Allosteric functioning of dimeric class C G-protein-coupled receptors

FEBS Journal

Volumn 272, Issue 12, 2005, Pages 2947-2955

  Pin, J P ^a,b,c,d   Kniazeff, J ^a,b,c,d   Liu, J ^a,b,c,d   Binet, V ^a,b,c,d   Goudet, C ^a,b,c,d   Rondard, P ^a,b,c,d   Prezeau L ^a,b,c,d  

^a INSTITUT DE GÉNOMIQUE FONCTIONNELLE   (France)

^b CNRS   (France)

^c INSERM   (France)

^d UNIV MONTPELLIER   (France)

Author keywords

Activation mechanism; Allosteric modulators; Dimerization; GPCR

Indexed keywords

G PROTEIN COUPLED RECEPTOR; G PROTEIN COUPLED RECEPTOR CLASS C; MEMBRANE RECEPTOR; MONOMER; OLIGOMER; RECEPTOR SUBUNIT; UNCLASSIFIED DRUG;

ALLOSTERISM; DIMERIZATION; DISULFIDE BOND; DRUG DESIGN; PRIORITY JOURNAL; PROTEIN ANALYSIS; PROTEIN DOMAIN; SHORT SURVEY; STRUCTURE ACTIVITY RELATION;

ANIMALS; DIMERIZATION; HUMANS; MODELS, MOLECULAR; PROTEIN CONFORMATION; PROTEIN STRUCTURE, TERTIARY; RECEPTORS, G-PROTEIN-COUPLED;

EID: 21344446100     PISSN: 1742464X     EISSN: None     Source Type: Journal    
DOI: 10.1111/j.1742-4658.2005.04728.x     Document Type: Short Survey

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