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Volumn 11, Issue 4, 2000, Pages 510-519

Synthesis, conjugation, and radiolabeling of a novel bifunctional chelating agent for 225Ac radioimmunotherapy applications

Author keywords

[No Author keywords available]

Indexed keywords

MONOCLONAL ANTIBODIES;

EID: 0033879250     PISSN: 10431802     EISSN: None     Source Type: Journal    
DOI: 10.1021/bc990153f     Document Type: Article
Times cited : (72)

References (43)
  • 5
    • 0030011011 scopus 로고    scopus 로고
    • Criteria for the selection of radionuclides for targeting nuclear antigens for cancer radioimmunotherapy
    • Srivastava, S. C. (1996) Criteria for the selection of radionuclides for targeting nuclear antigens for cancer radioimmunotherapy. Cancer Biother. Radiopharm. 11, 43-50.
    • (1996) Cancer Biother. Radiopharm. , vol.11 , pp. 43-50
    • Srivastava, S.C.1
  • 8
    • 0028842671 scopus 로고
    • Relationships between tumor size and curability for uniformly targeted therapy with beta-emitting radionuclides
    • O'Donoghue, J. A., Bardies, M., and Wheldon, T. E. (1995) Relationships between Tumor Size and Curability for Uniformly Targeted Therapy with Beta-Emitting Radionuclides. J. Nucl. Med. 36, 1902-1909.
    • (1995) J. Nucl. Med. , vol.36 , pp. 1902-1909
    • O'Donoghue, J.A.1    Bardies, M.2    Wheldon, T.E.3
  • 9
    • 0029443145 scopus 로고
    • Monoclonal antibody therapy of leukemia and lymphoma
    • (J. T. August, M. W. Anders, F. Murad, J. T. Coyle, Eds.) Academic Press, Inc., New York
    • Jurcic, J. G., Caron, P. C., and Scheinberg, D. A. (1995) Monoclonal Antibody Therapy of Leukemia and Lymphoma. In Advances in Pharmacology (J. T. August, M. W. Anders, F. Murad, J. T. Coyle, Eds.) Vol. 33, pp 287-314, Academic Press, Inc., New York.
    • (1995) Advances in Pharmacology , vol.33 , pp. 287-314
    • Jurcic, J.G.1    Caron, P.C.2    Scheinberg, D.A.3
  • 12
    • 0028017643 scopus 로고
    • Radioimmunotherapy of neoplastic meningitis in rats using an α-particle-emitting immunoconjugate
    • (a) Zalutsky, M. R., McLendon, R. E., Garg, P. K., Archer, G. E., Schuster, J. M., and Bigner, D. D. (1994) Radioimmunotherapy of neoplastic meningitis in rats using an α-particle-emitting immunoconjugate. Cancer Res. 54, 4719-4725.
    • (1994) Cancer Res. , vol.54 , pp. 4719-4725
    • Zalutsky, M.R.1    McLendon, R.E.2    Garg, P.K.3    Archer, G.E.4    Schuster, J.M.5    Bigner, D.D.6
  • 13
    • 0001042459 scopus 로고
    • 2 fragments with the α-particle emitting nuclide astatine-211: Preservation of the immunoreactivity and in vivo localization capacity
    • 2 fragments with the α-particle emitting nuclide astatine-211: Preservation of the immunoreactivity and in vivo localization capacity. Proc. Natl. Acad. Sci. 86, 7149-7153.
    • (1989) Proc. Natl. Acad. Sci. , vol.86 , pp. 7149-7153
    • Zalutsky, M.R.1    Garg, P.2    Friedman, H.S.3    Bigner, D.D.4
  • 15
    • 0002255839 scopus 로고    scopus 로고
    • Phase I trial of astatine-211 labeled human/mouse chimeric anti-tenascin antibody administered into malignant brain tumor resection cavities
    • Society of Neuro-Oncology Annual Meeting, San Francisco, CA
    • (11 ) Zalutsky, M. R., Akabani, G., Cokgor, I., Friedman, H. S., Coleman, R. E., Friedman, A. H., McLendon, R. E., Reist, C. J., Pegram, C. N., Zhao, X.-G., and Bigner, D. D. (1998) Phase I trial of astatine-211 labeled human/mouse chimeric anti-tenascin antibody administered into malignant brain tumor resection cavities. Society of Neuro-Oncology Annual Meeting, San Francisco, CA. Neuro-Oncology 1, S65-S66.
    • (1998) Neuro-oncology , vol.1
    • Zalutsky, M.R.1    Akabani, G.2    Cokgor, I.3    Friedman, H.S.4    Coleman, R.E.5    Friedman, A.H.6    McLendon, R.E.7    Reist, C.J.8    Pegram, C.N.9    Zhao, X.-G.10    Bigner, D.D.11
  • 19
    • 44949283598 scopus 로고
    • Newer approaches to the radiolabeling of monoclonal antibodies by the use of metal chelates
    • Gansow, O. A. (1991) Newer Approaches to the Radiolabeling of Monoclonal Antibodies by the Use of Metal Chelates. Nucl. Med. Biol. 18, 369-381.
    • (1991) Nucl. Med. Biol. , vol.18 , pp. 369-381
    • Gansow, O.A.1
  • 20
    • 0011764130 scopus 로고
    • Determination of the complex formation of actinium 1. Determination of the stability constants of ethylenediaminetetraacetate complexes of actinium and its separation from lanthanum in solutions of EDTA by the method of electromigration
    • (a) Makarova, T. P., Sinitsyna, G. S., Stepanov, A. V., Shestakova, I. A., and Shestkov, B. I. (1972) Determination of the Complex Formation of Actinium 1. Determination of the Stability constants of Ethylenediaminetetraacetate Complexes of Actinium and its Separation from Lanthanum in Solutions of EDTA by the Method of Electromigration. Radiochimiya 14, 538-541.
    • (1972) Radiochimiya , vol.14 , pp. 538-541
    • Makarova, T.P.1    Sinitsyna, G.S.2    Stepanov, A.V.3    Shestakova, I.A.4    Shestkov, B.I.5
  • 22
    • 0000593310 scopus 로고    scopus 로고
    • Carboxylate-derived calixarenes with high selectivity for actinium-225
    • (a) Chen, X., Ji, M., Fisher, D. R., and Wai, C. M. (1998) Carboxylate-derived calixarenes with high selectivity for actinium-225. Chem. Commun. 377-378.
    • (1998) Chem. Commun. , pp. 377-378
    • Chen, X.1    Ji, M.2    Fisher, D.R.3    Wai, C.M.4
  • 23
    • 0001590259 scopus 로고    scopus 로고
    • Conjugation, immunoreactivity, and immunogenicity of Calix[4]arenes; model study to potential Calix[4]-arene-based Ac3+ chelators
    • (b) Gansey, M. H. B. G., de Haan, A. S., Bos, E. S., Verboom, W., and Reinhoudt, D. N. (1999) Conjugation, Immunoreactivity, and Immunogenicity of Calix[4]arenes; Model Study to Potential Calix[4]-arene-Based Ac3+ Chelators. Bioconjugate Chem. 10, 613-623.
    • (1999) Bioconjugate Chem. , vol.10 , pp. 613-623
    • Gansey, M.H.B.G.1    De Haan, A.S.2    Bos, E.S.3    Verboom, W.4    Reinhoudt, D.N.5
  • 24
  • 25
    • 0000795358 scopus 로고
    • Metabolic characteristics within a chemical family
    • Durbin, P. W. (1960) Metabolic characteristics within a chemical family. Health Phys. 2, 225-238.
    • (1960) Health Phys. , vol.2 , pp. 225-238
    • Durbin, P.W.1
  • 26
    • 0344001700 scopus 로고    scopus 로고
    • personal communication
    • Kennel, S. J., personal communication.
    • Kennel, S.J.1
  • 27
    • 0022968394 scopus 로고
    • Synthesis of 1-(p-isothiocyanatobenzyl) derivatives of DTPA and EDTA. Antibody labeling and tumor-imaging studies
    • Brechbiel, M. W., Gansow, O. A., Atcher, R. W., Schlom, J., Esteban, J., Simpson, D. E., and Colcher, D. (1986) Synthesis of 1-(p-Isothiocyanatobenzyl) Derivatives of DTPA and EDTA. Antibody Labeling and Tumor-Imaging Studies. lnorg. Chem. 25, 2772.
    • (1986) Lnorg. Chem. , vol.25 , pp. 2772
    • Brechbiel, M.W.1    Gansow, O.A.2    Atcher, R.W.3    Schlom, J.4    Esteban, J.5    Simpson, D.E.6    Colcher, D.7
  • 30
    • 0023197202 scopus 로고
    • Complementation of intracavitary and intravenous administration of a monoclonal antibody (B72.3) in patients with carcinoma
    • (b) Colcher D., Esteban, J. E., Carrasquillo, J. A., Sugarbaker, P., Reynolds, J. C., Bryant, G., Larson, S. M., and Schlom, J. (1987) Complementation of intracavitary and intravenous administration of a monoclonal antibody (B72.3) in patients with carcinoma. Cancer Res. 47, 4218-4224.
    • (1987) Cancer Res. , vol.47 , pp. 4218-4224
    • Colcher, D.1    Esteban, J.E.2    Carrasquillo, J.A.3    Sugarbaker, P.4    Reynolds, J.C.5    Bryant, G.6    Larson, S.M.7    Schlom, J.8
  • 33
    • 0033380104 scopus 로고    scopus 로고
    • Spectrophotometric method for determination of bifunctional macrocyclic ligands in macrocyclic ligand-protein conjugates
    • Dadachova, E., Chappell, L. L., and Brechbiel, M. W. (1999) Spectrophotometric Method for Determination of Bifunctional Macrocyclic Ligands in Macrocyclic Ligand-Protein Conjugates. Nucl. Med. Biol. 26, 977-982.
    • (1999) Nucl. Med. Biol. , vol.26 , pp. 977-982
    • Dadachova, E.1    Chappell, L.L.2    Brechbiel, M.W.3
  • 34
    • 0010782540 scopus 로고    scopus 로고
    • 1,4,7,10,13,16,19,22-octaazacyclotetracosane-1,4,7,10,13, 16,19,22-octaacetic acid (H(8)OTEC) and 1,4,7,10,14,17, 20,23-octaazacyclohexacosane-1,4,7,10,14,17,20,23-octaacetic acid (H(8)OHEC): Synthesis and characterization of two large macrocyclic polyamine polycarboxylic ligands and some of their copper(II) and lanthanide(III) complexes
    • Schumann, H., Bottger, U. A., Zietzke, K., Hemling, H., Kociok-Kohn, G., Pickardt, J., Hahn, F. E., Zschunke, A., Schiefner, B., Gries, H., Raduchel, B., and Platzek, J. (1997) 1,4,7,10,13,16,19,22-Octaazacyclotetracosane-1,4,7,10,13, 16,19,22-octaacetic acid (H(8)OTEC) and 1,4,7,10,14,17, 20,23-octaazacyclohexacosane-1,4,7,10,14,17,20,23-octaacetic acid (H(8)OHEC): Synthesis and characterization of two large macrocyclic polyamine polycarboxylic ligands and some of their copper(II) and lanthanide(III) complexes. Chem. Ber.-Rec. 130, 267-277.
    • (1997) Chem. Ber.-rec. , vol.130 , pp. 267-277
    • Schumann, H.1    Bottger, U.A.2    Zietzke, K.3    Hemling, H.4    Kociok-Kohn, G.5    Pickardt, J.6    Hahn, F.E.7    Zschunke, A.8    Schiefner, B.9    Gries, H.10    Raduchel, B.11    Platzek, J.12
  • 36
    • 0031982801 scopus 로고    scopus 로고
    • Maleimidocysteineamido-DOTA derivatives: New reagents for radiometal chelate conjugation to antibody sulfhydryl groups undergo pH-dependent cleavage reactions
    • (b) Lewis, M. R., and Shively, J. E. (1998) Maleimidocysteineamido-DOTA Derivatives: New Reagents for Radiometal Chelate Conjugation to Antibody Sulfhydryl Groups Undergo pH-Dependent Cleavage Reactions. Bioconjugate Chem. 9, 72-86.
    • (1998) Bioconjugate Chem. , vol.9 , pp. 72-86
    • Lewis, M.R.1    Shively, J.E.2
  • 37
    • 0033136221 scopus 로고    scopus 로고
    • NMR studies of the metal-loading kinetics and acid-base chemistry of DOTA and butylamine-DOTA
    • Keire, D. A., and Kobayashi, M. (1999) NMR Studies of the Metal-Loading Kinetics and Acid-base Chemistry of DOTA and Butylamine-DOTA. Bioconjugate Chem. 10, 454-463.
    • (1999) Bioconjugate Chem. , vol.10 , pp. 454-463
    • Keire, D.A.1    Kobayashi, M.2
  • 39
    • 0001002121 scopus 로고
    • The peptide way to macrocyclic bifunctional chelating-agents -synthesis of 2-(p-nitrobenzyl)-1-1,4,7,10-tetraazacyclododecane-N,N′,N″, N‴-tetraacetic acid and study of its yttrium(III) complex
    • Moi, M. K., Meares, C. F., and DeNardo, S. J. (1988) The peptide way to macrocyclic bifunctional chelating-agents -synthesis of 2-(p-nitrobenzyl)-1-1,4,7,10-tetraazacyclododecane-N,N′,N″, N‴-tetraacetic acid and study of its yttrium(III) complex. J. Am. Chem. Soc. 110, 6266-6267.
    • (1988) J. Am. Chem. Soc. , vol.110 , pp. 6266-6267
    • Moi, M.K.1    Meares, C.F.2    DeNardo, S.J.3
  • 41
    • 0002521819 scopus 로고
    • Macrocyclic polyamines: 1,4,7,10,13,16-hexaazacyclooctadecane
    • (W. E. Noland, Ed.) John Wiley & Sons: New York, 1988
    • Atkins, T. J., Richman, J. E., and Oettlye, W. F., (1988) Macrocyclic Polyamines: 1,4,7,10,13,16-Hexaazacyclooctadecane. In Organic Synthesis Collective (W. E. Noland, Ed.) Vol. 6, pp 652-662, John Wiley & Sons: New York, 1988.
    • (1988) Organic Synthesis Collective , vol.6 , pp. 652-662
    • Atkins, T.J.1    Richman, J.E.2    Oettlye, W.F.3
  • 42
    • 84944648082 scopus 로고
    • Revised effective ionic radii and systematic studies of interatomic distances in halides and chalcogenides
    • Shannon, R. D. (1976) Revised Effective Ionic Radii and Systematic Studies of Interatomic Distances in Halides and Chalcogenides. Acta Crystallogr. 32, 751-767.
    • (1976) Acta Crystallogr. , vol.32 , pp. 751-767
    • Shannon, R.D.1
  • 43
    • 0008127787 scopus 로고    scopus 로고
    • Mapping an antibody binding site by nuclear decay
    • Mogul, R., and Meares, C. F. (1997) Mapping an Antibody Binding Site by Nuclear Decay J. Am. Chem. Soc. 119, 7169-7170.
    • (1997) J. Am. Chem. Soc. , vol.119 , pp. 7169-7170
    • Mogul, R.1    Meares, C.F.2


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