , vol.12 , pp. 7-34
    • Liu, S.1    Edwards, D.S.2
  • 42
    • 0030111464 scopus 로고    scopus 로고
    • Vehicles, chelators, and radionuclides: Choosing the "building blocks" of an effective therapeutic radioimmunoconjugate
    • Schubiger, P.A.; Alberto, R.; Smith, A. Vehicles, chelators, and radionuclides: Choosing the "building blocks" of an effective therapeutic radioimmunoconjugate. Bioconj. Chem., 1996, 7, 165-179.
    • (1996) Bioconj. Chem. , vol.7 , pp. 165-179
    • Schubiger, P.A.1    Alberto, R.2    Smith, A.3
  • 43
    • 0033402734 scopus 로고    scopus 로고
    • The role of inorganic chemistry in the development of radiometal agents for cancer therapy
    • Heeg, M.J.; Jurisson, S.S. The role of inorganic chemistry in the development of radiometal agents for cancer therapy. Acc. Chem. Res., 1999, 32, 1053-1060.
    • (1999) Acc. Chem. Res. , vol.32 , pp. 1053-1060
    • Heeg, M.J.1    Jurisson, S.S.2
  • 44
    • 0026008504 scopus 로고
    • Therapeutic radionuclides: Production and decay property considerations
    • Volkert, W.A.; Goeckeler, W.F.; Ehrhardt, G.J.; Ketring, A.R. Therapeutic radionuclides: Production and decay property considerations. J. Nucl. Med., 1991, 32, 174-185.
    • (1991) J. Nucl. Med. , vol.32 , pp. 174-185
    • Volkert, W.A.1    Goeckeler, W.F.2    Ehrhardt, G.J.3    Ketring, A.R.4
  • 45
    • 7744234136 scopus 로고    scopus 로고
    • The role of coordination chemistry in the development of target-specific radiopharmaceuticals
    • Liu, S. The role of coordination chemistry in the development of target-specific radiopharmaceuticals. Chem. Soc. Rev., 2004, 33, 445-461.
    • (2004) Chem. Soc. Rev. , vol.33 , pp. 445-461
    • Liu, S.1
  • 46
    • 84949404657 scopus 로고
    • Radiolabeling of monoclonal antibodies with metal chelates
    • Yuanfang, L.; Chuanchu, W. Radiolabeling of monoclonal antibodies with metal chelates. Pure Appl. Chem., 1991, 363, 427-463.
    • (1991) Pure Appl. Chem. , vol.363 , pp. 427-463
    • Yuanfang, L.1    Chuanchu, W.2
  • 47
    • 0035385136 scopus 로고    scopus 로고
    • 213Bi, and their decay chain related radionuclides, for therapeutic applications
    • 213Bi, and their decay chain related radionuclides, for therapeutic applications. Chem. Rev., 2001, 101, 2019-2036.
    • (2001) Chem. Rev. , vol.101 , pp. 2019-2036
    • Hassfjell, S.1    Brechbiel, M.W.2
  • 48
    • 33947365801 scopus 로고    scopus 로고
    • Conjugation of chelating agents to proteins and radiolabeling with trivalent metallic isotopes
    • Cooper, M.S.; Sabbah, E.; Mather, S.J. Conjugation of chelating agents to proteins and radiolabeling with trivalent metallic isotopes. Nat. Protoc., 2006, 1, 314-317.
    • (2006) Nat. Protoc. , vol.1 , pp. 314-317
    • Cooper, M.S.1    Sabbah, E.2    Mather, S.J.3
  • 49
    • 0033363494 scopus 로고    scopus 로고
    • Gadolinium(III) chelates as MRI contrast agents: Structure, dynamics, and applications
    • Caravan, P.; Ellison, J.J.; McMurry, T.J.; Lauffer, R.B. Gadolinium(III) chelates as MRI contrast agents: Structure, dynamics, and applications. Chem. Rev., 1999, 99, 2293-2352.
    • (1999) Chem. Rev. , vol.99 , pp. 2293-2352
    • Caravan, P.1    Ellison, J.J.2    McMurry, T.J.3    Lauffer, R.B.4
  • 50
    • 33845470656 scopus 로고
    • Metal chelates as probes of biological systems
    • Meares, C.F.; Wensel, T.G. Metal chelates as probes of biological systems. Acc. Chem. Res., 1984, 17, 202-209.
    • (1984) Acc. Chem. Res. , vol.17 , pp. 202-209
    • Meares, C.F.1    Wensel, T.G.2
  • 51
    • 0021512252 scopus 로고
    • Conjugation of antibodies with bifunctional chelating agents: Isothiocyanate and bromoacetamide reagents, methods of analysis, and subsequent addition of metal ions
    • Meares, C.F.; McCall, M.J.; Reardan, D.T.; Goodwin, D.A.; Diamanti, C.I.; McTigue, M. Conjugation of antibodies with bifunctional chelating agents: Isothiocyanate and bromoacetamide reagents, methods of analysis, and subsequent addition of metal ions. Anal. Biochem., 1984, 142 (1), 68-78.
    • (1984) Anal. Biochem. , vol.142 , Issue.1 , pp. 68-78
    • Meares, C.F.1    McCall, M.J.2    Reardan, D.T.3    Goodwin, D.A.4    Diamanti, C.I.5    McTigue, M.6
  • 52
    • 0022968394 scopus 로고
    • Synthesis of 1-(pisothiocyanatobenzyl) derivatives of DTPA and EDTA. Antibody labeling and tumor imaging
    • Brechbiel, M.W.; Gansow, O.A.; Atcher, R.W.; Schlom, J.; Esteban, J.; Simpson, D.E.; Colcher, D. Synthesis of 1-(pisothiocyanatobenzyl) derivatives of DTPA and EDTA. Antibody labeling and tumor imaging. Inorg. Chem., 1986, 25, 2772-2781.
    • (1986) Inorg. Chem. , vol.25 , pp. 2772-2781
    • Brechbiel, M.W.1    Gansow, O.A.2    Atcher, R.W.3    Schlom, J.4    Esteban, J.5    Simpson, D.E.6    Colcher, D.7
  • 54
    • 0024579002 scopus 로고
    • Synthesis of novel bifunctional chelators and their use in preparing monoclonal antibody conjugates for tumor targeting
    • Westerberg, D.A.; Carney, P.L.; Rogers, P.E.; Kline, S.J.; Johnson, D.K. Synthesis of novel bifunctional chelators and their use in preparing monoclonal antibody conjugates for tumor targeting. J. Med. Chem., 1989, 32, 236-243.
    • (1989) J. Med. Chem. , vol.32 , pp. 236-243
    • Westerberg, D.A.1    Carney, P.L.2    Rogers, P.E.3    Kline, S.J.4    Johnson, D.K.5
  • 57
    • 0002950518 scopus 로고
    • Kinetics and mechanisms of complex formation and ligand exchange
    • In, Martell, A.E., Ed. American Chemical Society: Washington, D. C
    • Margerum, D.W.; Cayley, G.R.; Weatherburn, D.C.; Pagenkopf, G.K., Kinetics and mechanisms of complex formation and ligand exchange. In Coordination Chemistry, Monograph 174, Martell, A.E., Ed. American Chemical Society: Washington, D.C., 1978, Vol. 2.
    • (1978) Coordination Chemistry, Monograph 174 , vol.2
    • Margerum, D.W.1    Cayley, G.R.2    Weatherburn, D.C.3    Pagenkopf, G.K.4
  • 59
    • 0025242732 scopus 로고
    • Radiometal labeling of immunoproteins: Covalent linkage of 2-(4-isothiocyanatobenzyl)diethylenetriaminepentaacetic acid ligands to immunoglobulin
    • Mirzadeh, S. Radiometal labeling of immunoproteins: Covalent linkage of 2-(4-isothiocyanatobenzyl)diethylenetriaminepentaacetic acid ligands to immunoglobulin. Bioconj. Chem., 1990, 1, 59-65.
    • (1990) Bioconj. Chem. , vol.1 , pp. 59-65
    • Mirzadeh, S.1
  • 60
    • 0026161977 scopus 로고
    • A convenient synthesis of bifunctional chelating agents based on diethylenetriaminepentaacetic acid and their coordination chemistry with yttrium(III)
    • Cummins, C.H.; Rutter, E.W., Jr.; Fordyce, W.A. A convenient synthesis of bifunctional chelating agents based on diethylenetriaminepentaacetic acid and their coordination chemistry with yttrium(III). Bioconj. Chem., 1991, 2 (3), 180-186.
    • (1991) Bioconj. Chem. , vol.2 , Issue.3 , pp. 180-186
    • Cummins, C.H.1    Rutter Jr., E.W.2    Fordyce, W.A.3
  • 61
    • 0028285302 scopus 로고
    • Comparative biodistribution of indium-and yttrium-labeled B3 monoclonal antibody conjugated to either 2-(p-SCN-Bz)-6-methyl-DTPA (1B4M-DTPA) or 2-(p-SCN-Bz)-1,4,7,10-tetraazacyclododecane tetraacetic acid (2B-DOTA)
    • Camera, L.; Kinuya, S.; Garmestani, K.; Brechbiel, M.W.; Wu, C.; Pai, L.H.; McMurry, T.J.; Gansow, O.A.; Pastan, I.; Paik, C.H.; Carrasquillo, J.A. Comparative biodistribution of indium-and yttrium-labeled B3 monoclonal antibody conjugated to either 2-(p-SCN-Bz)-6-methyl-DTPA (1B4M-DTPA) or 2-(p-SCN-Bz)-1,4,7,10-tetraazacyclododecane tetraacetic acid (2B-DOTA). Eur. J. Nucl. Med., 1994, 21, 640-646.
    • (1994) Eur. J. Nucl. Med. , vol.21 , pp. 640-646
    • Camera, L.1    Kinuya, S.2    Garmestani, K.3    Brechbiel, M.W.4    Wu, C.5    Pai, L.H.6    McMurry, T.J.7    Gansow, O.A.8    Pastan, I.9    Paik, C.H.10    Carrasquillo, J.A.11
  • 62
    • 0000051973 scopus 로고
    • Preparation and characterization of some aminopolycarboxylate complexes of manganese(III)
    • Hamm, R.E.; Suwyn, M.A. Preparation and characterization of some aminopolycarboxylate complexes of manganese(III). Inorg. Chem., 1967, 6, 139-142.
    • (1967) Inorg. Chem. , vol.6 , pp. 139-142
    • Hamm, R.E.1    Suwyn, M.A.2
  • 63
    • 33947334533 scopus 로고
    • Multidentate ligand kinetics. Xi. Polyamine reactions with copper complexes of ethylenediaminetetraacetate and cyclohexylene-diaminetetraacetate ions
    • Carr, J.D.; Libby, R.A.; Margerum, D.W. Multidentate ligand kinetics. Xi. Polyamine reactions with copper complexes of ethylenediaminetetraacetate and cyclohexylene-diaminetetraacetate ions. Inorg. Chem., 1967, 6, 1083-1088.
    • (1967) Inorg. Chem. , vol.6 , pp. 1083-1088
    • Carr, J.D.1    Libby, R.A.2    Margerum, D.W.3
  • 64
    • 3042784970 scopus 로고
    • Effect of cyclohexylene bridges on the metal ion size based selectivity of ligands in aqueous solution
    • de Sousa, A.S.; Graeme, J.B.; Croft, C.A.; Michael, J.P.; Hancock, R.D. Effect of cyclohexylene bridges on the metal ion size based selectivity of ligands in aqueous solution. Inorg. Chem., 1991, 30, 3525-3529.
    • (1991) Inorg. Chem. , vol.30 , pp. 3525-3529
    • de Sousa, A.S.1    Graeme, J.B.2    Croft, C.A.3    Michael, J.P.4    Hancock, R.D.5
  • 66
    • 37049066500 scopus 로고
    • Synthesis of c-functionalized trans-cyclohexyldiethylenetriamine-penta-acetic acids for labelling of monoclonal antibodies with the bismuth-212 o-particle emitter
    • Brechbiel, M.W.; Gansow, O.A. Synthesis of c-functionalized trans-cyclohexyldiethylenetriamine-penta-acetic acids for labelling of monoclonal antibodies with the bismuth-212 o-particle emitter. J. Chem. Soc. Perkin Trans. 1, 1992, 1173-1178.
    • (1992) J. Chem. Soc. Perkin Trans. , vol.1 , pp. 1173-1178
    • Brechbiel, M.W.1    Gansow, O.A.2
  • 68
    • 0032572835 scopus 로고    scopus 로고
    • Physical parameters and biological stability of yttrium(III) diethylenetriaminepentaacetic acid derivative conjugates
    • McMurry, T.J.; Pippin, C.G.; Wu, C.C.; Deal, K.A.; Brechbiel, M.W.; Mirzadeh, S.; Gansow, O.A. Physical parameters and biological stability of yttrium(III) diethylenetriaminepentaacetic acid derivative conjugates. J. Med. Chem., 1998, 41, 3546-3549.
    • (1998) J. Med. Chem. , vol.41 , pp. 3546-3549
    • McMurry, T.J.1    Pippin, C.G.2    Wu, C.C.3    Deal, K.A.4    Brechbiel, M.W.5    Mirzadeh, S.6    Gansow, O.A.7
  • 71
    • 0034733105 scopus 로고    scopus 로고
    • Preparation of functionalized, conformationally constrained DTPA analogues from l-or d-serine and trans-4-hydroxy-l-proline. Hydroxymethyl substituents on the central acetic acid and on the backbone
    • Pickersgill, I.F.; Rapoport, H. Preparation of functionalized, conformationally constrained DTPA analogues from l-or d-serine and trans-4-hydroxy-l-proline. Hydroxymethyl substituents on the central acetic acid and on the backbone. J. Org. Chem., 2000, 65, 4048-57.
    • (2000) J. Org. Chem. , vol.65 , pp. 4048-4057
    • Pickersgill, I.F.1    Rapoport, H.2
  • 73
    • 33845376023 scopus 로고
    • Coordination of lanthanides by two polyamino polycarboxylic macrocycles: Formation of highly stable lanthanide complexes
    • Loncin, M.F.; Desreux, J.F.; Merciny, E. Coordination of lanthanides by two polyamino polycarboxylic macrocycles: Formation of highly stable lanthanide complexes. Inorg. Chem., 1986, 25, 2646-2648.
    • (1986) Inorg. Chem. , vol.25 , pp. 2646-2648
    • Loncin, M.F.1    Desreux, J.F.2    Merciny, E.3
  • 74
    • 0001699465 scopus 로고
    • Thermodynamic study of lanthanide complexes of 1,4,7-triazacyclononane-N, Ń, Ń́-triacetic acid and 1,4,7,10-tetraazacyclododecane-N, Ń, Ń́, Ń́́-tetraacetic acid
    • Cacheris, W.P.; Nickle, S.K.; Sherry, A.D. Thermodynamic study of lanthanide complexes of 1,4,7-triazacyclononane-N, Ń, Ń́-triacetic acid and 1,4,7,10-tetraazacyclododecane-N, Ń, Ń́, Ń́́-tetraacetic acid. Inorg. Chem., 1987, 26, 958-960.
    • (1987) Inorg. Chem. , vol.26 , pp. 958-960
    • Cacheris, W.P.1    Nickle, S.K.2    Sherry, A.D.3
  • 75
    • 4243965213 scopus 로고
    • Stability constants of the lanthanide(III)-1,4,7,10-tetraazacyclododecane-N, Ń, Ń́, Ń́́-tetraacetate complexes
    • Toth, E.; Brucher, E. Stability constants of the lanthanide(III)-1,4,7,10-tetraazacyclododecane-N, Ń, Ń́, Ń́́-tetraacetate complexes. Inorganica Chimica Acta, 1994, 221, 165-167.
    • (1994) Inorganica Chimica Acta , vol.221 , pp. 165-167
    • Toth, E.1    Brucher, E.2
  • 81
    • 0011736580 scopus 로고
    • Bismuth-212-labeled anti-tac monoclonal antibody: M-particle-emitting radionuclides as modalities for radioimmunotherapy
    • Kozak, R.W.; Atcher, R.W.; Gansow, O.A.; Friedman, A.M.; Hines, J.J.; Waldmann, T.A. Bismuth-212-labeled anti-tac monoclonal antibody: m-particle-emitting radionuclides as modalities for radioimmunotherapy. Proc. Natl. Acad. Sci. USA, 1986, 83, 474-478.
    • (1986) Proc. Natl. Acad. Sci. USA , vol.83 , pp. 474-478
    • Kozak, R.W.1    Atcher, R.W.2    Gansow, O.A.3    Friedman, A.M.4    Hines, J.J.5    Waldmann, T.A.6
  • 88
    • 0033770164 scopus 로고    scopus 로고
    • Radioimmunoconjugates for targeted a therapy of malignant melanoma
    • Rizvi, S.M.A.; Sarkar, S.; Goozee, G.; Allen, B.J. Radioimmunoconjugates for targeted a therapy of malignant melanoma. Melanoma Res., 2000, 10, 281-289.
    • (2000) Melanoma Res. , vol.10 , pp. 281-289
    • Rizvi, S.M.A.1    Sarkar, S.2    Goozee, G.3    Allen, B.J.4
  • 90
    • 0035028492 scopus 로고    scopus 로고
    • Preclinical targeted alpha therapy for subcutaneous melanoma
    • Allen, B.J.; Rizvi, S.M.; Tian, Z. Preclinical targeted alpha therapy for subcutaneous melanoma. Melanoma Res., 2001, 11, 175-82.
    • (2001) Melanoma Res. , vol.11 , pp. 175-182
    • Allen, B.J.1    Rizvi, S.M.2    Tian, Z.3
  • 91
    • 0036167491 scopus 로고    scopus 로고
    • In vitro cytotoxicity of bismuth-213 (213bi)-labeled-plasminogen activator inhibitor type 2 (alpha-pai-2) on human breast cancer cells
    • Ranson, M.; Tian, Z.; Andronicos, N.M.; Rizvi, S.; Allen, B.J. In vitro cytotoxicity of bismuth-213 (213bi)-labeled-plasminogen activator inhibitor type 2 (alpha-pai-2) on human breast cancer cells. Breast Cancer Res. Treat., 2002, 71, 149-59.
    • (2002) Breast Cancer Res. Treat. , vol.71 , pp. 149-159
    • Ranson, M.1    Tian, Z.2    Andronicos, N.M.3    Rizvi, S.4    Allen, B.J.5
  • 92
    • 85047699075 scopus 로고    scopus 로고
    • In vitro and preclinical targeted alpha therapy of human prostate cancer with Bi-213 labeled J591 antibody against the prostate specific membrane antigen
    • Li, Y.; Tian, Z.; Rizvi, S.M.; Bander, N.H.; Allen, B.J. In vitro and preclinical targeted alpha therapy of human prostate cancer with Bi-213 labeled J591 antibody against the prostate specific membrane antigen. Prostate Cancer Prostatic Dis., 2002, 5, 36-46.
    • (2002) Prostate Cancer Prostatic Dis. , vol.5 , pp. 36-46
    • Li, Y.1    Tian, Z.2    Rizvi, S.M.3    Bander, N.H.4    Allen, B.J.5
  • 107
    • 0034922185 scopus 로고    scopus 로고
    • Rapid preparation of short-lived alpha particle emitting radioimmunopharmaceuticals
    • Ma, D.; McDevitt, M.R.; Finn, R.D.; Scheinberg, D.A. Rapid preparation of short-lived alpha particle emitting radioimmunopharmaceuticals. Appl. Radiat. Isot., 2001, 55, 463-470.
    • (2001) Appl. Radiat. Isot. , vol.55 , pp. 463-470
    • Ma, D.1    McDevitt, M.R.2    Finn, R.D.3    Scheinberg, D.A.4
  • 113
    • 1542609188 scopus 로고    scopus 로고
    • Susceptibility of the human pathogenic fungi cryptococcus neoformans and histoplasma capsulatum to gamma-radiation versus radioimmunotherapy with alpha-and beta-emitting radioisotopes
    • Dadachova, E.; Howell, R.W.; Bryan, R.A.; Frenkel, A.; Nosanchuk, J.D.; Casadevall, A. Susceptibility of the human pathogenic fungi cryptococcus neoformans and histoplasma capsulatum to gamma-radiation versus radioimmunotherapy with alpha-and beta-emitting radioisotopes. J. Nucl. Med., 2004, 45, 313-320.
    • (2004) J. Nucl. Med. , vol.45 , pp. 313-320
    • Dadachova, E.1    Howell, R.W.2    Bryan, R.A.3    Frenkel, A.4    Nosanchuk, J.D.5    Casadevall, A.6
  • 116
    • 34848840131 scopus 로고    scopus 로고
    • 213Bi-C-functionalized trans-cyclohexyl-diethylenetriaminepentaacetic acid-humanized 3S193 is enhanced by combination with paclitaxel chemotherapy
    • 213Bi-C-functionalized trans-cyclohexyl-diethylenetriaminepentaacetic acid-humanized 3S193 is enhanced by combination with paclitaxel chemotherapy. Clin. Cancer Res., 2007, 13 (18 Pt 2), 5604s-5612s.
    • (2007) Clin. Cancer Res. , vol.13 , Issue.18 PART 2
    • Kelly, M.P.1    Lee, F.T.2    Tahtis, K.3    Smyth, F.E.4    Brechbiel, M.W.5    Scott, A.M.6
  • 120
    • 0036660169 scopus 로고    scopus 로고
    • Bismuth 213-labeled anti-CD45 radioimmunoconjugate to condition dogs for nonmyeloablative allogeneic marrow grafts
    • Sandmaier, B.M.; Bethge, W.A.; Wilbur, D.S.; Hamlin, D.K.; Santos, E.B.; Brechbiel, M.W.; Fisher, D.R.; Storb, R. Bismuth 213-labeled anti-CD45 radioimmunoconjugate to condition dogs for nonmyeloablative allogeneic marrow grafts. Blood, 2002, 100, 318-26.
    • (2002) Blood , vol.100 , pp. 318-326
    • Sandmaier, B.M.1    Bethge, W.A.2    Wilbur, D.S.3    Hamlin, D.K.4    Santos, E.B.5    Brechbiel, M.W.6    Fisher, D.R.7    Storb, R.8
  • 121
    • 0038044865 scopus 로고    scopus 로고
    • Selective T-cell ablation with bismuth-213-labeled anti-TCRalphabeta as nonmyeloablative conditioning for allogeneic canine marrow transplantation
    • Bethge, W.A.; Wilbur, D.S.; Storb, R.; Hamlin, D.K.; Santos, E.B.; Brechbiel, M.W.; Fisher, D.R.; Sandmaier, B.M. Selective T-cell ablation with bismuth-213-labeled anti-TCRalphabeta as nonmyeloablative conditioning for allogeneic canine marrow transplantation. Blood, 2003, 101, 5068-5075.
    • (2003) Blood , vol.101 , pp. 5068-5075
    • Bethge, W.A.1    Wilbur, D.S.2    Storb, R.3    Hamlin, D.K.4    Santos, E.B.5    Brechbiel, M.W.6    Fisher, D.R.7    Sandmaier, B.M.8
  • 122
    • 4143134313 scopus 로고    scopus 로고
    • Radioimmunotherapy with bismuth-213 as conditioning for nonmyeloablative allogeneic hematopoietic cell transplantation in dogs: A dose deescalation study
    • Bethge, W.A.; Wilbur, D.S.; Storb, R.; Hamlin, D.K.; Santos, E.B.; Brechbiel, M.W.; Sandmaier, B.M. Radioimmunotherapy with bismuth-213 as conditioning for nonmyeloablative allogeneic hematopoietic cell transplantation in dogs: A dose deescalation study. Transplantation, 2004, 78, 352-359.
    • (2004) Transplantation , vol.78 , pp. 352-359
    • Bethge, W.A.1    Wilbur, D.S.2    Storb, R.3    Hamlin, D.K.4    Santos, E.B.5    Brechbiel, M.W.6    Sandmaier, B.M.7
  • 123
    • 65549097348 scopus 로고    scopus 로고
    • Biodistributions, myelosuppression, and toxicities in mice treated with an anti-CD45 antibody labeled with the alpha-emitting radionuclides bismuth-213 or astatine-211
    • Nakamae, H.; Wilbur, D.S.; Hamlin, D.K.; Thakar, M.S.; Santos, E.B.; Fisher, D.R.; Kenoyer, A.L.; Pagel, J.M.; Press, O.W.; Storb, R.; Sandmaier, B.M. Biodistributions, myelosuppression, and toxicities in mice treated with an anti-CD45 antibody labeled with the alpha-emitting radionuclides bismuth-213 or astatine-211. Cancer Res., 2009, 69, 2408-2415.
    • (2009) Cancer Res. , vol.69 , pp. 2408-2415
    • Nakamae, H.1    Wilbur, D.S.2    Hamlin, D.K.3    Thakar, M.S.4    Santos, E.B.5    Fisher, D.R.6    Kenoyer, A.L.7    Pagel, J.M.8    Press, O.W.9    Storb, R.10    Sandmaier, B.M.11
  • 125
    • 0030829956 scopus 로고    scopus 로고
    • Bi-labelled antibody and Bilabelled streptavidin. Comparison of targeting efficacy of a lymphoma cell line in vitro
    • Henriksen, G.; Funderud, S.; Hoff, P. Bi-labelled antibody and Bilabelled streptavidin. Comparison of targeting efficacy of a lymphoma cell line in vitro. J. Labl. Compd. Radiopharm., 1997, 39, 1039-1046.
    • (1997) J. Labl. Compd. Radiopharm. , vol.39 , pp. 1039-1046
    • Henriksen, G.1    Funderud, S.2    Hoff, P.3
  • 130
    • 0042870007 scopus 로고
    • Dissociation constants of the transplutonium element chelates of diethylene-pentaacetic acid (DTPA) and the application of DTPA chelates to solvent extraction separations of transplutionium elements from the lanthanide elements
    • Baybarz, R.D. Dissociation constants of the transplutonium element chelates of diethylene-pentaacetic acid (DTPA) and the application of DTPA chelates to solvent extraction separations of transplutionium elements from the lanthanide elements. J. Inorg. Nucl. Chem., 1965, 27, 1831-1839.
    • (1965) J. Inorg. Nucl. Chem. , vol.27 , pp. 1831-1839
    • Baybarz, R.D.1
  • 132
    • 1542582866 scopus 로고
    • Thermodyamic and kinetic data for macrocyclic interaction with cations and anions
    • Izatt, R.M.; Pawlak, K.; Bradshaw, J.S. Thermodyamic and kinetic data for macrocyclic interaction with cations and anions. Chem. Rev., 1991, 91, 1721-2085.
    • (1991) Chem. Rev. , vol.91 , pp. 1721-2085
    • Izatt, R.M.1    Pawlak, K.2    Bradshaw, J.S.3
  • 133
    • 84982474742 scopus 로고
    • Complex formation with tetraazaalkane-N, Ń, Ń́, Ń́́-tetraacetic acids as a funtion of ring size
    • Stetter, H.; Frank, W. Complex formation with tetraazaalkane-N, Ń, Ń́, Ń́́-tetraacetic acids as a funtion of ring size. Angew. Chem. Int. Ed. Engl., 1976, 15, 686.
    • (1976) Angew. Chem. Int. Ed. Engl. , vol.15 , pp. 686
    • Stetter, H.1    Frank, W.2
  • 134
    • 0021868224 scopus 로고
    • Copper chelates as probes of biological systems: Stable copper complexes with a macrocyclic bifunctional chelating agent
    • Moi, M.K.; Meares, C.F.; McCall, M.J.; Cole, W.C.; DeNardo, S.J. Copper chelates as probes of biological systems: Stable copper complexes with a macrocyclic bifunctional chelating agent. Anal. Biochem., 1985, 148, 249-53.
    • (1985) Anal. Biochem. , vol.148 , pp. 249-253
    • Moi, M.K.1    Meares, C.F.2    McCall, M.J.3    Cole, W.C.4    DeNardo, S.J.5
  • 137
    • 0023832349 scopus 로고
    • Copper-67-labeled monoclonal antibody lym-1, a potential radiopharmaceutical for cancer therapy: Labeling and biodistribution in Raji tumored mice
    • Deshpande, S.V.; DeNardo, S.J.; Meares, C.F.; McCall, M.J.; Adams, G.P.; Moi, M.K.; DeNardo, G.L. Copper-67-labeled monoclonal antibody lym-1, a potential radiopharmaceutical for cancer therapy: Labeling and biodistribution in Raji tumored mice. J. Nucl. Med., 1988, 29, 217-25.
    • (1988) J. Nucl. Med. , vol.29 , pp. 217-225
    • Deshpande, S.V.1    DeNardo, S.J.2    Meares, C.F.3    McCall, M.J.4    Adams, G.P.5    Moi, M.K.6    DeNardo, G.L.7
  • 138
    • 0035854927 scopus 로고    scopus 로고
    • Chelators for radioimmunotherapy: I. NMR and ab initio calculation studies on 1,4,7,10-tetra(carboxyethyl)-1,4,7,10-tetraazacyclododecane (DO4PR) and 1,4,7-tris(carboxymethyl)-10-(carboxyethyl)-1,4,7,10-tetraazacyclododeca ne (DO3A1PR)
    • Keire, D.A.; Jang, Y.H.; Li, L.; Dasgupta, S.; Goddard, W.A., III; Shively, J.E. Chelators for radioimmunotherapy: I. NMR and ab initio calculation studies on 1,4,7,10-tetra(carboxyethyl)-1,4,7,10-tetraazacyclododecane (DO4PR) and 1,4,7-tris(carboxymethyl)-10-(carboxyethyl)-1,4,7,10-tetraazacyclododeca ne (DO3A1PR). Inorg. Chem., 2001, 40, 4310-4318.
    • (2001) Inorg. Chem. , vol.40 , pp. 4310-4318
    • Keire, D.A.1    Jang, Y.H.2    Li, L.3    Dasgupta, S.4    Goddard III, W.A.5    Shively, J.E.6
  • 139
    • 0000019547 scopus 로고
    • 2O, and its relevance to NMR studies of the conformational behavior of the lanthanide complexes formed by macrocyclic ligand dota
    • 2O, and its relevance to NMR studies of the conformational behavior of the lanthanide complexes formed by macrocyclic ligand dota. Inorg. Chem., 1984, 23, 359-363.
    • (1984) Inorg. Chem. , vol.23 , pp. 359-363
    • Spirlet, M.-R.1    Rebizant, J.2    Desreux, J.F.3    Loncin, M.-F.4
  • 140
    • 33845471425 scopus 로고
    • Structural characteristics of a terbium(III) complex with 1,4,8,11-tetraazacyclo-tetradecane-1,4,8,11-tetraacetic acid. Lanthanide ions and the conformation of the 14-member macrocycles
    • Spirlet, M.-R.; Rebizant, J.; Loncin, M.-F.; Desreux, J.F. Structural characteristics of a terbium(III) complex with 1,4,8,11-tetraazacyclo-tetradecane-1,4,8,11-tetraacetic acid. Lanthanide ions and the conformation of the 14-member macrocycles. Inorg. Chem., 1984, 23, 4278-4283.
    • (1984) Inorg. Chem. , vol.23 , pp. 4278-4283
    • Spirlet, M.-R.1    Rebizant, J.2    Loncin, M.-F.3    Desreux, J.F.4
  • 141
    • 33748880706 scopus 로고
    • Synthesis, characterization, and crystal structures of M(DO3A) (M = Fe, Gd) and Na[M(DOTA)] (M = Fe, Y, Gd)
    • Chang, C.A.; Fancesconi, L.C.; Malley, M.F.; Kumar, K.; Gougoutas, J.Z.; Tweedle, M.F. Synthesis, characterization, and crystal structures of M(DO3A) (M = Fe, Gd) and Na[M(DOTA)] (M = Fe, Y, Gd). Inorg. Chem., 1993, 332, 3501-3508.
    • (1993) Inorg. Chem. , vol.332 , pp. 3501-3508
    • Chang, C.A.1    Fancesconi, L.C.2    Malley, M.F.3    Kumar, K.4    Gougoutas, J.Z.5    Tweedle, M.F.6
  • 143
    • 0347211651 scopus 로고    scopus 로고
    • Mechanistic studies of some macrocyclic complexes
    • Lincoln, S.F. Mechanistic studies of some macrocyclic complexes. Coordination Chem. Rev., 1997, 166, 255-289.
    • (1997) Coordination Chem. Rev. , vol.166 , pp. 255-289
    • Lincoln, S.F.1
  • 144
    • 33751391354 scopus 로고
    • NMR study of solution structures and dynamics of lanthanide(III) complexes of DOTA
    • Aime, S.; Botta, M.; Ermondi, G. NMR study of solution structures and dynamics of lanthanide(III) complexes of DOTA. Inorg. Chem., 1992, 31, 4291-4299.
    • (1992) Inorg. Chem. , vol.31 , pp. 4291-4299
    • Aime, S.1    Botta, M.2    Ermondi, G.3
  • 147
    • 0001002121 scopus 로고
    • The peptide way to macrocyclic bifunctional chelating agents: Synthesis of 2-(pnitrobenzyl)-1,4,7,10-tetraazacyclododecane-N, N', N", N"'-tetraacetic acid and study of its yttrium(III) complex
    • Moi, M.K.; Meares, C.F.; DeNardo, S.J. The peptide way to macrocyclic bifunctional chelating agents: Synthesis of 2-(pnitrobenzyl)-1,4,7,10-tetraazacyclododecane-N, N', N", N"'-tetraacetic acid and study of its yttrium(III) complex. J. Am. Chem. Soc., 1988, 110, 6266-6267.
    • (1988) J. Am. Chem. Soc. , vol.110 , pp. 6266-6267
    • Moi, M.K.1    Meares, C.F.2    DeNardo, S.J.3
  • 148
    • 0035083298 scopus 로고    scopus 로고
    • An improved method for conjugating monoclonal antibodies with N-hydroxysulfosuccinimidyl DOTA
    • Lewis, M.R.; Kao, J.Y.; Anderson, A.-L.J.; Shively, J.E.; Raubitschek, A. An improved method for conjugating monoclonal antibodies with N-hydroxysulfosuccinimidyl DOTA. Bioconj. Chem., 2001, 12 (2), 320-324.
    • (2001) Bioconj. Chem. , vol.12 , Issue.2 , pp. 320-324
    • Lewis, M.R.1    Kao, J.Y.2    Anderson, A.-L.J.3    Shively, J.E.4    Raubitschek, A.5
  • 150
    • 37049085190 scopus 로고
    • Synthesis of C-and N-functionalized derivatives of 1,4,7-triazacyclononane-1,4,7-triylacetic acid (NOTA), 1,4,7,10-tetraazacyclododecane-1,4,7,10-tetrayl-tetra-acetic acid (DOTA), and diethylene-triaminepenta-acetic acid (DTPA): Bifunctional complexing agents for the derivatisation of antibodies
    • Cox, J.P.L.; Craig, A.S.; Helps, I.M.; Jankowski, K.J.; Parker, D.; Eaton, M.A.W.; Millican, A.T.; Millar, K.; Beeley, N.R.A.; Boyce, B.A. Synthesis of C-and N-functionalized derivatives of 1,4,7-triazacyclononane-1,4,7-triylacetic acid (NOTA), 1,4,7,10-tetraazacyclododecane-1,4,7,10-tetrayl-tetra-acetic acid (DOTA), and diethylene-triaminepenta-acetic acid (DTPA): Bifunctional complexing agents for the derivatisation of antibodies. J. Chem. Soc. Perkin Trans. I, 1990, 2567-2576.
    • (1990) J. Chem. Soc. Perkin Trans. , vol.I , pp. 2567-2576
    • Cox, J.P.L.1    Craig, A.S.2    Helps, I.M.3    Jankowski, K.J.4    Parker, D.5    Eaton, M.A.W.6    Millican, A.T.7    Millar, K.8    Beeley, N.R.A.9    Boyce, B.A.10
  • 151
    • 0031982801 scopus 로고    scopus 로고
    • Maleimidocysteine-amido-DOTA derivatives: New reagents for radiometal chelate conjugation to antibody sulfhydryl groups undergo pH-dependent cleavage reactions
    • Lewis, M.R.; Shively, J.E. Maleimidocysteine-amido-DOTA derivatives: New reagents for radiometal chelate conjugation to antibody sulfhydryl groups undergo pH-dependent cleavage reactions. Bioconj. Chem., 1998, 9, 72-86.
    • (1998) Bioconj. Chem. , vol.9 , pp. 72-86
    • Lewis, M.R.1    Shively, J.E.2
  • 152
    • 0031594362 scopus 로고    scopus 로고
    • 90Y-labeled DOTA and maleimidocysteineamido-DOTA conjugated to chimeric anticarcinoembryonic antigen antibody in xenograft-bearing nude mice: Comparison of stable and chemically labile linker systems
    • 90Y-labeled DOTA and maleimidocysteineamido-DOTA conjugated to chimeric anticarcinoembryonic antigen antibody in xenograft-bearing nude mice: Comparison of stable and chemically labile linker systems. Bioconj. Chem., 1998, 9, 87-93.
    • (1998) Bioconj. Chem. , vol.9 , pp. 87-93
    • Williams, L.E.1    Lewis, M.R.2    Bebb, G.G.3    Clarke, K.G.4    Odom-Maryon, T.L.5    Shively, J.E.6    Raubitschek, A.A.7
  • 154
    • 0026951113 scopus 로고
    • Radiohalogenation of proteins: An overview of radionuclides, labeling methods, and reagents for conjugate labeling
    • Wilbur, D.S. Radiohalogenation of proteins: An overview of radionuclides, labeling methods, and reagents for conjugate labeling. Bioconj. Chem., 1992, 3, 433-70.
    • (1992) Bioconj. Chem. , vol.3 , pp. 433-470
    • Wilbur, D.S.1
  • 157
    • 0025935998 scopus 로고
    • Carboxymethylsubstituted bifunctional chelators: Preparation of aryl isothiocyanate derivatives of 3-(carboxymethyl)-3-azapentanedioic acid, 3,12-bis(carboxymethyl)-6,9-dioxa-3,12-diazatetra-decanedioic acid, and 1,4,7,10-tetraazacyclo-dodecane-N, N', N", N"'-tetraacetic acid for use as protein labels
    • Kline, S.J.; Betebenner, D.A.; Johnson, D.K. Carboxymethylsubstituted bifunctional chelators: Preparation of aryl isothiocyanate derivatives of 3-(carboxymethyl)-3-azapentanedioic acid, 3,12-bis(carboxymethyl)-6,9-dioxa-3,12-diazatetra-decanedioic acid, and 1,4,7,10-tetraazacyclo-dodecane-N, N', N", N"'-tetraacetic acid for use as protein labels. Bioconj. Chem., 1991, 2, 26-31.
    • (1991) Bioconj. Chem. , vol.2 , pp. 26-31
    • Kline, S.J.1    Betebenner, D.A.2    Johnson, D.K.3
  • 158
    • 79959566996 scopus 로고
    • Process for preparing mono-N-alkylated polyazamacrocycles
    • Kruper, W.J. Process for preparing mono-N-alkylated polyazamacrocycles. US Patent 5,064,956, 1991.
    • (1991) US Patent 5,064,956
    • Kruper, W.J.1
  • 159
    • 0033490521 scopus 로고    scopus 로고
    • Improved synthesis of the bifunctional chelating agent 1,4,7,10-tetraaza-N-(1-carboxy-3-(4-nitrophenyl)propyl)-N ', N ", N "'-tris(acetic acid)-cyclododecane (PA-DOTA)
    • Chappell, L.L.; Rogers, B.E.; Khazaeli, M.B.; Mayo, M.S.; Buchsbaum, D.J.; Brechbiel, M.W. Improved synthesis of the bifunctional chelating agent 1,4,7,10-tetraaza-N-(1-carboxy-3-(4-nitrophenyl)propyl)-N ', N ", N "'-tris(acetic acid)-cyclododecane (PA-DOTA). Bioorg. Med. Chem., 1999, 7, 2313-2320.
    • (1999) Bioorg. Med. Chem. , vol.7 , pp. 2313-2320
    • Chappell, L.L.1    Rogers, B.E.2    Khazaeli, M.B.3    Mayo, M.S.4    Buchsbaum, D.J.5    Brechbiel, M.W.6
  • 160
    • 0029261677 scopus 로고
    • Yttrium-90 chelation properties of tetraazatetraacetic acid macrocycles, diethylenetriaminepentaacetic acid analogues, and a novel terpyridine acyclic chelator
    • Stimmel, J.B.; Stockstill, M.E.; Kull, F.C. Yttrium-90 chelation properties of tetraazatetraacetic acid macrocycles, diethylenetriaminepentaacetic acid analogues, and a novel terpyridine acyclic chelator. Bioconj. Chem., 1995, 5, 219-225.
    • (1995) Bioconj. Chem. , vol.5 , pp. 219-225
    • Stimmel, J.B.1    Stockstill, M.E.2    Kull, F.C.3
  • 162
    • 0142043358 scopus 로고    scopus 로고
    • Synthesis and evaluation of novel bifunctional chelating agents based on 1,4,7,10-tetraazacyclo-dodecane-N, N', N", N"'-tetraacetic acid for radiolabeling proteins
    • Chappell, L.L.; Ma, D.; Milenic, D.E.; Garmestani, K.; Venditto, V.; Beitzel, M.P.; Brechbiel, M.W. Synthesis and evaluation of novel bifunctional chelating agents based on 1,4,7,10-tetraazacyclo-dodecane-N, N', N", N"'-tetraacetic acid for radiolabeling proteins. Nucl. Med. Bio., 2003, 30, 581-595.
    • (2003) Nucl. Med. Bio. , vol.30 , pp. 581-595
    • Chappell, L.L.1    Ma, D.2    Milenic, D.E.3    Garmestani, K.4    Venditto, V.5    Beitzel, M.P.6    Brechbiel, M.W.7
  • 163
    • 0037121891 scopus 로고    scopus 로고
    • Polymethylated DOTA ligands. 1. Synthesis of rigidified ligands and studies on the effects of alkyl substitution on acid-base properties and conformational mobility
    • Ranganathan, R.S.; Pillai, R.K.; Raju, N.; Fan, H.; Nguyen, H.; Tweedle, M.F.; Desreux, J.F.; Jacques, V. Polymethylated DOTA ligands. 1. Synthesis of rigidified ligands and studies on the effects of alkyl substitution on acid-base properties and conformational mobility. Inorg. Chem., 2002, 41, 6846-55.
    • (2002) Inorg. Chem. , vol.41 , pp. 6846-6855
    • Ranganathan, R.S.1    Pillai, R.K.2    Raju, N.3    Fan, H.4    Nguyen, H.5    Tweedle, M.F.6    Desreux, J.F.7    Jacques, V.8
  • 165
    • 37049078590 scopus 로고
    • Structure and solution stability of indium and gallium complexes of 1,4,7-triazacyclononane-triacetate and of yttrium complexes of 1,4,7,10-tetraazacyclododecanetetraacetate and related ligands: Kinetically stable complexes for use in imaging and radioimmunotherapy, xray molecular structure of the indium and gallium complexes of 1,4,7-triazacyclononane-1,4,7-triacetic acid
    • Broan, C.F.; Cox, J.P.L.; Craig, A.S.; Kataky, R.; Parker, D.; Harrison, A.; Randall, A.M.; Ferguson, G. Structure and solution stability of indium and gallium complexes of 1,4,7-triazacyclononane-triacetate and of yttrium complexes of 1,4,7,10-tetraazacyclododecanetetraacetate and related ligands: Kinetically stable complexes for use in imaging and radioimmunotherapy, xray molecular structure of the indium and gallium complexes of 1,4,7-triazacyclononane-1,4,7-triacetic acid. J. Chem. Soc. Perkin Trans. 2, 1991, 87-99.
    • (1991) J. Chem. Soc. Perkin Trans. , vol.2 , pp. 87-99
    • Broan, C.F.1    Cox, J.P.L.2    Craig, A.S.3    Kataky, R.4    Parker, D.5    Harrison, A.6    Randall, A.M.7    Ferguson, G.8
  • 167
    • 0025490926 scopus 로고
    • Synthesis and evaluation of two new bifunctional carboxy-methylated tetraazamacrocyclic chelating agents for protein labeling with indium-111
    • Ruser, G.; Ritter, W.; Maecke, H.R. Synthesis and evaluation of two new bifunctional carboxy-methylated tetraazamacrocyclic chelating agents for protein labeling with indium-111. Bioconj. Chem., 1990, 1, 345-349.
    • (1990) Bioconj. Chem. , vol.1 , pp. 345-349
    • Ruser, G.1    Ritter, W.2    Maecke, H.R.3
  • 169
    • 0027716160 scopus 로고
    • Novel pendant-type macrocyclic bifunctional chelating agents: (carboxymethyl)amino deriva-tives of 2-(4-nitrobenzyl)-1,4,7,10-tetraazacyclo-dodecane-N, N', N", N"'-tetraacetic acid and their complex formation with yttrium (III)
    • Takenouchi, K.; Tabe, M.; Watanabe, K.; Hazato, A.; Kato, Y.; Shionaya, M.; Koike, T.; Kimura, E. Novel pendant-type macrocyclic bifunctional chelating agents: (carboxymethyl)amino deriva-tives of 2-(4-nitrobenzyl)-1,4,7,10-tetraazacyclo-dodecane-N, N', N", N"'-tetraacetic acid and their complex formation with yttrium (III). J. Org. Chem., 1993, 58, 6895-6899.
    • (1993) J. Org. Chem. , vol.58 , pp. 6895-6899
    • Takenouchi, K.1    Tabe, M.2    Watanabe, K.3    Hazato, A.4    Kato, Y.5    Shionaya, M.6    Koike, T.7    Kimura, E.8
  • 170
    • 33751500226 scopus 로고
    • Thermodynamic and kinetic studies of lanthanide complexes of 1,4,7,10,13-pentaaza-cyclopentadecane-N, Ń, Ń́, Ń́́, Ń́́́-pentaacetic acid and 1,4,7,10,13,16-hexaazacyclooctadecane-N, Ń, Ń́, Ń́́, Ń́́́, Ń́́́́-hexaacetic acid
    • Kodama, M.; Koike, T.; Mahatma, A.B.; Kimura, E. Thermodynamic and kinetic studies of lanthanide complexes of 1,4,7,10,13-pentaaza-cyclopentadecane-N, Ń, Ń́, Ń́́, Ń́́́-pentaacetic acid and 1,4,7,10,13,16-hexaazacyclooctadecane-N, Ń, Ń́, Ń́́, Ń́́́, Ń́́́́-hexaacetic acid. Inorg. Chem., 1991, 30, 1270-1273.
    • (1991) Inorg. Chem. , vol.30 , pp. 1270-1273
    • Kodama, M.1    Koike, T.2    Mahatma, A.B.3    Kimura, E.4
  • 172
    • 0026889151 scopus 로고
    • Synthesis of novel 1,4,7-triazacyclononane-N, N', N"-triacetic acid deriva-tives suitable for protein labeling
    • Studer, M.; Meares, C.F. Synthesis of novel 1,4,7-triazacyclononane-N, N', N"-triacetic acid deriva-tives suitable for protein labeling. Bioconj. Chem., 1992, 3, 337-341.
    • (1992) Bioconj. Chem. , vol.3 , pp. 337-341
    • Studer, M.1    Meares, C.F.2
  • 173
    • 0024792586 scopus 로고
    • 71Ga NMR, and crystal structure of a neutral gallium(III) complex of 1,4,7-triazacyclo-nonanetriacetate: A potential radiopharmaceutical?
    • 71Ga NMR, and crystal structure of a neutral gallium(III) complex of 1,4,7-triazacyclo-nonanetriacetate: A potential radiopharmaceutical? J. Chem. Soc. Chem. Commun., 1989, 1793-1794.
    • (1989) J. Chem. Soc. Chem. Commun. , pp. 1793-1794
    • Craig, A.S.1    Parker, D.2    Adams, H.3    Bailey, N.A.4
  • 178
    • 0036682172 scopus 로고    scopus 로고
    • Synthesis and biological evaluation of novel macrocyclic ligands with pendent donor groups as potential yttrium chelators for radioimmunotherapy with improved complex formation kinetics
    • Chong, H.S.; Garmestani, K.; Ma, D.; Milenic, D.E.; Overstreet, T.; Brechbiel, M.W. Synthesis and biological evaluation of novel macrocyclic ligands with pendent donor groups as potential yttrium chelators for radioimmunotherapy with improved complex formation kinetics. J. Med. Chem., 2002, 45, 3458-64.
    • (2002) J. Med. Chem. , vol.45 , pp. 3458-3464
    • Chong, H.S.1    Garmestani, K.2    Ma, D.3    Milenic, D.E.4    Overstreet, T.5    Brechbiel, M.W.6
  • 179
    • 37849053994 scopus 로고    scopus 로고
    • Rational design and generation of a bimodal bifunctional ligand for antibody-targeted radiation cancer therapy
    • Chong, H.S.; Ma, X.; Le, T.; Kwamena, B.; Milenic, D.E.; Brady, E.D.; Song, H.A.; Brechbiel, M.W. Rational design and generation of a bimodal bifunctional ligand for antibody-targeted radiation cancer therapy. J. Med. Chem., 2008, 51, 118-125.
    • (2008) J. Med. Chem. , vol.51 , pp. 118-125
    • Chong, H.S.1    Ma, X.2    Le, T.3    Kwamena, B.4    Milenic, D.E.5    Brady, E.D.6    Song, H.A.7    Brechbiel, M.W.8
  • 181
    • 0000614265 scopus 로고
    • Darstellung und komplexbildung von polyazacycloalkan-N-essigsauren
    • Stetter, H.; Frank, W.; Mertens, R. Darstellung und komplexbildung von polyazacycloalkan-N-essigsauren. Tertrahedron, 1981, 37, 767-772.
    • (1981) Tertrahedron , vol.37 , pp. 767-772
    • Stetter, H.1    Frank, W.2    Mertens, R.3
  • 182
    • 0034706364 scopus 로고    scopus 로고
    • An efficient synthesis of pyridine containing triaza-macrocyclic triacetate ligand and luminescence properties of its europium(III) complex
    • Siaugue, J.-M.; Segat-Dioury, F.; Favre-Reguillon, A.; Madic, C.; Foos, J.; Guy, A. An efficient synthesis of pyridine containing triaza-macrocyclic triacetate ligand and luminescence properties of its europium(III) complex. Tetrahedron Lett., 2000, 41, 7443-7446.
    • (2000) Tetrahedron Lett. , vol.41 , pp. 7443-7446
    • Siaugue, J.-M.1    Segat-Dioury, F.2    Favre-Reguillon, A.3    Madic, C.4    Foos, J.5    Guy, A.6
  • 183
    • 0000808322 scopus 로고
    • Synthesis, crystal structure, and potentiometry of pyridine-containing tetraaza macrocycle ligands with acetate pendant arms
    • Kim, W.D.; Hrncir, D.C.; Kiefer, G.E.; Sherry, A.D. Synthesis, crystal structure, and potentiometry of pyridine-containing tetraaza macrocycle ligands with acetate pendant arms. Inorg. Chem., 1995, 34, 2225-2232.
    • (1995) Inorg. Chem. , vol.34 , pp. 2225-2232
    • Kim, W.D.1    Hrncir, D.C.2    Kiefer, G.E.3    Sherry, A.D.4
  • 184
    • 33751155242 scopus 로고
    • Relaxometry, luminescence measurements, electrophoresis, and animal biodistribution of lanthanide(III) complexes of some polyaza macrocyclic acetates containing pyridine
    • Kim, W.D.; Kiefer, G.E.; Maton, F.; McMillan, K.; Muller, R.N.; Sherry, A.D. Relaxometry, luminescence measurements, electrophoresis, and animal biodistribution of lanthanide(III) complexes of some polyaza macrocyclic acetates containing pyridine. Inorg. Chem., 1995, 34, 2225-2232.
    • (1995) Inorg. Chem. , vol.34 , pp. 2225-2232
    • Kim, W.D.1    Kiefer, G.E.2    Maton, F.3    McMillan, K.4    Muller, R.N.5    Sherry, A.D.6
  • 185
    • 33751267978 scopus 로고    scopus 로고
    • Equilibrium and formation/dissociation kinetics of some Ln(III)PCTA complexes
    • Tircso, G.; Kovacs, Z.; Sherry, A.D. Equilibrium and formation/dissociation kinetics of some Ln(III)PCTA complexes. Inorg Chem, 2006, 45, 9269-80.
    • (2006) Inorg Chem , vol.45 , pp. 9269-9280
    • Tircso, G.1    Kovacs, Z.2    Sherry, A.D.3
  • 186
    • 56249102760 scopus 로고    scopus 로고
    • Evaluation of novel bifunctional chelates for the development of Cu-64-based radiopharmaceuticals
    • Ferreira, C.L.; Yapp, D.T.; Lamsa, E.; Gleave, M.; Bensimon, C.; Jurek, P.; Kiefer, G.E. Evaluation of novel bifunctional chelates for the development of Cu-64-based radiopharmaceuticals. Nucl. Med. Biol., 2008, 35, 875-82.
    • (2008) Nucl. Med. Biol. , vol.35 , pp. 875-882
    • Ferreira, C.L.1    Yapp, D.T.2    Lamsa, E.3    Gleave, M.4    Bensimon, C.5    Jurek, P.6    Kiefer, G.E.7
  • 188
    • 63749104476 scopus 로고    scopus 로고
    • (S)-5-(p-nitrobenzyl)-PCTA, a promising bifunctional ligand with advantageous metal ion complexation kinetics
    • Tircso, G.; Benyo, E.T.; Suh, E.H.; Jurek, P.; Kiefer, G.E.; Sherry, A.D.; Kovacs, Z. (S)-5-(p-nitrobenzyl)-PCTA, a promising bifunctional ligand with advantageous metal ion complexation kinetics. Bioconj. Chem., 2009, 20, 565-575.
    • (2009) Bioconj. Chem. , vol.20 , pp. 565-575
    • Tircso, G.1    Benyo, E.T.2    Suh, E.H.3    Jurek, P.4    Kiefer, G.E.5    Sherry, A.D.6    Kovacs, Z.7
  • 190
    • 0037467468 scopus 로고    scopus 로고
    • A rare earth-DOTA-binding antibody: Probe properties and binding affinity across the lanthanide series
    • Corneillie, T.M.; Whetstone, P.A.; Fisher, A.J.; Meares, C.F. A rare earth-DOTA-binding antibody: Probe properties and binding affinity across the lanthanide series. J. Am. Chem. Soc., 2003, 125, 3436-3437.
    • (2003) J. Am. Chem. Soc. , vol.125 , pp. 3436-3437
    • Corneillie, T.M.1    Whetstone, P.A.2    Fisher, A.J.3    Meares, C.F.4
  • 191
    • 33646126500 scopus 로고    scopus 로고
    • Irreversibly binding anti-metal chelate antibodies: Artificial receptors for pretargeting
    • Corneillie, T.M.; Whetstone, P.A.; Meares, C.F. Irreversibly binding anti-metal chelate antibodies: Artificial receptors for pretargeting. J. Inorg. Biochem., 2006, 100, 882-90.
    • (2006) J. Inorg. Biochem. , vol.100 , pp. 882-890
    • Corneillie, T.M.1    Whetstone, P.A.2    Meares, C.F.3
  • 192
    • 33750604650 scopus 로고    scopus 로고
    • Antibodies with infinite affinity: Origins and applications
    • Butlin, N.G.; Meares, C.F. Antibodies with infinite affinity: Origins and applications. Acc. Chem. Res., 2006, 39, 780-787.
    • (2006) Acc. Chem. Res. , vol.39 , pp. 780-787
    • Butlin, N.G.1    Meares, C.F.2
  • 194
    • 16444385850 scopus 로고    scopus 로고
    • A comparison of high-versus low-linear energy transfer somatostatin receptor targeted radionuclide therapy in vitro
    • Nayak, T.; Norenberg, J.; Anderson, T.; Atcher, R. A comparison of high-versus low-linear energy transfer somatostatin receptor targeted radionuclide therapy in vitro. Cancer Biother. Radiopharm., 2005, 20 (1), 52-7.
    • (2005) Cancer Biother. Radiopharm. , vol.20 , Issue.1 , pp. 52-57
    • Nayak, T.1    Norenberg, J.2    Anderson, T.3    Atcher, R.4
  • 200
    • 0030611218 scopus 로고    scopus 로고
    • 212Bi-DOTMP: An alpha particle emitting bone-seeking agent for targeted radiotherapy
    • 212Bi-DOTMP: An alpha particle emitting bone-seeking agent for targeted radiotherapy. Nucl. Med. Biol., 1997, 24, 231-237.
    • (1997) Nucl. Med. Biol. , vol.24 , pp. 231-237
    • Hassfjell, S.P.1    Bruland, Ø.S.2    Hoff, P.3
  • 202
    • 26744445230 scopus 로고
    • Lead(II) and bismuth(III) complexes of the polyazacycloalkane-N-acetic acids NOTA, DOTA, and TETA
    • Kumar, K.; Magerstädt, M.; Gansow, O.A. Lead(II) and bismuth(III) complexes of the polyazacycloalkane-N-acetic acids NOTA, DOTA, and TETA. J. Chem. Soc., Chem. Commun., 1989, 3, 145-146.
    • (1989) J. Chem. Soc., Chem. Commun. , vol.3 , pp. 145-146
    • Kumar, K.1    Magerstädt, M.2    Gansow, O.A.3
  • 204
    • 69749100336 scopus 로고    scopus 로고
    • Coordination of bismuth and lead in porphyrins: Towards an in-situ generator for alpharadiotherapy?
    • Halime, Z.; Lachkar, M.; Boitrel, B. Coordination of bismuth and lead in porphyrins: Towards an in-situ generator for alpharadiotherapy? Biochimie, 2009, 91, 1318-20.
    • (2009) Biochimie , vol.91 , pp. 1318-1320
    • Halime, Z.1    Lachkar, M.2    Boitrel, B.3
  • 206
    • 0035979480 scopus 로고    scopus 로고
    • Generation of lead-212 and radioimmunoconjugates for use in cancer therapy and the 'emanating power' of stearates
    • Wrasidlo, W.; Mysels, K.J. Generation of lead-212 and radioimmunoconjugates for use in cancer therapy and the 'emanating power' of stearates. Colloids Surf., A, 2001, 186, 123-128.
    • (2001) Colloids Surf., A , vol.186 , pp. 123-128
    • Wrasidlo, W.1    Mysels, K.J.2
  • 210
    • 37049083654 scopus 로고
    • Stability enhancement of heavy-metal-macrocycle complexes via pendant amide coordination
    • Carlton, L.; Hancock, R.D.; Maumela, H.; Wainright, K.P. Stability enhancement of heavy-metal-macrocycle complexes via pendant amide coordination. J. Chem. Soc. Chem. Commun., 1994, 1007-1008.
    • (1994) J. Chem. Soc. Chem. Commun. , pp. 1007-1008
    • Carlton, L.1    Hancock, R.D.2    Maumela, H.3    Wainright, K.P.4
  • 211
    • 0001497634 scopus 로고
    • The amide oxygen as a donor group. Metal ion complexing properties of tetra-N-acetamide substituted cyclen: A crystallographic, nmr, molecular mechanics, and thermodynamic study
    • Maumela, H.; Hancock, R.D.; Carlton, L.; Reibenspies, J.H.; Wainwright, K.P. The amide oxygen as a donor group. Metal ion complexing properties of tetra-N-acetamide substituted cyclen: A crystallographic, nmr, molecular mechanics, and thermodynamic study. J. Am. Chem. Soc., 1995, 117, 6698-6707.
    • (1995) J. Am. Chem. Soc. , vol.117 , pp. 6698-6707
    • Maumela, H.1    Hancock, R.D.2    Carlton, L.3    Reibenspies, J.H.4    Wainwright, K.P.5
  • 212
    • 0019451116 scopus 로고
    • Accumulation of weak bases in relation to intralysosomal pH in cultured human skin fibroblasts
    • Hollemans, M.; Elferink, R.O.; De Groot, P.G.; Strijland, A.; Tager, J.M. Accumulation of weak bases in relation to intralysosomal pH in cultured human skin fibroblasts. Biochim. Biophys. Acta, 1981, 643, 140-51.
    • (1981) Biochim. Biophys. Acta , vol.643 , pp. 140-151
    • Hollemans, M.1    Elferink, R.O.2    de Groot, P.G.3    Strijland, A.4    Tager, J.M.5
  • 213
    • 2642714342 scopus 로고
    • Fluorescence probe measurement of the intralysosomal pH in living cells and the perturbation of pH by various agents
    • Ohkuma, S.; Poole, B. Fluorescence probe measurement of the intralysosomal pH in living cells and the perturbation of pH by various agents. Proc. Natl. Acad. Sci. USA, 1978, 75, 3327-31.
    • (1978) Proc. Natl. Acad. Sci. USA , vol.75 , pp. 3327-3331
    • Ohkuma, S.1    Poole, B.2
  • 215
    • 34250217093 scopus 로고    scopus 로고
    • Potentiation of high-LET radiation by gemcitabine: Targeting HER2 with trastuzumab to treat disseminated peritoneal disease
    • Milenic, D.E.; Garmestani, K.; Brady, E.D.; Albert, P.S.; Abdulla, A.; Flynn, J.; Brechbiel, M.W. Potentiation of high-LET radiation by gemcitabine: Targeting HER2 with trastuzumab to treat disseminated peritoneal disease. Clin. Cancer Res., 2007, 13, 1926-35.
    • (2007) Clin. Cancer Res. , vol.13 , pp. 1926-1935
    • Milenic, D.E.1    Garmestani, K.2    Brady, E.D.3    Albert, P.S.4    Abdulla, A.5    Flynn, J.6    Brechbiel, M.W.7
  • 218
    • 0024091184 scopus 로고
    • Investigations of ionsize-selective synergism in solvent extraction
    • McDowell, W.J.; Case, G.N.; Aldrup, D.W. Investigations of ionsize-selective synergism in solvent extraction. Separation Sci. Technol., 1988, 23, 1251-1268.
    • (1988) Separation Sci. Technol. , vol.23 , pp. 1251-1268
    • McDowell, W.J.1    Case, G.N.2    Aldrup, D.W.3
  • 221
    • 0000593310 scopus 로고    scopus 로고
    • Carboxylate-derived calixarenes with high selectivity for actinium-225
    • Chen, X.; Ji, M.; Fisher, D.R.; Wai, C.M. Carboxylate-derived calixarenes with high selectivity for actinium-225. Chem. Commun., 1998, 377-378.
    • (1998) Chem. Commun. , pp. 377-378
    • Chen, X.1    Ji, M.2    Fisher, D.R.3    Wai, C.M.4
  • 222
    • 0032706530 scopus 로고    scopus 로고
    • Monofunctionalization of calix[4]arene tetra-carboxylic acid at the upper rim with isothiocyanate group: First bifunctional chelating agent for alphaemitter Ac-225
    • Chen, X.Y.; Ji, M.; Fisher, D.R.; Wai, C.M. Monofunctionalization of calix[4]arene tetra-carboxylic acid at the upper rim with isothiocyanate group: First bifunctional chelating agent for alphaemitter Ac-225. Synlett, 1999, 11, 1784-1786.
    • (1999) Synlett , vol.11 , pp. 1784-1786
    • Chen, X.Y.1    Ji, M.2    Fisher, D.R.3    Wai, C.M.4
  • 232
    • 3042729733 scopus 로고    scopus 로고
    • Alpha-particle emitting atomic generator (actinium-225)-labeled trastuzumab (herceptin) targeting of breast cancer spheroids: Efficacy versus HER2/neu expression
    • Ballangrud, A.M.; Yang, W.H.; Palm, S.; Enmon, R.; Borchardt, P.E.; Pellegrini, V.A.; McDevitt, M.R.; Scheinberg, D.A.; Sgouros, G. Alpha-particle emitting atomic generator (actinium-225)-labeled trastuzumab (herceptin) targeting of breast cancer spheroids: Efficacy versus HER2/neu expression. Clin. Cancer Res., 2004, 10, 4489-4497.
    • (2004) Clin. Cancer Res. , vol.10 , pp. 4489-4497
    • Ballangrud, A.M.1    Yang, W.H.2    Palm, S.3    Enmon, R.4    Borchardt, P.E.5    Pellegrini, V.A.6    McDevitt, M.R.7    Scheinberg, D.A.8    Sgouros, G.9
  • 234
    • 33845205546 scopus 로고    scopus 로고
    • Influence of the linker on the biodistribution and catabolism of actinium-225 self-immolative tumor-targeted isotope generators
    • Antczak, C.; Jaggi, J.S.; LeFave, C.V.; Curcio, M.J.; McDevitt, M.R.; Scheinberg, D.A. Influence of the linker on the biodistribution and catabolism of actinium-225 self-immolative tumor-targeted isotope generators. Bioconj. Chem, 2006, 17, 1551-60.
    • (2006) Bioconj. Chem , vol.17 , pp. 1551-1560
    • Antczak, C.1    Jaggi, J.S.2    LeFave, C.V.3    Curcio, M.J.4    McDevitt, M.R.5    Scheinberg, D.A.6
  • 238
    • 1442351111 scopus 로고    scopus 로고
    • Thorium and actinium polyphosphonate compounds as bone-seeking alpha particleemitting agents
    • Henriksen, G.; Bruland, O.S.; Larsen, R.H. Thorium and actinium polyphosphonate compounds as bone-seeking alpha particleemitting agents. Anticancer Res., 2004, 24, 101-5.
    • (2004) Anticancer Res. , vol.24 , pp. 101-105
    • Henriksen, G.1    Bruland, O.S.2    Larsen, R.H.3
  • 242
    • 84872186397 scopus 로고
    • No-carrier-added radiohalogenation methods with heavy halogens
    • Coenen, H.H.; Moerlein, S.M.; Stöcklin, G. No-carrier-added radiohalogenation methods with heavy halogens. Radiochimica Acta, 1983, 34, 47-68.
    • (1983) Radiochimica Acta , vol.34 , pp. 47-68
    • Coenen, H.H.1    Moerlein, S.M.2    Stöcklin, G.3
  • 243
    • 0002008091 scopus 로고
    • Astatine: Its organonuclear chemistry and biomedical applications
    • Brown, I. Astatine: Its organonuclear chemistry and biomedical applications. Adv. Org. Chem., 1987, 31, 43-88.
    • (1987) Adv. Org. Chem. , vol.31 , pp. 43-88
    • Brown, I.1
  • 244
    • 0001826224 scopus 로고
    • Recent advances in the organic chemistry of astatine
    • In, Patai, S.; Rappoport, Z., Eds. John Wiley & Sons Ltd: New York
    • Berei, K.; Vasáros, L., Recent advances in the organic chemistry of astatine. In Supplement 2: The chemistry of halides, pseudo-halides and azides., Patai, S.; Rappoport, Z., Eds. John Wiley & Sons Ltd: New York, 1995, pp 787-819.
    • (1995) Supplement 2: The chemistry of halides, pseudo-halides and azides , pp. 787-819
    • Berei, K.1    Vasáros, L.2
  • 246
    • 0001236972 scopus 로고
    • Artificially radioactive element 85
    • Corson, D.R.; Mackenzie, K.R.; Segre, E. Artificially radioactive element 85. Phys. Rev., 1940, 58, 672-678.
    • (1940) Phys. Rev. , vol.58 , pp. 672-678
    • Corson, D.R.1    Mackenzie, K.R.2    Segre, E.3
  • 248
    • 0001628817 scopus 로고
    • A comparison of the metabolism of iodine and of element 85 (eka-iodine)
    • Hamilton, J.G.; Soley, M.H. A comparison of the metabolism of iodine and of element 85 (eka-iodine). Proc. Natl. Acad. Sci, USA, 1940, 26, 483-489.
    • (1940) Proc. Natl. Acad. Sci, USA , vol.26 , pp. 483-489
    • Hamilton, J.G.1    Soley, M.H.2
  • 250
  • 251
    • 0031913296 scopus 로고    scopus 로고
    • Preparation and preliminary evaluation of astatine-211 labeled IgG via DTPA anhydride
    • Ning, L.; Jiannan, J.; Shangwu, M.; Hengliu, C.; Yanping, Y. Preparation and preliminary evaluation of astatine-211 labeled IgG via DTPA anhydride. J. Radioanal. Nucl. Chem., 1998, 227, 187-190.
    • (1998) J. Radioanal. Nucl. Chem. , vol.227 , pp. 187-190
    • Ning, L.1    Jiannan, J.2    Shangwu, M.3    Hengliu, C.4    Yanping, Y.5
  • 254
    • 43149087101 scopus 로고    scopus 로고
    • 211At complexes as potential precursors for astatine radiopharmaceuticals. Part I: Synthesis
    • 211At complexes as potential precursors for astatine radiopharmaceuticals. Part I: Synthesis. Bioconj. Chem., 2008, 19, 958-65.
    • (2008) Bioconj. Chem. , vol.19 , pp. 958-965
    • Pruszynski, M.1    Bilewicz, A.2    Zalutsky, M.R.3
  • 256
    • 0018232828 scopus 로고
    • The preparation of astatine labelled proteins using an electrophilic reaction
    • Vaughan, A.T.M.; Fremlin, J.H. The preparation of astatine labelled proteins using an electrophilic reaction. Int. J. Nucl. Med. Biol., 1978, 5, 229-230.
    • (1978) Int. J. Nucl. Med. Biol. , vol.5 , pp. 229-230
    • Vaughan, A.T.M.1    Fremlin, J.H.2
  • 257
    • 0023854518 scopus 로고
    • Astatination of proteins using an Nsuccinimidyl tri-n-butylstannyl benzoate intermediate
    • Zalutsky, M.R.; Narula, A.S. Astatination of proteins using an Nsuccinimidyl tri-n-butylstannyl benzoate intermediate. Appl. Radiat. Isot., 1988, 39, 227-232.
    • (1988) Appl. Radiat. Isot. , vol.39 , pp. 227-232
    • Zalutsky, M.R.1    Narula, A.S.2
  • 260
    • 33645737114 scopus 로고    scopus 로고
    • Astatinated trastuzumab, a putative agent for radionuclide immunotherapy of ErbB2-expressing tumours
    • Persson, M.I.; Gedda, L.; Jensen, H.J.; Lundqvist, H.; Malmstrom, P.U.; Tolmachev, V. Astatinated trastuzumab, a putative agent for radionuclide immunotherapy of ErbB2-expressing tumours. Oncol. Rep., 2006, 15, 673-80.
    • (2006) Oncol. Rep. , vol.15 , pp. 673-680
    • Persson, M.I.1    Gedda, L.2    Jensen, H.J.3    Lundqvist, H.4    Malmstrom, P.U.5    Tolmachev, V.6
  • 261
    • 34547379205 scopus 로고    scopus 로고
    • Reagents for astatination of biomolecules. 2. Conjugation of anionic boron cage pendant groups to a protein provides a method for direct labeling that is stable to in vivo deastatination
    • Wilbur, D.S.; Chyan, M.K.; Hamlin, D.K.; Vessella, R.L.; Wedge, T.J.; Hawthorne, M.F. Reagents for astatination of biomolecules. 2. Conjugation of anionic boron cage pendant groups to a protein provides a method for direct labeling that is stable to in vivo deastatination. Bioconj. Chem., 2007, 18, 1226-40.
    • (2007) Bioconj. Chem. , vol.18 , pp. 1226-1240
    • Wilbur, D.S.1    Chyan, M.K.2    Hamlin, D.K.3    Vessella, R.L.4    Wedge, T.J.5    Hawthorne, M.F.6
  • 265
    • 0031105498 scopus 로고    scopus 로고
    • Synthesis and preliminary biological evaluation of (3-iodobenzoyl)norbiotinamide and (5-iodo-3-pyridinyl)carbonyl)norbiotinamide: Two radio-iodinated biotin conjugates with improved stability
    • Foulon, C.F.; Alston, K.L.; Zalutsky, M.R. Synthesis and preliminary biological evaluation of (3-iodobenzoyl)norbiotinamide and (5-iodo-3-pyridinyl)carbonyl)norbiotinamide: Two radio-iodinated biotin conjugates with improved stability. Bioconj. Chem., 1997, 8, 179-186.
    • (1997) Bioconj. Chem. , vol.8 , pp. 179-186
    • Foulon, C.F.1    Alston, K.L.2    Zalutsky, M.R.3
  • 267
    • 0004150764 scopus 로고
    • Academic Press: New York
    • Grimes, R.N., Carboranes. Academic Press: New York, 1970.
    • (1970) Carboranes
    • Grimes, R.N.1
  • 268
    • 0000338437 scopus 로고
    • 12 and their derivatives
    • 12 and their derivatives. Chem. Rev., 1992, 92, 209-223.
    • (1992) Chem. Rev. , vol.92 , pp. 209-223
    • Bregadze, V.I.1
  • 270
    • 0000527594 scopus 로고
    • Halodicarba-undecaborate(II) ions
    • Olsen, F.P.; Hawthorne, M.F. Halodicarba-undecaborate(II) ions. Inorg. Chem., 1965, 4, 1839-1840.
    • (1965) Inorg. Chem. , vol.4 , pp. 1839-1840
    • Olsen, F.P.1    Hawthorne, M.F.2
  • 273
    • 33745945620 scopus 로고
    • The role of chemistry in the development of boron neutron capture therapy of cancer
    • Hawthorne, M.F. The role of chemistry in the development of boron neutron capture therapy of cancer. Angew. Chem. Int. Ed., 1993, 32, 950-984.
    • (1993) Angew. Chem. Int. Ed. , vol.32 , pp. 950-984
    • Hawthorne, M.F.1
  • 275
    • 0001329148 scopus 로고    scopus 로고
    • Synthesis of highly iodinated icosahedral mono-and dicarbon carboranes
    • Srivastava, R.R.; Hamlin, D.K.; Wilbur, D.S. Synthesis of highly iodinated icosahedral mono-and dicarbon carboranes. J. Org. Chem., 1996, 61, 9041-9044.
    • (1996) J. Org. Chem. , vol.61 , pp. 9041-9044
    • Srivastava, R.R.1    Hamlin, D.K.2    Wilbur, D.S.3
  • 277
    • 1842861595 scopus 로고    scopus 로고
    • Synthesis, radioiodination, and biodistribution of some nido-and closo-monocarbon carborane derivatives
    • Wilbur, D.S.; Hamlin, D.K.; Srivastava, R.R.; Chyan, M.K. Synthesis, radioiodination, and biodistribution of some nido-and closo-monocarbon carborane derivatives. Nucl. Med. Biol., 2004, 31, 523-30.
    • (2004) Nucl. Med. Biol. , vol.31 , pp. 523-530
    • Wilbur, D.S.1    Hamlin, D.K.2    Srivastava, R.R.3    Chyan, M.K.4
  • 278
  • 280
    • 63749103279 scopus 로고    scopus 로고
    • Reagents for astatination of biomolecules. 3. Comparison of closodecaborate(2-) and closo-dodecaborate(2-) moieties as reactive groups for labeling with astatine-211
    • Wilbur, D.S.; Chyan, M.K.; Hamlin, D.K.; Perry, M.A. Reagents for astatination of biomolecules. 3. Comparison of closodecaborate(2-) and closo-dodecaborate(2-) moieties as reactive groups for labeling with astatine-211. Bioconj. Chem., 2009, 20, 591-602.
    • (2009) Bioconj. Chem. , vol.20 , pp. 591-602
    • Wilbur, D.S.1    Chyan, M.K.2    Hamlin, D.K.3    Perry, M.A.4
  • 281
    • 76949084254 scopus 로고    scopus 로고
    • Preparation and in vivo evaluation of radioiodinated closo-decaborate(2-) derivatives to identify structural components that provide low retention in tissues
    • Wilbur, D.S.; Chyan, M.K.; Hamlin, D.K.; Perry, M.A. Preparation and in vivo evaluation of radioiodinated closo-decaborate(2-) derivatives to identify structural components that provide low retention in tissues. Nucl. Med. Biol., 2010, 37, 167-78.
    • (2010) Nucl. Med. Biol. , vol.37 , pp. 167-178
    • Wilbur, D.S.1    Chyan, M.K.2    Hamlin, D.K.3    Perry, M.A.4
  • 283
    • 0026130211 scopus 로고
    • Conjugation of phenyl isothiocyanate derivatives of carborane to antitumor antibody and in vivo lacalization of conjugates in nude mice
    • Varadarajan, A.; Sharkey, R.M.; Goldenberg, D.M.; Hawthorne, M.F. Conjugation of phenyl isothiocyanate derivatives of carborane to antitumor antibody and in vivo lacalization of conjugates in nude mice. Bioconj. Chem., 1991, 2, 102-110.
    • (1991) Bioconj. Chem. , vol.2 , pp. 102-110
    • Varadarajan, A.1    Sharkey, R.M.2    Goldenberg, D.M.3    Hawthorne, M.F.4
  • 284
    • 0026861943 scopus 로고
    • Carboranyl peptide-antibody conjugates for neutron-capture therapy: Preparation, characterization, and in vivo evaluation
    • Paxton, R.J.; Beatty, B.G.; Varadarajan, A.; Hawthorne, M.F. Carboranyl peptide-antibody conjugates for neutron-capture therapy: Preparation, characterization, and in vivo evaluation. Biocon. Chem., 1992, 3, 241-247.
    • (1992) Biocon. Chem. , vol.3 , pp. 241-247
    • Paxton, R.J.1    Beatty, B.G.2    Varadarajan, A.3    Hawthorne, M.F.4
  • 287
    • 0030250865 scopus 로고    scopus 로고
    • Development and in vitro studies of epidermal growth factor-dextran conjugates for boron neutron capture therapy
    • Gedda, L.; Olsson, P.; Pontén, J.; Carlsson, J. Development and in vitro studies of epidermal growth factor-dextran conjugates for boron neutron capture therapy. Bioconj. Chem., 1996, 7, 584-591.
    • (1996) Bioconj. Chem. , vol.7 , pp. 584-591
    • Gedda, L.1    Olsson, P.2    Pontén, J.3    Carlsson, J.4
  • 290
    • 0038793484 scopus 로고    scopus 로고
    • Biodistribution of the chimeric monoclonal antibody U36 radioiodinated with a closododecaborate-containing linker. Comparison with other radioiodination methods
    • Nestor, M.; Persson, M.; Cheng, J.; Tolmachev, V.; Van Dongen, G.; Anniko, M.; Kairemo, K. Biodistribution of the chimeric monoclonal antibody U36 radioiodinated with a closododecaborate-containing linker. Comparison with other radioiodination methods. Bioconj. Chem., 2003, 14, 805-810.
    • (2003) Bioconj. Chem. , vol.14 , pp. 805-810
    • Nestor, M.1    Persson, M.2    Cheng, J.3    Tolmachev, V.4    van Dongen, G.5    Anniko, M.6    Kairemo, K.7
  • 291
    • 35848963867 scopus 로고    scopus 로고
    • In vitro evaluation of two polyhedral boron anion derivatives as linkers for attachment of radioiodine to the anti-HER2 monoclonal antibody trastuzumab
    • Persson, M.; Sivaev, I.; Winberg, K.J.; Gedda, L.; Malmstrom, P.U.; Tolmachev, V. In vitro evaluation of two polyhedral boron anion derivatives as linkers for attachment of radioiodine to the anti-HER2 monoclonal antibody trastuzumab. Cancer Biother. Radiopharm., 2007, 22, 585-96.
    • (2007) Cancer Biother. Radiopharm. , vol.22 , pp. 585-596
    • Persson, M.1    Sivaev, I.2    Winberg, K.J.3    Gedda, L.4    Malmstrom, P.U.5    Tolmachev, V.6
  • 293
    • 34247487372 scopus 로고    scopus 로고
    • 212Pb@C(60) and its water-soluble derivatives: Synthesis, stability, and suitability for radioimmunotherapy
    • 212Pb@C(60) and its water-soluble derivatives: Synthesis, stability, and suitability for radioimmunotherapy. J. Am. Chem. Soc., 2007, 129, 5131-8.
    • (2007) J. Am. Chem. Soc. , vol.129 , pp. 5131-5138
    • Diener, M.D.1    Alford, J.M.2    Kennel, S.J.3    Mirzadeh, S.4
  • 295
    • 34548811410 scopus 로고    scopus 로고
    • 211AtCl@us-tube nanocapsules: A new concept in radiotherapeuticagent design
    • 211AtCl@us-tube nanocapsules: A new concept in radiotherapeuticagent design. Small, 2007, 3, 1496-1499.
    • (2007) Small , vol.3 , pp. 1496-1499
    • Hartman, K.B.1    Hamlin, D.K.2    Wilbur, D.S.3    Wilson, L.J.4
  • 296
    • 46249128521 scopus 로고    scopus 로고
    • Synthesis and evalation of a watersoluble polymer to reduce Ac-225 daughter migration
    • Fitzsimmons, J.; Atcher, R. Synthesis and evalation of a watersoluble polymer to reduce Ac-225 daughter migration. J. Label. Compds. Radiopharm., 2007, 50, 147-153.
    • (2007) J. Label. Compds. Radiopharm. , vol.50 , pp. 147-153
    • Fitzsimmons, J.1    Atcher, R.2
  • 298
    • 0026060897 scopus 로고
    • Influence of surface hydrophilicity of liposomes on their interaction with plasma protein and clearance from the circulation: Studies with poly(ethyleneglycol)-coated vesicles
    • Senior, J.; Delgado, C.; Fisher, D.; Tilcock, C.; Gregoriadis, G. Influence of surface hydrophilicity of liposomes on their interaction with plasma protein and clearance from the circulation: Studies with poly(ethyleneglycol)-coated vesicles. Biochim. Biophy. s Acta, 1991, 1062, 77-82.
    • (1991) Biochim. Biophy. s Acta , vol.1062 , pp. 77-82
    • Senior, J.1    Delgado, C.2    Fisher, D.3    Tilcock, C.4    Gregoriadis, G.5
  • 300
    • 1842850605 scopus 로고    scopus 로고
    • Sterically stabilized liposomes as a carrier for alphaemitting radium and actinium radionuclides
    • Henriksen, G.; Schoultz, B.W.; Michaelsen, T.E.; Bruland, O.S.; Larsen, R.H. Sterically stabilized liposomes as a carrier for alphaemitting radium and actinium radionuclides. Nucl. Med. Biol., 2004, 31, 441-9.
    • (2004) Nucl. Med. Biol. , vol.31 , pp. 441-449
    • Henriksen, G.1    Schoultz, B.W.2    Michaelsen, T.E.3    Bruland, O.S.4    Larsen, R.H.5
  • 302
    • 36849037503 scopus 로고    scopus 로고
    • Enhanced retention of the alpha-particleemitting daughters of actinium-225 by liposome carriers
    • Sofou, S.; Kappel, B.J.; Jaggi, J.S.; McDevitt, M.R.; Scheinberg, D.A.; Sgouros, G. Enhanced retention of the alpha-particleemitting daughters of actinium-225 by liposome carriers. Bioconj. Chem., 2007, 18, 2061-7.
    • (2007) Bioconj. Chem. , vol.18 , pp. 2061-2067
    • Sofou, S.1    Kappel, B.J.2    Jaggi, J.S.3    McDevitt, M.R.4    Scheinberg, D.A.5    Sgouros, G.6
  • 303
    • 45749101319 scopus 로고    scopus 로고
    • 225Ac in rigid liposomes for potential targeted therapy of micrometastases
    • 225Ac in rigid liposomes for potential targeted therapy of micrometastases. Bioconj. Chem., 2008, 19, 1274-82.
    • (2008) Bioconj. Chem. , vol.19 , pp. 1274-1282
    • Chang, M.Y.1    Seideman, J.2    Sofou, S.3
  • 304
    • 0003131542 scopus 로고    scopus 로고
    • Repair of radiation damage and the dose rate effect
    • In, Lippencott Williams & Wilkins: Philadelphia
    • Hall, E.J.; Giaccia, A.J., Repair of radiation damage and the dose rate effect. In Radiobiology for the radiologist., Lippencott Williams & Wilkins: Philadelphia, 2006, pp 60-84.
    • (2006) Radiobiology for the radiologist , pp. 60-84
    • Hall, E.J.1    Giaccia, A.J.2
  • 305
    • 33749266047 scopus 로고    scopus 로고
    • Requirements regarding dose rate and exposure time for killing of tumour cells in beta particle radionuclide therapy
    • Carlsson, J.; Eriksson, V.; Stenerlow, B.; Lundqvist, H. Requirements regarding dose rate and exposure time for killing of tumour cells in beta particle radionuclide therapy. Eur. J Nucl. Med. Mol. Imaging, 2006, 33 (10), 1185-1195.
    • (2006) Eur. J Nucl. Med. Mol. Imaging , vol.33 , Issue.10 , pp. 1185-1195
    • Carlsson, J.1    Eriksson, V.2    Stenerlow, B.3    Lundqvist, H.4
  • 306
    • 34248649003 scopus 로고    scopus 로고
    • Oxygen effect and reoxygenation
    • In, Sixth Edition ed.; Lippincott Williams & Wilkins: Philadelpha
    • Hall, E.J.; Giaccia, A.J., Oxygen effect and reoxygenation. In Radiobiology for the radiologist., Sixth Edition ed.; Lippincott Williams & Wilkins: Philadelpha, 2006, pp 85-105.
    • (2006) Radiobiology for the radiologist , pp. 85-105
    • Hall, E.J.1    Giaccia, A.J.2
  • 307
    • 33747666734 scopus 로고    scopus 로고
    • Radioimmunotherapy as non-myeloablative conditioning for allogeneic marrow transplantation
    • Bethge, W.A.; Wilbur, D.S.; Sandmaier, B.M. Radioimmunotherapy as non-myeloablative conditioning for allogeneic marrow transplantation. Leuk. Lymphoma, 2006, 47, 1205-14.
    • (2006) Leuk. Lymphoma , vol.47 , pp. 1205-1214
    • Bethge, W.A.1    Wilbur, D.S.2    Sandmaier, B.M.3
  • 308
    • 0028197111 scopus 로고
    • Approaches to improved antibody-and peptide-mediated targeting for imaging and therapy of cancer
    • Fritzberg, A.R.; Beaumier, P.L.; Bottino, B.J.; Reno, J.M. Approaches to improved antibody-and peptide-mediated targeting for imaging and therapy of cancer. J. Controlled Release, 1994, 28, 167-173.
    • (1994) J. Controlled Release , vol.28 , pp. 167-173
    • Fritzberg, A.R.1    Beaumier, P.L.2    Bottino, B.J.3    Reno, J.M.4
  • 310
    • 0000302143 scopus 로고
    • Reaction mechanisms in the radiolysis of peptides, polypeptides, and proteins
    • Garrison, W.M. Reaction mechanisms in the radiolysis of peptides, polypeptides, and proteins. Chem. Rev., 1985, 87, 381-398.
    • (1985) Chem. Rev. , vol.87 , pp. 381-398
    • Garrison, W.M.1
  • 312
    • 0031901579 scopus 로고    scopus 로고
    • Effects of radiolysis on yttrium-90-labeled Lym-1 antibody preparations
    • Salako, Q.A.; O'Donnell, R.T.; DeNardo, S.J. Effects of radiolysis on yttrium-90-labeled Lym-1 antibody preparations. J. Nucl. Med., 1998, 39, 667-70.
    • (1998) J. Nucl. Med. , vol.39 , pp. 667-670
    • Salako, Q.A.1    O'Donnell, R.T.2    DeNardo, S.J.3
  • 314
    • 0024286990 scopus 로고
    • Albumin-an important extracellular antioxidant?
    • Halliwell, B. Albumin-an important extracellular antioxidant? Biochem. Pharm., 1988, 37, 569-571.
    • (1988) Biochem. Pharm. , vol.37 , pp. 569-571
    • Halliwell, B.1
  • 315
    • 0034923735 scopus 로고    scopus 로고
    • 90Y-labeled DOTAbiomolecule conjugates using gentisic acid and ascorbic acid
    • 90Y-labeled DOTAbiomolecule conjugates using gentisic acid and ascorbic acid. Bioconj. Chem., 2001, 12, 554-558.
    • (2001) Bioconj. Chem. , vol.12 , pp. 554-558
    • Liu, S.1    Edwards, D.S.2
  • 316
    • 0141792922 scopus 로고    scopus 로고
    • Ascorbic acid used as a buffer agent and radiolytic stabilizer for metalloradiopharmaceuticals
    • Liu, S.; Ellars, C.E.; Edwards, D.S. Ascorbic acid used as a buffer agent and radiolytic stabilizer for metalloradiopharmaceuticals. Bioconj. Chem., 2003, 14, 1052-1056.
    • (2003) Bioconj. Chem. , vol.14 , pp. 1052-1056
    • Liu, S.1    Ellars, C.E.2    Edwards, D.S.3
  • 317
    • 0025124512 scopus 로고
    • Inhibition of autoradiolysis of radiolabeled monoclonal antibodies by cryopreservation
    • Wahl, R.L.; Wissing, J.; del Rosario, R.; Zasadny, K.R. Inhibition of autoradiolysis of radiolabeled monoclonal antibodies by cryopreservation. J. Nucl. Med., 1990, 31, 84-89.
    • (1990) J. Nucl. Med. , vol.31 , pp. 84-89
    • Wahl, R.L.1    Wissing, J.2    del Rosario, R.3    Zasadny, K.R.4
  • 322
    • 25444498863 scopus 로고    scopus 로고
    • 211At-astatobenzoate synthesis
    • 211At-astatobenzoate synthesis. J. Nucl. Med., 2005, 46 (8), 1393-400.
    • (2005) J. Nucl. Med. , vol.46 , Issue.8 , pp. 1393-1400
    • Pozzi, O.R.1    Zalutsky, M.R.2
  • 326
    • 0000169039 scopus 로고
    • Time-resolved fluorescence of a new europium chelate complex: Demonstration of highly sensitive detection of protein and DNA samples
    • Saha, A.K.; Kross, K.; Kloszewski, E.D.; Upson, D.A.; Toner, J.L.; Snow, R.A.; Black, C.D.V.; Desai, V.C. Time-resolved fluorescence of a new europium chelate complex: Demonstration of highly sensitive detection of protein and DNA samples. J. Am. Chem. Soc., 1993, 115, 11032-11033.
    • (1993) J. Am. Chem. Soc. , vol.115 , pp. 11032-11033
    • Saha, A.K.1    Kross, K.2    Kloszewski, E.D.3    Upson, D.A.4    Toner, J.L.5    Snow, R.A.6    Black, C.D.V.7    Desai, V.C.8
  • 327
    • 79959565618 scopus 로고
    • Complexing agents and targeting radioactive immunoreagents useful in therapeutic and diagnostic imaging compositions and methods
    • November 22
    • Toner, J.L.; Hilborn, D.A.; Murray, B.J.; Hossain, T.Z. Complexing agents and targeting radioactive immunoreagents useful in therapeutic and diagnostic imaging compositions and methods. U.S. Patent 5,367,080, November 22, 1994.
    • (1994) U.S. Patent 5,367,080
    • Toner, J.L.1    Hilborn, D.A.2    Murray, B.J.3    Hossain, T.Z.4
  • 329
    • 11444270384 scopus 로고    scopus 로고
    • Time gating improves sensitivity in energy transfer assays with terbium chelate/dark quencher oligonucleotide probes
    • Johansson, M.K.; Cook, R.M.; Xu, J.; Raymond, K.N. Time gating improves sensitivity in energy transfer assays with terbium chelate/dark quencher oligonucleotide probes. J. Am. Chem. Soc., 2004, 126, 16451-16455.
    • (2004) J. Am. Chem. Soc. , vol.126 , pp. 16451-16455
    • Johansson, M.K.1    Cook, R.M.2    Xu, J.3    Raymond, K.N.4


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