Synthesis and biological evaluation of a novel decadentate ligand DEPA

Bioorganic and Medicinal Chemistry Letters

Volumn 18, Issue 21, 2008, Pages 5792-5795

  Chong, Hyun Soon ^a   Lim, Sooyoun ^a   Baidoo, Kwamena E ^b   Milenic, Diane E ^b   Ma, Xiang ^a   Jia, Fang ^c   Song, Hyun A ^a   Brechbiel, Martin W ^b   Lewis, Michael R ^c  

^a Illinois Institute of Technology   (United States)

^b NATIONAL CANCER INSTITUTE   (United States)

^c Nuclear Science and Engineering Institute   (United States)

Author keywords

177Lu; 212Bi; 213Bi; Bimodal ligand; DEPA; Radioimmunotherapy

Indexed keywords

1,4,7 TRIS(TERT BUTOXYCARBONYLMETHYL)TETRAAZACYCLODODECANE; 7 [2 (BISCARBOXYMETHYLAMINO)ETHYL] 4,10 BISCARBOXYMETHYL 1,4,7,10 TETRAAZACYCLODODEC 1 YL ACETIC ACID; ARSENAZO 3; BISMUTH 212; BISMUTH 213; HETEROCYCLIC COMPOUND; LUTETIUM 177; MACROCYCLIC COMPOUND; UNCLASSIFIED DRUG;

ANIMAL EXPERIMENT; ARTICLE; CANCER THERAPY; COMPLEX FORMATION; DRUG DISTRIBUTION; DRUG SCREENING; DRUG STABILITY; DRUG SYNTHESIS; MOUSE; NONHUMAN; RADIOIMMUNOTHERAPY;

CHELATING AGENTS; GLYCINE; HETEROCYCLIC COMPOUNDS, 1-RING; LIGANDS; REPRODUCIBILITY OF RESULTS;

EID: 54049084113     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmcl.2008.09.063     Document Type: Article

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