Constitutive activity at serotonin 5-HT(1D) receptors: Detection by homologous GTPγS versus [35S]-GTPγS binding isotherms

Neuropharmacology

Volumn 40, Issue 1, 2001, Pages 57-64

  Audinot, Valérie ^a   Newman Tancredi, Adrian ^a   Millan, Mark J ^a  

^a INSTITUT DE RECHERCHES INTERNATIONALES SERVIER   (France)

Author keywords

5 HT(1D) receptor; Constitutive activity; Inverse agonist; 35S GTP S

Indexed keywords

2,3,6,7 TETRAHYDRO 1' METHYL 5 [[2' METHYL 4' (5 METHYL 1,2,4 OXADIAZOL 3 YL) 4 BIPHENYLYL]CARBONYL]SPIRO[FURO[2,3 F]INDOLE 3,4' PIPERIDINE]; G PROTEIN COUPLED RECEPTOR; GUANOSINE 5' O (3 THIOTRIPHOSPHATE); METITEPINE; N [1 (2,3 DIHYDRO[1,4]DIOXIN 5 YL)PIPERID 4 YL]INDAN 2 YL AMINE DICHLOROHYDRATE; S 18127; SEROTONIN; SEROTONIN 1B AGONIST; SEROTONIN 1D AGONIST; SEROTONIN 1D ANTAGONIST; SEROTONIN 1D RECEPTOR; UNCLASSIFIED DRUG;

ANIMAL CELL; ARTICLE; BINDING AFFINITY; BINDING COMPETITION; BINDING SITE; CONCENTRATION RESPONSE; CONTROLLED STUDY; DRUG EFFECT; MEMBRANE BINDING; NONHUMAN; PRIORITY JOURNAL; RECEPTOR BINDING; RECEPTOR UPREGULATION;

EID: 0033765247     PISSN: 00283908     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0028-3908(00)00104-0     Document Type: Article

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