-
1
-
-
50449091972
-
Alpha-particle radioimmunotherapy with astatine-211 and bismuth-213
-
Lucignani G. Alpha-particle radioimmunotherapy with astatine-211 and bismuth-213. Eur J Nucl Med Mol Imaging 35 (2008) 1729-1733
-
(2008)
Eur J Nucl Med Mol Imaging
, vol.35
, pp. 1729-1733
-
-
Lucignani, G.1
-
3
-
-
14844340282
-
The promise of targeted alpha-particle therapy
-
Mulford D.A., Scheinberg D.A., and Jurcic J.G. The promise of targeted alpha-particle therapy. J Nucl Med 46 Suppl 1 (2005) 199S-204S
-
(2005)
J Nucl Med
, vol.46
, Issue.SUPPL. 1
-
-
Mulford, D.A.1
Scheinberg, D.A.2
Jurcic, J.G.3
-
4
-
-
24044539916
-
Cancer radioimmunotherapy with alpha-emitting nuclides
-
Couturier O., Supiot S., Degraef-Mougin M., Faivre-Chauvet A., Carlier T., Chatal J.F., et al. Cancer radioimmunotherapy with alpha-emitting nuclides. Eur J Nucl Med Mol Imaging 32 (2005) 601-614
-
(2005)
Eur J Nucl Med Mol Imaging
, vol.32
, pp. 601-614
-
-
Couturier, O.1
Supiot, S.2
Degraef-Mougin, M.3
Faivre-Chauvet, A.4
Carlier, T.5
Chatal, J.F.6
-
5
-
-
0035451674
-
Advancements in cancer therapy with alpha-emitters: a review
-
Imam S.K. Advancements in cancer therapy with alpha-emitters: a review. Int J Rad Oncol Biol Phys 51 (2001) 271-278
-
(2001)
Int J Rad Oncol Biol Phys
, vol.51
, pp. 271-278
-
-
Imam, S.K.1
-
6
-
-
35549000927
-
Targeted alpha-therapy: past, present, future?
-
Brechbiel M.W. Targeted alpha-therapy: past, present, future?. Dalton Trans (2007) 4918-4928
-
(2007)
Dalton Trans
, pp. 4918-4928
-
-
Brechbiel, M.W.1
-
7
-
-
0026951113
-
Radiohalogenation of proteins: an overview of radionuclides, labeling methods, and reagents for conjugate labeling
-
Wilbur D.S. Radiohalogenation of proteins: an overview of radionuclides, labeling methods, and reagents for conjugate labeling. Bioconjug Chem 3 (1992) 433-470
-
(1992)
Bioconjug Chem
, vol.3
, pp. 433-470
-
-
Wilbur, D.S.1
-
8
-
-
0000508399
-
The synthesis of radiolabeled compounds via organometallic intermediates
-
Kabalka G.W., and Varma R.S. The synthesis of radiolabeled compounds via organometallic intermediates. Tetrahedron 45 (1989) 6601-6621
-
(1989)
Tetrahedron
, vol.45
, pp. 6601-6621
-
-
Kabalka, G.W.1
Varma, R.S.2
-
9
-
-
0007396871
-
Regiospecific incorporation of no-carrier-added radiobromine and radioiodine into aromatic rings via halogenodegermylation
-
Moerlein S.M. Regiospecific incorporation of no-carrier-added radiobromine and radioiodine into aromatic rings via halogenodegermylation. J Chem Soc Perkin Trans I (1985) 1687-1692
-
(1985)
J Chem Soc Perkin Trans I
, pp. 1687-1692
-
-
Moerlein, S.M.1
-
10
-
-
63749118446
-
211At]astatide and development of labeling reagents to increase stability
-
211At]astatide and development of labeling reagents to increase stability. Curr Radiopharm 1 (2008) 144-176
-
(2008)
Curr Radiopharm
, vol.1
, pp. 144-176
-
-
Wilbur, D.S.1
-
11
-
-
34547379205
-
Reagents for astatination of biomolecules: 2. Conjugation of anionic boron cage pendant groups to a protein provides a method for direct labeling that is stable to in vivo deastatination
-
Wilbur D.S., Chyan M.K., Hamlin D.K., Vessella R.L., Wedge T.J., and Hawthorne M.F. Reagents for astatination of biomolecules: 2. Conjugation of anionic boron cage pendant groups to a protein provides a method for direct labeling that is stable to in vivo deastatination. Bioconjug Chem 18 (2007) 1226-1240
-
(2007)
Bioconjug Chem
, vol.18
, pp. 1226-1240
-
-
Wilbur, D.S.1
Chyan, M.K.2
Hamlin, D.K.3
Vessella, R.L.4
Wedge, T.J.5
Hawthorne, M.F.6
-
12
-
-
10744222244
-
Reagents for astatination of biomolecules: comparison of the in vivo distribution and stability of some radioiodinated/astatinated benzamidyl and nido-carboranyl compounds
-
Wilbur D.S., Chyan M.K., Hamlin D.K., Kegley B.B., Risler R., Pathare P.M., et al. Reagents for astatination of biomolecules: comparison of the in vivo distribution and stability of some radioiodinated/astatinated benzamidyl and nido-carboranyl compounds. Bioconjug Chem 15 (2004) 203-223
-
(2004)
Bioconjug Chem
, vol.15
, pp. 203-223
-
-
Wilbur, D.S.1
Chyan, M.K.2
Hamlin, D.K.3
Kegley, B.B.4
Risler, R.5
Pathare, P.M.6
-
13
-
-
2542447254
-
Biotin reagents in antibody pretargeting: 6. Synthesis and in vivo evaluation of astatinated and radioiodinated aryl- and nido-carboranyl-biotin derivatives
-
Wilbur D.S., Hamlin D.K., Chyan M.K., Kegley B.B., Quinn J., and Vessella R.L. Biotin reagents in antibody pretargeting: 6. Synthesis and in vivo evaluation of astatinated and radioiodinated aryl- and nido-carboranyl-biotin derivatives. Bioconjug Chem 15 (2004) 601-616
-
(2004)
Bioconjug Chem
, vol.15
, pp. 601-616
-
-
Wilbur, D.S.1
Hamlin, D.K.2
Chyan, M.K.3
Kegley, B.B.4
Quinn, J.5
Vessella, R.L.6
-
14
-
-
1842861595
-
Synthesis, radioiodination, and biodistribution of some nido- and closo-monocarbon carborane derivatives
-
Wilbur D.S., Hamlin D.K., Srivastava R.R., and Chyan M.K. Synthesis, radioiodination, and biodistribution of some nido- and closo-monocarbon carborane derivatives. Nucl Med Biol 31 (2004) 523-530
-
(2004)
Nucl Med Biol
, vol.31
, pp. 523-530
-
-
Wilbur, D.S.1
Hamlin, D.K.2
Srivastava, R.R.3
Chyan, M.K.4
-
15
-
-
9244224115
-
Comparative metabolism and retention of iodine-125, yttrium-90, indium-111 radioimmunoconjugates by cancer cells
-
Press O.W., Shan D., Howell-Clark J., Eary J., Appelbaum F.R., Matthews D., et al. Comparative metabolism and retention of iodine-125, yttrium-90, indium-111 radioimmunoconjugates by cancer cells. Cancer Res 56 (1996) 2123-2129
-
(1996)
Cancer Res
, vol.56
, pp. 2123-2129
-
-
Press, O.W.1
Shan, D.2
Howell-Clark, J.3
Eary, J.4
Appelbaum, F.R.5
Matthews, D.6
-
16
-
-
0027368237
-
Intracellular metabolism of indium-111-DTPA-labeled receptor targeted proteins
-
Duncan J.R., and Welch M.J. Intracellular metabolism of indium-111-DTPA-labeled receptor targeted proteins. J Nucl Med 34 (1993) 1728-1738
-
(1993)
J Nucl Med
, vol.34
, pp. 1728-1738
-
-
Duncan, J.R.1
Welch, M.J.2
-
17
-
-
0029058307
-
Effects of radiolabeling monoclonal antibodies with a residualizing iodine radiolabel on the accretion of radioisotope in tumors
-
Stein R., Goldenberg D.M., Thorpe S.R., Basu A., and Mattes M.J. Effects of radiolabeling monoclonal antibodies with a residualizing iodine radiolabel on the accretion of radioisotope in tumors. Cancer Res 55 (1995) 3132-3139
-
(1995)
Cancer Res
, vol.55
, pp. 3132-3139
-
-
Stein, R.1
Goldenberg, D.M.2
Thorpe, S.R.3
Basu, A.4
Mattes, M.J.5
-
18
-
-
0000229150
-
Applications of radiolabeled boron clusters to the diagnosis and treatment of cancer
-
Hawthorne M.F., and Maderna A. Applications of radiolabeled boron clusters to the diagnosis and treatment of cancer. Chem Rev 99 (1999) 3421-3434
-
(1999)
Chem Rev
, vol.99
, pp. 3421-3434
-
-
Hawthorne, M.F.1
Maderna, A.2
-
19
-
-
0000323139
-
The chemistry of neutron capture therapy
-
Soloway A.H., Tjarks W., Barnum B.A., Rong F.G., Barth R.F., Codogni I.M., et al. The chemistry of neutron capture therapy. Chem Rev 98 (1998) 1515-1562
-
(1998)
Chem Rev
, vol.98
, pp. 1515-1562
-
-
Soloway, A.H.1
Tjarks, W.2
Barnum, B.A.3
Rong, F.G.4
Barth, R.F.5
Codogni, I.M.6
-
20
-
-
46849106280
-
Renal uptake and metabolism of radiopharmaceuticals derived from peptides and proteins
-
Akizawa H., Uehara T., and Arano Y. Renal uptake and metabolism of radiopharmaceuticals derived from peptides and proteins. Adv Drug Deliv Rev 60 (2008) 1319-1328
-
(2008)
Adv Drug Deliv Rev
, vol.60
, pp. 1319-1328
-
-
Akizawa, H.1
Uehara, T.2
Arano, Y.3
-
21
-
-
0036749889
-
Altering pharmacokinetics of radiolabeled antibodies by the interposition of metabolizable linkages. Metabolizable linkers and pharmacokinetics of monoclonal antibodies
-
Akizawa H., and Arano Y. Altering pharmacokinetics of radiolabeled antibodies by the interposition of metabolizable linkages. Metabolizable linkers and pharmacokinetics of monoclonal antibodies. Q J Nucl Med 46 (2002) 206-223
-
(2002)
Q J Nucl Med
, vol.46
, pp. 206-223
-
-
Akizawa, H.1
Arano, Y.2
-
22
-
-
63749103279
-
Reagents for astatination of biomolecules: 3. Comparison of closo-decaborate(2-) and closo-dodecaborate(2-) moieties as reactive groups for labeling with astatine-211
-
Wilbur D.S., Chyan M.K., Hamlin D.K., and Perry M.A. Reagents for astatination of biomolecules: 3. Comparison of closo-decaborate(2-) and closo-dodecaborate(2-) moieties as reactive groups for labeling with astatine-211. Bioconjug Chem 20 (2009) 591-602
-
(2009)
Bioconjug Chem
, vol.20
, pp. 591-602
-
-
Wilbur, D.S.1
Chyan, M.K.2
Hamlin, D.K.3
Perry, M.A.4
-
23
-
-
12944252114
-
Chemistry of boranes: XXXI. 1,10-Bis(hydroxymethyl)octachlorodecaborate (2-)
-
Knoth W.H. Chemistry of boranes: XXXI. 1,10-Bis(hydroxymethyl)octachlorodecaborate (2-). J Am Chem Soc 89 (1967) 4850-4852
-
(1967)
J Am Chem Soc
, vol.89
, pp. 4850-4852
-
-
Knoth, W.H.1
-
24
-
-
0000832049
-
Physiology
-
Foster H.L., Small J.D., and Fox J.G. (Eds), Academic Press, New York
-
Kaplan H.M., Brewer N.R., and Blair W.H. Physiology. In: Foster H.L., Small J.D., and Fox J.G. (Eds). The Mouse in Biomedical Research (1983), Academic Press, New York 248-292
-
(1983)
The Mouse in Biomedical Research
, pp. 248-292
-
-
Kaplan, H.M.1
Brewer, N.R.2
Blair, W.H.3
-
27
-
-
65549097348
-
Biodistributions, myelosuppression and toxicities in mice treated with an anti-CD45 antibody labeled with the α-emitting radionuclides bismuth-213 or astatine-211
-
Nakamae H., Wilbur D.S., Hamlin D.K., Thakar M.S., Santos E.B., Fisher D.R., et al. Biodistributions, myelosuppression and toxicities in mice treated with an anti-CD45 antibody labeled with the α-emitting radionuclides bismuth-213 or astatine-211. Cancer Res 69 (2009) 2408-2415
-
(2009)
Cancer Res
, vol.69
, pp. 2408-2415
-
-
Nakamae, H.1
Wilbur, D.S.2
Hamlin, D.K.3
Thakar, M.S.4
Santos, E.B.5
Fisher, D.R.6
-
28
-
-
0024458164
-
Reduction of background activities by introduction of a diester linkage between antibody and a chelate in radioimmunodetection of tumor
-
Paik C.H., Yokoyama K., Reynolds J.C., Quadri S.M., Min C.Y., Shin S.Y., et al. Reduction of background activities by introduction of a diester linkage between antibody and a chelate in radioimmunodetection of tumor. J Nucl Med 30 (1989) 1693-1701
-
(1989)
J Nucl Med
, vol.30
, pp. 1693-1701
-
-
Paik, C.H.1
Yokoyama, K.2
Reynolds, J.C.3
Quadri, S.M.4
Min, C.Y.5
Shin, S.Y.6
-
30
-
-
0026130704
-
A novel bifunctional metabolizable linker for the conjugation of antibodies with radionuclides
-
Arano Y., Matsushima H., Tagawa M., Koizumi M., Endo K., Konishi J., et al. A novel bifunctional metabolizable linker for the conjugation of antibodies with radionuclides. Bioconjug Chem 2 (1991) 71-76
-
(1991)
Bioconjug Chem
, vol.2
, pp. 71-76
-
-
Arano, Y.1
Matsushima, H.2
Tagawa, M.3
Koizumi, M.4
Endo, K.5
Konishi, J.6
-
31
-
-
0028156807
-
Decreased kidney uptake of technetium-99m-labelled Fab′ fragments in ovarian carcinoma bearing nude mice using a cleavable chelator
-
Tibben J.G., Massuger L.F.A.G., Boerman O.C., Claessens R.A.M.J., Borm G.F., Pak K.Y., et al. Decreased kidney uptake of technetium-99m-labelled Fab′ fragments in ovarian carcinoma bearing nude mice using a cleavable chelator. Nucl Med Biol 21 (1994) 17-24
-
(1994)
Nucl Med Biol
, vol.21
, pp. 17-24
-
-
Tibben, J.G.1
Massuger, L.F.A.G.2
Boerman, O.C.3
Claessens, R.A.M.J.4
Borm, G.F.5
Pak, K.Y.6
-
32
-
-
84987453854
-
Chelate radiochemistry: cleavable linkers lead to altered levels of radioactivity in the liver
-
Meares C.F., McCall M.J., Deshpande S.V., DeNardo S.J., and Goodwin D.A. Chelate radiochemistry: cleavable linkers lead to altered levels of radioactivity in the liver. Int J Cancer 2 (1988) 99-102
-
(1988)
Int J Cancer
, vol.2
, pp. 99-102
-
-
Meares, C.F.1
McCall, M.J.2
Deshpande, S.V.3
DeNardo, S.J.4
Goodwin, D.A.5
-
33
-
-
0032170893
-
Cathepsin substrates as cleavable peptide linkers in bioconjugates, selected from a fluorescence quench combinatorial library
-
Peterson J.J., and Meares C.F. Cathepsin substrates as cleavable peptide linkers in bioconjugates, selected from a fluorescence quench combinatorial library. Bioconjug Chem 9 (1998) 618-626
-
(1998)
Bioconjug Chem
, vol.9
, pp. 618-626
-
-
Peterson, J.J.1
Meares, C.F.2
-
34
-
-
33846435172
-
Development of tissue plasminogen activator specific "on demand cleavable" (odc) linkers for radioimmunotherapy by screening one-bead-one-compound combinatorial peptide libraries
-
Kumaresan P.R., Natarajan A., Song A., Wang X., Liu R., DeNardo G., et al. Development of tissue plasminogen activator specific "on demand cleavable" (odc) linkers for radioimmunotherapy by screening one-bead-one-compound combinatorial peptide libraries. Bioconjug Chem 18 (2007) 175-182
-
(2007)
Bioconjug Chem
, vol.18
, pp. 175-182
-
-
Kumaresan, P.R.1
Natarajan, A.2
Song, A.3
Wang, X.4
Liu, R.5
DeNardo, G.6
-
35
-
-
24144489048
-
Reversible covalent chemistry in drug delivery
-
West K.R., and Otto S. Reversible covalent chemistry in drug delivery. Curr Drug Discov Technol 2 (2005) 123-160
-
(2005)
Curr Drug Discov Technol
, vol.2
, pp. 123-160
-
-
West, K.R.1
Otto, S.2
-
36
-
-
1942438684
-
Polymeric anticancer drugs with pH-controlled activation
-
Ulbrich K., and Subr V. Polymeric anticancer drugs with pH-controlled activation. Adv Drug Deliv Rev 56 (2004) 1023-1050
-
(2004)
Adv Drug Deliv Rev
, vol.56
, pp. 1023-1050
-
-
Ulbrich, K.1
Subr, V.2
-
38
-
-
33646184196
-
Aryldithioethyloxycarbonyl (Ardec): a new family of amine protecting groups removable under mild reducing conditions and their applications to peptide synthesis
-
Lapeyre M., Leprince J., Massonneau M., Oulyadi H., Renard P.Y., Romieu A., et al. Aryldithioethyloxycarbonyl (Ardec): a new family of amine protecting groups removable under mild reducing conditions and their applications to peptide synthesis. Chemistry 12 (2006) 3655-3671
-
(2006)
Chemistry
, vol.12
, pp. 3655-3671
-
-
Lapeyre, M.1
Leprince, J.2
Massonneau, M.3
Oulyadi, H.4
Renard, P.Y.5
Romieu, A.6
-
39
-
-
0015694487
-
131I-labelled m-iodohippuric acid and its behaviour in kidney function studies compared to o-iodohippuric acid
-
131I-labelled m-iodohippuric acid and its behaviour in kidney function studies compared to o-iodohippuric acid. Int J Appl Radiat Isot 24 (1973) 463-469
-
(1973)
Int J Appl Radiat Isot
, vol.24
, pp. 463-469
-
-
Elias, H.1
Arnold, C.2
Kloss, G.3
-
40
-
-
0016260069
-
Lysosomotropic agents
-
De Duve C., De Barsy T., Polle B., Trouet A., Tulkens P., and Van Hoof F. Lysosomotropic agents. Biochem Pharm 23 (1974) 2495-2531
-
(1974)
Biochem Pharm
, vol.23
, pp. 2495-2531
-
-
De Duve, C.1
De Barsy, T.2
Polle, B.3
Trouet, A.4
Tulkens, P.5
Van Hoof, F.6
-
41
-
-
0025491169
-
Antibody conjugates with morpholinodoxorubicin and acid-cleavable linkers
-
Mueller B.M., Wrasidlo W.A., and Reisfeld R.A. Antibody conjugates with morpholinodoxorubicin and acid-cleavable linkers. Bioconjug Chem 1 (1990) 325-330
-
(1990)
Bioconjug Chem
, vol.1
, pp. 325-330
-
-
Mueller, B.M.1
Wrasidlo, W.A.2
Reisfeld, R.A.3
-
42
-
-
0026164319
-
New hydrazone derivatives of adriamycin and their immunoconjugates - a correlation between acid stability and cytotoxicity
-
Kaneko T., Willner D., Monkovic I., Knipe J.O., Braslawsky G.R., Greenfield R.S., et al. New hydrazone derivatives of adriamycin and their immunoconjugates - a correlation between acid stability and cytotoxicity. Bioconjug Chem 2 (1991) 133-141
-
(1991)
Bioconjug Chem
, vol.2
, pp. 133-141
-
-
Kaneko, T.1
Willner, D.2
Monkovic, I.3
Knipe, J.O.4
Braslawsky, G.R.5
Greenfield, R.S.6
|