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European Journal of Pharmaceutical Sciences

Volumn 15, Issue 3, 2002, Pages 307-310

Synthesis of 1,3-thiazine derivatives and their evaluation as potential antimycobacterial agents

(5) Koketsu, Mamoru a Tanaka, Kohsuke a Takenaka, Yuichi a Kwong, Cecil D b Ishihara, Hideharu a

a GIFU UNIVERSITY (Japan)

b SOUTHERN RESEARCH INSTITUTE (United States)

Author keywords

5,6 Dihydro 4H 1,3 thiazine; Antimycobacterial agents; Mycobacterium tuberculosis

Indexed keywords

BACTERIA; ENZYME INHIBITION; LEAD; SYNTHESIS (CHEMICAL);

ANTIMYCOBACTERIAL AGENTS;

DRUG PRODUCTS PLANTS;

1,3 THIAZINE DERIVATIVE; 4 ETHYL 4 HYDROXY 2 PHENYL 5,6 DIHYDRO 4H 1,3 THIAZINE; 4 HYDROXY 4 METHYL 6 PENTYL 2 PHENYL 5,6 DIHYDRO 4H 1,3 THIAZINE; 5 HYDROXY 3 PHENYL 4 AZA 2 THIABICYCLO[3.3.1]NONE 3 ENE; 5,6 DIHYDRO 4H 1,3 THIAZINE DERIVATIVE; ALAMAR BLUE; ANTIMYCOBACTERIAL AGENT; DYE; ETHAMBUTOL; ISONIAZID; KETONE DERIVATIVE; RIFAMPICIN; STREPTOMYCIN; THIOBENZAMIDE; UNCLASSIFIED DRUG;

ANTIBACTERIAL ACTIVITY; ARTICLE; ASSAY; CARBON NUCLEAR MAGNETIC RESONANCE; CATALYSIS; CHEMICAL REACTION; CONCENTRATION RESPONSE; CONTROLLED STUDY; DRUG SENSITIVITY; DRUG SYNTHESIS; MINIMUM INHIBITORY CONCENTRATION; MYCOBACTERIUM TUBERCULOSIS; NONHUMAN; PRIORITY JOURNAL; PROTON NUCLEAR MAGNETIC RESONANCE; ROOM TEMPERATURE; TECHNIQUE;

ANTITUBERCULAR AGENTS; DRUG EVALUATION, PRECLINICAL; MICROBIAL SENSITIVITY TESTS; MYCOBACTERIUM TUBERCULOSIS; THIAZINES;

EID: 0036121495 PISSN: 09280987 EISSN: None Source Type: Journal
DOI: 10.1016/S0928-0987(02)00014-3 Document Type: Article

Times cited : (148)

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