SCOPUS 정보 검색 플랫폼

Volumn 8, Issue 12, 2013, Pages 2036-2046

Effect of linker length and composition on heterobivalent ligand-mediated receptor cross-talk between the A1 adenosine and β2 adrenergic receptors

(3) Barlow, Nicholas a Baker, Stephen P b Scammells, Peter J a

a MONASH UNIVERSITY (Australia)

b UNIVERSITY OF FLORIDA COLLEGE OF MEDICINE (United States)

Author keywords

2 adrenergic receptors; A1 adenosine receptors; combined pharmacophores; heterobivalent ligands; structure activity relationships

Indexed keywords

6 N CYCLOPENTYLADENOSINE; 8 CYCLOPENTYL 1,3 DIPROPYLXANTHINE; ADENOSINE; ADENOSINE A1 RECEPTOR; ADENOSINE A1 RECEPTOR AGONIST; ADENOSINE TRIPHOSPHATE; ADENYLATE CYCLASE; BETA 2 ADRENERGIC RECEPTOR; BETA 2 ADRENERGIC RECEPTOR STIMULATING AGENT; CYCLIC AMP; ETHANOLAMINE; G PROTEIN COUPLED RECEPTOR; HETEROBIVALENT LIGAND; IODINE 125; IODOPINDOLOL; ISOPRENALINE; LIGAND; N6 (11 ((2 (2 (2 (12 ((2 HYDROXY 2 (4 HYDROXY 3 (HYDROXYMETHYL)PHENYL)ETHYL)AMINO)DODECANAMIDO)ETHYLOXY)ETHOXY)ETHYLAMINO)FORMYL)UNDECYL)ADENOSINE ACETATE; N6 (11 ((6 (12 ((2 HYDROXY 2 (4 HYDROXY 3 (HYDROXYMETHYL)PHENYL)ETHYL)AMINO)DODECANAMIDO)HEXYLAMINO)FORMYL)UNDECYL)ADENOSINE ACETATE; N6 (5 ((2 (2 (2 (12 ((2 HYDROXY 2 (4 HYDROXY 3 (HYDROXYMETHYL)PHENYL)ETHYL)AMINO)DODECANAMIDO)ETHYLOXY)ETHOXY)ETHYLAMINO)FORMYL)PENTYL)ADENOSINE ACETATE; PERTUSSIS TOXIN; SALBUTAMOL; SALIGENIN; TRITIUM; UNCLASSIFIED DRUG;

ANIMAL CELL; ARTICLE; BINDING AFFINITY; CARBON NUCLEAR MAGNETIC RESONANCE; CELL CULTURE; CHEMICAL STRUCTURE; CONTROLLED STUDY; DRUG RECEPTOR BINDING; DRUG SELECTIVITY; ISOTOPE LABELING; LIGAND BINDING; NONHUMAN; PHARMACOPHORE; PRIORITY JOURNAL; PROTON NUCLEAR MAGNETIC RESONANCE; RECEPTOR AFFINITY; RECEPTOR CROSS TALK; SECOND MESSENGER; STRUCTURE ACTIVITY RELATION;

A1 ADENOSINE RECEPTORS; COMBINED PHARMACOPHORES; HETEROBIVALENT LIGANDS; STRUCTURE-ACTIVITY RELATIONSHIPS; Β2 ADRENERGIC RECEPTORS;

ADRENERGIC BETA-1 RECEPTOR AGONISTS; ANIMALS; CELL LINE; CRICETINAE; KINETICS; LIGANDS; PERTUSSIS TOXIN; PROTEIN BINDING; RECEPTOR CROSS-TALK; RECEPTORS, ADRENERGIC, BETA-1; RECEPTORS, ADRENERGIC, BETA-2; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 84889884758 PISSN: 18607179 EISSN: 18607187 Source Type: Journal
DOI: 10.1002/cmdc.201300286 Document Type: Article

Times cited : (9)

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