Binding profile of the novel 5-HT(1B/1D) receptor antagonist,[3H]GR 125,743, in guinea-pig brain: a comparison with [3H]5-carboxamidotryptamine

European Journal of Pharmacology

Volumn 327, Issue 2-3, 1997, Pages 247-256

  Audinot, Valérie ^a   Lochon, Sonia ^a   Newman Tancredi, Adrian ^a   Lavielle, Gilbert ^a   Millan, Mark J ^a  

^a INSTITUT DE RECHERCHES SERVIER   (France)

Author keywords

5 HT (5 hydroxytryptamine, serotonin); 5 HT(1D) receptor; 3H 5 CT; 3H GR 125,743; Ginea pig

Indexed keywords

5 CARBAMOYLTRYPTAMINE; DIHYDROERGOTAMINE; KETANSERIN; MESULERGINE; METERGOLINE; METHYSERGIDE; METITEPINE; N [4 METHOXY 3 (4 METHYL 1 PIPERAZINYL)PHENYL] 2' METHYL 4' (5 METHYL 1,2,4 OXADIAZOL 3 YL)[1,1' BIPHENYL] 4 CARBOXAMIDE; N [4 METHOXY 3 (4 METHYL 1 PIPERAZINYL)PHENYL] 3 METHYL 4 (4 PYRIDYL)BENZAMIDE; PROPRANOLOL; RITANSERIN; SEROTONIN; SEROTONIN 1B RECEPTOR; SEROTONIN 1D RECEPTOR; SEROTONIN ANTAGONIST; SUMATRIPTAN; UNCLASSIFIED DRUG;

ANIMAL CELL; ANIMAL TISSUE; ARTICLE; BINDING SITE; CATTLE; CONTROLLED STUDY; DRUG RECEPTOR BINDING; FRONTAL CORTEX; GUINEA PIG; NONHUMAN; PRIORITY JOURNAL; RECEPTOR AFFINITY;

ANIMALS; BENZAMIDES; BINDING, COMPETITIVE; BRAIN; GUINEA PIGS; KINETICS; PYRIDINES; SEROTONIN; SEROTONIN AGONISTS; SEROTONIN ANTAGONISTS;

EID: 0031009595     PISSN: 00142999     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0014-2999(97)89668-9     Document Type: Article

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