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Current Medicinal Chemistry - Anti-Cancer Agents

Volumn 2, Issue 2, 2002, Pages 155-185

Design of selectively activated anticancer prodrugs: Elimination and cyclization strategies

(5) Papot, S a Tranoy, I a Tillequin, F a Florent, J C a Gesson, J P a

a UNIVERSITÉ DE POITIERS (France)

Author keywords

[No Author keywords available]

Indexed keywords

9 AMINOCAMPTOTHECIN; ACIVICIN; ACROLEIN; ACROLEIN DERIVATIVE; AMIDE; ANTHRACYCLINE DERIVATIVE; ANTINEOPLASTIC AGENT; BENZIMIDAZOLE DERIVATIVE; BENZODIAZEPINE DERIVATIVE; BETA GLUCURONIDASE; CARBAMIC ACID DERIVATIVE; CARBONIC ACID; CHLORMETHINE DERIVATIVE; CYCLOPHOSPHAMIDE; CYTOTOXIC AGENT; DACTINOMYCIN; DAUNORUBICIN; DAUNORUBICIN DERIVATIVE; DICHLORODIETHYLAMINE; DOXORUBICIN DERIVATIVE; MITOMYCIN C; N (4 BETA GLUCURONYL 3 NITROBENZYLOXYCARBONYL)DOXORUBICIN; NAPHTHOQUINONE; OXAZOLIDINONE DERIVATIVE; PHOSPHORAMIDE MUSTARD; PLASMIN; PRODRUG; TALLIMUSTINE; TUMOR ANTIGEN; UNINDEXED DRUG;

ANTIBODY DIRECTED ENZYME PRODRUG THERAPY; ANTIGEN RECOGNITION; CANCER CELL; CANCER LOCALIZATION; CELL HYPOXIA; CONTROLLED STUDY; COVALENT BOND; CYCLIZATION; DRUG ACTIVATION; DRUG BLOOD LEVEL; DRUG DESIGN; DRUG ELIMINATION; DRUG FORMULATION; DRUG HALF LIFE; DRUG HYDROLYSIS; DRUG MECHANISM; DRUG RELEASE; DRUG SELECTIVITY; DRUG STABILITY; DRUG STRUCTURE; HUMAN; MACROMOLECULE; MICROENVIRONMENT; NONHUMAN; REDUCTION; REVIEW;

ANIMALS; ANTINEOPLASTIC AGENTS; CROSS-LINKING REAGENTS; CYCLIZATION; HUMANS; PRODRUGS; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 0036080057 PISSN: 15680118 EISSN: None Source Type: Journal
DOI: 10.2174/1568011023354173 Document Type: Review

Times cited : (63)

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