CAR2 displays unique ligand binding and RXRα heterodimerization characteristics

Drug Metabolism and Disposition

Volumn 35, Issue 3, 2007, Pages 428-439

  Auerbach, Scott S ^a   DeKeyser, Joshua G ^b   Stoner, Matthew A ^b   Omiecinski, Curtis J ^b  

^a UNIVERSITY OF WASHINGTON SCHOOL OF MEDICINE   (United States)

^b PENNSYLVANIA STATE UNIVERSITY   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

ANDROSTANE DERIVATIVE; ASPARTIC ACID; CLOTRIMAZOLE; CONSTITUTIVE ANDROSTANE RECEPTOR; CONSTITUTIVE ANDROSTANE RECEPTOR 2; CYTOCHROME P450 2B6; CYTOCHROME P450 3A4; RETINOID X RECEPTOR ALPHA; SERINE; STEROID RECEPTOR COACTIVATOR 1; UNCLASSIFIED DRUG;

ANIMAL CELL; ARTICLE; CONTROLLED STUDY; DIMERIZATION; DRUG RECEPTOR BINDING; GENE MUTATION; GENE OVEREXPRESSION; LIGAND BINDING; NONHUMAN; NUCLEOTIDE SEQUENCE; PRIORITY JOURNAL; PROTEIN EXPRESSION; PROTEIN PROTEIN INTERACTION; SITE DIRECTED MUTAGENESIS; TRANSACTIVATION;

ANDROSTANOLS; ANIMALS; BINDING SITES; CERCOPITHECUS AETHIOPS; CLOTRIMAZOLE; COS CELLS; GENES, REPORTER; HUMANS; LIGANDS; LUCIFERASES; MUTAGENESIS, SITE-DIRECTED; OXIMES; RECEPTORS, CYTOPLASMIC AND NUCLEAR; RESPONSE ELEMENTS; RETINOID X RECEPTOR ALPHA; THIAZOLES; TRANSCRIPTION FACTORS; TRANSFECTION;

EID: 33847388435     PISSN: 00909556     EISSN: 1521009X     Source Type: Journal    
DOI: 10.1124/dmd.106.012641     Document Type: Article

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