Vehicles, chelators, and radionuclides: Choosing the "building blocks" of an effective therapeutic radioimmunoconjugate

Bioconjugate Chemistry

Volumn 7, Issue 2, 1996, Pages

  August Schubiger, P ^a   Alberto, Roger ^a   Smith, Alan ^a  

^a PAUL SCHERRER INSTITUTE   (Switzerland)

Author keywords

[No Author keywords available]

Indexed keywords

BUILDING BLOCKES; RADIOIMMUNOCONJUGATES;

EID: 0030111464     PISSN: 10431802     EISSN: None     Source Type: Journal    
DOI: None     Document Type: Review

References (12)

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6. 2: Chemistry and animal biodistribution. Tenth International Symposium on Radiopharmacy Chemistry Abstracts, p 313.
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8. Annunziato, M. E., Patel, U. S., Ranade, M., and Palumbo, P. S. (1993) p-Maleimidophenyl Isocyanate: A novel Heterobi-functional Linker for Hydroxyl to Thiol Coupling. Bioconjugate Chem. 4, 212-218.
9. 16Re Radioimmunotherapy of small cell lung carcinoma xenografts in Nude mice. Cancer Res. 51, 676-681.
10. Bischof-Delaloye, A., Buchegger, F., Delaloye, B., Smith, A., Poncioni, M., Mach, J.-P., and Schubiger, P. A. (1996) Clinical evaluation of a Cu-67 labeled anti-CEA MAb (manuscript in preparation).
11. Wheldon, T. E. (1993) Radionuclide therapy of cancer particle range and therapeutic effectiveness Nucl. Med. Commun. 14, 408-410.
12. Wong, S. S. (1993) Chemistry of protein conjugation and cross-linking. ISBN 0-6493-5866-8. CRC Press Inc., Boca Raton, Florida.