메뉴 건너뛰기




Volumn 66, Issue 3, 2007, Pages 191-208

Emerging trends in tuberculosis therapy - A review

Author keywords

Antimycobacterial agents; Cell envelope; Drugs; MIC; Mycobacterium tuberculosis; Targets; Therapeutic agents

Indexed keywords

ANTIGEN-ANTIBODY REACTIONS; BACTERIOPHAGES; CELLS; DRUG PRODUCTS; PULMONARY DISEASES;

EID: 33947214354     PISSN: 00224456     EISSN: None     Source Type: Journal    
DOI: None     Document Type: Review
Times cited : (12)

References (101)
  • 1
    • 67650238578 scopus 로고    scopus 로고
    • in by T L Lemke & D A Williams, 5th edn (Lippincott Williams & Wilkins, USA)
    • Lemke T L, in Foye's Principles of Medicinal Chemistry by T L Lemke & D A Williams, 5th edn (Lippincott Williams & Wilkins, USA) 2002, 904-906.
    • Foye's Principles of Medicinal Chemistry , vol.2002 , pp. 904-906
    • Lemke, T.L.1
  • 2
  • 3
    • 33947200513 scopus 로고    scopus 로고
    • www.who.org
  • 6
    • 0030298489 scopus 로고    scopus 로고
    • Enzymatic synthesis of UDP-galactofuranose and an assay for UDP-galactopyranose mutase based on high-performance liquid chromatography
    • Lee R, Monsey D, Weston A, Duncan K, Rithner C & McNeil M, Enzymatic synthesis of UDP-galactofuranose and an assay for UDP-galactopyranose mutase based on high-performance liquid chromatography, Anal Biochem, 242 (1996) 1-7.
    • (1996) Anal Biochem , vol.242 , pp. 1-7
    • Lee, R.1    Monsey, D.2    Weston, A.3    Duncan, K.4    Rithner, C.5    McNeil, M.6
  • 7
    • 0031444647 scopus 로고    scopus 로고
    • Mycobacterial arabinan biosynthesis: The use of synthetic arabinoside acceptors in the development of an arabinosyl transfer assay
    • Lee R E, Brennan P J &Besra G S, Mycobacterial arabinan biosynthesis: The use of synthetic arabinoside acceptors in the development of an arabinosyl transfer assay, Glycobiology, 7 (1997) 1121-1128.
    • (1997) Glycobiology , vol.7 , pp. 1121-1128
    • Lee, R.E.1    Brennan, P.J.2    Besra, G.S.3
  • 8
    • 0030950127 scopus 로고    scopus 로고
    • Determination of the pathway for rhamnose biosynthesis in mycobacteria: Cloning, sequencing and expression of the Mycobacterium tuberculosis gene encoding alpha-D-glucose-1-phosphate thymidylyltransferase
    • Ma Y, Mills J A, Belisle J T, Vissa V, Howell M, Bowlin K, Scherman M S & McNeil M, Determination of the pathway for rhamnose biosynthesis in mycobacteria: Cloning, sequencing and expression of the Mycobacterium tuberculosis gene encoding alpha-D-glucose-1-phosphate thymidylyltransferase, Microbiology, 143 (1997) 937-945.
    • (1997) Microbiology , vol.143 , pp. 937-945
    • Ma, Y.1    Mills, J.A.2    Belisle, J.T.3    Vissa, V.4    Howell, M.5    Bowlin, K.6    Scherman, M.S.7    McNeil, M.8
  • 9
    • 0030029877 scopus 로고    scopus 로고
    • Galactofuranose biosynthesis in Escherichia coli K-12: Identification and cloning of UDP-galactopyranose mutase
    • Nassau P M, Martin S L, Brown R E, Weston A, Honsey D, McNeil M R & Duncan K, Galactofuranose biosynthesis in Escherichia coli K-12: Identification and cloning of UDP-galactopyranose mutase, J Bacteriol, 178 (1996) 1047-1052.
    • (1996) J Bacteriol , vol.178 , pp. 1047-1052
    • Nassau, P.M.1    Martin, S.L.2    Brown, R.E.3    Weston, A.4    Honsey, D.5    McNeil, M.R.6    Duncan, K.7
  • 10
    • 12844278679 scopus 로고    scopus 로고
    • Pathway to synthesis and processing of mycolic acids in Mycobacterium tuberculosis
    • Takayama K, Wang C & Besra G S, Pathway to synthesis and processing of mycolic acids in Mycobacterium tuberculosis, Clin Microbiol Rev, 18 (2005) 81-101.
    • (2005) Clin Microbiol Rev , vol.18 , pp. 81-101
    • Takayama, K.1    Wang, C.2    Besra, G.S.3
  • 11
    • 33947246829 scopus 로고    scopus 로고
    • http://www.chemsoc.org/chembytes/ezine/1998/evans.htm
  • 16
    • 0031879709 scopus 로고    scopus 로고
    • In vitro and in vivo activities of moxifloxacin and clinafloxacin against Mycobacterium tuberculosis
    • Ji B, Lounis N, Maslo C, Truffot-Pernot C, Bonnafous P & Grosset J, In vitro and in vivo activities of moxifloxacin and clinafloxacin against Mycobacterium tuberculosis, Antimicrob Ag Chemother, 42 (1998) 2066-2069.
    • (1998) Antimicrob Ag Chemother , vol.42 , pp. 2066-2069
    • Ji, B.1    Lounis, N.2    Maslo, C.3    Truffot-Pernot, C.4    Bonnafous, P.5    Grosset, J.6
  • 17
    • 0032910406 scopus 로고    scopus 로고
    • Moxifloxacin (BAY12-8039), a new 8-methoxyquinolone is active in a mouse model of tuberculosis
    • Miyazaki E, Miyazaki M, Chen J M, Chaisson R E & Bishai W R, Moxifloxacin (BAY12-8039), a new 8-methoxyquinolone is active in a mouse model of tuberculosis, Antimicrob Ag Chemother, 43 (1999) 85-89.
    • (1999) Antimicrob Ag Chemother , vol.43 , pp. 85-89
    • Miyazaki, E.1    Miyazaki, M.2    Chen, J.M.3    Chaisson, R.E.4    Bishai, W.R.5
  • 19
    • 0029100035 scopus 로고
    • Antimicrobial activity of CS-940, a new trifluorinated quinolone
    • Biedenbach D J, Sutton L D & Jones R N, Antimicrobial activity of CS-940, a new trifluorinated quinolone, Antimicrob Ag Chemother, 39 (1995) 2325-2330.
    • (1995) Antimicrob Ag Chemother , vol.39 , pp. 2325-2330
    • Biedenbach, D.J.1    Sutton, L.D.2    Jones, R.N.3
  • 20
    • 0033011810 scopus 로고    scopus 로고
    • Fluoroquinolone action against clinical isolates of Mycobacterium tuberculosis: Effects of a C-8 methoxyl Group on survival in liquid media and in human macrophages
    • Zhao B Y, Pine R, Domagala J & Drlica K, Fluoroquinolone action against clinical isolates of Mycobacterium tuberculosis: Effects of a C-8 methoxyl Group on survival in liquid media and in human macrophages, Antimicrob Ag Chemother, 43 (1999) 661-666.
    • (1999) Antimicrob Ag Chemother , vol.43 , pp. 661-666
    • Zhao, B.Y.1    Pine, R.2    Domagala, J.3    Drlica, K.4
  • 21
    • 0032881134 scopus 로고    scopus 로고
    • Dual inhibitory activity of sitafloxacin(DU-6859a) against DNA gyrase and topoisomerase IV of Streptococcus pneumoniae
    • Onodera Y, Uchida Y, Tanaka M & Sato K, Dual inhibitory activity of sitafloxacin(DU-6859a) against DNA gyrase and topoisomerase IV of Streptococcus pneumoniae, J Antimicrob Chemother, 44 (1999) 533-536.
    • (1999) J Antimicrob Chemother , vol.44 , pp. 533-536
    • Onodera, Y.1    Uchida, Y.2    Tanaka, M.3    Sato, K.4
  • 22
    • 0042864697 scopus 로고    scopus 로고
    • Recent advances in research on antituberculars
    • Roy B N, Karnik M A & Sankaran R, Recent advances in research on antituberculars, J Ind Chem Soc, 79 (2002) 320-335.
    • (2002) J Ind Chem Soc , vol.79 , pp. 320-335
    • Roy, B.N.1    Karnik, M.A.2    Sankaran, R.3
  • 23
    • 0042515174 scopus 로고    scopus 로고
    • Synthesis, and antimycobacterial and cytotoxic evaluation of certain fluoroquinolone derivatives
    • Chem Abstr, 140 (2004) 16634
    • Sheu J Y, Chen Y L, Tzeng C C, Hsu S L, Fang K C & Wang T C, Synthesis, and antimycobacterial and cytotoxic evaluation of certain fluoroquinolone derivatives, Helv Chem Acta(Eng), 86 (2003) 2481-2489; Chem Abstr, 140 (2004) 16634.
    • (2003) Helv Chem Acta(Eng) , vol.86 , pp. 2481-2489
    • Sheu, J.Y.1    Chen, Y.L.2    Tzeng, C.C.3    Hsu, S.L.4    Fang, K.C.5    Wang, T.C.6
  • 24
    • 0034026489 scopus 로고    scopus 로고
    • Antimicrobial activities of mefloquine and a series of related compounds
    • Kunin C M & Ellis W Y, Antimicrobial activities of mefloquine and a series of related compounds, Antimicrob Ag Chemother, 44 (2000) 848-852.
    • (2000) Antimicrob Ag Chemother , vol.44 , pp. 848-852
    • Kunin, C.M.1    Ellis, W.Y.2
  • 26
    • 0036661719 scopus 로고    scopus 로고
    • Synthesis of novel 3-N-[(substitutedaryl/heterotryl)methylene]- imino-2-methyl-5-thienyl-thieno[2,3-d]pyrimidine4-(3H)-ones as possible antimicrobial agents
    • Chambhare R V, Bobade A S & Khasde B G, Synthesis of novel 3-N-[(substitutedaryl/heterotryl)methylene]- imino-2-methyl-5-thienyl-thieno[2,3-d]pyrimidine4-(3H)-ones as possible antimicrobial agents, Ind J Het Chem, 12 (2002) 67-68.
    • (2002) Ind J Het Chem , vol.12 , pp. 67-68
    • Chambhare, R.V.1    Bobade, A.S.2    Khasde, B.G.3
  • 27
    • 0037196950 scopus 로고    scopus 로고
    • Synthesis and antituberculous activity of n-mannich bases of 3-[4-(4-chlorophenyl)-6-(4-methylphenyl)pyrimidin-2-yl]iminoisatin derivatives
    • Chem Abstr, 138 (2003) 89754
    • Sriram D, Yogeeswari P, Pandeya S N & Ananthan S, Synthesis and antituberculous activity of n-mannich bases of 3-[4-(4-chlorophenyl)-6-(4-methylphenyl)pyrimidin-2-yl]iminoisatin derivatives, Scientia Pharmaceutica (Eng), 70 (2002) 39-48; Chem Abstr, 138 (2003) 89754.
    • (2002) Scientia Pharmaceutica (Eng) , vol.70 , pp. 39-48
    • Sriram, D.1    Yogeeswari, P.2    Pandeya, S.N.3    Ananthan, S.4
  • 31
    • 33947217608 scopus 로고    scopus 로고
    • US Pat 6, 087, 358 Chem Abstrt, 133 (2000) 89525
    • Baker W R, Shaopei C & Keeler E L, US Pat 6, 087, 358 (2000); Chem Abstrt, 133 (2000) 89525.
    • (2000)
    • Baker, W.R.1    Shaopei, C.2    Keeler, E.L.3
  • 34
    • 0035038011 scopus 로고    scopus 로고
    • Drug targeting Mycobacterium tuberculosis cell wall synthesis: Genetics of dTDP-rhamnose synthetic enzymes and development of a microtiter plate-based screen for inhibitors of conversion of dTDP-glucose to
    • Ma Y, Stern R J, Scherman M S, Vissa V D, Yan W, Jones V C, Zhang F, Franzblau S G, Lewis W H & McNeil M R, Drug targeting Mycobacterium tuberculosis cell wall synthesis: genetics of dTDP-rhamnose synthetic enzymes and development of a microtiter plate-based screen for inhibitors of conversion of dTDP-glucose to dTDP-rhamnose, Antimicrob Ag Chemother, 5 (2001) 1407-1416.
    • (2001) DTDP-rhamnose Antimicrob Ag Chemother , vol.5 , pp. 1407-1416
    • Ma, Y.1    Stern, R.J.2    Scherman, M.S.3    Vissa, V.D.4    Yan, W.5    Jones, V.C.6    Zhang, F.7    Franzblau, S.G.8    Lewis, W.H.9    McNeil, M.R.10
  • 38
    • 0036157457 scopus 로고    scopus 로고
    • Synthesis and biological evaluation of trehalose analogs as potential inhibitors of mycobacterial cell wall biosynthesis
    • Rose J D, Maddry J A, Comber R N, Suling W J, Wilson L N & Reynolds R C, Synthesis and biological evaluation of trehalose analogs as potential inhibitors of mycobacterial cell wall biosynthesis, Carbohydr Res, 337 (2002) 105-120.
    • (2002) Carbohydr Res , vol.337 , pp. 105-120
    • Rose, J.D.1    Maddry, J.A.2    Comber, R.N.3    Suling, W.J.4    Wilson, L.N.5    Reynolds, R.C.6
  • 39
    • 0028064838 scopus 로고
    • Recognition of the lipid intermediate for arabinogalactan/arabinomannan biosynthesis and its relation to the mode of action of ethambutol on mycobacteria
    • Wolucka B A, McNeil M R, deHoffman E, Chojnaki T & Brennan P J, Recognition of the lipid intermediate for arabinogalactan/arabinomannan biosynthesis and its relation to the mode of action of ethambutol on mycobacteria, J Biol Chem, 269 (1994) 23328-23335.
    • (1994) J Biol Chem , vol.269 , pp. 23328-23335
    • Wolucka, B.A.1    McNeil, M.R.2    deHoffman, E.3    Chojnaki, T.4    Brennan, P.J.5
  • 40
    • 0029977936 scopus 로고    scopus 로고
    • Polyprenylphosphate-pentoses in mycobacteria are synthesized from 5-phosphoribose pyrophosphate
    • Scherman M S, Kalbe-Bournonville L, Bush D, Xin Y, Deng L & McNeil M, Polyprenylphosphate-pentoses in mycobacteria are synthesized from 5-phosphoribose pyrophosphate, J Biol Chem, 271 (1996) 29652-29658.
    • (1996) J Biol Chem , vol.271 , pp. 29652-29658
    • Scherman, M.S.1    Kalbe-Bournonville, L.2    Bush, D.3    Xin, Y.4    Deng, L.5    McNeil, M.6
  • 41
    • 0037073950 scopus 로고    scopus 로고
    • Synthesis and antituberculosis activity of C-phosphonate analogues of decaprenolphosphoarabinose, a key intermediate in the biosynthesis of mycobactedal arabinogalactan and lipoarabinomannan
    • Centrone C A & Lowary T L, Synthesis and antituberculosis activity of C-phosphonate analogues of decaprenolphosphoarabinose, a key intermediate in the biosynthesis of mycobactedal arabinogalactan and lipoarabinomannan. J Org Chem, 67 (2002) 8862-8870.
    • (2002) J Org Chem , vol.67 , pp. 8862-8870
    • Centrone, C.A.1    Lowary, T.L.2
  • 44
    • 0005690525 scopus 로고    scopus 로고
    • in by C Curius, S Ghisla & N Blau (Walter de Gruyter, Berlin, Germany)
    • Temple C G, in Chemistry and Biology of Pteridines, by C Curius, S Ghisla & N Blau (Walter de Gruyter, Berlin, Germany) 1990, 1009-1014.
    • Chemistry and Biology of Pteridines , vol.1990 , pp. 1009-1014
    • Temple, C.G.1
  • 49
    • 0022479574 scopus 로고
    • Single amino acid substitutions in the enzyme acetolactate synthase confer resistance to the herbicide sulfometuron methyl
    • Yadav N, McDevitt R E, Benard S & Falco S C, Single amino acid substitutions in the enzyme acetolactate synthase confer resistance to the herbicide sulfometuron methyl, Proc Natl Acad Sci, 83 (1986) 4418-4422.
    • (1986) Proc Natl Acad Sci , vol.83 , pp. 4418-4422
    • Yadav, N.1    McDevitt, R.E.2    Benard, S.3    Falco, S.C.4
  • 52
    • 19944429772 scopus 로고    scopus 로고
    • A diarylquinoline drug active on the ATP synthase of Mycobacterium tuberculosis
    • Andries K, A diarylquinoline drug active on the ATP synthase of Mycobacterium tuberculosis, Science, 307 (2005) 223-227.
    • (2005) Science , vol.307 , pp. 223-227
    • Andries, K.1
  • 53
    • 0037075792 scopus 로고    scopus 로고
    • Synthesis and antimycobacterial activity of 6-arylpurines: The requirements for the N-9 substituent in active anti-mycobacterial purines
    • Gundersen L, Nissen-Meyer J & Spilsberg B, Synthesis and antimycobacterial activity of 6-arylpurines: The requirements for the N-9 substituent in active anti-mycobacterial purines, J Med Chem, 45 (2002) 1383-1386.
    • (2002) J Med Chem , vol.45 , pp. 1383-1386
    • Gundersen, L.1    Nissen-Meyer, J.2    Spilsberg, B.3
  • 56
    • 0031753303 scopus 로고    scopus 로고
    • Bactericidal activities of the pyrrole derivative BM212 against multidrug-resistant and intramacrophagic Mycobacterium tuberculosis strains
    • Deidda D, Lampis G, Fioravanti R, Biava M, Portea G, Zanetti S & Pompei R, Bactericidal activities of the pyrrole derivative BM212 against multidrug-resistant and intramacrophagic Mycobacterium tuberculosis strains, Antimicrob Ag Chemother, 42 (1998) 3035-3037.
    • (1998) Antimicrob Ag Chemother , vol.42 , pp. 3035-3037
    • Deidda, D.1    Lampis, G.2    Fioravanti, R.3    Biava, M.4    Portea, G.5    Zanetti, S.6    Pompei, R.7
  • 57
    • 0036029005 scopus 로고
    • BM 212 and its derivatives as a new class of anti-mycobacterial active agents
    • Biava M, BM 212 and its derivatives as a new class of anti-mycobacterial active agents, Curr Med Chem, 9 (1995) 1859-1869.
    • (1995) Curr Med Chem , vol.9 , pp. 1859-1869
    • Biava, M.1
  • 58
    • 0035833112 scopus 로고    scopus 로고
    • Anti-mycobacterial activity of 9-sulfonylated/ sulfenylated-6-mercaptopurine derivatives
    • Scozzafava A, Mastrolenzo A & Supuran C T, Anti-mycobacterial activity of 9-sulfonylated/sulfenylated-6-mercaptopurine derivatives, Bioorg Med Chem Lett, 11 (2001) 1675-1678.
    • (2001) Bioorg Med Chem Lett , vol.11 , pp. 1675-1678
    • Scozzafava, A.1    Mastrolenzo, A.2    Supuran, C.T.3
  • 61
    • 0033594440 scopus 로고    scopus 로고
    • Synthesis and antimalarial activity of 11 dispiro-1,2,4,5-tetraoxane analogues of WR 148999. 7,8,15,16-tetraoxadispiro[5.2.5.2]hexadecanes substituted at the 1 and 10 positions with unsaturated and polar functional groups
    • Dong Y, Matile H, Chollet J, Kaminsky R, Wood K & Vennerstrom J L, Synthesis and antimalarial activity of 11 dispiro-1,2,4,5-tetraoxane analogues of WR 148999. 7,8,15,16-tetraoxadispiro[5.2.5.2]hexadecanes substituted at the 1 and 10 positions with unsaturated and polar functional groups, J Med Chem, 42 (1999) 1477-1480.
    • (1999) J Med Chem , vol.42 , pp. 1477-1480
    • Dong, Y.1    Matile, H.2    Chollet, J.3    Kaminsky, R.4    Wood, K.5    Vennerstrom, J.L.6
  • 62
    • 0018101097 scopus 로고
    • Chemical constituents of Gentianaceae. XXIV. Anti-Mycobacterium tuberculosis activity of naturally occurring xanthones and synthetic analogs
    • Ghosal S, Biswas K & Chauduri R K, Chemical constituents of Gentianaceae. XXIV. Anti-Mycobacterium tuberculosis activity of naturally occurring xanthones and synthetic analogs, J Pharm Sci, 67 (1978) 721-722.
    • (1978) J Pharm Sci , vol.67 , pp. 721-722
    • Ghosal, S.1    Biswas, K.2    Chauduri, R.K.3
  • 63
    • 0036241998 scopus 로고    scopus 로고
    • Synthesis and anti-tubercular evaluation of 4-quinolylhydrazones
    • Savini L, Chiasserini L, Gaeta A & Pellerano C, Synthesis and anti-tubercular evaluation of 4-quinolylhydrazones, Bioorg Med Chem, 10 (2002) 2193-2198.
    • (2002) Bioorg Med Chem , vol.10 , pp. 2193-2198
    • Savini, L.1    Chiasserini, L.2    Gaeta, A.3    Pellerano, C.4
  • 64
    • 0035445139 scopus 로고    scopus 로고
    • Influence of the replacement of the oxo function with the thioxo group on the antimycobacterial activity of 3-aryl-6,8-dichloro-2H-1,3-benzoxazine-2,4(3H)-diones and 3-arylquinazoline-2,4(1H,3H)-diones
    • Waisser K, Gregor J, Dostál H, Kubicová L, Klimeǒvá V & Kaustová J, Influence of the replacement of the oxo function with the thioxo group on the antimycobacterial activity of 3-aryl-6,8-dichloro-2H-1,3-benzoxazine-2,4(3H)-diones and 3-arylquinazoline-2,4(1H,3H)-diones, Farmaco. 56 (2001) 803-807.
    • (2001) Farmaco , vol.56 , pp. 803-807
    • Waisser, K.1    Gregor, J.2    Dostál, H.3    Kubicová, L.4    Klimeǒvá, V.5    Kaustová, J.6
  • 66
    • 0034830902 scopus 로고    scopus 로고
    • Redox-activated, hypoxia-selective DNA cleavage by quinoxaline 1,4-di-N-oxide
    • Ganley B, Chowdhury G, Bhansali J, Daniels J S & Gates K S, Redox-activated, hypoxia-selective DNA cleavage by quinoxaline 1,4-di-N-oxide, Bioorg Med Chem, 9 (2001) 2395-2401.
    • (2001) Bioorg Med Chem , vol.9 , pp. 2395-2401
    • Ganley, B.1    Chowdhury, G.2    Bhansali, J.3    Daniels, J.S.4    Gates, K.S.5
  • 67
    • 1342324049 scopus 로고    scopus 로고
    • Synthesis, anti-mycobacterial, anti-trichomonas and anti-candida in vitro activities of 2-substituted-6,7-difluoro-3-methylquinoxaline 1,4-dioxides
    • Carta A, Loriga M, Paglietti G, Mattana A, Fiori P L, Mollicotti P, Sechi L & Zannetti S, Synthesis, anti-mycobacterial, anti-trichomonas and anti-candida in vitro activities of 2-substituted-6,7-difluoro-3-methylquinoxaline 1,4-dioxides, Eur J Med Chem, 39 (2004) 195-203.
    • (2004) Eur J Med Chem , vol.39 , pp. 195-203
    • Carta, A.1    Loriga, M.2    Paglietti, G.3    Mattana, A.4    Fiori, P.L.5    Mollicotti, P.6    Sechi, L.7    Zannetti, S.8
  • 68
    • 0035093384 scopus 로고    scopus 로고
    • Anti-mycobacterial activity of new quinoxaline-2-carbonitrile and quinoxaline-2-carbonitrile 1,4-di-N-oxide derivatives
    • Ortega M A, Montoya M E, Jaso A, Zarranz B, Tirapu I, Aldana I & Monge A, Anti-mycobacterial activity of new quinoxaline-2-carbonitrile and quinoxaline-2-carbonitrile 1,4-di-N-oxide derivatives, Pharmazie, 56 (2001) 205-207.
    • (2001) Pharmazie , vol.56 , pp. 205-207
    • Ortega, M.A.1    Montoya, M.E.2    Jaso, A.3    Zarranz, B.4    Tirapu, I.5    Aldana, I.6    Monge, A.7
  • 69
    • 0037447952 scopus 로고    scopus 로고
    • Synthesis and antimycobacterial activity of new quinoxaline-2-carboxamide 1,4-di-N-oxide derivatives
    • Zarranz B, Jaso A, Aldana I & Monge A, Synthesis and antimycobacterial activity of new quinoxaline-2-carboxamide 1,4-di-N-oxide derivatives, Bioorg Med Chem, 11 (2003) 2149-2156.
    • (2003) Bioorg Med Chem , vol.11 , pp. 2149-2156
    • Zarranz, B.1    Jaso, A.2    Aldana, I.3    Monge, A.4
  • 70
    • 0001945179 scopus 로고
    • Design of compounds active against Mycobacterium tuberculosis
    • Waisser K, Klimesova V & Odlerová Z, Design of compounds active against Mycobacterium tuberculosis, Folia Pharm Univ Carol, 18 (1995) 31-37.
    • (1995) Folia Pharm Univ Carol , vol.18 , pp. 31-37
    • Waisser, K.1    Klimesova, V.2    Odlerová, Z.3
  • 71
    • 0030762464 scopus 로고    scopus 로고
    • Synthesis and antimycobacterial activity of some new 3-heterocyclic substituted chromones
    • Gasparova R, Lacova M, El-Shaaer H M & Odlerová Z, Synthesis and antimycobacterial activity of some new 3-heterocyclic substituted chromones, Farmaco, 52 (1997) 251-253.
    • (1997) Farmaco , vol.52 , pp. 251-253
    • Gasparova, R.1    Lacova, M.2    El-Shaaer, H.M.3    Odlerová, Z.4
  • 73
    • 0036241998 scopus 로고    scopus 로고
    • Synthesis and anti-tubercular evaluation of 4-quinolylhydrazones
    • Savini L, Chiasserini L, Gaeta A & Pellerano C, Synthesis and anti-tubercular evaluation of 4-quinolylhydrazones, Bioorg Med Chem, 10 (2002) 2193-2198.
    • (2002) Bioorg Med Chem , vol.10 , pp. 2193-2198
    • Savini, L.1    Chiasserini, L.2    Gaeta, A.3    Pellerano, C.4
  • 74
    • 0036121495 scopus 로고    scopus 로고
    • Synthesis of 1,3-thiazine derivatives and their evaluation as potential antimycobacterial agents
    • Koketsu M, Tanaka K, Takenaka Y, Kwong C D & Ishihara H, Synthesis of 1,3-thiazine derivatives and their evaluation as potential antimycobacterial agents, Eur J Pharm Sci, 15 (2002) 307-310.
    • (2002) Eur J Pharm Sci , vol.15 , pp. 307-310
    • Koketsu, M.1    Tanaka, K.2    Takenaka, Y.3    Kwong, C.D.4    Ishihara, H.5
  • 76
    • 0035492471 scopus 로고    scopus 로고
    • Synthesis, antimycobacterial activities and cytotoxicity on V79 of 3-[4′-Y-(1,1′-biphenyl)-4-yl]-N,N-dimethyl-3-(4-X-phenyl)-2- propen-1-amine derivatives
    • De Souza A O, Santos R R Jr, Ferreira-Julio J F, Rodríguez J A, Melo P S, Haun M, Sato D N & Durán N, Synthesis, antimycobacterial activities and cytotoxicity on V79 of 3-[4′-Y-(1,1′-biphenyl)-4-yl]-N,N-dimethyl-3-(4-X-phenyl)-2- propen-1-amine derivatives. Eur J Med Chem, 36 (2001) 843-850.
    • (2001) Eur J Med Chem , vol.36 , pp. 843-850
    • De Souza, A.O.1    Santos Jr., R.R.2    Ferreira-Julio, J.F.3    Rodríguez, J.A.4    Melo, P.S.5    Haun, M.6    Sato, D.N.7    Durán, N.8
  • 77
    • 0034633853 scopus 로고    scopus 로고
    • Combination of molecular modeling and quantitative structure-activity relationship analysis in the study of antimycobacterial activity of pyridine derivatives
    • Klimesova V, Palat K, Waisser K & Klimes J, Combination of molecular modeling and quantitative structure-activity relationship analysis in the study of antimycobacterial activity of pyridine derivatives, Int J Pharm, 207 (2000) 1-6.
    • (2000) Int J Pharm , vol.207 , pp. 1-6
    • Klimesova, V.1    Palat, K.2    Waisser, K.3    Klimes, J.4
  • 81
    • 0035048959 scopus 로고    scopus 로고
    • Antimycobacterial activity of 1-deaza-7,8-dihydropteridine derivatives against Mycobacterium tuberculosis and Mycobacterium avium complex in vitro
    • Suling W J & Maddry J A, Antimycobacterial activity of 1-deaza-7,8-dihydropteridine derivatives against Mycobacterium tuberculosis and Mycobacterium avium complex in vitro, J Antimicrob Chemother, 47 (2001) 451-454.
    • (2001) J Antimicrob Chemother , vol.47 , pp. 451-454
    • Suling, W.J.1    Maddry, J.A.2
  • 82
    • 0034058145 scopus 로고    scopus 로고
    • Oxazolidinones, A review
    • Diekema D J & Jones R N, Oxazolidinones, A review, Drugs, 59 (2000) 7-16.
    • (2000) Drugs , vol.59 , pp. 7-16
    • Diekema, D.J.1    Jones, R.N.2
  • 85
    • 0013797020 scopus 로고
    • Studies on pyrrolnitrin, a new antibiotic. I. Isolation and properties of pyrrolnitri
    • Arima K, Imanaka H, Kousaka M, Fukuda A & Tamura G, Studies on pyrrolnitrin, a new antibiotic. I. Isolation and properties of pyrrolnitri, J Antibiot Ser A, 18 (1968) 201-204.
    • (1968) J Antibiot Ser A , vol.18 , pp. 201-204
    • Arima, K.1    Imanaka, H.2    Kousaka, M.3    Fukuda, A.4    Tamura, G.5
  • 86
    • 1842630349 scopus 로고    scopus 로고
    • Synthesis and preliminary evaluation of some pyrazine containing thiazolines and thiazolidinones as antimicrobial agents
    • Bonde C G & Gaikwad N J, Synthesis and preliminary evaluation of some pyrazine containing thiazolines and thiazolidinones as antimicrobial agents, Bioorg Med Chem, 12 (2004) 2151-2161.
    • (2004) Bioorg Med Chem , vol.12 , pp. 2151-2161
    • Bonde, C.G.1    Gaikwad, N.J.2
  • 87
    • 0033913636 scopus 로고    scopus 로고
    • New groups of antimycobacterial agents: 6-chloro-3-phenyl-4-thioxo-2H-1,3-benzoxazine-2(3H)-ones and 6-chloro-3-phenyl-2H-1,3-benzoxazine-2,4(3H)-dithiones
    • Waisser K, Gregor J, Kubicova L, Klimesova V, Kunes J, Machacek M & Kaustova J, New groups of antimycobacterial agents: 6-chloro-3-phenyl-4-thioxo-2H-1,3-benzoxazine-2(3H)-ones and 6-chloro-3-phenyl-2H-1,3-benzoxazine-2,4(3H)-dithiones, Eur J Med Chem, 35 (2000) 733-741.
    • (2000) Eur J Med Chem , vol.35 , pp. 733-741
    • Waisser, K.1    Gregor, J.2    Kubicova, L.3    Klimesova, V.4    Kunes, J.5    Machacek, M.6    Kaustova, J.7
  • 88
    • 0033549680 scopus 로고    scopus 로고
    • Novel antimycobacterial benzoxazole alkaloids from the West Indian Sea whip Pseudopterogorgia elisabethae
    • Rodriguez A D, Ramirez C, Rodriguez II & Gonzalez E, Novel antimycobacterial benzoxazole alkaloids from the West Indian Sea whip Pseudopterogorgia elisabethae, Org Letts, 1 (1999) 527-530.
    • (1999) Org Letts , vol.1 , pp. 527-530
    • Rodriguez, A.D.1    Ramirez, C.2    Rodriguez, I.I.3    Gonzalez, E.4
  • 89
    • 0031734041 scopus 로고    scopus 로고
    • Tuberculosis: A search for novel therapy starting with natural products
    • Mitscher L A & Baker W, Tuberculosis: A search for novel therapy starting with natural products, Med Res Rev, 18 (1997) 363-374.
    • (1997) Med Res Rev , vol.18 , pp. 363-374
    • Mitscher, L.A.1    Baker, W.2
  • 90
    • 0033987119 scopus 로고    scopus 로고
    • In vitro Investigation of the Antimicrobial Activities of Novel Tetramethylpiperidine-Substituted Phenazines against Mycobacterium tuberculosis
    • Van Rensburg C E J, Joone G K, Sirgel F A, Matlola N M & O'Sullivan J F, In vitro Investigation of the Antimicrobial Activities of Novel Tetramethylpiperidine-Substituted Phenazines against Mycobacterium tuberculosis, Chemother, 46 (2000) 43-48.
    • (2000) Chemother , vol.46 , pp. 43-48
    • Van Rensburg, C.E.J.1    Joone, G.K.2    Sirgel, F.A.3    Matlola, N.M.4    O'Sullivan, J.F.5
  • 93
    • 0031806247 scopus 로고    scopus 로고
    • Inhibition of human immunodeficiency virus type 1 reverse transcriptase activity by cordatolides isolated from Calophyllum cordato-oblongum
    • Dharmaratne H R, Wanigasekera W M, Mata-Greenwood E & Pezzuto J M, Inhibition of human immunodeficiency virus type 1 reverse transcriptase activity by cordatolides isolated from Calophyllum cordato-oblongum, Planta Medica, 64 (1998) 460-461.
    • (1998) Planta Medica , vol.64 , pp. 460-461
    • Dharmaratne, H.R.1    Wanigasekera, W.M.2    Mata-Greenwood, E.3    Pezzuto, J.M.4
  • 96
    • 0033971447 scopus 로고    scopus 로고
    • Pharmacokinetics and tissue distribution of rifametane, a new 3-azinomethyl-rifamycin derivative, in several animal species
    • Bruzzese T, Rimaroli C, Bonabello A, Mozzi G, Ajay S & Cooverj N D, Pharmacokinetics and tissue distribution of rifametane, a new 3-azinomethyl-rifamycin derivative, in several animal species, Arzneimittel-Forschung, 50 (2000) 60-71.
    • (2000) Arzneimittel-Forschung , vol.50 , pp. 60-71
    • Bruzzese, T.1    Rimaroli, C.2    Bonabello, A.3    Mozzi, G.4    Ajay, S.5    Cooverj, N.D.6
  • 98
    • 0030961425 scopus 로고    scopus 로고
    • Treatment of multidrug-resistant pulmonary tuberculosis with interferon-gamma via aerosol
    • Condos R, Rom W M & Schluger N W, Treatment of multidrug-resistant pulmonary tuberculosis with interferon-gamma via aerosol, Lancet, 349 (1997) 1513-1515.
    • (1997) Lancet , vol.349 , pp. 1513-1515
    • Condos, R.1    Rom, W.M.2    Schluger, N.W.3
  • 100
    • 0034679958 scopus 로고    scopus 로고
    • Lipid lunch for persistent pathogen
    • Bishai W, Lipid lunch for persistent pathogen, Nature, 406 (2000) 683-685.
    • (2000) Nature , vol.406 , pp. 683-685
    • Bishai, W.1


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.