Novel inhibitors of HIV-1 integration

Current Drug Metabolism

Volumn 5, Issue 4, 2004, Pages 291-304

  Witvrouw, M ^a   Van Maele, B ^a   Vercammen, J ^b   Hantson, A ^a   Engelborghs, Y ^b   De Clercq, E ^a   Pannecouque, C ^a   Debyser, Z ^a  

^a REGA INSTITUTE FOR MEDICAL RESEARCH   (Belgium)

^b UNIVERSITY OF LEUVEN   (Belgium)

Author keywords

Diketo acids; HIV; Inhibitors; Integrase; LEDGF; Pyranodipyrimidines; Resistance

Indexed keywords

1 (5 CHLOROINDOL 3 YL) 3 HYDROXY 3 (2H TETRAZOL 5 YL)PROPENONE; 1 [5 (4 FLUOROBENZYL) 2 FURYL] 3 (1,2,4 TRIAZOL 3 YL) 1,3 PROPANEDIONE; 4 [1 (4 FLUOROBENZYL) 2 PYRROLYL] 2,4 DIOXOBUTYRIC ACID; ANTIRETROVIRUS AGENT; CAFFEIC ACID PHENETHYL ESTER; CICHORIC ACID; CYNARINE; GLYCOPROTEIN GP 120; GRANULATINE; HYDRAZIDE DERIVATIVE; INTEGRASE; INTEGRASE INHIBITOR; INTEGRIC ACID; L 708906; N (4 FLUOROBENZYL) 8 HYDROXY 5 (TETRAHYDRO 2H 1,2 THIAZIN 2 YL) 1,6 NAPHTHYRIDINE 7 CARBOXAMIDE S,S DIOXIDE; NAPTHTOTHIAZEPINE; OXOACID; PROTEINASE; PROTEINASE INHIBITOR; PYRIMIDINE DERIVATIVE; RNA DIRECTED DNA POLYMERASE; RNA DIRECTED DNA POLYMERASE INHIBITOR; SALICYLHYDRAZIDE; THIAZEPINE DERIVATIVE; UNCLASSIFIED DRUG; V 165; VIRUS DNA; VIRUS ENVELOPE PROTEIN;

ACQUIRED IMMUNE DEFICIENCY SYNDROME; ANTIBIOTIC RESISTANCE; ANTIVIRAL ACTIVITY; CLINICAL TRIAL; DEATH; DRUG APPROVAL; DRUG STRUCTURE; DRUG TARGETING; ENZYME ASSAY; FLUORESCENCE SPECTROSCOPY; FOOD AND DRUG ADMINISTRATION; GENE MUTATION; GENOTYPE PHENOTYPE CORRELATION; HIGHLY ACTIVE ANTIRETROVIRAL THERAPY; HUMAN; HUMAN IMMUNODEFICIENCY VIRUS 1; HUMAN IMMUNODEFICIENCY VIRUS INFECTION; LIFE CYCLE; MOLECULAR MECHANICS; PATHOGENESIS; POLYMERIZATION; REAL TIME POLYMERASE CHAIN REACTION; RETROVIRUS; REVIEW; VIRUS CULTURE; VIRUS DNA CELL DNA INTERACTION; VIRUS INHIBITION; VIRUS REPLICATION; VIRUS STRAIN; VIRUS TRANSMISSION;

ANIMALS; HIV INFECTIONS; HIV INTEGRASE; HIV INTEGRASE INHIBITORS; HIV-1; HUMANS; VIRUS INTEGRATION;

EID: 3242886580     PISSN: 13892002     EISSN: None     Source Type: Journal    
DOI: 10.2174/1389200043335487     Document Type: Review

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