Acyclic chelate with ideal properties for 68Ga PET imaging agent elaboration

Journal of the American Chemical Society

Volumn 132, Issue 44, 2010, Pages 15726-15733

  Boros, Eszter ^a,c   Ferreira, Cara L ^b   Cawthray, Jacqueline F ^a,c   Price, Eric W ^a   Patrick, Brian O ^a   Wester, Dennis W ^b   Adam, Michael J ^c   Orvig, Chris ^a  

^a UNIVERSITY OF BRITISH COLUMBIA   (Canada)

^b MDS Inc   (Canada)

^c TRIUMF   (Canada)

Author keywords

[No Author keywords available]

Indexed keywords

BIFUNCTIONAL; BIODISTRIBUTIONS; CONCENTRATION-DEPENDENT; LIGAND CONCENTRATION; MACROCYCLES; NO DECOMPOSITION; PET IMAGING; SPECIFIC ACTIVITY;

CHELATION; NUCLEAR MEDICINE;

GALLIUM;

1,4,7,10 TETRAAZACYCLODODECANE 1,4,7,10 TETRAACETIC ACID; APOTRANSFERRIN; CHELATING AGENT; GALLIUM 67; GALLIUM 68; NOTA; RADIOPHARMACEUTICAL AGENT; UNCLASSIFIED DRUG;

ANIMAL EXPERIMENT; ANIMAL TISSUE; ARTICLE; CONCENTRATION RESPONSE; DECOMPOSITION; DRUG DISTRIBUTION; DRUG SYNTHESIS; FEMALE; ISOTOPE LABELING; MOUSE; NONHUMAN; POSITRON EMISSION TOMOGRAPHY; PURIFICATION; QUANTITATIVE ANALYSIS; RADIATION DOSE DISTRIBUTION;

ANIMALS; CHELATING AGENTS; GALLIUM RADIOISOTOPES; HETEROCYCLIC COMPOUNDS; HUMANS; MOLECULAR STRUCTURE; POSITRON-EMISSION TOMOGRAPHY;

EID: 78149264198     PISSN: 00027863     EISSN: 15205126     Source Type: Journal    
DOI: 10.1021/ja106399h     Document Type: Article

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