SCOPUS 정보 검색 플랫폼

Volumn 348, Issue 8, 2015, Pages 531-540

Rational Modification of the Biological Profile of GPCR Ligands through Combination with Other Biologically Active Moieties

(3) Huang, Guozheng a Nimczick, Martin a Decker, Michael a

a UNIVERSITY OF WÜRZBURG (Germany)

Author keywords

Bivalent ligand; Drug design; Hybrid molecule; Multifunctional ligand

Indexed keywords

BIOLOGICAL PRODUCT; CANNABINOID 1 RECEPTOR; CANNABINOID 1 RECEPTOR ANTAGONIST; CANNABINOID 2 RECEPTOR; CANNABINOID 2 RECEPTOR ANTAGONIST; CANNABINOID RECEPTOR ANTAGONIST; CHOLINESTERASE INHIBITOR; DOPAMINE RECEPTOR BLOCKING AGENT; G PROTEIN COUPLED RECEPTOR; HISTAMINE H3 RECEPTOR ANTAGONIST; LIGAND; OPIATE ANTAGONIST; OPIATE RECEPTOR; TACRINE; UNCLASSIFIED DRUG; DRUG; PROTEIN BINDING;

ALLOSTERISM; ARTICLE; BIOLOGICAL ACTIVITY; DRUG DESIGN; DRUG EFFICACY; DRUG RECEPTOR BINDING; HUMAN; LIGAND BINDING; PHARMACOPHORE; PRIORITY JOURNAL; PROTEIN PROTEIN INTERACTION; RECEPTOR BINDING ASSAY; STRUCTURE ACTIVITY RELATION; ANIMAL; BINDING SITE; CHEMISTRY; DRUG EFFECTS; METABOLISM; MOLECULARLY TARGETED THERAPY; PROTEIN CONFORMATION; SIGNAL TRANSDUCTION;

ANIMALS; BINDING SITES; DRUG DESIGN; HUMANS; LIGANDS; MOLECULAR TARGETED THERAPY; PHARMACEUTICAL PREPARATIONS; PROTEIN BINDING; PROTEIN CONFORMATION; RECEPTORS, G-PROTEIN-COUPLED; SIGNAL TRANSDUCTION; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 84938417797 PISSN: 03656233 EISSN: 15214184 Source Type: Journal
DOI: 10.1002/ardp.201500079 Document Type: Article

Times cited : (6)

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