Structural and biophysical characterisation of G protein-coupled receptor ligand binding using resonance energy transfer and fluorescent labelling techniques

Biochimica et Biophysica Acta - Biomembranes

Volumn 1838, Issue 1 PARTA, 2014, Pages 3-14

  Ward, Richard J ^a   Milligan, Graeme ^a  

^a UNIVERSITY OF GLASGOW   (United Kingdom)

Author keywords

FlAsH labelling; Fluorescent ligand; FRET sensor; G protein coupled receptor; Ligand binding

Indexed keywords

FLUORESCENT DYE; G PROTEIN COUPLED RECEPTOR; LIGAND; PROTEIN SERINE THREONINE KINASE;

BIOSENSOR; CELL MEMBRANE; CONFORMATIONAL TRANSITION; DRUG DESIGN; DRUG IDENTIFICATION; DRUG TARGETING; ENERGY TRANSFER; FLUORESCENCE ANALYSIS; FLUORESCENCE RESONANCE ENERGY TRANSFER; HUMAN; INTERMETHOD COMPARISON; ISOTOPE LABELING; LIGAND BINDING; MICROSCOPY; NONHUMAN; PRIORITY JOURNAL; PROTEIN STABILITY; RECEPTOR BINDING; RECEPTOR LIGAND INTERACTION; RESONANCE ENERGY TRANSFER; REVIEW; SIGNAL TRANSDUCTION; STRUCTURE BASED LIGAND DESIGN; X RAY CRYSTALLOGRAPHY;

FLASH LABELLING; FLUORESCENT LIGAND; FRET SENSOR; G PROTEIN-COUPLED RECEPTOR; LIGAND BINDING;

BIOPHYSICS; CRYSTALLOGRAPHY, X-RAY; FLUORESCENCE RESONANCE ENERGY TRANSFER; FLUORESCENT DYES; LIGANDS; PROTEIN BINDING; PROTEIN CONFORMATION; RECEPTORS, G-PROTEIN-COUPLED;

EID: 84888376322     PISSN: 00052736     EISSN: 18792642     Source Type: Journal    
DOI: 10.1016/j.bbamem.2013.04.007     Document Type: Review

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