Probing biased/partial agonism at the G protein-coupled A2B adenosine receptor

Biochemical Pharmacology

Volumn 90, Issue 3, 2014, Pages 297-306

  Gao, Zhan Guo ^a   Balasubramanian, Ramachandran ^a   Kiselev, Evgeny ^a   Wei, Qiang ^a   Jacobson, Kenneth A ^a  

^a NATIONAL INSTITUTE OF DIABETES AND DIGESTIVE AND KIDNEY DISEASES   (United States)

Author keywords

Adenosine receptor; Arrestin; Calcium; Cyclic AMP; GPCR; Purines

Indexed keywords

2 ANILINOADENOSINE; 2 [4 (2 CARBOXYETHYL)PHENETHYLAMINO]ADENOSINE 5' (N ETHYLCARBOXAMIDE); ADENOSINE 5' (N ETHYLCARBOXAMIDE); ADENOSINE A2B RECEPTOR; ADENOSINE RECEPTOR STIMULATING AGENT; BAY 606583; BETA ARRESTIN; CALCIUM; CYCLIC AMP; G PROTEIN COUPLED RECEPTOR; INSULIN; LUF 5833; MITOGEN ACTIVATED PROTEIN KINASE 1; MITOGEN ACTIVATED PROTEIN KINASE 3; MRS 3534; MRS 3997; MRS 5911; SMALL INTERFERING RNA; UNCLASSIFIED DRUG;

ANIMAL CELL; ARTICLE; BLADDER CANCER CELL LINE; CALCIUM MOBILIZATION; CONTROLLED STUDY; DRUG POTENCY; DRUG RECEPTOR BINDING; GENE OVEREXPRESSION; GENE SILENCING; HEK293 CELL LINE; HUMAN; HUMAN CELL; INSULIN RELEASE; MOUSE; NONHUMAN; PANCREAS ISLET BETA CELL; PRIORITY JOURNAL; PROTEIN EXPRESSION; PROTEIN PHOSPHORYLATION; QUANTITATIVE ANALYSIS;

EID: 84903887192     PISSN: 00062952     EISSN: 18732968     Source Type: Journal    
DOI: 10.1016/j.bcp.2014.05.008     Document Type: Article

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