Interfacial peptide inhibitors of HIV-1 integrase activity and dimerization

Bioorganic and Medicinal Chemistry Letters

Volumn 13, Issue 6, 2003, Pages 1175-1177

  Zhao, Lei ^a   O'Reilly, Mary K ^a   Shultz, Michael D ^a   Chmielewski, Jean ^a  

^a PURDUE UNIVERSITY   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

DIMER; INTEGRASE; INTEGRASE INHIBITOR; VIRUS ENZYME;

AMINO ACID SEQUENCE; ARTICLE; CONCENTRATION RESPONSE; DIMERIZATION; DRUG MECHANISM; DRUG POTENCY; ENZYME ACTIVE SITE; ENZYME ACTIVITY; ENZYME INHIBITION; ENZYME SUBUNIT; HUMAN IMMUNODEFICIENCY VIRUS 1; IC 50; NONHUMAN; PEPTIDE ANALYSIS; PROTEIN CROSS LINKING; PROTEIN SECONDARY STRUCTURE;

CHROMATOGRAPHY, HIGH PRESSURE LIQUID; CROSS-LINKING REAGENTS; ELECTROPHORESIS, POLYACRYLAMIDE GEL; HIV INTEGRASE; HIV INTEGRASE INHIBITORS; MODELS, MOLECULAR; MUTATION; PEPTIDES; PROTEIN DENATURATION;

HUMAN IMMUNODEFICIENCY VIRUS 1;

EID: 0037463767     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0960-894X(03)00040-4     Document Type: Article

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