Structure-guided discovery of a novel aminoglycoside conjugate targeting HIV-1 RNA viral genome

ACS Chemical Biology

Volumn 8, Issue 11, 2013, Pages 2509-2517

  Ennifar, Eric ^a   Aslam, Muhammad Waqar ^b   Strasser, Perrine ^a   Hoffmann, Guillaume ^a   Dumas, Philippe ^a   Van Delft, Floris L ^b  

^a INST DE BIOL MOLEC ET CELLULAIRE   (France)

^b RADBOUD UNIVERSITY NIJMEGEN   (Netherlands)

Author keywords

[No Author keywords available]

Indexed keywords

DIMER; NEOMYCIN; THYMINE; VIRUS RNA; AMINOGLYCOSIDE; ANTI HUMAN IMMUNODEFICIENCY VIRUS AGENT; GLYCOCONJUGATE;

ANTIVIRAL ACTIVITY; ARTICLE; BINDING AFFINITY; CHEMICAL STRUCTURE; CONJUGATE; CRYSTAL STRUCTURE; DRUG BINDING; DRUG DESIGN; DRUG SYNTHESIS; DRUG TARGETING; HUMAN IMMUNODEFICIENCY VIRUS 1; IN VITRO STUDY; ISOTHERMAL TITRATION CALORIMETRY; NONHUMAN; PRIORITY JOURNAL; VIRUS GENOME; CHEMISTRY; DRUG DELIVERY SYSTEM; HUMAN;

AMINOGLYCOSIDES; ANTI-HIV AGENTS; DRUG DELIVERY SYSTEMS; GENOME, VIRAL; GLYCOCONJUGATES; HIV-1; HUMANS; MODELS, MOLECULAR; RNA, VIRAL;

EID: 84887893190     PISSN: 15548929     EISSN: 15548937     Source Type: Journal    
DOI: 10.1021/cb400498n     Document Type: Article

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