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Volumn 38, Issue , 2017, Pages 8-16

Cyclotides as drug design scaffolds

Author keywords

[No Author keywords available]

Indexed keywords

CYCLOTIDE; MOLECULAR SCAFFOLD;

EID: 85013986653     PISSN: 13675931     EISSN: 18790402     Source Type: Journal    
DOI: 10.1016/j.cbpa.2017.01.018     Document Type: Review
Times cited : (102)

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    • Design, synthesis, structural and functional characterization of novel melanocortin agonists based on the cyclotide kalata B1
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    • Design of a cyclotide antagonist of neuropilin-1 and -2 that potently inhibits endothelial cell migration
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    • Recombinant expression and phenotypic screening of a bioactive cyclotide against α-synuclein-induced cytotoxicity in baker's yeast
    • The first paper to report the recombinant expression of cyclotides inside live yeast cells.
    • 64• Jagadish, K., Gould, A., Borra, R., Majumder, S., Mushtaq, Z., Shekhtman, A., Camarero, J.A., Recombinant expression and phenotypic screening of a bioactive cyclotide against α-synuclein-induced cytotoxicity in baker's yeast. Angew Chem Int Ed 54 (2015), 8390–8394 The first paper to report the recombinant expression of cyclotides inside live yeast cells.
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