Mechanisms of agonism and inverse agonism at serotonin 5-HT(1A) receptors

Journal of Neurochemistry

Volumn 74, Issue 1, 2000, Pages 347-357

  McLoughlin, David J ^b   Strange, Philip G ^a  

^a UNIVERSITY OF READING   (United Kingdom)

^b The University   (United Kingdom)

Author keywords

35S GTP S binding; Agonist; Inverse agonist; Mechanisms of action; Serotonin 5 HT(1A) receptor

Indexed keywords

2 DIPROPYLAMINO 8 HYDROXYTETRALIN; 5 CARBAMOYLTRYPTAMINE; EMONAPRIDE; GUANINE NUCLEOTIDE BINDING PROTEIN; GUANOSINE 5' O (3 THIOTRIPHOSPHATE); METITEPINE; SEROTONIN; SEROTONIN 1A AGONIST; SEROTONIN 1A ANTAGONIST; SEROTONIN 1A RECEPTOR; SPIPERONE;

ANIMAL CELL; ARTICLE; CHO CELL; DRUG MECHANISM; DRUG POTENCY; DRUG RECEPTOR BINDING; NONHUMAN; PRIORITY JOURNAL; PROTEIN STABILITY; SEROTONINERGIC SYSTEM;

8-HYDROXY-2-(DI-N-PROPYLAMINO)TETRALIN; ANIMALS; CHO CELLS; CRICETINAE; GUANOSINE 5'-O-(3-THIOTRIPHOSPHATE); GUANOSINE DIPHOSPHATE; OSMOLAR CONCENTRATION; RECEPTORS, SEROTONIN; RECEPTORS, SEROTONIN, 5-HT1; SEROTONIN AGONISTS; SODIUM;

ANIMALIA; CRICETINAE; CRICETULUS GRISEUS;

EID: 0033983969     PISSN: 00223042     EISSN: None     Source Type: Journal    
DOI: 10.1046/j.1471-4159.2000.0740347.x     Document Type: Article

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