Inverse agonists and neutral antagonists of recombinant human A1 adenosine receptors stably expressed in Chinese hamster ovary cells

Molecular Pharmacology

Volumn 53, Issue 5, 1998, Pages 886-893

  Shryock, John C ^a   Ozeck, Mark J ^b   Belardinelli, Luiz ^a,b  

^a UNIVERSITY OF FLORIDA COLLEGE OF MEDICINE   (United States)

^b UNIVERSITY OF FLORIDA   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

2 AMINO 4,5 DIMETHYL 3 (3 TRIFLUOROMETHYLBENZOYL)THIOPHENE; 6 N CYCLOPENTYLADENOSINE; 9 CHLORO 2 (2 FURYL) 5,6 DIHYDRO 5 IMINO 1,2,4 TRIAZOLO[2,3 C]QUINAZOLINE; 9 METHYL 6 N (2 NORBORNYL)ADENINE; ADENOSINE; ADENOSINE A1 RECEPTOR; ADENOSINE DEAMINASE; ADENYLATE CYCLASE; CYCLIC AMP; FORSKOLIN; GUANINE NUCLEOTIDE BINDING PROTEIN; GUANOSINE TRIPHOSPHATE; PHOSPHODIESTERASE;

ANIMAL CELL; ARTICLE; CHO CELL; ENZYME ACTIVITY; LIGAND BINDING; NONHUMAN; PRIORITY JOURNAL; PROTEIN CONFORMATION; PROTEIN EXPRESSION; RECEPTOR DENSITY;

ANIMALS; CHO CELLS; CRICETINAE; CYCLIC AMP; GTP-BINDING PROTEINS; GUANOSINE 5'-O-(3-THIOTRIPHOSPHATE); HUMANS; RECEPTORS, PURINERGIC P1; RECOMBINANT PROTEINS;

EID: 0031777856     PISSN: 0026895X     EISSN: None     Source Type: Journal    
DOI: None     Document Type: Article

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