SCOPUS 정보 검색 플랫폼

Volumn 12, Issue 1, 2014, Pages 156-161

Reaction site-driven regioselective synthesis of AChE inhibitors

(12) Oueis, Emilia a Santoni, Gianluca b,c Ronco, Cyril a Syzgantseva, Olga a Tognetti, Vincent a Joubert, Laurent a Romieu, Anthony a Weik, Martin b,c Jean, Ludovic a Sabot, Cyrille a Nachon, Florian d Renard, Pierre Yves a

a UNIVERSITÉ DE ROUEN (France)

b INSTITUT DE BIOLOGIE STRUCTURALE (France)

c CEA GRENOBLE (France)

d INSTITUT DE RECHERCHE BIOMÉDICALE DES ARMÉES (France)

Author keywords

[No Author keywords available]

Indexed keywords

CHELATION; ENZYMES; REGIOSELECTIVITY; SYNTHESIS (CHEMICAL);

BIOLOGICAL TARGETS; BUILDING BLOCKES; CLICK CHEMISTRY; COMPUTATIONAL MODELLING; HUISGEN CYCLOADDITION; HUMAN ACETYLCHOLINESTERASE; MULTIDENTATE LIGANDS; REGIOSELECTIVE SYNTHESIS;

LIGANDS;

ACETYLCHOLINESTERASE; AMINOQUINOLINE DERIVATIVE; CHOLINESTERASE INHIBITOR; LIGAND; RECOMBINANT PROTEIN;

ARTICLE; CHEMICAL STRUCTURE; CHEMISTRY; CLICK CHEMISTRY; CYCLIZATION; HUMAN; METABOLISM; STEREOISOMERISM;

ACETYLCHOLINESTERASE; AMINOQUINOLINES; CHOLINESTERASE INHIBITORS; CLICK CHEMISTRY; CYCLIZATION; HUMANS; LIGANDS; MODELS, MOLECULAR; MOLECULAR STRUCTURE; RECOMBINANT PROTEINS; STEREOISOMERISM;

EID: 84889069748 PISSN: 14770520 EISSN: None Source Type: Journal
DOI: 10.1039/c3ob42109k Document Type: Article

Times cited : (27)

References (36)

1
- 0025117445
- D. Rideout T. Calogeropoulou J. Jaworski M. Mccarthy Biopolymers 1990 29 247 262
- (1990) Biopolymers , vol.29 , pp. 247-262
- Rideout, D.¹ Calogeropoulou, T.² Jaworski, J.³ McCarthy, M.⁴

2
- 77949816947
- G. E. Boldt T. J. Dicherson K. D. Janda Drug Discovery Today 2004 9 143 148
- (2004) Drug Discovery Today , vol.9 , pp. 143-148
- Boldt, G.E.¹ Dicherson, T.J.² Janda, K.D.³

3
- 1842635467
- A. V. Eliseev Drug Discovery Today 2004 9 348 349
- (2004) Drug Discovery Today , vol.9 , pp. 348-349
- Eliseev, A.V.¹

4
- 34447562439
- K. B. Sharpless R. Manetsh Expert Opin. Drug Discovery 2006 1 525 538
- (2006) Expert Opin. Drug Discovery , vol.1 , pp. 525-538
- Sharpless, K.B.¹ Manetsh, R.²

5
- 0037087516
- W. G. Lewis L. G. Green F. Grynszpan Z. Radič P. R. Carlier P. Taylor M. G. Finn K. B. Sharpless Angew. Chem., Int. Ed. 2002 41 1053 1057
- (2002) Angew. Chem., Int. Ed. , vol.41 , pp. 1053-1057
- Lewis, W.G.¹ Green, L.G.² Grynszpan, F.³ Radič, Z.⁴ Carlier, P.R.⁵ Taylor, P.⁶ Finn, M.G.⁷ Sharpless, K.B.⁸

6
- 5644276317
- R. Manetsch A. Krasinski Z. Radič J. Raushel P. Taylor K. B. Sharpless H. C. Kolb J. Am. Chem. Soc. 2004 126 12809 12818
- (2004) J. Am. Chem. Soc. , vol.126 , pp. 12809-12818
- Manetsch, R.¹ Krasinski, A.² Radič, Z.³ Raushel, J.⁴ Taylor, P.⁵ Sharpless, K.B.⁶ Kolb, H.C.⁷

7
- 77956609618
- T. Suzuki Y. Ota Y. Kasuya M. Mutsuga Y. Kawamura H. Tsumoto H. Nakagawa M. G. Finn N. Miyata Angew. Chem., Int. Ed. 2010 49 6817 6820
- (2010) Angew. Chem., Int. Ed. , vol.49 , pp. 6817-6820
- Suzuki, T.¹ Ota, Y.² Kasuya, Y.³ Mutsuga, M.⁴ Kawamura, Y.⁵ Tsumoto, H.⁶ Nakagawa, H.⁷ Finn, M.G.⁸ Miyata, N.⁹

8
- 84888995031
- T. Suzuki Y. Ota Y. Kasuya M. Mutsuga Y. Kawamura H. Tsumoto H. Nakagawa M. G. Finn N. Miyata Angew. Chem., Int. Ed. 2010 122 6969 6972
- (2010) Angew. Chem., Int. Ed. , vol.122 , pp. 6969-6972
- Suzuki, T.¹ Ota, Y.² Kasuya, Y.³ Mutsuga, M.⁴ Kawamura, Y.⁵ Tsumoto, H.⁶ Nakagawa, H.⁷ Finn, M.G.⁸ Miyata, N.⁹

9
- 77949786732
- S. K. Mamidyala M. G. Finn Chem. Soc. Rev. 2010 39 1252 1261
- (2010) Chem. Soc. Rev. , vol.39 , pp. 1252-1261
- Mamidyala, S.K.¹ Finn, M.G.²

10
- 77949858836
- X. Hu R. Manetsch Chem. Soc. Rev. 2010 39 1316 1324
- (2010) Chem. Soc. Rev. , vol.39 , pp. 1316-1324
- Hu, X.¹ Manetsch, R.²

11
- 80755172538
- S. W. Millward R. K. Henning G. A. Kwong S. M. Pitram H. D. Agnew K. M. Deyle A. Nag J. E. Hein S. S. Lee J. Lim J. A. Pfeilsticker K. B. Sharpless J. R. Heath J. Am. Chem. Soc. 2011 133 18280 18288
- (2011) J. Am. Chem. Soc. , vol.133 , pp. 18280-18288
- Millward, S.W.¹ Henning, R.K.² Kwong, G.A.³ Pitram, S.M.⁴ Agnew, H.D.⁵ Deyle, K.M.⁶ Nag, A.⁷ Hein, J.E.⁸ Lee, S.S.⁹ Lim, J.¹⁰ Pfeilsticker, J.A.¹¹ Sharpless, K.B.¹² Heath, J.R.¹³

12
- 84873976921
- C. Peruzzotti S. Borrelli M. Ventura R. Pantano G. Fumagalli M. S. Christodoulou D. Monticelli M. Luzzani A. L. Fallacara C. Tintori M. Botta D. Passarella ACS Med. Chem. Lett. 2013 4 274 277
- (2013) ACS Med. Chem. Lett. , vol.4 , pp. 274-277
- Peruzzotti, C.¹ Borrelli, S.² Ventura, M.³ Pantano, R.⁴ Fumagalli, G.⁵ Christodoulou, M.S.⁶ Monticelli, D.⁷ Luzzani, M.⁸ Fallacara, A.L.⁹ Tintori, C.¹⁰ Botta, M.¹¹ Passarella, D.¹²

13
- 84886810370
- W. Tieu T. P. Soares da Costa M. Y. Yap K. L. Keeling M. C. J. Wilce J. C. Wallace G. W. Booker S. W. Polyak A. D. Abell Chem. Sci. 2013 4 3533 3537
- (2013) Chem. Sci. , vol.4 , pp. 3533-3537
- Tieu, W.¹ Soares Da Costa, T.P.² Yap, M.Y.³ Keeling, K.L.⁴ Wilce, M.C.J.⁵ Wallace, J.C.⁶ Booker, G.W.⁷ Polyak, S.W.⁸ Abell, A.D.⁹

14
- 84877873373
- P. Anand B. Singh Arch. Pharmacal. Res. 2013 36 375 399
- (2013) Arch. Pharmacal. Res. , vol.36 , pp. 375-399
- Anand, P.¹ Singh, B.²

15
- 18644384979
- A. Krasinski Z. Radič R. Manetsch J. Raushel P. Taylor K. B. Sharpless H. C. Kolb J. Am. Chem. Soc. 2005 127 6686 6692
- (2005) J. Am. Chem. Soc. , vol.127 , pp. 6686-6692
- Krasinski, A.¹ Radič, Z.² Manetsch, R.³ Raushel, J.⁴ Taylor, P.⁵ Sharpless, K.B.⁶ Kolb, H.C.⁷

16
- 1242342257
- Y. Bourne H. C. Kolbe Z. Radic K. B. Sharpless P. Taylor P. Marchot Proc. Natl. Acad. Sci. U. S. A. 2004 101 1449 1454
- (2004) Proc. Natl. Acad. Sci. U. S. A. , vol.101 , pp. 1449-1454
- Bourne, Y.¹ Kolbe, H.C.² Radic, Z.³ Sharpless, K.B.⁴ Taylor, P.⁵ Marchot, P.⁶

17
- 33746210083
- M. Whiting J. Muldoon Y.-C. Lin S. M. Silverman W. Lindstrom A. J. Olson H. C. Kolb M. G. Finn K. B. Sharpless J. H. Elder V. V. Fokin Angew. Chem., Int. Ed. 2006 45 1435 1439
- (2006) Angew. Chem., Int. Ed. , vol.45 , pp. 1435-1439
- Whiting, M.¹ Muldoon, J.² Lin, Y.-C.³ Silverman, S.M.⁴ Lindstrom, W.⁵ Olson, A.J.⁶ Kolb, H.C.⁷ Finn, M.G.⁸ Sharpless, K.B.⁹ Elder, J.H.¹⁰ Fokin, V.V.¹¹

18
- 11244252206
- V. P. Mocharla B. Colasson L. V. Lee S. Röper K. B. Sharpless C.-H. Wong H. C. Kolb Angew. Chem., Int. Ed. 2005 44 116 120
- (2005) Angew. Chem., Int. Ed. , vol.44 , pp. 116-120
- Mocharla, V.P.¹ Colasson, B.² Lee, L.V.³ Röper, S.⁴ Sharpless, K.B.⁵ Wong, C.-H.⁶ Kolb, H.C.⁷

19
- 78649645179
- N. Willand M. Desroses P. Toto B. Dirié Z. Lens V. Villeret P. Rucktooa C. Locht A. Baulard B. Deprez ACS Chem. Biol. 2010 5 1007 1013
- (2010) ACS Chem. Biol. , vol.5 , pp. 1007-1013
- Willand, N.¹ Desroses, M.² Toto, P.³ Dirié, B.⁴ Lens, Z.⁵ Villeret, V.⁶ Rucktooa, P.⁷ Locht, C.⁸ Baulard, A.⁹ Deprez, B.¹⁰

20
- 84859994538
- N. P. Grimster B. Stump J. R. Fotsing T. Weide T. T. Talley J. G. Yamauchi Á. Nemecz C. Kim K.-Y. Ho K. B. Sharpless P. Taylor V. V. Fokin J. Am. Chem. Soc. 2012 134 6732 6740
- (2012) J. Am. Chem. Soc. , vol.134 , pp. 6732-6740
- Grimster, N.P.¹ Stump, B.² Fotsing, J.R.³ Weide, T.⁴ Talley, T.T.⁵ Yamauchi, J.G.⁶ Nemecz, Á.⁷ Kim, C.⁸ Ho, K.-Y.⁹ Sharpless, K.B.¹⁰ Taylor, P.¹¹ Fokin, V.V.¹²

21
- 84857720222
- C. Ronco E. Carletti J.-P. Colletier M. Weik F. Nachon L. Jean P.-Y. Renard ChemMedChem 2012 7 400 405
- (2012) ChemMedChem , vol.7 , pp. 400-405
- Ronco, C.¹ Carletti, E.² Colletier, J.-P.³ Weik, M.⁴ Nachon, F.⁵ Jean, L.⁶ Renard, P.-Y.⁷

22
- 13044253491
- P. Camps R. El Achab D. M. Görbig J. Morral D. Muñoz-Torrero A. Badia J. E. Baños N. M. Vivas X. Barril M. Orozco F. J. Luque J. Med. Chem. 1999 42 3227 3242
- (1999) J. Med. Chem. , vol.42 , pp. 3227-3242
- Camps, P.¹ El Achab, R.² Görbig, D.M.³ Morral, J.⁴ Muñoz-Torrero, D.⁵ Badia, A.⁶ Baños, J.E.⁷ Vivas, N.M.⁸ Barril, X.⁹ Orozco, M.¹⁰ Luque, F.J.¹¹

23
- 0034736034
- P. Camps R. El Achab J. Morral D. Muñoz-Torrero A. Badia J. E. Baños N. M. Vivas X. Barril M. Orozco F. J. Luque J. Med. Chem. 2000 43 4657 4666
- (2000) J. Med. Chem. , vol.43 , pp. 4657-4666
- Camps, P.¹ El Achab, R.² Morral, J.³ Muñoz-Torrero, D.⁴ Badia, A.⁵ Baños, J.E.⁶ Vivas, N.M.⁷ Barril, X.⁸ Orozco, M.⁹ Luque, F.J.¹⁰

24
- 66449109554
- C. Ronco G. Sorin F. Nachon R. Foucault L. Jean A. Romieu P.-Y. Renard Bioorg. Med. Chem. 2009 17 4523 4536
- (2009) Bioorg. Med. Chem. , vol.17 , pp. 4523-4536
- Ronco, C.¹ Sorin, G.² Nachon, F.³ Foucault, R.⁴ Jean, L.⁵ Romieu, A.⁶ Renard, P.-Y.⁷

25
- 77955850312
- C. Ronco L. Jean P.-Y. Renard Tetrahedron 2010 66 7399 7404
- (2010) Tetrahedron , vol.66 , pp. 7399-7404
- Ronco, C.¹ Jean, L.² Renard, P.-Y.³

26
- 78650901081
- C. Ronco L. Jean H. Outaabout P.-Y. Renard Eur. J. Org. Chem. 2011 302 310
- (2011) Eur. J. Org. Chem. , pp. 302-310
- Ronco, C.¹ Jean, L.² Outaabout, H.³ Renard, P.-Y.⁴

27
- 79955068835
- C. Ronco R. Foucault E. Gillon P. Bohn F. Nachon L. Jean P.-Y. Renard ChemMedChem 2011 6 876 888
- (2011) ChemMedChem , vol.6 , pp. 876-888
- Ronco, C.¹ Foucault, R.² Gillon, E.³ Bohn, P.⁴ Nachon, F.⁵ Jean, L.⁶ Renard, P.-Y.⁷

28
- 84880070992
- F. Nachon E. Carletti C. Ronco M. Trovaslet Y. Nicolet L. Jean P.-Y. Renard Biochem. J. 2013 453 393 399
- (2013) Biochem. J. , vol.453 , pp. 393-399
- Nachon, F.¹ Carletti, E.² Ronco, C.³ Trovaslet, M.⁴ Nicolet, Y.⁵ Jean, L.⁶ Renard, P.-Y.⁷

29
- 39149091398
- A. Cavalli M. L. Bolognesi A. Minarini M. Rosini V. Tumiatti M. Recanatini C. Melchiorre J. Med. Chem. 2008 51 347 371
- (2008) J. Med. Chem. , vol.51 , pp. 347-371
- Cavalli, A.¹ Bolognesi, M.L.² Minarini, A.³ Rosini, M.⁴ Tumiatti, V.⁵ Recanatini, M.⁶ Melchiorre, C.⁷

30
- 15444378025
- P. Camps X. Formosa D. Muñoz-Torrero J. Petrignet A. Badia M. V. Clos J. Med. Chem. 2005 48 1701 1704
- (2005) J. Med. Chem. , vol.48 , pp. 1701-1704
- Camps, P.¹ Formosa, X.² Muñoz-Torrero, D.³ Petrignet, J.⁴ Badia, A.⁵ Clos, M.V.⁶

31
- 45749135895
- P. Camps X. Formosa C. Galdeano T. Gómez D. Muñoz-Torrero M. Scarpellini E. Viayna A. Badia M. V. Clos A. Camins M. Pallàs M. Bartolini F. Mancini V. Andrisano J. Estelrich M. Lizondo A. Bidon-Chanal F. J. Luque J. Med. Chem. 2008 51 3588 3598
- (2008) J. Med. Chem. , vol.51 , pp. 3588-3598
- Camps, P.¹ Formosa, X.² Galdeano, C.³ Gómez, T.⁴ Muñoz-Torrero, D.⁵ Scarpellini, M.⁶ Viayna, E.⁷ Badia, A.⁸ Clos, M.V.⁹ Camins, A.¹⁰ Pallàs, M.¹¹ Bartolini, M.¹² Mancini, F.¹³ Andrisano, V.¹⁴ Estelrich, J.¹⁵ Lizondo, M.¹⁶ Bidon-Chanal, A.¹⁷ Luque, F.J.¹⁸

32
- 78349232410
- E. Viayna T. Gómez C. Galdeano L. Ramírez M. Ratia A. Badia M. V. Clos E. Verdaguer F. Junyent A. Camins M. Pallàs M. Bartolini F. Mancini V. Andrisano M. P. Arce M. I. Rodríguez-Franco A. Bidon-Chanal F. J. Luque P. Camps D. Muñoz-Torrero ChemMedChem 2010 5 1855 1870
- (2010) ChemMedChem , vol.5 , pp. 1855-1870
- Viayna, E.¹ Gómez, T.² Galdeano, C.³ Ramírez, L.⁴ Ratia, M.⁵ Badia, A.⁶ Clos, M.V.⁷ Verdaguer, E.⁸ Junyent, F.⁹ Camins, A.¹⁰ Pallàs, M.¹¹ Bartolini, M.¹² Mancini, F.¹³ Andrisano, V.¹⁴ Arce, M.P.¹⁵ Rodríguez-Franco, M.I.¹⁶ Bidon-Chanal, A.¹⁷ Luque, F.J.¹⁸ Camps, P.¹⁹ Muñoz-Torrero, D.²⁰ more..

33
- 84860376939
- J. Peters M. Trovaslet M. Trapp F. Nachon F. Hill E. Royer F. Gabel L. van Eijck P. Masson M. Tehei Phys. Chem. Chem. Phys. 2012 19 6764 6770
- (2012) Phys. Chem. Chem. Phys. , vol.19 , pp. 6764-6770
- Peters, J.¹ Trovaslet, M.² Trapp, M.³ Nachon, F.⁴ Hill, F.⁵ Royer, E.⁶ Gabel, F.⁷ Van Eijck, L.⁸ Masson, P.⁹ Tehei, M.¹⁰

34
- 84875806859
- M. Trovaslet M. Trapp M. Weik F. Nachon P. Masson M. Tehei J. Peters Chem.-Biol. Interact. 2013 1 14 18
- (2013) Chem.-Biol. Interact. , vol.1 , pp. 14-18
- Trovaslet, M.¹ Trapp, M.² Weik, M.³ Nachon, F.⁴ Masson, P.⁵ Tehei, M.⁶ Peters, J.⁷

35
- 50649094935
- Z. Radič R. Manetsch D. Fournier K. B. Sharpless P. Taylor Chem. Biol. Interact. 2008 175 161 165
- (2008) Chem. Biol. Interact. , vol.175 , pp. 161-165
- Radič, Z.¹ Manetsch, R.² Fournier, D.³ Sharpless, K.B.⁴ Taylor, P.⁵

36
- 33750139049
- S. Senapati Y. Cheng J. A. McCammon J. Med. Chem. 2006 49 6222 6230
- (2006) J. Med. Chem. , vol.49 , pp. 6222-6230
- Senapati, S.¹ Cheng, Y.² McCammon, J.A.³

* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.