메뉴 건너뛰기




Volumn 157, Issue 1-2, 2008, Pages 117-122

Ketoconazole increases the plasma levels of ivermectin in sheep

Author keywords

Drug drug interaction; Ketoconazole; Macrocyclic lactone; P glycoprotein; Resistance; Sheep

Indexed keywords

DRUG METABOLITE; GLYCOPROTEIN P; IVERMECTIN; KETOCONAZOLE; LACTONE;

EID: 51249101705     PISSN: 03044017     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.vetpar.2008.06.017     Document Type: Article
Times cited : (50)

References (33)
  • 1
    • 0032860581 scopus 로고    scopus 로고
    • Enhanced absorption of pour-on ivermectin formulation in rats by co-administration of the multidrug-resistant-reversing agent verapamil
    • Alvinerie M., Dupuy J., Eeckhoutte C., and Sutra J.F. Enhanced absorption of pour-on ivermectin formulation in rats by co-administration of the multidrug-resistant-reversing agent verapamil. Parasitol. Res. 85 (1999) 920-922
    • (1999) Parasitol. Res. , vol.85 , pp. 920-922
    • Alvinerie, M.1    Dupuy, J.2    Eeckhoutte, C.3    Sutra, J.F.4
  • 2
    • 51249091474 scopus 로고    scopus 로고
    • Alvinerie, M., Tardieu, D., Sutra, J., D, Bojensen, G., Galtier, P., 1994. Metabolic profile of ivermectin in goats: an "in vivo" and "in vitro" evaluation (ed.) 1994. EAVPT International Congress, Edinburgh, Scotland. August 7-11, 1994.
    • Alvinerie, M., Tardieu, D., Sutra, J., D, Bojensen, G., Galtier, P., 1994. Metabolic profile of ivermectin in goats: an "in vivo" and "in vitro" evaluation (ed.) 1994. EAVPT International Congress, Edinburgh, Scotland. August 7-11, 1994.
  • 3
    • 33344474213 scopus 로고    scopus 로고
    • Modulation of the P-glycoprotein-mediated intestinal secretion of ivermectin: in vitro and in vivo assessments
    • Ballent M., Lifschitz A., Virkel G., Sallovitz J., and Lanusse C. Modulation of the P-glycoprotein-mediated intestinal secretion of ivermectin: in vitro and in vivo assessments. Drug Metab. Dispos. 34 (2006) 457-463
    • (2006) Drug Metab. Dispos. , vol.34 , pp. 457-463
    • Ballent, M.1    Lifschitz, A.2    Virkel, G.3    Sallovitz, J.4    Lanusse, C.5
  • 4
    • 34247591496 scopus 로고    scopus 로고
    • Involvement of P-glycoprotein on ivermectin kinetic behaviour in sheep: itraconazole-mediated changes on gastrointestinal disposition
    • Ballent M., Lifschitz A., Virkel G., Sallovitz J., and Lanusse C. Involvement of P-glycoprotein on ivermectin kinetic behaviour in sheep: itraconazole-mediated changes on gastrointestinal disposition. J. Vet. Pharmacol. Ther. 30 (2007) 242-248
    • (2007) J. Vet. Pharmacol. Ther. , vol.30 , pp. 242-248
    • Ballent, M.1    Lifschitz, A.2    Virkel, G.3    Sallovitz, J.4    Lanusse, C.5
  • 5
    • 0030430033 scopus 로고    scopus 로고
    • Cytochrome P450 isoform inhibitors as a tool for the investigation of metabolic reactions catalyzed by human liver microsomes
    • Bourrie M., Meunier V., Berger Y., and Fabre G. Cytochrome P450 isoform inhibitors as a tool for the investigation of metabolic reactions catalyzed by human liver microsomes. J. Pharmacol. Exp. Ther. 277 (1996) 321-332
    • (1996) J. Pharmacol. Exp. Ther. , vol.277 , pp. 321-332
    • Bourrie, M.1    Meunier, V.2    Berger, Y.3    Fabre, G.4
  • 6
    • 0023550895 scopus 로고
    • Comparative in vivo and in vitro metabolism of ivermectin in steers, sheep, swine, and rat
    • Chiu S.H., Taub R., Sestokas E., Lu A.Y., and Jacob T.A. Comparative in vivo and in vitro metabolism of ivermectin in steers, sheep, swine, and rat. Drug Metab. Rev. 18 (1987) 289-302
    • (1987) Drug Metab. Rev. , vol.18 , pp. 289-302
    • Chiu, S.H.1    Taub, R.2    Sestokas, E.3    Lu, A.Y.4    Jacob, T.A.5
  • 8
    • 33644898140 scopus 로고    scopus 로고
    • Effects of cytochrome P450 3A modulators ketoconazole and carbamazepine on quetiapine pharmacokinetics
    • Grimm S.W., Richtand N.M., Winter H.R., Stams K.R., and Reele S.B. Effects of cytochrome P450 3A modulators ketoconazole and carbamazepine on quetiapine pharmacokinetics. Br. J. Clin. Pharmacol. 61 (2006) 58-69
    • (2006) Br. J. Clin. Pharmacol. , vol.61 , pp. 58-69
    • Grimm, S.W.1    Richtand, N.M.2    Winter, H.R.3    Stams, K.R.4    Reele, S.B.5
  • 9
    • 34848924630 scopus 로고    scopus 로고
    • Multiple oral dosing of ketoconazole increases dog exposure to ivermectin
    • Hugnet C., Lespine A., and Alvinerie M. Multiple oral dosing of ketoconazole increases dog exposure to ivermectin. J. Pharm. Pharm. Sci. 10 (2007) 311-318
    • (2007) J. Pharm. Pharm. Sci. , vol.10 , pp. 311-318
    • Hugnet, C.1    Lespine, A.2    Alvinerie, M.3
  • 10
    • 19444367783 scopus 로고    scopus 로고
    • In vivo effects of cyclosporin A and ketoconazole on the pharmacokinetics of representative substrates for P-glycoprotein and cytochrome P450 (CYP) 3A in rats
    • Kageyama M., Namiki H., Fukushima H., Ito Y., Shibata N., and Takada K. In vivo effects of cyclosporin A and ketoconazole on the pharmacokinetics of representative substrates for P-glycoprotein and cytochrome P450 (CYP) 3A in rats. Biol. Pharm. Bull. 28 (2005) 316-322
    • (2005) Biol. Pharm. Bull. , vol.28 , pp. 316-322
    • Kageyama, M.1    Namiki, H.2    Fukushima, H.3    Ito, Y.4    Shibata, N.5    Takada, K.6
  • 11
    • 4444375921 scopus 로고    scopus 로고
    • Drug resistance in nematodes of veterinary importance: a status report
    • Kaplan R.M. Drug resistance in nematodes of veterinary importance: a status report. Trends Parasitol. 20 (2004) 477-481
    • (2004) Trends Parasitol. , vol.20 , pp. 477-481
    • Kaplan, R.M.1
  • 13
    • 8344226085 scopus 로고    scopus 로고
    • Multiple oral dosing of ketoconazole influences pharmacokinetics of quinidine after intravenous and oral administration in beagle dogs
    • Kuroha M., Shirai Y., and Shimoda M. Multiple oral dosing of ketoconazole influences pharmacokinetics of quinidine after intravenous and oral administration in beagle dogs. J. Vet. Pharmacol. Ther. 27 (2004) 355-359
    • (2004) J. Vet. Pharmacol. Ther. , vol.27 , pp. 355-359
    • Kuroha, M.1    Shirai, Y.2    Shimoda, M.3
  • 15
    • 0036263229 scopus 로고    scopus 로고
    • Intestinal secretion is a major route for parent ivermectin elimination in the rat
    • Laffont C.M., Toutain P.L., Alvinerie M., and Bousquet-Melou A. Intestinal secretion is a major route for parent ivermectin elimination in the rat. Drug Metab. Dispos. 30 (2002) 626-630
    • (2002) Drug Metab. Dispos. , vol.30 , pp. 626-630
    • Laffont, C.M.1    Toutain, P.L.2    Alvinerie, M.3    Bousquet-Melou, A.4
  • 18
    • 0026595179 scopus 로고
    • Effects of imidazole derivatives on cytochromes P450 from human hepatocytes in primary culture
    • Maurice M., Pichard L., Daujat M., Fabre I., Joyeux H., Domergue J., and Maurel P. Effects of imidazole derivatives on cytochromes P450 from human hepatocytes in primary culture. FASEB J. 6 (1992) 752-758
    • (1992) FASEB J. , vol.6 , pp. 752-758
    • Maurice, M.1    Pichard, L.2    Daujat, M.3    Fabre, I.4    Joyeux, H.5    Domergue, J.6    Maurel, P.7
  • 20
    • 0035164622 scopus 로고    scopus 로고
    • Ivermectin sensitivity in collies is associated with a deletion mutation of the mdr1 gene
    • Mealey K.L., Bentjen S.A., Gay J.M., and Cantor G.H. Ivermectin sensitivity in collies is associated with a deletion mutation of the mdr1 gene. Pharmacogenetics 11 (2001) 727-733
    • (2001) Pharmacogenetics , vol.11 , pp. 727-733
    • Mealey, K.L.1    Bentjen, S.A.2    Gay, J.M.3    Cantor, G.H.4
  • 21
    • 0442298029 scopus 로고    scopus 로고
    • Influence of verapamil on the pharmacokinetics of the antiparasitic drugs ivermectin and moxidectin in sheep
    • Molento M.B., Lifschitz A., Sallovitz J., Lanusse C., and Prichard R. Influence of verapamil on the pharmacokinetics of the antiparasitic drugs ivermectin and moxidectin in sheep. Parasitol. Res. 92 (2004) 121-127
    • (2004) Parasitol. Res. , vol.92 , pp. 121-127
    • Molento, M.B.1    Lifschitz, A.2    Sallovitz, J.3    Lanusse, C.4    Prichard, R.5
  • 23
    • 33847343857 scopus 로고    scopus 로고
    • Ogasawara, A., Kume, T., Kazama, E., 2007. Effect of oral ketoconazole on intestinal first-pass effect of midazolam and fexofenadine in cynomolgus monkeys. Drug Metab. Dispos. 35, 410-418.
    • Ogasawara, A., Kume, T., Kazama, E., 2007. Effect of oral ketoconazole on intestinal first-pass effect of midazolam and fexofenadine in cynomolgus monkeys. Drug Metab. Dispos. 35, 410-418.
  • 24
    • 0019974468 scopus 로고
    • Noncompartmental determination of the steady-state volume of distribution for any mode of administration
    • Perrier D., and Mayersohn M. Noncompartmental determination of the steady-state volume of distribution for any mode of administration. J. Pharm. Sci. 71 (1982) 372-373
    • (1982) J. Pharm. Sci. , vol.71 , pp. 372-373
    • Perrier, D.1    Mayersohn, M.2
  • 26
    • 34347399591 scopus 로고    scopus 로고
    • ABC transporters and beta-tubulin in macrocyclic lactone resistance: prospects for marker development
    • Prichard R.K., and Roulet A. ABC transporters and beta-tubulin in macrocyclic lactone resistance: prospects for marker development. Parasitology 134 (2007) 1123-1132
    • (2007) Parasitology , vol.134 , pp. 1123-1132
    • Prichard, R.K.1    Roulet, A.2
  • 27
    • 23844442993 scopus 로고    scopus 로고
    • Ketoconazole increases plasma concentrations of antimalarial mefloquine in healthy human volunteers
    • Ridtitid W., Wongnawa M., Mahatthanatrakul W., Raungsri N., and Sunbhanich M. Ketoconazole increases plasma concentrations of antimalarial mefloquine in healthy human volunteers. J. Clin. Pharm. Ther. 30 (2005) 285-290
    • (2005) J. Clin. Pharm. Ther. , vol.30 , pp. 285-290
    • Ridtitid, W.1    Wongnawa, M.2    Mahatthanatrakul, W.3    Raungsri, N.4    Sunbhanich, M.5
  • 29
    • 0032789210 scopus 로고    scopus 로고
    • Haemonchus contortus: sequence heterogeneity of internucleotide binding domains from P-glycoproteins
    • Sangster N.C., Bannan S.C., Weiss A.S., Nulf S.C., Klein R.D., and Geary T.G. Haemonchus contortus: sequence heterogeneity of internucleotide binding domains from P-glycoproteins. Exp. Parasitol. 91 (1999) 250-257
    • (1999) Exp. Parasitol. , vol.91 , pp. 250-257
    • Sangster, N.C.1    Bannan, S.C.2    Weiss, A.S.3    Nulf, S.C.4    Klein, R.D.5    Geary, T.G.6
  • 31
    • 0842347428 scopus 로고    scopus 로고
    • Development of an in vivo preclinical screen model to estimate absorption and first-pass hepatic extraction of xenobiotics. II. Use of ketoconazole to identify P-glycoprotein/CYP3A-limited bioavailability in the monkey
    • Ward K.W., Stelman G.J., Morgan J.A., Zeigler K.S., Azzarano L.M., Kehler J.R., McSurdy-Freed J.E., Proksch J.W., and Smith B.R. Development of an in vivo preclinical screen model to estimate absorption and first-pass hepatic extraction of xenobiotics. II. Use of ketoconazole to identify P-glycoprotein/CYP3A-limited bioavailability in the monkey. Drug Metab. Dispos. 32 (2004) 172-177
    • (2004) Drug Metab. Dispos. , vol.32 , pp. 172-177
    • Ward, K.W.1    Stelman, G.J.2    Morgan, J.A.3    Zeigler, K.S.4    Azzarano, L.M.5    Kehler, J.R.6    McSurdy-Freed, J.E.7    Proksch, J.W.8    Smith, B.R.9


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.