SCOPUS 정보 검색 플랫폼

MedChemComm

Volumn 2, Issue 10, 2011, Pages 1011-1015

Design, synthesis and antiproliferative activity of urocanic-chalcone hybrid derivatives

(5) Ciupa, Alexander a Griffiths, Natalie J a Light, Stephanie K a Wood, Pauline J a Caggiano, Lorenzo a

a University of Bath (United Kingdom)

Author keywords

[No Author keywords available]

Indexed keywords

ANTINEOPLASTIC AGENT; DOXORUBICIN; UNCLASSIFIED DRUG; UROCANIC CHALCONE HYBRID DERIVATIVE;

ANTIPROLIFERATIVE ACTIVITY; ARTICLE; BREAST CARCINOMA; CELL PROLIFERATION; CELL STRAIN HT29; COLON CANCER; CONTROLLED STUDY; DRUG ACTIVITY; DRUG DESIGN; DRUG POTENCY; DRUG STRUCTURE; DRUG SYNTHESIS; HUMAN; HUMAN CELL; IC 50; METASTASIS POTENTIAL; PRIORITY JOURNAL;

EID: 80053595120 PISSN: 20402503 EISSN: 20402511 Source Type: Journal
DOI: 10.1039/c1md00155h Document Type: Article

Times cited : (17)

References (55)

1
- 80053595136
- US Patent 5473057
- W. H. Fenical, P. R. Jensen and T. Lindel, 1995, US Patent 5473057
- (1995)
- Fenical, W.H.¹ Jensen, P.R.² Lindel, T.³

2
- 0030984058
- T. Lindel P. R. Jensen W. Fenical B. H. Long A. M. Casazza J. Carboni C. R. Fairchild J. Am. Chem. Soc. 1997 119 8744
- (1997) J. Am. Chem. Soc. , vol.119 , pp. 8744
- Lindel, T.¹ Jensen, P.R.² Fenical, W.³ Long, B.H.⁴ Casazza, A.M.⁵ Carboni, J.⁶ Fairchild, C.R.⁷

3
- 84928704587
- M. D'Ambrosio A. Guerriero F. Pietra Helv. Chim. Acta 1987 70 2019
- (1987) Helv. Chim. Acta , vol.70 , pp. 2019
- D'Ambrosio, M.¹ Guerriero, A.² Pietra, F.³

4
- 84986348031
- M. D'Ambrosio A. Guerriero F. Pietra Helv. Chim. Acta 1988 71 964
- (1988) Helv. Chim. Acta , vol.71 , pp. 964
- D'Ambrosio, M.¹ Guerriero, A.² Pietra, F.³

5
- 0002551688
- M. Ciomei C. Albanese W. Pastori M. Grandi F. Pietra M. D'Ambrosio A. Guerriero C. Battistini Proc. Amer. Ass. Can. Res. 1997 38 5
- (1997) Proc. Amer. Ass. Can. Res. , vol.38 , pp. 5
- Ciomei, M.¹ Albanese, C.² Pastori, W.³ Grandi, M.⁴ Pietra, F.⁵ D'Ambrosio, M.⁶ Guerriero, A.⁷ Battistini, C.⁸

6
- 33947717002
- K.-H. Altmann J. Gertsch Nat. Prod. Rep. 2007 24 327
- (2007) Nat. Prod. Rep. , vol.24 , pp. 327
- Altmann, K.-H.¹ Gertsch, J.²

7
- 67649344837
- Y. Zhao W.-S. Fang K. Pors Expert Opin. Ther. Pat. 2009 19 607
- (2009) Expert Opin. Ther. Pat. , vol.19 , pp. 607
- Zhao, Y.¹ Fang, W.-S.² Pors, K.³

8
- 0032862624
- K. C. Nicolaou J. Pfefferkorn J. Xu N. Winssinger T. Ohshima S. Kim S. Hosokawa D. Vourloumis F. van Delft T. Li Chem. Pharm. Bull. 1999 47 1199
- (1999) Chem. Pharm. Bull. , vol.47 , pp. 1199
- Nicolaou, K.C.¹ Pfefferkorn, J.² Xu, J.³ Winssinger, N.⁴ Ohshima, T.⁵ Kim, S.⁶ Hosokawa, S.⁷ Vourloumis, D.⁸ Van Delft, F.⁹ Li, T.¹⁰

9
- 0032520890
- B. H. Long J. M. Carboni A. J. Wasserman L. A. Cornell A. M. Casazza P. R. Jensen T. Lindel W. Fenical C. R. Fairchild Cancer Res. 1998 58 1111
- (1998) Cancer Res. , vol.58 , pp. 1111
- Long, B.H.¹ Carboni, J.M.² Wasserman, A.J.³ Cornell, L.A.⁴ Casazza, A.M.⁵ Jensen, P.R.⁶ Lindel, T.⁷ Fenical, W.⁸ Fairchild, C.R.⁹

10
- 0033609037
- E. Hamel D. L. Sackett D. Vourloumis K. C. Nicolaou Biochemistry 1999 38 5490
- (1999) Biochemistry , vol.38 , pp. 5490
- Hamel, E.¹ Sackett, D.L.² Vourloumis, D.³ Nicolaou, K.C.⁴

11
- 0031470265
- K. C. Nicolaou F. van Delft T. Ohshima D. Vourloumis J. Xu S. Hosokawa J. Pfefferkorn S. Kim T. Li Angew. Chem., Int. Ed. Engl. 1997 36 2520
- (1997) Angew. Chem., Int. Ed. Engl. , vol.36 , pp. 2520
- Nicolaou, K.C.¹ Van Delft, F.² Ohshima, T.³ Vourloumis, D.⁴ Xu, J.⁵ Hosokawa, S.⁶ Pfefferkorn, J.⁷ Kim, S.⁸ Li, T.⁹

12
- 0032475452
- K. C. Nicolaou T. Ohshima S. Hosokawa F. L. van Delft D. Vourloumis J. Y. Xu J. Pfefferkorn S. Kim J. Am. Chem. Soc. 1998 120 8674
- (1998) J. Am. Chem. Soc. , vol.120 , pp. 8674
- Nicolaou, K.C.¹ Ohshima, T.² Hosokawa, S.³ Van Delft, F.L.⁴ Vourloumis, D.⁵ Xu, J.Y.⁶ Pfefferkorn, J.⁷ Kim, S.⁸

13
- 0031882649
- X.-T. Chen C. E. Gutteridge S. K. Bhattacharya B. Zhou T. R. R. Pettus T. Hascall S. J. Danishefsky Angew. Chem., Int. Ed. 1998 37 185
- (1998) Angew. Chem., Int. Ed. , vol.37 , pp. 185
- Chen, X.-T.¹ Gutteridge, C.E.² Bhattacharya, S.K.³ Zhou, B.⁴ Pettus, T.R.R.⁵ Hascall, T.⁶ Danishefsky, S.J.⁷

14
- 0031924818
- X.-T. Chen B. Zhou S. K. Bhattacharya C. E. Gutteridge T. R. R. Pettus S. J. Danishefsky Angew. Chem., Int. Ed. 1998 37 789
- (1998) Angew. Chem., Int. Ed. , vol.37 , pp. 789
- Chen, X.-T.¹ Zhou, B.² Bhattacharya, S.K.³ Gutteridge, C.E.⁴ Pettus, T.R.R.⁵ Danishefsky, S.J.⁶

15
- 0030723674
- K. C. Nicolaou J. Y. Xu S. Kim T. Ohshima S. Hosokawa J. Pfefferkorn J. Am. Chem. Soc. 1997 119 11353
- (1997) J. Am. Chem. Soc. , vol.119 , pp. 11353
- Nicolaou, K.C.¹ Xu, J.Y.² Kim, S.³ Ohshima, T.⁴ Hosokawa, S.⁵ Pfefferkorn, J.⁶

16
- 0032475416
- K. C. Nicolaou J. Y. Xu S. Kim J. Pfefferkorn T. Ohshima D. Vourloumis S. Hosokawa J. Am. Chem. Soc. 1998 120 8661
- (1998) J. Am. Chem. Soc. , vol.120 , pp. 8661
- Nicolaou, K.C.¹ Xu, J.Y.² Kim, S.³ Pfefferkorn, J.⁴ Ohshima, T.⁵ Vourloumis, D.⁶ Hosokawa, S.⁷

17
- 0032486436
- K. C. Nicolaou S. Kim J. Pfefferkorn J. Xu T. Ohshima S. Hosokawa D. Vourloumis T. Li Angew. Chem., Int. Ed. 1998 37 1418
- (1998) Angew. Chem., Int. Ed. , vol.37 , pp. 1418
- Nicolaou, K.C.¹ Kim, S.² Pfefferkorn, J.³ Xu, J.⁴ Ohshima, T.⁵ Hosokawa, S.⁶ Vourloumis, D.⁷ Li, T.⁸

18
- 0032576190
- K. C. Nicolaou N. Winssinger D. Vourloumis T. Ohshima S. Kim J. Pfefferkorn J. Y. Xu T. Li J. Am. Chem. Soc. 1998 120 10814
- (1998) J. Am. Chem. Soc. , vol.120 , pp. 10814
- Nicolaou, K.C.¹ Winssinger, N.² Vourloumis, D.³ Ohshima, T.⁴ Kim, S.⁵ Pfefferkorn, J.⁶ Xu, J.Y.⁷ Li, T.⁸

19
- 0035944995
- J. Telser R. Beumer A. A. Bell S. M. Ceccarelli D. Monti C. Gennari Tetrahedron Lett. 2001 42 9187
- (2001) Tetrahedron Lett. , vol.42 , pp. 9187
- Telser, J.¹ Beumer, R.² Bell, A.A.³ Ceccarelli, S.M.⁴ Monti, D.⁵ Gennari, C.⁶

20
- 0037454986
- R. Beumer P. Bayón P. Bugada S. Ducki N. Mongelli F. R. Sirtori J. Telser C. Gennari Tetrahedron Lett. 2003 44 681
- (2003) Tetrahedron Lett. , vol.44 , pp. 681
- Beumer, R.¹ Bayón, P.² Bugada, P.³ Ducki, S.⁴ Mongelli, N.⁵ Sirtori, F.R.⁶ Telser, J.⁷ Gennari, C.⁸

21
- 0141961790
- R. Beumer P. Bayón P. Bugada S. Ducki N. Mongelli F. R. Sirtori J. Telser C. Gennari Tetrahedron 2003 59 8803
- (2003) Tetrahedron , vol.59 , pp. 8803
- Beumer, R.¹ Bayón, P.² Bugada, P.³ Ducki, S.⁴ Mongelli, N.⁵ Sirtori, F.R.⁶ Telser, J.⁷ Gennari, C.⁸

22
- 0141760258
- L. Caggiano D. Castoldi R. Beumer P. Bayón J. Tesler C. Gennari Tetrahedron Lett. 2003 44 7913
- (2003) Tetrahedron Lett. , vol.44 , pp. 7913
- Caggiano, L.¹ Castoldi, D.² Beumer, R.³ Bayón, P.⁴ Tesler, J.⁵ Gennari, C.⁶

23
- 13444273184
- D. Castoldi L. Caggiano P. Bayón A. M. Costa P. Cappella O. Sharon C. Gennari Tetrahedron 2005 61 2123
- (2005) Tetrahedron , vol.61 , pp. 2123
- Castoldi, D.¹ Caggiano, L.² Bayón, P.³ Costa, A.M.⁴ Cappella, P.⁵ Sharon, O.⁶ Gennari, C.⁷

24
- 13244291529
- D. Castoldi L. Caggiano L. Panigada O. Sharon A. M. Costa C. Gennari Angew. Chem., Int. Ed. 2005 44 588
- (2005) Angew. Chem., Int. Ed. , vol.44 , pp. 588
- Castoldi, D.¹ Caggiano, L.² Panigada, L.³ Sharon, O.⁴ Costa, A.M.⁵ Gennari, C.⁶

25
- 29344446565
- D. Castoldi L. Caggiano L. Panigada O. Sharon A. M. Costa C. Gennari Chem.-Eur. J. 2006 12 51
- (2006) Chem.-Eur. J. , vol.12 , pp. 51
- Castoldi, D.¹ Caggiano, L.² Panigada, L.³ Sharon, O.⁴ Costa, A.M.⁵ Gennari, C.⁶

26
- 17444408490
- G. C. H. Chiang A. D. Bond A. Ayscough G. Pain S. Ducki A. B. Holmes Chem. Commun. 2005 1860
- (2005) Chem. Commun. , pp. 1860
- Chiang, G.C.H.¹ Bond, A.D.² Ayscough, A.³ Pain, G.⁴ Ducki, S.⁵ Holmes, A.B.⁶

27
- 65549108181
- S. Y. Frankie Mak G. C. H. Chiang J. E. P. Davidson J. E. Davies A. Ayscough G. Pain J. W. Burton A. B. Holmes Tetrahedron: Asymmetry 2009 20 921
- (2009) Tetrahedron: Asymmetry , vol.20 , pp. 921
- Frankie Mak, S.Y.¹ Chiang, G.C.H.² Davidson, J.E.P.³ Davies, J.E.⁴ Ayscough, A.⁵ Pain, G.⁶ Burton, J.W.⁷ Holmes, A.B.⁸

28
- 77950854525
- D. I. Batovska I. T. Todorova Curr. Clin. Pharmacol. 2010 5 1
- (2010) Curr. Clin. Pharmacol. , vol.5 , pp. 1
- Batovska, D.I.¹ Todorova, I.T.²

29
- 0030014602
- C. W. G. Fishwick R. J. Foster R. E. Carr Tetrahedron Lett. 1996 37 3915
- (1996) Tetrahedron Lett. , vol.37 , pp. 3915
- Fishwick, C.W.G.¹ Foster, R.J.² Carr, R.E.³

30
- 0030006607
- R. W. Hartmann M. Frotscher D. Ledergerber G. A. Wächter G. L. Grün T. F. Sergejew Arch. Pharm. 1996 329 251
- (1996) Arch. Pharm. , vol.329 , pp. 251
- Hartmann, R.W.¹ Frotscher, M.² Ledergerber, D.³ Wächter, G.A.⁴ Grün, G.L.⁵ Sergejew, T.F.⁶

31
- 0030059847
- G. A. Wächter R. W. Hartmann T. Sergejew G. L. Grün D. Ledergerber J. Med. Chem. 1996 39 834
- (1996) J. Med. Chem. , vol.39 , pp. 834
- Wächter, G.A.¹ Hartmann, R.W.² Sergejew, T.³ Grün, G.L.⁴ Ledergerber, D.⁵

32
- 80053590272
- R. W. Hartmann, B. Wachall, M. Yoshihama, M. Nakakoshi, S. Nomoto and Y. Ikeda, 2003, US 6559157
- R. W. Hartmann, B. Wachall, M. Yoshihama, M. Nakakoshi, S. Nomoto and Y. Ikeda, 2003, US 6559157

33
- 0036238085
- M. Recanatini A. Cavalli P. Valenti Med. Res. Rev. 2002 22 282
- (2002) Med. Res. Rev. , vol.22 , pp. 282
- Recanatini, M.¹ Cavalli, A.² Valenti, P.³

34
- 0036848634
- S. Grubjesic R. M. Moriarty J. M. Pezzuto Expert Opin. Ther. Pat. 2002 12 1647
- (2002) Expert Opin. Ther. Pat. , vol.12 , pp. 1647
- Grubjesic, S.¹ Moriarty, R.M.² Pezzuto, J.M.³

35
- 80053598181
- D. W. Gil and J. E. Donello, 2003, WO 03/099289
- D. W. Gil and J. E. Donello, 2003, WO 03/099289

36
- 80053598933
- K. Chow, T. Heidelbaugh, D. Gil, M. Garst, L. A. Wheeler, P. X. Nguyen and D. G. Gomez, 2003, WO 03/099795
- K. Chow, T. Heidelbaugh, D. Gil, M. Garst, L. A. Wheeler, P. X. Nguyen and D. G. Gomez, 2003, WO 03/099795

37
- 10344262032
- L. M. Ni C. Q. Meng J. A. Sikorski Expert Opin. Ther. Pat. 2004 14 1669
- (2004) Expert Opin. Ther. Pat. , vol.14 , pp. 1669
- Ni, L.M.¹ Meng, C.Q.² Sikorski, J.A.³

38
- 71849101913
- Y. K. Rao S.-H. Fang Y.-M. Tzeng Bioorg. Med. Chem. 2009 17 7909
- (2009) Bioorg. Med. Chem. , vol.17 , pp. 7909
- Rao, Y.K.¹ Fang, S.-H.² Tzeng, Y.-M.³

39
- 72049087235
- S. Ducki D. Rennison M. Woo A. Kendall J. F. D. Chabert A. T. McGown N. J. Lawrence Bioorg. Med. Chem. 2009 17 7698
- (2009) Bioorg. Med. Chem. , vol.17 , pp. 7698
- Ducki, S.¹ Rennison, D.² Woo, M.³ Kendall, A.⁴ Chabert, J.F.D.⁵ McGown, A.T.⁶ Lawrence, N.J.⁷

40
- 77954316234
- D. Kumar N. M. Kumar K. Akamatsu E. Kusaka H. Harada T. Ito Bioorg. Med. Chem. Lett. 2010 20 3916
- (2010) Bioorg. Med. Chem. Lett. , vol.20 , pp. 3916
- Kumar, D.¹ Kumar, N.M.² Akamatsu, K.³ Kusaka, E.⁴ Harada, H.⁵ Ito, T.⁶

41
- 64049097460
- A. L. Risinger F. J. Giles S. L. Mooberry Cancer Treat. Rev. 2009 35 255
- (2009) Cancer Treat. Rev. , vol.35 , pp. 255
- Risinger, A.L.¹ Giles, F.J.² Mooberry, S.L.³

42
- 33744820579
- G. C. Tron T. Pirali G. Sorba F. Pagliai S. Busacca A. A. Genazzani J. Med. Chem. 2006 49 3033
- (2006) J. Med. Chem. , vol.49 , pp. 3033
- Tron, G.C.¹ Pirali, T.² Sorba, G.³ Pagliai, F.⁴ Busacca, S.⁵ Genazzani, A.A.⁶

43
- 0027330403
- D. L. Sackett Pharmacol. Ther. 1993 59 163
- (1993) Pharmacol. Ther. , vol.59 , pp. 163
- Sackett, D.L.¹

44
- 25844502482
- V. Srivastava A. S. Negi J. K. Kumar M. M. Gupta S. P. S. Khanuja Bioorg. Med. Chem. 2005 13 5892
- (2005) Bioorg. Med. Chem. , vol.13 , pp. 5892
- Srivastava, V.¹ Negi, A.S.² Kumar, J.K.³ Gupta, M.M.⁴ Khanuja, S.P.S.⁵

45
- 65549090459
- D. W. Siemann D. J. Chaplin P. A. Walicke Expert Opin. Invest. Drugs 2009 18 189
- (2009) Expert Opin. Invest. Drugs , vol.18 , pp. 189
- Siemann, D.W.¹ Chaplin, D.J.² Walicke, P.A.³

46
- 33745713018
- J. Bourdron L. Commeiras P. Barbier V. Bourgarel-Rey E. Pasquier N. Vanthuyne J. C. Hubaud V. Peyrot J. L. Parrain Bioorg. Med. Chem. 2006 14 5540
- (2006) Bioorg. Med. Chem. , vol.14 , pp. 5540
- Bourdron, J.¹ Commeiras, L.² Barbier, P.³ Bourgarel-Rey, V.⁴ Pasquier, E.⁵ Vanthuyne, N.⁶ Hubaud, J.C.⁷ Peyrot, V.⁸ Parrain, J.L.⁹

47
- 77950939804
- M. P. Leese F. Jourdan M. R. Kimberley G. E. Cozier N. Thiyagarajan C. Stengel S. Regis-Lydi P. A. Foster S. P. Newman K. R. Acharya E. Ferrandis A. Purohit M. J. Reed B. V. L. Potter Chem. Commun. 2010 46 2907
- (2010) Chem. Commun. , vol.46 , pp. 2907
- Leese, M.P.¹ Jourdan, F.² Kimberley, M.R.³ Cozier, G.E.⁴ Thiyagarajan, N.⁵ Stengel, C.⁶ Regis-Lydi, S.⁷ Foster, P.A.⁸ Newman, S.P.⁹ Acharya, K.R.¹⁰ Ferrandis, E.¹¹ Purohit, A.¹² Reed, M.J.¹³ Potter, B.V.L.¹⁴

48
- 77950654528
- E. C. Breen J. J. Walsh Curr. Med. Chem. 2010 17 609
- (2010) Curr. Med. Chem. , vol.17 , pp. 609
- Breen, E.C.¹ Walsh, J.J.²

49
- 34547583281
- Z. Wang E. M. Bennett D. J. Wilson C. Salomon R. Vince J. Med. Chem. 2007 50 3416
- (2007) J. Med. Chem. , vol.50 , pp. 3416
- Wang, Z.¹ Bennett, E.M.² Wilson, D.J.³ Salomon, C.⁴ Vince, R.⁵

50
- 79551489157
- H. S. Bodiwala S. Sabde P. Gupta R. Mukherjee R. Kumar P. Garg K. K. Bhutani D. Mitra I. P. Singh Bioorg. Med. Chem. 2011 19 1256
- (2011) Bioorg. Med. Chem. , vol.19 , pp. 1256
- Bodiwala, H.S.¹ Sabde, S.² Gupta, P.³ Mukherjee, R.⁴ Kumar, R.⁵ Garg, P.⁶ Bhutani, K.K.⁷ Mitra, D.⁸ Singh, I.P.⁹

51
- 31044435734
- S. Bhagat R. Sharma D. M. Sawant L. Sharma A. K. Chakraborti J. Mol. Catal. A: Chem. 2006 244 20
- (2006) J. Mol. Catal. A: Chem. , vol.244 , pp. 20
- Bhagat, S.¹ Sharma, R.² Sawant, D.M.³ Sharma, L.⁴ Chakraborti, A.K.⁵

52
- 67650318246
- N. M. Rateb H. F. Zohdi Synth. Commun. 2009 39 2789
- (2009) Synth. Commun. , vol.39 , pp. 2789
- Rateb, N.M.¹ Zohdi, H.F.²

53
- 34047174521
- T. Narender K. Papi Reddy Tetrahedron Lett. 2007 48 3177
- (2007) Tetrahedron Lett. , vol.48 , pp. 3177
- Narender, T.¹ Papi Reddy, K.²

54
- 0001269610
- MTS is 3-(4,5-dimethylthiazol-2-yl)-5-(3-carboxymethoxyphenyl)-2-(4- sulfophenyl)-2H-tetrazolium
- N. Lauth-de Viguerie N. Sergueeva M. Damiot H. Mawlawi M. Riviere A. Lattes Heterocycles 1994 37 1561
- (1994) Heterocycles , vol.37 , pp. 1561
- Lauth-De Viguerie, N.¹ Sergueeva, N.² Damiot, M.³ Mawlawi, H.⁴ Riviere, M.⁵ Lattes, A.⁶

55
- 0025899234
- A. H. Cory T. C. Owen J. A. Barltrop J. G. Cory Cancer Commun. 1991 3 207
- (1991) Cancer Commun. , vol.3 , pp. 207
- Cory, A.H.¹ Owen, T.C.² Barltrop, J.A.³ Cory, J.G.⁴

* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.