A KV2.1 gating modifier binding assay suitable for highthroughput screening

Channels

Volumn 3, Issue 6, 2009, Pages

  Schmalhofer, William A ^a   Ratliff, Kevin S ^a   Weinglass, Adam B ^a   Kaczorowski, Gregory J ^a   Garcia, Maria L ^a   Herrington, James ^a  

^a MERCK RESEARCH LABORATORIES   (United States)

Author keywords

Automated electrophysiology; Binding assay; Gating modifier; High throughput screen; KV2.1; Potassium channel; Tarantula toxin; Voltage gated

Indexed keywords

CHARYBDOTOXIN; IBERIOTOXIN; LARGE CONDUCTANCE CALCIUM ACTIVATED POTASSIUM CHANNEL; POTASSIUM; SHAB POTASSIUM CHANNEL; VOLTAGE GATED SODIUM CHANNEL;

ANIMAL CELL; ANIMAL CELL CULTURE; ARTICLE; BINDING AFFINITY; BINDING ASSAY; CHO CELL; DEPOLARIZATION; FEMALE; HIGH THROUGHPUT SCREENING; MEMBRANE POTENTIAL; NONHUMAN; PROTEIN BINDING; PROTEIN EXPRESSION;

TARANTULA;

EID: 72449189610     PISSN: 19336950     EISSN: 19336969     Source Type: Journal    
DOI: 10.4161/chan.3.6.10201     Document Type: Article

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