Drug-transporter mediated interactions between anthelminthic and antiretroviral drugs across the Caco-2 cell monolayers

BMC Pharmacology and Toxicology

Volumn 18, Issue 1, 2017, Pages

  Kigen, Gabriel ^a,b   Edwards, Geoffrey ^b  

^a MOI UNIVERSITY   (Kenya)

^b UNIVERSITY OF LIVERPOOL   (United Kingdom)

Author keywords

Antiparasitic; Antiretroviral; Caco 2 cell monolayers; Drug interactions; Drug transport; Intestinal epithelium; TEER

Indexed keywords

ANTHELMINTIC AGENT; ANTIRETROVIRUS AGENT; EFAVIRENZ; IVERMECTIN; LOPINAVIR; NEVIRAPINE; PRAZIQUANTEL; SAQUINAVIR;

APICAL MEMBRANE; APPARENT PERMEABILITY; ARTICLE; BASOLATERAL MEMBRANE; CACO-2 CELL LINE; CONTROLLED STUDY; DRUG EFFECT; DRUG PENETRATION; DRUG TRANSPORT; EFFLUX RATE CONSTANT; HIGH PERFORMANCE LIQUID CHROMATOGRAPHY; HUMAN; HUMAN CELL; IN VITRO STUDY; TRANSEPITHELIAL RESISTANCE; ACTIVE TRANSPORT; DRUG INTERACTION; METABOLISM;

ANTHELMINTICS; ANTI-RETROVIRAL AGENTS; BIOLOGICAL TRANSPORT, ACTIVE; CACO-2 CELLS; DRUG INTERACTIONS; HUMANS; IVERMECTIN; PRAZIQUANTEL;

EID: 85018252279     PISSN: None     EISSN: 20506511     Source Type: Journal    
DOI: 10.1186/s40360-017-0129-6     Document Type: Article

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