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Bioorganic and Medicinal Chemistry Letters

Volumn 21, Issue 16, 2011, Pages 4884-4887

Carbonic anhydrase i and II activation with mono- and dihalogenated histamine derivatives

(6) Saada, Mohamed Chiheb a Vullo, Daniela b Montero, Jean Louis a Scozzafava, Andrea b Winum, Jean Yves a Supuran, Claudiu T b

a INSTITUT CHARLES GERHARDT (France)

b UNIVERSITY OF FLORENCE (Italy)

Author keywords

Carbonic anhydrase; Cytosolic isoforms I and II; Enzyme activator; Halogenated histamine; Histamine

Indexed keywords

BROMINE; CARBONATE DEHYDRATASE I; CARBONATE DEHYDRATASE II; CHLORINE; FLUORINE; HISTAMINE DERIVATIVE;

ARTICLE; BINDING SITE; ENZYME ACTIVATION; ENZYME ACTIVITY; HALOGENATION; STRUCTURE ACTIVITY RELATION;

CARBONIC ANHYDRASE I; CARBONIC ANHYDRASE II; DOSE-RESPONSE RELATIONSHIP, DRUG; ENZYME ACTIVATION; HALOGENS; HISTAMINE; HUMANS; MODELS, MOLECULAR; MOLECULAR STRUCTURE; STEREOISOMERISM; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 79960929731 PISSN: 0960894X EISSN: 14643405 Source Type: Journal
DOI: 10.1016/j.bmcl.2011.06.030 Document Type: Article

Times cited : (23)

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