HIV-1 integrase inhibitors that compete with the target DNA substrate define a unique strand transfer conformation for integrase

Proceedings of the National Academy of Sciences of the United States of America

Volumn 97, Issue 21, 2000, Pages 11244-11249

  Espeseth, Amy S ^a   Felock, Peter ^a   Wolfe, Abigail ^a   Witmer, Marc ^a   Grobler, Jay ^a   Anthony, Neville ^a   Egbertson, Melissa ^a   Melamed, Jeffrey Y ^a   Young, Steve ^a   Hamill, Terence ^a   Cole, James L ^a   Hazuda, Daria J ^a  

^a MERCK RESEARCH LABORATORIES   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

4 [1 (4 FLUOROBENZYL) 2 PYRROLYL] 2,4 DIOXOBUTYRIC ACID; DNA; INTEGRASE; INTEGRASE INHIBITOR; UNCLASSIFIED DRUG;

BINDING AFFINITY; BINDING SITE; COMPLEX FORMATION; CONFERENCE PAPER; DRUG BINDING; DRUG PROTEIN BINDING; ENZYME ACTIVE SITE; ENZYME ACTIVITY; ENZYME CONFORMATION; ENZYME INHIBITION; HUMAN IMMUNODEFICIENCY VIRUS 1; NONHUMAN; PRIORITY JOURNAL;

HUMAN IMMUNODEFICIENCY VIRUS; HUMAN IMMUNODEFICIENCY VIRUS 1;

EID: 12944270496     PISSN: 00278424     EISSN: None     Source Type: Journal    
DOI: 10.1073/pnas.200139397     Document Type: Article

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