Pharmacological analysis of G-protein activation mediated by guinea-pig recombinant 5-HT(1B) receptors in C6-glial cells: Similarities with the human 5-HT(1B) receptor

British Journal of Pharmacology

Volumn 123, Issue 1, 1998, Pages 51-62

  Pauwels, Petrus J ^a   Wurch, Thierry ^a   Palmier, Christiane ^a   Colpaert, Francis C ^a  

^a INSTITUT DE RECHERCHE PIERRE FABRE   (France)

Author keywords

35S GTP S binding response; Agonist inverse agonist; Guinea pig recombinant 5 HT(1B) receptor; Human 5 HT(1B) receptor; Rat C6 glial cell line

Indexed keywords

5 CARBAMOYLTRYPTAMINE; CP 122638; CYCLIC AMP; DIHYDROERGOTAMINE; FORSKOLIN; GUANINE NUCLEOTIDE BINDING PROTEIN; GUANOSINE 5' O (3 THIOTRIPHOSPHATE); KETANSERIN; LIGAND; METITEPINE; N [4 METHOXY 3 (4 METHYL 1 PIPERAZINYL)PHENYL] 2' METHYL 4' (5 METHYL 1,2,4 OXADIAZOL 3 YL)[1,1' BIPHENYL] 4 CARBOXAMIDE; NARATRIPTAN; RECOMBINANT RECEPTOR; RITANSERIN; RIZATRIPTAN; SEROTONIN 1B RECEPTOR; SP 224289; SUMATRIPTAN; UNCLASSIFIED DRUG; ZOLMITRIPTAN;

ANIMAL CELL; ARTICLE; BINDING AFFINITY; BINDING SITE; CONCENTRATION RESPONSE; CONTROLLED STUDY; DRUG POTENCY; GLIA CELL; GUINEA PIG; MEMBRANE BINDING; NONHUMAN; PRIORITY JOURNAL; RAT; RECEPTOR AFFINITY; SPECIES DIFFERENCE;

AMINO ACID SEQUENCE; ANIMALS; CELL LINE; CELL MEMBRANE; CLONING, MOLECULAR; CYCLIC AMP; GTP-BINDING PROTEINS; GUANOSINE 5'-O-(3-THIOTRIPHOSPHATE); GUINEA PIGS; HUMANS; MOLECULAR SEQUENCE DATA; NEUROGLIA; POLYMERASE CHAIN REACTION; RATS; RECEPTORS, SEROTONIN; RNA, MESSENGER;

EID: 0031964030     PISSN: 00071188     EISSN: None     Source Type: Journal    
DOI: 10.1038/sj.bjp.0701584     Document Type: Article

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