SCOPUS 정보 검색 플랫폼

Organic and Biomolecular Chemistry

Volumn 9, Issue 7, 2011, Pages 2251-2257

An straightforward entry to new pyrazolo-fused dibenzo[1,4]diazepines

(5) Hernández, Susana a Moreno, Isabel a Sanmartin, Raul a Teresa Herrero, María a Domínguez, Esther a

a UNIVERSITY OF THE BASQUE COUNTRY UPV EHU (Spain)

Author keywords

[No Author keywords available]

Indexed keywords

ARYLHYDRAZINES; CELECOXIB; ENAMINONES; HETEROCYCLIZATIONS; HETEROGENEOUS CATALYST; N-ARYLATION REACTIONS; POLYMER-SUPPORTED; RIMONABANT; STRUCTURE SIMILARITY; TANDEM SEQUENCE;

BENZODIAZEPINE DERIVATIVE; NITROGEN DERIVATIVE; PYRAZOLE DERIVATIVE;

ARTICLE; CATALYSIS; CHEMICAL STRUCTURE; CHEMISTRY; OXIDATION REDUCTION REACTION;

BENZODIAZEPINES; CATALYSIS; MOLECULAR STRUCTURE; NITROGEN COMPOUNDS; OXIDATION-REDUCTION; PYRAZOLES;

EID: 79952764529 PISSN: 14770520 EISSN: None Source Type: Journal
DOI: 10.1039/c0ob00812e Document Type: Article

Times cited : (27)

References (88)

1
- 0003799357
- M. V. Wolf and A. Burger, ed.; Wiley: New York
- J. A. Vida, in Medicinal Chemistry Part III, M. V. Wolf, and, A. Burger, ed.; Wiley: New York, 1981
- (1981) Medicinal Chemistry Part III
- Vida In, J.A.¹

2
- 0003607021
- A. R. Katrizky and C. W. Rees, Eds; Pergamon: Oxford, Ch. 1/06
- J. K. Landquist, in Comprehensive Heterocyclic Chemistry, A. R. Katrizky, and, C. W. Rees, Eds; Pergamon: Oxford, 1984; Vol 1., Ch. 1/06
- (1984) Comprehensive Heterocyclic Chemistry
- Landquist, J.K.¹

3
- 0003607021
- A. R. Katrizky and C. W. Rees, Eds; Pergamon: Oxford, Ch. 5/18
- J. T. Sharp, in Comprehensive Heterocyclic Chemistry, A. R. Katrizky, and, C. W. Rees, Eds; Pergamon: Oxford, 1984; Vol 7., Ch. 5/18
- (1984) Comprehensive Heterocyclic Chemistry
- Sharp In, J.T.¹

4
- 0003680152
- A. G. Gilman, L. S. Goodman, T. W. Ralland and F. Murand, ed.; MacMillan: New York, 391-413
- R. Baldessarini, in The Pharmacologic Basis of Therapeutics, A. G. Gilman, L. S. Goodman, T. W. Ralland, and, F. Murand, ed.; MacMillan: New York, 1985; Vol 1, pp 391-413
- (1985) The Pharmacologic Basis of Therapeutics
- Baldessarini In, R.¹

5
- 34548155962
- R. Ramajayan R. Girdhar M. R. Yadav Mini-Rev. Med. Chem. 2007 7 793 812
- (2007) Mini-Rev. Med. Chem. , vol.7 , pp. 793-812
- Ramajayan, R.¹ Girdhar, R.² Yadav, M.R.³

6
- 0033647332
- Y. Shimada N. Taniguchi A. Matsuhisa K. Sakamoto T. Yatsu A. Tanaka Chem Pharm. Bull 2000 48 1644 1651
- (2000) Chem Pharm. Bull , vol.48 , pp. 1644-1651
- Shimada, Y.¹ Taniguchi, N.² Matsuhisa, A.³ Sakamoto, K.⁴ Yatsu, T.⁵ Tanaka, A.⁶

7
- 1942438459
- See for example:
- A. L. Sabb R. L. Vogel G. S. Welmaker J. E. Sabalski J. Coupet J. Dunlop S. Rosenzweig-Lipson B. Harrison Bioorg. Med. Chem. Lett. 2004 14 2603 2607
- (2004) Bioorg. Med. Chem. Lett. , vol.14 , pp. 2603-2607
- Sabb, A.L.¹ Vogel, R.L.² Welmaker, G.S.³ Sabalski, J.E.⁴ Coupet, J.⁵ Dunlop, J.⁶ Rosenzweig-Lipson, S.⁷ Harrison, B.⁸

8
- 67849133186
- B. Petit-Demouliere F. Masse N. Cogrel M. Hascoet M. Bourin Behav. Brain Res. 2009 204 200 205
- (2009) Behav. Brain Res. , vol.204 , pp. 200-205
- Petit-Demouliere, B.¹ Masse, F.² Cogrel, N.³ Hascoet, M.⁴ Bourin, M.⁵

9
- 0003594838
- S. Needle and M. J. Waring, ed.; The Macmillan Press Ltd.: London, UK, 54-88
- D. E. Thurston, in Molecular Aspects of Anticancer Drug-DNA Interactions, S. Needle, and, M. J. Waring, ed.; The Macmillan Press Ltd.: London, UK, 1993; Vol. 1, pp 54-88
- (1993) Molecular Aspects of Anticancer Drug-DNA Interactions
- Thurston In, D.E.¹

10
- 41249094767
- A. Kamal N. Shankaraiah S. Prabhakar C. R. Reddy N. Markandeya K. Laxma X. Devaiah Bioorg. Med. Chem. Lett. 2008 18 2434 2439
- (2008) Bioorg. Med. Chem. Lett. , vol.18 , pp. 2434-2439
- Kamal, A.¹ Shankaraiah, N.² Prabhakar, S.³ Reddy, C.R.⁴ Markandeya, N.⁵ Laxma, K.⁶ Devaiah, X.⁷

11
- 43349083517
- J. Ip J. X. Wilson J. P. Uetrecht Chem. Res. Toxicol. 2008 21 869 873
- (2008) Chem. Res. Toxicol. , vol.21 , pp. 869-873
- Ip, J.¹ Wilson, J.X.² Uetrecht, J.P.³

12
- 65149105853
- A. Bali S. Malhotra H. Dhir A. Kumar A. Sharma Bioorg. Med. Chem. Lett. 2009 19 3041 3044
- (2009) Bioorg. Med. Chem. Lett. , vol.19 , pp. 3041-3044
- Bali, A.¹ Malhotra, S.² Dhir, H.³ Kumar, A.⁴ Sharma, A.⁵

13
- 36549013145
- C. Lamberth Heterocycles 2007 71 1467 1502
- (2007) Heterocycles , vol.71 , pp. 1467-1502
- Lamberth, C.¹

14
- 51649116082
- Diaryl heterocycles in general are a selective class of COX-2 inhibitors. See:
- W. Zheng S. R. Yates S. K. Papiernik J. Agric. Food Chem. 2008 56 7367 7372
- (2008) J. Agric. Food Chem. , vol.56 , pp. 7367-7372
- Zheng, W.¹ Yates, S.R.² Papiernik, S.K.³

15
- 0035960062
- P. Chavatte S. Yous C. Marot N. Baurin D. Lesieur J. Med. Chem. 2001 44 3223 3230
- (2001) J. Med. Chem. , vol.44 , pp. 3223-3230
- Chavatte, P.¹ Yous, S.² Marot, C.³ Baurin, N.⁴ Lesieur, D.⁵

16
- 67649644733
- J. Kelsey O. Harris J. Cassin Behav. Brain Res. 2009 203 304 307
- (2009) Behav. Brain Res. , vol.203 , pp. 304-307
- Kelsey, J.¹ Harris, O.² Cassin, J.³

17
- 35348833742
- Other applications of Celecoxib include treatment of preterm labour, osteoarthritis and rheumatoid arthritis, inflammatory bowel disease and duodenal polyposis in familial adenomatous polyposis. See
- V. K. Kotagiri S. Suthrapu J. M. Reddy C. P. Rao V. Bollugoddu A. Bhattacharya R. Bandichhor Org. Process Res. Dev. 2007 11 910 912
- (2007) Org. Process Res. Dev. , vol.11 , pp. 910-912
- Kotagiri, V.K.¹ Suthrapu, S.² Reddy, J.M.³ Rao, C.P.⁴ Bollugoddu, V.⁵ Bhattacharya, A.⁶ Bandichhor, R.⁷

18
- 0036739034
- C. S. Stika G. A. Gross G. Leguizamon S. Gerber R. Levy A. Mathur L. M. Bernhard D. M. Nelson Y. Sadovsky Am. J. Obstet. Gynecol. 2002 187 653 660
- (2002) Am. J. Obstet. Gynecol. , vol.187 , pp. 653-660
- Stika, C.S.¹ Gross, G.A.² Leguizamon, G.³ Gerber, S.⁴ Levy, R.⁵ Mathur, A.⁶ Bernhard, L.M.⁷ Nelson, D.M.⁸ Sadovsky, Y.⁹

19
- 0036708025
- K. Dilger C. Herrlinger J. Peters H. W. Seyberth H. Scheweer U. Klotz J. Clin. Pharmacol. 2002 42 985 994
- (2002) J. Clin. Pharmacol. , vol.42 , pp. 985-994
- Dilger, K.¹ Herrlinger, C.² Peters, J.³ Seyberth, H.W.⁴ Scheweer, H.⁵ Klotz, U.⁶

20
- 0036676087
- This type of compounds comprises a class of non-steroidal anti-inflammatory drugs (NSAID). See for example:
- K. M. Woessner R. A. Simon D. D. Stevenson Arthritis Rheum. 2002 46 2201 2206
- (2002) Arthritis Rheum. , vol.46 , pp. 2201-2206
- Woessner, K.M.¹ Simon, R.A.² Stevenson, D.D.³

21
- 57649121700
- J. P. O'Connor T. Lysz Drugs of Today 2008 44 693 709
- (2008) Drugs of Today , vol.44 , pp. 693-709
- O'Connor, J.P.¹ Lysz, T.²

22
- 0025370568
- U. Taeuber Drugs Exp. Clin. Res. 1990 16 7 15
- (1990) Drugs Exp. Clin. Res. , vol.16 , pp. 7-15
- Taeuber, U.¹

23
- 0035974649
- A. G. Habeeb P. N. Praveen E. E. Knaus J. Med. Chem. 2001 44 3039 3042
- (2001) J. Med. Chem. , vol.44 , pp. 3039-3042
- Habeeb, A.G.¹ Praveen, P.N.² Knaus, E.E.³

24
- 0037168053
- H. Liu X. Huang J. M. Shen X. Luo M. Li B. Xiong G. Chen J. Shen Y. Yang H. Jiang K. Chen J. Med. Chem. 2002 45 4816 4827
- (2002) J. Med. Chem. , vol.45 , pp. 4816-4827
- Liu, H.¹ Huang, X.² Shen, J.M.³ Luo, X.⁴ Li, M.⁵ Xiong, B.⁶ Chen, G.⁷ Shen, J.⁸ Yang, Y.⁹ Jiang, H.¹⁰ Chen, K.¹¹

25
- 1542613875
- S. K. Singh S. Vobbalareddy S. Shivaramakrishna A. Krishnamraju S. A. Rajjak S. R. Casturi V. Akhila Y. K. Rao Bioorg. Med. Chem. Lett. 2004 14 1683 1688
- (2004) Bioorg. Med. Chem. Lett. , vol.14 , pp. 1683-1688
- Singh, S.K.¹ Vobbalareddy, S.² Shivaramakrishna, S.³ Krishnamraju, A.⁴ Rajjak, S.A.⁵ Casturi, S.R.⁶ Akhila, V.⁷ Rao, Y.K.⁸

26
- 1642540579
- Narayama et al. reported the synthesis and anticonvulsant activity of a series of triazolo-fused benzodiapepine derivatives. See:
- A. Weber A. Casini A. Heine D. Kuhn C. T. Sapuran A. Scozzafava G. Klebe J. Med. Chem. 2004 47 550 557
- (2004) J. Med. Chem. , vol.47 , pp. 550-557
- Weber, A.¹ Casini, A.² Heine, A.³ Kuhn, D.⁴ Sapuran, C.T.⁵ Scozzafava, A.⁶ Klebe, G.⁷

27
- 33645963789
- Later, the same authors described the antianxiety properties and the anticancer activity of some of these derivatives:
- B. Narayana K. K. V. Raj B. V. Ashalatha N. S. Kumari Eur. J. Med. Chem. 2006 41 417 422
- (2006) Eur. J. Med. Chem. , vol.41 , pp. 417-422
- Narayana, B.¹ Raj, K.K.V.² Ashalatha, B.V.³ Kumari, N.S.⁴

28
- 79952770997
- It is well known the pharmacological activity of some thieno-fused diazepines such as clotiazepam, brotizolam and etizolam. See for example:
- K. K. V. Raj B. Narayana N. S. Kumari B. V. Ashalatha B. K. Sarojini Journal of Pharmacology and Toxicology 2006 1 471 477
- (2006) Journal of Pharmacology and Toxicology , vol.1 , pp. 471-477
- Raj, K.K.V.¹ Narayana, B.² Kumari, N.S.³ Ashalatha, B.V.⁴ Sarojini, B.K.⁵

29
- 0036949423
- Some pyrrolo[2,1-c][1,4]benzodiazepines (PBDs) such us DC-81, tomamycin and anthramycin are naturally occurring anticancer antibiotics produced by some species of Streptomyces bacteria. See:
- V. Lisowsky F. Fabis A. Pierre D. H. Caignard P. Renard S. Rault J. Enzyme Inhib. Med. Chem. 2002 17 403 407
- (2002) J. Enzyme Inhib. Med. Chem. , vol.17 , pp. 403-407
- Lisowsky, V.¹ Fabis, F.² Pierre, A.³ Caignard, D.H.⁴ Renard, P.⁵ Rault, S.⁶

30
- 60049086079
- A. Kamal D. Rajender D. R. Reddy M. K. Reddy G. Balakishan T. B. Shaik M. Chourasia G. N. Sastry Bioorg. Med. Chem. 2009 17 1557 1572
- (2009) Bioorg. Med. Chem. , vol.17 , pp. 1557-1572
- Kamal, A.¹ Rajender, D.² Reddy, D.R.³ Reddy, M.K.⁴ Balakishan, G.⁵ Shaik, T.B.⁶ Chourasia, M.⁷ Sastry, G.N.⁸

31
- 58949091407
- See for example:
- W. P. Hu J. J. Liang Ch. L. Kao Y. Ch. Chen Ch. Y. Chung F. Y. Tsai M. J. Wu L. S. Chang Y. L. Chen J. J. Wang Bioorg. Med. Chem. 2009 17 1172 1182
- (2009) Bioorg. Med. Chem. , vol.17 , pp. 1172-1182
- Hu, W.P.¹ Liang, J.J.² Kao, Ch.L.³ Ch., C.Y.⁴ Chung, Ch.Y.⁵ Tsai, F.Y.⁶ Wu, M.J.⁷ Chang, L.S.⁸ Chen, Y.L.⁹ Wang, J.J.¹⁰

32
- 54049091217
- and references cited therein Pirenzepine is a pyridobenzodiazepine with multiple biological activities. See for example:
- Y. Ohta H. Chiba S. Oishi N. Fujii H. Ohno Org. Lett. 2008 10 3535 3538
- (2008) Org. Lett. , vol.10 , pp. 3535-3538
- Ohta, Y.¹ Chiba, H.² Oishi, S.³ Fujii, N.⁴ Ohno, H.⁵

33
- 67749116459
- B. Ilien N. Glasser J.-P. Clamme P. Didier E. Piemont R. Chinnappan S. B. Daval J.-L. Galzi Y. Mely J. Biol. Chem. 2009 284 19533 19543
- (2009) J. Biol. Chem. , vol.284 , pp. 19533-19543
- Ilien, B.¹ Glasser, N.² Clamme, J.-P.³ Didier, P.⁴ Piemont, E.⁵ Chinnappan, R.⁶ Daval, S.B.⁷ Galzi, J.-L.⁸ Mely, Y.⁹

34
- 51149095394
- B. Insuasty F. Orozco J. Quiroga R. Abonia M. Nogueras J. Cobo Eur. J. Med. Chem. 2008 43 1955 1962
- (2008) Eur. J. Med. Chem. , vol.43 , pp. 1955-1962
- Insuasty, B.¹ Orozco, F.² Quiroga, J.³ Abonia, R.⁴ Nogueras, M.⁵ Cobo, J.⁶

35
- 51449111470
- B. Insuasty F. Orozco C. Lizarazu J. Quiroga R. Abonia M. Hursthouse M. Nogueras J. Cobo Bioorg. Med. Chem. 2008 16 8492 8500
- (2008) Bioorg. Med. Chem. , vol.16 , pp. 8492-8500
- Insuasty, B.¹ Orozco, F.² Lizarazu, C.³ Quiroga, J.⁴ Abonia, R.⁵ Hursthouse, M.⁶ Nogueras, M.⁷ Cobo, J.⁸

36
- 33748621833
- A. Guram R. A. Rennels S. L. Buchwald Angew. Chem., Int. Ed. Engl. 1995 34 1348 1350
- (1995) Angew. Chem., Int. Ed. Engl. , vol.34 , pp. 1348-1350
- Guram, A.¹ Rennels, R.A.² Buchwald, S.L.³

37
- 0029044538
- For a revision on the Buchwald-Hartwig reaction see:
- J. Louis J. F. Hartwig Tetrahedron Lett. 1995 36 3609 3612
- (1995) Tetrahedron Lett. , vol.36 , pp. 3609-3612
- Louis, J.¹ Hartwig, J.F.²

38
- 0037060980
- 2041-2075
- D. Prim, J.-M. Campagne, D. Joseph and B. Andrioletti, Tetrahedron 2002, 58, 2041-2075
- (2002) Tetrahedron , vol.58
- Prim, D.¹ Campagne, J.-M.² Joseph, D.³ Andrioletti, B.⁴

39
- 0000157513
- The Buchwald-Hartwig amination from an industrial point of view is described in:
- A. R. Muci S. L. Buchwald Top. Curr. Chem. 219 131 209
- Top. Curr. Chem. , vol.219 , pp. 131-209
- Muci, A.R.¹ Buchwald, S.L.²

40
- 12344337315
- The Buchwald-Hartwig cross-coupling reaction has been used in pharmaceutical synthesis, natural product synthesis, and material science. A very good revision of these applications in:
- B. Schlummer U. Scholz Adv. Synth. Catal. 2004 346 1599 1626
- (2004) Adv. Synth. Catal. , vol.346 , pp. 1599-1626
- Schlummer, B.¹ Scholz, U.²

41
- 52049105452
- The synthesis of indoles or indolines by the Buchwald-Hartwig aimantion is described in:
- D. S. Surry S. L. Buchwald Angew. Chem., Int. Ed. 2008 47 6338 6361
- (2008) Angew. Chem., Int. Ed. , vol.47 , pp. 6338-6361
- Surry, D.S.¹ Buchwald, S.L.²

42
- 0034603363
- J. A. Brown Tetrahedron Lett. 2000 41 1623 1626
- (2000) Tetrahedron Lett. , vol.41 , pp. 1623-1626
- Brown, J.A.¹

43
- 0034679492
- M. Watanabe T. Yamamoto M. Nishiyama Angew. Chem., Int. Ed. 2000 39 2501 2504
- (2000) Angew. Chem., Int. Ed. , vol.39 , pp. 2501-2504
- Watanabe, M.¹ Yamamoto, T.² Nishiyama, M.³

44
- 0029874188
- J. P. Wolfe R. A. Rennels S. L. Buchwald Tetrahedron 1996 52 7525 7546
- (1996) Tetrahedron , vol.52 , pp. 7525-7546
- Wolfe, J.P.¹ Rennels, R.A.² Buchwald, S.L.³

45
- 0033564994
- Preparation of indazoles by this methodology:
- B. H. Yang S. L. Buchwald Org. Lett. 1999 1 35 37
- (1999) Org. Lett. , vol.1 , pp. 35-37
- Yang, B.H.¹ Buchwald, S.L.²

46
- 0037029838
- Y.-M. Zhu Y. Kiyu H. Katayama Tetrahedron Lett. 2002 43 3577 3580
- (2002) Tetrahedron Lett. , vol.43 , pp. 3577-3580
- Zhu, Y.-M.¹ Kiyu, Y.² Katayama, H.³

47
- 0035897164
- J. J. Song N. K. Yee Tetrahedron Lett. 2001 42 2937 2940
- (2001) Tetrahedron Lett. , vol.42 , pp. 2937-2940
- Song, J.J.¹ Yee, N.K.²

48
- 0034707984
- The access to phenazines by this procedure is described in:
- J. J. Song N. K. Yee Org. Lett. 2000 2 519 521
- (2000) Org. Lett. , vol.2 , pp. 519-521
- Song, J.J.¹ Yee, N.K.²

49
- 0034650815
- Synthesis of benzimidazoles:
- T. Emoto N. Kubosaki Y. Yamagiwa T. Kamikawa Tetrahedron Lett. 2000 41 355 358
- (2000) Tetrahedron Lett. , vol.41 , pp. 355-358
- Emoto, T.¹ Kubosaki, N.² Yamagiwa, Y.³ Kamikawa, T.⁴

50
- 0037017716
- C. T. Brian S. A. Brunton Tetrahedron Lett. 2002 43 1893 1895
- (2002) Tetrahedron Lett. , vol.43 , pp. 1893-1895
- Brian, C.T.¹ Brunton, S.A.²

51
- 0000401303
- T. Iwaki A. Yasuhara T. Sakamoto J. Chem. Soc., Perkin Trans. 1 1999 1505 1510
- (1999) J. Chem. Soc., Perkin Trans. 1 , pp. 1505-1510
- Iwaki, T.¹ Yasuhara, A.² Sakamoto, T.³

52
- 32144431909
- C. Venkatesh G. S. M. Sundaram H. Ila H. Junjappa J. Org. Chem. 2006 71 1280 1283
- (2006) J. Org. Chem. , vol.71 , pp. 1280-1283
- Venkatesh, C.¹ Sundaram, G.S.M.² Ila, H.³ Junjappa, H.⁴

53
- 0043009828
- Synthesis of oxazepines an thiazepines:
- C. T. Brian J. T. Steer J. Org. Chem. 2003 68 6814 6816
- (2003) J. Org. Chem. , vol.68 , pp. 6814-6816
- Brian, C.T.¹ Steer, J.T.²

54
- 0037462378
- Preparation of imidazoles and its benzo- and aza- analogues:
- B. J. Margolis J. J. Swisorski B. N. Rogers J. Org. Chem. 2003 68 644 647
- (2003) J. Org. Chem. , vol.68 , pp. 644-647
- Margolis, B.J.¹ Swisorski, J.J.² Rogers, B.N.³

55
- 9444290796
- Preparation of oxindoles:
- K. T. J. Loones B. U. W. Maes R. A. Dommisse G. L. F. Lemiere Chem. Commun. 2004 2466 2467
- (2004) Chem. Commun. , pp. 2466-2467
- Loones, K.T.J.¹ Maes, B.U.W.² Dommisse, R.A.³ Lemiere, G.L.F.⁴

56
- 33749023851
- An elegant synthetic route for the access to a series of dibenzodiazepine-11-ones based on an intramolecular amination process was reported in:
- F. Bonnaterre M. Bois-Choussy J. Zhu Org. Lett. 2006 8 4351 4354
- (2006) Org. Lett. , vol.8 , pp. 4351-4354
- Bonnaterre, F.¹ Bois-Choussy, M.² Zhu, J.³

57
- 9644304518
- For the synthesis of 1,4-benzodiazepine-2,5-diones by the combination of an Ugi multicomponent reaction and a palladium catalyzed N-arylation, see:
- E. M. Beccalli G. Broggini G. Paladino C. Zoni Tetrahedron 2005 61 61 68
- (2005) Tetrahedron , vol.61 , pp. 61-68
- Beccalli, E.M.¹ Broggini, G.² Paladino, G.³ Zoni, C.⁴

58
- 7744222516
- G. Cuny M. Bois-Choussy J. Zhu J. Am. Chem. Soc. 2004 126 14475 14484
- (2004) J. Am. Chem. Soc. , vol.126 , pp. 14475-14484
- Cuny, G.¹ Bois-Choussy, M.² Zhu, J.³

59
- 33646036709
- A recent application of the modified Vilsmeier-Haak reagent DMFDMA is described in:
- C. Kalinsky M. Umkehrer G. Ross J. Kolb C. Burdack W. Hiller Tetrahedron Lett. 2006 47 3423 3426
- (2006) Tetrahedron Lett. , vol.47 , pp. 3423-3426
- Kalinsky, C.¹ Umkehrer, M.² Ross, G.³ Kolb, J.⁴ Burdack, C.⁵ Hiller, W.⁶

60
- 70350680826
- Ortho-bromoarylhydrazines 4b-d were prepared by diazotization/reduction of the corresponding anilines. For a related procedure, see:
- F. M. Abdelrazek N. H. Metwally Synth. Commun. 2009 39 4088 4099
- (2009) Synth. Commun. , vol.39 , pp. 4088-4099
- Abdelrazek, F.M.¹ Metwally, N.H.²

61
- 0034091818
- This tandem has been successfully applied by our group to the synthesis of different heterocycles. See for example:
- D. Gennet P. Michel A. Rassat Synthesis 2000 447 451
- (2000) Synthesis , pp. 447-451
- Gennet, D.¹ Michel, P.² Rassat, A.³

62
- 0000228798
- E. Domínguez E. Ibeas E. Martinez de Marigorta J. K. Palacios R. SanMartin J. Org. Chem. 1996 61 5435 5439
- (1996) J. Org. Chem. , vol.61 , pp. 5435-5439
- Domínguez, E.¹ Ibeas, E.² Martinez De Marigorta, E.³ Palacios, J.K.⁴ Sanmartin, R.⁵

63
- 0037131141
- R. Olivera R. SanMartin F. Churruca E. Domínguez J. Org. Chem. 2002 67 7215 7225
- (2002) J. Org. Chem. , vol.67 , pp. 7215-7225
- Olivera, R.¹ Sanmartin, R.² Churruca, F.³ Domínguez, E.⁴

64
- 0141742132
- S. Hernández R. SanMartin I. Tellitu E. Domínguez Org. Lett. 2003 5 1095 1098
- (2003) Org. Lett. , vol.5 , pp. 1095-1098
- Hernández, S.¹ Sanmartin, R.² Tellitu, I.³ Domínguez, E.⁴

65
- 0023217546
- V. T. Bandurco C. F. Schewender S. C. Bell D. W. Combs R. M. Kanojia S. D. Levine D. M. Mulvey M. A. Appollina M. S. Reed E. A. Malloy R. Falotico J. B. Moore A. J. Tobia J. Med. Chem. 1987 30 1421 1426
- (1987) J. Med. Chem. , vol.30 , pp. 1421-1426
- Bandurco, V.T.¹ Schewender, C.F.² Bell, S.C.³ Combs, D.W.⁴ Kanojia, R.M.⁵ Levine, S.D.⁶ Mulvey, D.M.⁷ Appollina, M.A.⁸ Reed, M.S.⁹ Malloy, E.A.¹⁰ Falotico, R.¹¹ Moore, J.B.¹² Tobia, A.J.¹³

66
- 0033522729
- G. Broggini L. Garanti G. Molteni T. Pilati A. Ponti G. Zecchi Tetrahedron: Asymmetry 1999 10 2203 2212
- (1999) Tetrahedron: Asymmetry , vol.10 , pp. 2203-2212
- Broggini, G.¹ Garanti, L.² Molteni, G.³ Pilati, T.⁴ Ponti, A.⁵ Zecchi, G.⁶

67
- 0000418343
- J. P. Wolfe S. L. Buchwald J. Org. Chem. 1997 62 1264 1267
- (1997) J. Org. Chem. , vol.62 , pp. 1264-1267
- Wolfe, J.P.¹ Buchwald, S.L.²

68
- 0000777908
- J. L. Louie M. S. Driver B. C. Hamann J. F. Hartwing J. Org. Chem. 1997 62 1268 1273
- (1997) J. Org. Chem. , vol.62 , pp. 1268-1273
- Louie, J.L.¹ Driver, M.S.² Hamann, B.C.³ Hartwing, J.F.⁴

69
- 0034712161
- Copper catalyzed N-arylation reactions are reported in:
- J. P. Wolfe S. L. Buchwald J. Org. Chem. 2000 65 1144 1157
- (2000) J. Org. Chem. , vol.65 , pp. 1144-1157
- Wolfe, J.P.¹ Buchwald, S.L.²

70
- 0033593282
- H. B. Goodbrand N.-X. Hu J. Org. Chem. 1999 64 670 674
- (1999) J. Org. Chem. , vol.64 , pp. 670-674
- Goodbrand, H.B.¹ Hu, N.-X.²

71
- 0033515805
- A. Kiyomori J.-F. Marcoux S. L. Buchwald Tetrahedron Lett. 1999 40 2657 2660
- (1999) Tetrahedron Lett. , vol.40 , pp. 2657-2660
- Kiyomori, A.¹ Marcoux, J.-F.² Buchwald, S.L.³

72
- 0035898818
- R. Gujadhur D. Venkataraman J. T. Kintigh Tetrahedron Lett. 2001 42 4791 4793
- (2001) Tetrahedron Lett. , vol.42 , pp. 4791-4793
- Gujadhur, R.¹ Venkataraman, D.² Kintigh, J.T.³

73
- 0037149057
- 3)Br and other copper derivatives soluble in organic solvents is described in:
- F. Y. Kwong A. Klapars S. L. Buchwald Org. Lett. 2002 4 581 584
- (2002) Org. Lett. , vol.4 , pp. 581-584
- Kwong, F.Y.¹ Klapars, A.² Buchwald, S.L.³

74
- 0001572402
- R. K. Gujadhur C. G. Bates D. Venkataraman Org. Lett. 2001 3 4315 4317
- (2001) Org. Lett. , vol.3 , pp. 4315-4317
- Gujadhur, R.K.¹ Bates, C.G.² Venkataraman, D.³

75
- 0034659728
- J. Schward V. P. W. Bohm M. G. Gardiner M. Grosche W. A. Herrmann W. Hieringer G. Raudaschl-Sieber Chem.-Eur. J. 2000 6 1773 1780
- (2000) Chem.-Eur. J. , vol.6 , pp. 1773-1780
- Schward, J.¹ Bohm, V.P.W.² Gardiner, M.G.³ Grosche, M.⁴ Herrmann, W.A.⁵ Hieringer, W.⁶ Raudaschl-Sieber, G.⁷

76
- 33645802202
- L. Djakovitch V. Dufaud R. Zaide Adv. Synth. Catal. 2006 348 715 724
- (2006) Adv. Synth. Catal. , vol.348 , pp. 715-724
- Djakovitch, L.¹ Dufaud, V.² Zaide, R.³

77
- 62649107110
- J. Demel X. Sujandi S.-E. Park J. Cejka P. Stepnicka J. Mol. Catal. A: Chem. 2009 302 28 35
- (2009) J. Mol. Catal. A: Chem. , vol.302 , pp. 28-35
- Demel, J.¹ Sujandi, X.² Park, S.-E.³ Cejka, J.⁴ Stepnicka, P.⁵

78
- 0037060753
- S. Fugita Y. Yoshida B. M. Bhanage M. Shirai M. Arai J. Mol. Catal. A: Chem. 2002 180 277 284
- (2002) J. Mol. Catal. A: Chem. , vol.180 , pp. 277-284
- Fugita, S.¹ Yoshida, Y.² Bhanage, B.M.³ Shirai, M.⁴ Arai, M.⁵

79
- 0033536404
- B. M. Bhanage M. Shirai M. Arai J. Mol. Catal. A: Chem. 1999 145 69 74
- (1999) J. Mol. Catal. A: Chem. , vol.145 , pp. 69-74
- Bhanage, B.M.¹ Shirai, M.² Arai, M.³

80
- 0029639927
- R. V. Chaudhari B. M. Bhanage R. M. Deshpande H. Delmas Nature 1995 373 501 503
- (1995) Nature , vol.373 , pp. 501-503
- Chaudhari, R.V.¹ Bhanage, B.M.² Deshpande, R.M.³ Delmas, H.⁴

81
- 0033609838
- B. M. Bhanage Y. Ikushima M. Shirai M. Arai Tetrahedron Lett. 1999 40 6427 6430
- (1999) Tetrahedron Lett. , vol.40 , pp. 6427-6430
- Bhanage, B.M.¹ Ikushima, Y.² Shirai, M.³ Arai, M.⁴

82
- 40249114677
- and references cited therein The FibreCat 1000 series is commercialized by Johnson Matthey Chemicals. Futher information about FibreCat catalysts, including their application in Suzuki-Miyaura and Mizoroki-Heck coupling reactions, can be found at
- P. J. Tambade Y. P. Patil M. J. Bhanushali B. M. Bhanage Tetrahedron Lett. 2008 49 2221 2224
- (2008) Tetrahedron Lett. , vol.49 , pp. 2221-2224
- Tambade, P.J.¹ Patil, Y.P.² Bhanushali, M.J.³ Bhanage, B.M.⁴

83
- 0001560006
- T. J. Colacot E. S. Gore A. Kuber Organometallics 2002 21 3301 3304
- (2002) Organometallics , vol.21 , pp. 3301-3304
- Colacot, T.J.¹ Gore, E.S.² Kuber, A.³

84
- 75349095976
- T. J. Colacot Top. Catal. 2008 48 91 98
- (2008) Top. Catal. , vol.48 , pp. 91-98
- Colacot, T.J.¹

85
- 56049104219
- Our group has reported the application of FibreCat catalysts in arylation of ketone enolates:
- T. J. Colacot W. A. Carole B. A. Neide A. Harad Organometallics 2008 27 5605 4611
- (2008) Organometallics , vol.27 , pp. 5605-4611
- Colacot, T.J.¹ Carole, W.A.² Neide, B.A.³ Harad, A.⁴

86
- 1242351219
- F. Churruca R. SanMartin M. Carril I. Tellitu E. Domínguez Tetrahedron 2004 60 2393 2408
- (2004) Tetrahedron , vol.60 , pp. 2393-2408
- Churruca, F.¹ Sanmartin, R.² Carril, M.³ Tellitu, I.⁴ Domínguez, E.⁵

87
- 20744456158
- In the direct C-H activation reaction:
- F. Churruca R. SanMartin I. Tellitu E. Dominguez Eur. J. Org. Chem. 2005 2481 2490
- (2005) Eur. J. Org. Chem. , pp. 2481-2490
- Churruca, F.¹ Sanmartin, R.² Tellitu, I.³ Dominguez, E.⁴

88
- 75349095055
- 3CN. For, more details see reference 37a The limit of thermal stability of FibreCat™ series is at around 120 °C. A partial loss of activity on recycling this type of heterogeneous catalyst has been observed in other cross-coupling reactions. See for example references 36-37
- S. Hernández I. Moreno R. SanMartin G. Gómez M. T. Herrero E. Domínguez J. Org. Chem. 2010 75 434 441
- (2010) J. Org. Chem. , vol.75 , pp. 434-441
- Hernández, S.¹ Moreno, I.² Sanmartin, R.³ Gómez, G.⁴ Herrero, M.T.⁵ Domínguez, E.⁶

* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.